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Joseph Pontillo, Ph.D.

Affiliations: 
2001 University of California, Los Angeles, Los Angeles, CA 
Area:
Biologically Active Compounds
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"Joseph Pontillo"
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Michael E. Jung grad student 2001 UCLA
 (Approaches toward the synthesis of two families of cytotoxic natural products: The Otteliones and the Sclerophytins.)

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Publications

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Chen C, Wu D, Guo Z, et al. (2008) Discovery of sodium R-(+)-4-{2-[5-(2-Fluoro-3-methoxyphenyl)-3-(2-fluoro-6- [trifluoromethyl]-benzyl)-4-methyl-2,6-dioxo-3,6-dihydro-2H-pyrimidin-1-yl] -1-phenylethylamino}butyrate (elagolix), a potent and orally available nonpeptide antagonist of the human gonadotropin-releasing hormone receptor Journal of Medicinal Chemistry. 51: 7478-7485
Pontillo J, Wu D, Ching B, et al. (2008) Synthesis and structure-activity relationships of selective norepinephrine reuptake inhibitors (sNRI) with improved pharmaceutical characteristics. Bioorganic & Medicinal Chemistry Letters. 18: 6151-5
Wu D, Pontillo J, Ching B, et al. (2008) Discovery of a potent, selective, and less flexible selective norepinephrine reuptake inhibitor (sNRI). Bioorganic & Medicinal Chemistry Letters. 18: 4224-7
Chen C, Chen Y, Pontillo J, et al. (2008) Potent and orally bioavailable zwitterion GnRH antagonists with low CYP3A4 inhibitory activity Bioorganic and Medicinal Chemistry Letters. 18: 3301-3305
Tran JA, Arellano M, Fleck BA, et al. (2008) Studies on the structure-activity relationship of the basic amine of phenylpiperazines as melanocortin-4 receptor antagonists Medicinal Chemistry. 4: 67-74
Tran JA, Tucci FC, Jiang W, et al. (2007) Pyrrolidinones as orally bioavailable antagonists of the human melanocortin-4 receptor with anti-cachectic activity. Bioorganic & Medicinal Chemistry. 15: 5166-76
Chen CW, Tran JA, Jiang W, et al. (2006) Propionylpiperazines as human melanocortin-4 receptor ligands. Bioorganic & Medicinal Chemistry Letters. 16: 4800-3
Hudson S, Kiankarimi M, Rowbottom MW, et al. (2006) Synthesis and structure-activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 2. Bioorganic & Medicinal Chemistry Letters. 16: 4922-30
Jiang W, Tucci FC, Chen CW, et al. (2006) Arylpropionylpiperazines as antagonists of the human melanocortin-4 receptor. Bioorganic & Medicinal Chemistry Letters. 16: 4674-8
Dyck B, Zhao L, Tamiya J, et al. (2006) Substituted chromones and quinolones as potent melanin-concentrating hormone receptor 1 antagonists. Bioorganic & Medicinal Chemistry Letters. 16: 4237-42
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