Hiroshi Hiasa
Affiliations: | University of Minnesota, Twin Cities, Minneapolis, MN |
Area:
Pharmacology, BiochemistryGoogle:
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Publications
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| Aguirre AL, Chheda PR, Lentz SRC, et al. (2020) Identification of an ethyl 5,6-dihydropyrazolo[1,5-c]quinazoline-1-carboxylate as a catalytic inhibitor of DNA gyrase. Bioorganic & Medicinal Chemistry. 115439 |
| Fan BZ, Hiasa H, Lv W, et al. (2020) Design, synthesis and structure-activity relationships of novel 15-membered macrolides: Quinolone/quinoline-containing sidechains tethered to the C-6 position of azithromycin acylides. European Journal of Medicinal Chemistry. 193: 112222 |
| Delgado JL, Lentz SRC, Kulkarni CA, et al. (2019) Probing structural requirements for human topoisomerase I inhibition by a novel N1-Biphenyl fluoroquinolone. European Journal of Medicinal Chemistry. 172: 109-130 |
| Lentz SRC, Chheda PR, Oppegard LM, et al. (2019) The C7-aminomethylpyrrolidine group rescues the activity of a thio-fluoroquinolone. Biochimie. 160: 24-27 |
| Ostrer L, Khodursky RF, Johnson JR, et al. (2018) Analysis of Mutational Patterns in Quinolone Resistance-Determining Regions of GyrA and ParC of Clinical Isolates. International Journal of Antimicrobial Agents |
| Oppegard LM, Delgado JL, Kulkarni CA, et al. (2018) Novel N-1 substituted fluoroquinolones inhibit human topoisomerase I activity and exhibit anti-proliferative activity. Investigational New Drugs |
| Towle TR, Kulkarni CA, Oppegard LM, et al. (2018) Design, synthesis, and evaluation of novel N-1 fluoroquinolone derivatives: Probing for binding contact with the active site tyrosine of gyrase. Bioorganic & Medicinal Chemistry Letters |
| Delgado JL, Hsieh CM, Chan NL, et al. (2018) Topoisomerases as anticancer targets. The Biochemical Journal. 475: 373-398 |
| Hiasa H. (2018) DNA Topoisomerases as Targets for Antibacterial Agents. Methods in Molecular Biology (Clifton, N.J.). 1703: 47-62 |
| Malik M, Mustaev A, Schwanz HA, et al. (2016) Suppression of gyrase-mediated resistance by C7 aryl fluoroquinolones. Nucleic Acids Research |