Michael Zengerle
Affiliations: | Michael Zengerle |
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| Klein VG, Townsend CE, Testa A, et al. (2020) Understanding and Improving the Membrane Permeability of VH032-Based PROTACs. Acs Medicinal Chemistry Letters. 11: 1732-1738 |
| Runcie AC, Zengerle M, Chan KH, et al. (2018) Optimization of a "bump-and-hole" approach to allele-selective BET bromodomain inhibition. Chemical Science. 9: 2452-2468 |
| Chan KH, Zengerle M, Testa A, et al. (2017) Impact of target warhead and linkage vector on inducing protein degradation: comparison of Bromodomain and Extra-Terminal (BET) degraders derived from triazolodiazepine (JQ1) and tetrahydroquinoline (I-BET726) BET inhibitor scaffolds. Journal of Medicinal Chemistry |
| Gadd MS, Testa A, Lucas X, et al. (2017) Structural basis of PROTAC cooperative recognition for selective protein degradation. Nature Chemical Biology |
| Runcie AC, Chan KH, Zengerle M, et al. (2016) Chemical genetics approaches for selective intervention in epigenetics. Current Opinion in Chemical Biology. 33: 186-194 |
| Baud MGJ, Lin-Shiao E, Zengerle M, et al. (2016) New Synthetic Routes to Triazolo-benzodiazepine Analogues: Expanding the Scope of the Bump-and-Hole Approach for Selective Bromo and Extra-Terminal (BET) Bromodomain Inhibition. Journal of Medicinal Chemistry. 59: 1492-1500 |
| Zengerle M, Chan KH, Ciulli A. (2015) Selective Small Molecule Induced Degradation of the BET Bromodomain Protein BRD4. Acs Chemical Biology |
| Baud MG, Lin-Shiao E, Cardote T, et al. (2014) Chemical biology. A bump-and-hole approach to engineer controlled selectivity of BET bromodomain chemical probes. Science (New York, N.Y.). 346: 638-41 |
| Bierwisch A, Zengerle M, Thiermann H, et al. (2014) Detoxification of alkyl methylphosphonofluoridates by an oxime-substituted β-cyclodextrin--an in vitro structure-activity study. Toxicology Letters. 224: 209-14 |
| Brandhuber F, Zengerle M, Porwol L, et al. (2012) Detoxification of tabun at physiological pH mediated by substituted β-cyclodextrin and glucose derivatives containing oxime groups. Toxicology. 302: 163-71 |