Mauro Mileni, Ph.D.
Affiliations: | 2006-2011 | Scripps Research Institute | |
| 2011-2013 | Receptos | ||
| 2014- | Abilita Bio |
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Publications
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| Chrencik JE, Roth CB, Terakado M, et al. (2015) Crystal Structure of Antagonist Bound Human Lysophosphatidic Acid Receptor 1. Cell. 161: 1633-43 |
| Skjevik AA, Mileni M, Baumann A, et al. (2014) The N-terminal sequence of tyrosine hydroxylase is a conformationally versatile motif that binds 14-3-3 proteins and membranes. Journal of Molecular Biology. 426: 150-68 |
| Wu H, Wacker D, Mileni M, et al. (2012) Structure of the human κ-opioid receptor in complex with JDTic. Nature. 485: 327-32 |
| Miller MT, Mileni M, Comoletti D, et al. (2011) The crystal structure of the α-neurexin-1 extracellular region reveals a hinge point for mediating synaptic adhesion and function. Structure (London, England : 1993). 19: 767-78 |
| Ezzili C, Mileni M, McGlinchey N, et al. (2011) Reversible competitive α-ketoheterocycle inhibitors of fatty acid amide hydrolase containing additional conformational constraints in the acyl side chain: orally active, long-acting analgesics. Journal of Medicinal Chemistry. 54: 2805-22 |
| Baksh MM, Kussrow AK, Mileni M, et al. (2011) Label-free quantification of membrane-ligand interactions using backscattering interferometry. Nature Biotechnology. 29: 357-60 |
| Mileni M, Garfunkle J, Ezzili C, et al. (2011) Fluoride-mediated capture of a noncovalent bound state of a reversible covalent enzyme inhibitor: X-ray crystallographic analysis of an exceptionally potent α-ketoheterocycle inhibitor of fatty acid amide hydrolase. Journal of the American Chemical Society. 133: 4092-100 |
| Lodola A, Capoferri L, Rivara S, et al. (2011) Understanding the role of carbamate reactivity in fatty acid amide hydrolase inhibition by QM/MM mechanistic modelling. Chemical Communications (Cambridge, England). 47: 2517-9 |
| Ezzili C, Mileni M, McGlinchey N, et al. (2011) alpha-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Containing Additional Conformational Contraints in the Acyl Side Chain Journal of Medicinal Chemistry. 54: 2805-2822 |
| Mileni M, Kamtekar S, Wood DC, et al. (2010) Crystal structure of fatty acid amide hydrolase bound to the carbamate inhibitor URB597: discovery of a deacylating water molecule and insight into enzyme inactivation. Journal of Molecular Biology. 400: 743-54 |