| Year |
Citation |
Score |
| 2019 |
Khodair AI, Awad MK, Gesson JP, Elshaier YAMM. New N-ribosides and N-mannosides of rhodanine derivatives with anticancer activity on leukemia cell line: Design, synthesis, DFT and molecular modelling studies. Carbohydrate Research. 487: 107894. PMID 31865252 DOI: 10.1016/J.Carres.2019.107894 |
0.341 |
|
| 2011 |
Khodair AI, Gesson JP. A new approach for the N- and S-galactosylation of 5-arylidene-2-thioxo-4-thiazolidinones. Carbohydrate Research. 346: 2831-7. PMID 22088884 DOI: 10.1016/J.Carres.2011.09.035 |
0.362 |
|
| 2010 |
Fonteneau N, Martin P, Mondon M, Ficheux H, Gesson J. ChemInform Abstract: Synthesis of Quinone and Xanthone Analogues of Rhein. Cheminform. 33: no-no. DOI: 10.1002/CHIN.200207058 |
0.317 |
|
| 2010 |
PAPOT S, COMBAUD D, GESSON J. ChemInform Abstract: A New Spacer Group Derived from Arylmalonaldehydes for Glucuronylated Prodrugs. Cheminform. 30: no-no. DOI: 10.1002/CHIN.199902251 |
0.597 |
|
| 2010 |
GESSON J, MONDON M, POKROVSKA N. ChemInform Abstract: Synthesis of Fused Aromatic [1,3]Dioxoles from 2-Hydroxymethylphenols. Cheminform. 29: no-no. DOI: 10.1002/CHIN.199813108 |
0.301 |
|
| 2009 |
Charrier C, Clarhaut J, Gesson JP, Estiu G, Wiest O, Roche J, Bertrand P. Synthesis and modeling of new benzofuranone histone deacetylase inhibitors that stimulate tumor suppressor gene expression. Journal of Medicinal Chemistry. 52: 3112-5. PMID 19385600 DOI: 10.1021/Jm9002439 |
0.327 |
|
| 2009 |
Charrier C, Roche J, Gesson J, Bertrand P. Biological activities of substituted trichostatic acid derivatives Journal of Chemical Sciences. 121: 471-479. DOI: 10.1007/S12039-009-0056-1 |
0.379 |
|
| 2008 |
Thomas M, Clarhaut J, Tranoy-Opalinski I, Gesson JP, Roche J, Papot S. Synthesis and biological evaluation of glucuronide prodrugs of the histone deacetylase inhibitor CI-994 for application in selective cancer chemotherapy. Bioorganic & Medicinal Chemistry. 16: 8109-16. PMID 18692397 DOI: 10.1016/J.Bmc.2008.07.048 |
0.615 |
|
| 2008 |
Cantet AC, Carreyre H, Gesson JP, Jouannetaud MP, Renoux B. Gem-difluorination of aminoalkynes via highly reactive dicationic species in superacid HF-SbF5: application to the efficient synthesis of difluorinated cinchona alkaloid derivatives. The Journal of Organic Chemistry. 73: 2875-8. PMID 18315004 DOI: 10.1021/Jo702441P |
0.435 |
|
| 2007 |
Charrier C, Roche J, Gesson JP, Bertrand P. Antiproliferative activities of a library of hybrids between indanones and HDAC inhibitor SAHA and MS-275 analogues. Bioorganic & Medicinal Chemistry Letters. 17: 6142-6. PMID 17897824 DOI: 10.1016/J.Bmcl.2007.09.041 |
0.377 |
|
| 2007 |
Loudni L, Roche J, Potiron V, Clarhaut J, Bachmann C, Gesson JP, Tranoy-Opalinski I. Design, synthesis and biological evaluation of 1,4-benzodiazepine-2,5-dione-based HDAC inhibitors. Bioorganic & Medicinal Chemistry Letters. 17: 4819-23. PMID 17624773 DOI: 10.1016/J.Bmcl.2007.06.067 |
0.363 |
|
| 2007 |
Thomas M, Gesson JP, Papot S. First O-glycosylation of hydroxamic acids. The Journal of Organic Chemistry. 72: 4262-4. PMID 17465568 DOI: 10.1021/Jo0701839 |
0.638 |
|
| 2007 |
Thomas M, Rivault F, Tranoy-Opalinski I, Roche J, Gesson JP, Papot S. Synthesis and biological evaluation of the suberoylanilide hydroxamic acid (SAHA) beta-glucuronide and beta-galactoside for application in selective prodrug chemotherapy. Bioorganic & Medicinal Chemistry Letters. 17: 983-6. PMID 17157009 DOI: 10.1016/J.Bmcl.2006.11.042 |
0.623 |
|
| 2007 |
Papot S, Thomas M, Gesson J. Efficient Regio- and Stereoselective Synthesis of 1-β-O-Glucuronyl Carbamates and Carbonates from Unprotected 1,2,3,4-Hydroxyl Glucuronates Synlett. 2007: 1966-1968. DOI: 10.1055/S-2007-984534 |
0.623 |
|
| 2007 |
Cantet A, Gesson J, Renoux B, Jouannetaud M. A New Synthesis of Trifluorinated Compounds via 1,1-Dichloro-1-alkenes in Superacid. Cheminform. 38. DOI: 10.1016/J.Tetlet.2007.05.137 |
0.42 |
|
| 2007 |
Thomas M, Gesson J, Papot S. Efficient Regio- and Stereoselective Synthesis of 1-β-O-Glucuronyl Carbamates and Carbonates from Unprotected 1,2,3,4-Hydroxyl Glucuronates. Cheminform. 38. DOI: 10.1002/chin.200750198 |
0.596 |
|
| 2006 |
Charrier C, Bertrand P, Gesson JP, Roche J. Synthesis of rigid trichostatin A analogs as HDAC inhibitors. Bioorganic & Medicinal Chemistry Letters. 16: 5339-44. PMID 16904890 DOI: 10.1016/J.Bmcl.2006.07.080 |
0.408 |
|
| 2006 |
Faveau C, Mondon M, Gesson J, Mahnke T, Gebhardt S, Koert U. Synthetic studies on a phenyl-laulimalide analogue Tetrahedron Letters. 47: 8305-8308. DOI: 10.1016/J.Tetlet.2006.09.104 |
0.338 |
|
| 2006 |
Fernandes A, Marrot J, Gesson J, Papot S. A New Simple and Convenient Method for the Synthesis of Substituted 2,6,9-Trioxabicyclo[3.3.1]-nona-3,7-dienes from Arylmalondialdehydes. Cheminform. 37. DOI: 10.1016/J.Tetlet.2006.06.043 |
0.661 |
|
| 2006 |
Fernandes A, Marrot J, Gesson J, Papot S. A new simple and convenient method for the synthesis of substituted 2,6,9-trioxabicyclo[3.3.1]-nona-3,7-dienes from arylmalondialdehydes Tetrahedron Letters. 47: 5961-5964. DOI: 10.1016/J.TETLET.2006.06.043 |
0.626 |
|
| 2005 |
Combaud D, Thomas M, Papot S, Gesson J. Synthesis and Evaluation of p-Nitrophenylβ-D-Glucopyranosiduronic Analogues as New Triggers for β-Glucuronidase Mediated Prodrug Mono- Therapy Letters in Drug Design & Discovery. 2: 631-637. DOI: 10.2174/157018005774717271 |
0.61 |
|
| 2005 |
Quintard D, Bertrand P, Bachmann C, Gesson J. Synthesis and Conformational Analysis of Macrocycles Related to 10-Oxa-epothilone. Cheminform. 36. DOI: 10.1002/Ejoc.200400212 |
0.403 |
|
| 2004 |
Rivault F, Tranoy-Opalinski I, Gesson JP. A new linker for glucuronylated anticancer prodrugs. Bioorganic & Medicinal Chemistry. 12: 675-82. PMID 14759728 DOI: 10.1016/J.Bmc.2003.11.026 |
0.338 |
|
| 2003 |
Khodair AI, Al-Masoudi NA, Gesson JP. A new approach to the synthesis of benzothiazole, benzoxazole, and pyridine nucleosides as potential antitumor agents. Nucleosides, Nucleotides & Nucleic Acids. 22: 2061-76. PMID 14680028 DOI: 10.1081/Ncn-120026407 |
0.366 |
|
| 2003 |
Bouazza F, Renoux B, Bachmann C, Gesson JP. Total synthesis and conformational analysis of the antifungal agent (-)-PF1163B. Organic Letters. 5: 4049-52. PMID 14572246 DOI: 10.1021/Ol035309C |
0.423 |
|
| 2003 |
Papot S, Tranoy I, Tillequin F, Florent JC, Gesson JP. Design of selectively activated anticancer prodrugs: elimination and cyclization strategies. Current Medicinal Chemistry. Anti-Cancer Agents. 2: 155-85. PMID 12678742 DOI: 10.2174/1568011023354173 |
0.58 |
|
| 2003 |
Quintard D, Bertrand P, Vielle S, Raimbaud E, Renard P, Pfeiffer B, Gesson J. Enantioselective synthesis of 2,3-dehydro-3-desoxy-10-oxa epothilone D Synlett. 2003: 2033-2036. DOI: 10.1055/S-2003-42034 |
0.41 |
|
| 2002 |
Papot S, Rivault F, Tranoy I, Gesson J. Synthesis and β-Glucuronidase Mediated Cleavage of an Alcohol Prodrug Incorporating a Double Spacer Moiety Synlett. 2002: 0164-0166. DOI: 10.1055/S-2002-19327 |
0.599 |
|
| 2002 |
Vielle S, Raimbaud E, Bertrand P, Quintard D, Renard P, Pfeiffer B, Gesson J. Design and synthesis of tubulin ligands based on epothilones: a preliminary study Tetrahedron Letters. 43: 9213-9216. DOI: 10.1016/S0040-4039(02)02242-6 |
0.306 |
|
| 2001 |
Azoulay M, Chalard F, Gesson JP, Florent JC, Monneret C. 2-Nitro and 4-nitro-quinone-methides are not irreversible inhibitors of bovine beta-glucuronidase. Carbohydrate Research. 332: 151-6. PMID 11434372 DOI: 10.1016/S0008-6215(01)00083-0 |
0.371 |
|
| 2001 |
Papot S, Combaud D, Bosslet K, Gerken M, Czech J, Gesson JP. Synthesis and cytotoxic activity of a glucuronylated prodrug of nornitrogen mustard. Bioorganic & Medicinal Chemistry Letters. 10: 1835-7. PMID 10969980 DOI: 10.1016/S0960-894X(00)00353-X |
0.658 |
|
| 2001 |
Forget-Champagne D, Mondon M, Fonteneau N, Gesson J. Selective cross-metathesis of 2-allylphenols with styrenes Tetrahedron Letters. 42: 7229-7231. DOI: 10.1016/S0040-4039(01)01376-4 |
0.313 |
|
| 2001 |
Fonteneau N, Martin P, Mondon M, Ficheux H, Gesson J. Synthesis of quinone and xanthone analogs of rhein Tetrahedron. 57: 9131-9135. DOI: 10.1016/S0040-4020(01)00918-8 |
0.419 |
|
| 2000 |
Rodier S, Le Huérou Y, Renoux B, Doyon J, Renard P, Pierré A, Gesson JP, Grée R. Synthesis and cytotoxic activity of acetogenin analogues Bioorganic and Medicinal Chemistry Letters. 10: 1373-1375. PMID 10890167 DOI: 10.1016/S0960-894X(00)00236-5 |
0.387 |
|
| 2000 |
Gesson J, Mondon M, Pokrovska N. Synthesis of Fused Aromatic [1,3]Dioxoles from 2-Hydroxymethylphenols Synlett. 12: 1395-1396. DOI: 10.1055/S-1997-1037 |
0.406 |
|
| 1999 |
Papot S, Combaud D, Gesson JP. A new spacer group derived from arylmalonaldehydes for glucuronylated prodrugs. Bioorganic & Medicinal Chemistry Letters. 8: 2545-8. PMID 9873577 DOI: 10.1016/S0960-894X(98)00454-5 |
0.65 |
|
| 1999 |
Bertrand P, El Sukkari H, Gesson J, Renoux B. Bis-Tetrahydrofurans from Carbohydrates via Iodoetherification and Iodine Substitution Synthesis. 1999: 330-335. DOI: 10.1055/S-1999-3392 |
0.373 |
|
| 1999 |
Sukkari HE, Renoux B, Bertrand P, Gesson J. Synthesis of Bis-THF Compounds from D-Glucose Journal of Chemical Research-S. 482-483. DOI: 10.1039/A902756D |
0.301 |
|
| 1999 |
Mondon M, Boeker N, Gesson J. Cycloaddition of Ketene Acetals with 4-Bromo-6-spiroepoxycyclohexa-2,4-dienone Journal of Chemical Research-S. 484-485. DOI: 10.1039/A902751C |
0.32 |
|
| 1999 |
Bonnarme V, Mondon M, Gesson J, Cousson A. Cyclodimerization and Diels–Alder reaction of a spiroepoxycyclohexadienone with an o-quinodimethane structure Chemical Communications. 1143-1144. DOI: 10.1039/A901914F |
0.304 |
|
| 1999 |
Papot S, Bachmann C, Combaud D, Gesson J. Study of biscarbamates derived from 2-aminobenzylamines as models for alcohol prodrugs Tetrahedron. 55: 4699-4708. DOI: 10.1016/S0040-4020(99)00139-8 |
0.62 |
|
| 1999 |
Bonnarme V, Bachmann C, Cousson A, Mondon M, Gesson J. Diels-Alder reaction of 4-bromo-6-spiroepoxycyclohexa-2,4-dienone with electron-rich and neutral dienophiles Tetrahedron. 55: 433-448. DOI: 10.1016/S0040-4020(98)01041-2 |
0.345 |
|
| 1998 |
Florent JC, Dong X, Gaudel G, Mitaku S, Monneret C, Gesson JP, Jacquesy JC, Mondon M, Renoux B, Andrianomenjanahary S, Michel S, Koch M, Tillequin F, Gerken M, Czech J, et al. Prodrugs of anthracyclines for use in antibody-directed enzyme prodrug therapy. Journal of Medicinal Chemistry. 41: 3572-81. PMID 9733483 DOI: 10.1021/Jm970589L |
0.335 |
|
| 1998 |
Khodair AI, Gesson J. SULFUR GLYCOSYLATION REACTIONS INVOLVING 3-ALLYL-2-THIOHYDANTOIN NUCLEOSIDE BASES AS POTENTIAL ANTIVIRAL AND ANTITUMOR AGENTS Phosphorus, Sulfur, and Silicon and the Related Elements. 142: 167-190. DOI: 10.1080/10426509808029674 |
0.358 |
|
| 1998 |
Sukkari HE, Gesson J, Renoux B. Ring closing metathesis and cross metathesis of carbohydrate derivatives Tetrahedron Letters. 39: 4043-4046. DOI: 10.1016/S0040-4039(98)00692-3 |
0.395 |
|
| 1998 |
Gesson J, Renoux B, Tranoy I. Annonaceous acetogenins: Preparation of new methoxy substituted THF synthons from D-glucose Tetrahedron. 54: 6739-6750. DOI: 10.1016/S0040-4020(98)00336-6 |
0.375 |
|
| 1997 |
Gesson J, Renoux B, Schulten E. Synthesis of the THF moiety of annonacin based on aldolisation and Baeyer-Villiger oxidation Tetrahedron Letters. 38: 5811-5814. DOI: 10.1016/S0040-4039(97)01292-6 |
0.348 |
|
| 1992 |
Bertrand P, Gesson J. Stereoselective Synthesis of the trans 2,4-Disubstituted Butyrolactone Moiety of Annonaceous Acetogenins Synlett. 1992: 889-890. DOI: 10.1055/S-1992-21529 |
0.426 |
|
| 1986 |
Gesson J, Jacquesy J, Renoux B. A new annulation of carvone to chiral trans and cis fused bicyclic ketones Tetrahedron Letters. 27: 4461-4464. DOI: 10.1016/S0040-4039(00)84979-5 |
0.402 |
|
| 1984 |
BERRIER C, JACQUESY JC, GESSON JP, RENOUX A. ChemInform Abstract: CYCLIZATION OF DIARYLALKANES IN A SUPERACIDIC MEDIUM: SYNTHESIS OF TRICYCLIC KETONES CONTAINING AN ANGULAR METHYL GROUP AND THEIR ISOMERIZATION MECHANISM Chemischer Informationsdienst. 15. DOI: 10.1002/CHIN.198439146 |
0.301 |
|
| 1982 |
Gesson J, Mondon M. Total synthesis of 11-deoxydaunomycinone Journal of the Chemical Society, Chemical Communications. 421-423. DOI: 10.1039/C39820000421 |
0.366 |
|
| 1981 |
Gesson J, Jacquesy J, Mondon M. Anthracyclines. II - regiospecific synthesis of 6-deoxyanthracycline intermediates Tetrahedron Letters. 22: 1337-1340. DOI: 10.1016/S0040-4039(01)90311-9 |
0.406 |
|
| 1980 |
Gesson J, Jacquesy J, Jouannetaud M. A novel route to resorcinols Journal of the Chemical Society, Chemical Communications. 1128-1129. DOI: 10.1039/C39800001128 |
0.336 |
|
| 1980 |
Gesson J, Jacquesy J, Mondon M. Regioselective dienolate formation and alkylation of alkyl 2-methyl cyclohexene-1 carboxylates Tetrahedron Letters. 21: 2509-2512. DOI: 10.1016/0040-4039(80)80113-4 |
0.403 |
|
| 1976 |
Gesson J, Jacquesy J. Synthesis of tricyclic ketones containing an angular methyl group in ‘superacid’ media Journal of the Chemical Society, Chemical Communications. 652-653. DOI: 10.1039/C39760000652 |
0.387 |
|
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