Hiroaki Sasai - Publications

Affiliations: 
Osaka University, Toyonaka-shi, Ōsaka-fu, Japan 

162 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2024 Zhao R, Zhou DY, Asano K, Suzuki T, Sasai H, Suzuki T. General Synthesis of -1,4-Dialdehydes and Their Application in Ir-Catalyzed Asymmetric Tishchenko Reactions. Acs Omega. 9: 17945-17955. PMID 38680320 DOI: 10.1021/acsomega.3c09381  0.417
2023 Krishnan CG, Kondo M, Yasuda O, Fan D, Nakamura K, Wakabayashi Y, Sasai H, Takizawa S. Light-controlled p value of chiral Brønsted acid catalysts in enantioselective aza-Friedel-Crafts reaction. Chemical Communications (Cambridge, England). 59: 9956-9959. PMID 37526022 DOI: 10.1039/d3cc02719h  0.319
2023 Kondo M, Nakamura K, Krishnan CG, Sasai H, Takizawa S. Photoswitchable Chiral Organocatalysts: Photocontrol of Enantioselective Reactions. Chemical Record (New York, N.Y.). e202300040. PMID 37010445 DOI: 10.1002/tcr.202300040  0.414
2022 Khalid MI, Salem MSH, Sako M, Kondo M, Sasai H, Takizawa S. Electrochemical synthesis of heterodehydro[7]helicenes. Communications Chemistry. 5: 166. PMID 36697698 DOI: 10.1038/s42004-022-00780-7  0.385
2022 Kumar A, Sasai H, Takizawa S. Atroposelective Synthesis of C-C Axially Chiral Compounds via Mono- and Dinuclear Vanadium Catalysis. Accounts of Chemical Research. PMID 36206455 DOI: 10.1021/acs.accounts.2c00545  0.461
2022 Krishnan CG, Kondo M, Nakamura K, Sasai H, Takizawa S. Photoswitchable Chiral Cation-Binding Catalyst: Photocontrol of Catalytic Activity on Enantioselective Aminal Synthesis. Organic Letters. 24: 2670-2674. PMID 35353533 DOI: 10.1021/acs.orglett.2c00741  0.359
2021 Kishi N, Adachi Y, Jiang R, Doi T, Zhou DY, Asano K, Obora Y, Suzuki T, Sasai H, Suzuki T. Catalytic enantioselective intramolecular Tishchenko reaction of -dialdehyde: synthesis of ()-cedarmycins. Rsc Advances. 11: 11606-11609. PMID 35423664 DOI: 10.1039/d1ra00915j  0.481
2021 Nakamura K, Kondo M, Krishnan CG, Takizawa S, Sasai H. Azopyridine-based chiral oxazolines with rare-earth metals for photoswitchable catalysis. Chemical Communications (Cambridge, England). PMID 34231579 DOI: 10.1039/d1cc02602j  0.334
2020 Schober L, Sako M, Takizawa S, Gröger H, Sasai H. Catalytic and enantioselective oxa-Piancatelli reaction using a chiral vanadium complex. Chemical Communications (Cambridge, England). PMID 32735309 DOI: 10.1039/D0Cc02621B  0.518
2020 Kondo M, Wathsala HDP, Sako M, Hanatani Y, Ishikawa K, Hara S, Takaai T, Washio T, Takizawa S, Sasai H. Exploration of flow reaction conditions using machine-learning for enantioselective organocatalyzed Rauhut-Currier and [3+2] annulation sequence. Chemical Communications (Cambridge, England). PMID 31903462 DOI: 10.1039/C9Cc08526B  0.337
2020 Sako M, Losa R, Takiishi T, Vo-Thanh G, Takizawa S, Sasai H. Vanadium(V) Complex-Catalyzed One-Pot Synthesis of Phenanthridines via a Pictet-Spengler-Dehydrogenative Aromatization Sequence Catalysts. 10: 860. DOI: 10.3390/Catal10080860  0.401
2020 Sen A, Zhu L, Takizawa S, Takenaka K, Sasai H. Synthesis of Allylamine Derivatives via Intermolecular Aza‐Wacker‐Type Reaction Promoted by Palladium‐SPRIX Catalyst Advanced Synthesis & Catalysis. 362: 3558-3563. DOI: 10.1002/Adsc.202000644  0.471
2020 Chaki BM, Takenaka K, Zhu L, Tsujihara T, Takizawa S, Sasai H. Enantioselective One‐pot Synthesis of 3‐Azabicyclo[3.1.0]hexanes via Allylic Substitution and Oxidative Cyclization Advanced Synthesis & Catalysis. 362: 1537-1547. DOI: 10.1002/Adsc.202000044  0.474
2019 Ito Y, Kusakabe T, Dhage YD, Takahashi K, Sakata K, Sasai H, Kato K. TOTAL SYNTHESIS OF (-)-GRAMININ A BASED ON ASYMMETRIC CYCLIZATION CARBONYLATION OF PROPARGYL ACETATE. The Journal of Organic Chemistry. PMID 31789031 DOI: 10.1021/Acs.Joc.9B02886  0.472
2019 Kondo M, Takizawa S, Jiang Y, Sasai H. Room-Temperature, Metal-Free and One-Pot Preparation of 2H-Indazoles via Mills Reaction and Cyclization Sequence Masaru Kondo,* Shinobu Takizawa, Yuzhao Jiang, Hiroaki Sasai. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 31150138 DOI: 10.1002/Chem.201902242  0.395
2018 Sako M, Aoki T, Zumbrägel N, Schober L, Gröger H, Takizawa S, Sasai H. Chiral Dinuclear Vanadium Complex-mediated Oxidative Coupling of Resorcinols. The Journal of Organic Chemistry. PMID 30501179 DOI: 10.1021/Acs.Joc.8B02494  0.479
2018 Peng CP, Kusakabe T, Kikkawa S, Mochida T, Azumaya I, Dhage YD, Takahashi K, Sasai H, Kato K. Asymmetric Cyclizative Dimerization of (ortho-Alkynyl Phenyl) (Methoxymethyl) Sulfides with Palladium(II) Bisoxazoline Catalyst. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 30412336 DOI: 10.1002/Chem.201804779  0.484
2018 Sen A, Takenaka K, Sasai H. Enantioselective Aza-Wacker-Type Cyclization Promoted by Pd-SPRIX Catalyst. Organic Letters. PMID 30354176 DOI: 10.1021/Acs.Orglett.8B02946  0.481
2018 Zumbrägel N, Sako M, Takizawa S, Sasai H, Gröger H. Vanadium-Catalyzed Dehydrogenation of N-Heterocycles in Water. Organic Letters. PMID 30067034 DOI: 10.1021/Acs.Orglett.8B01484  0.368
2018 Sako M, Takizawa S, Sasai H. Chiral Vanadium Complex-catalyzed Enantioselective Oxidative Coupling Reactions Journal of Synthetic Organic Chemistry, Japan. 76: 874-884. DOI: 10.5059/Yukigoseikyokaishi.76.874  0.499
2018 Sasai H, Chaki BM, Wakita K, Takizawa S, Takenaka K. Enantioselective Synthesis of Spiro (Isoxazole-Isoxazoline) Hybrid Ligand Heterocycles. 97: 493. DOI: 10.3987/Com-18-S(T)41  0.438
2018 Kishi K, Takizawa S, Sasai H. Phosphine-Catalyzed Dual Umpolung Domino Michael Reaction: Facile Synthesis of Hydroindole- and Hydrobenzofuran-2-Carboxylates Acs Catalysis. 8: 5228-5232. DOI: 10.1021/Acscatal.8B01011  0.476
2017 Takizawa S, Sako M, Kishi K, Shigenobu M, Vo-Thanh G, Sasai H. Chiral Organocatalyzed Intermolecular Rauhut-Currier Reaction of Nitroalkenes with Ethyl Allenoate. Chemical & Pharmaceutical Bulletin. 65: 997-999. PMID 29093299 DOI: 10.1248/Cpb.C17-00554  0.474
2017 Sairenji S, Kikuchi T, Abozeid MA, Takizawa S, Sasai H, Ando Y, Ohmatsu K, Ooi T, Fujita M. Determination of the absolute configuration of compounds bearing chiral quaternary carbon centers using the crystalline sponge method. Chemical Science. 8: 5132-5136. PMID 28970900 DOI: 10.1039/C7Sc01524K  0.766
2017 Takizawa S, Sako M, Abozeid MA, Kishi K, Wathsala HDP, Hirata S, Murai K, Fujioka H, Sasai H. Enantio- and Diastereoselective Betti/aza-Michael Sequence: Single Operated Preparation of Chiral 1,3-Disubstituted Isoindolines. Organic Letters. PMID 28956612 DOI: 10.1021/Acs.Orglett.7B02693  0.772
2017 Kim HY, Takizawa S, Sasai H, Oh K. Reversal of Enantioselectivity Approach to BINOLs via Single and Dual 2-Naphthol Activation Modes. Organic Letters. PMID 28696128 DOI: 10.1021/Acs.Orglett.7B01734  0.676
2017 Abozeid MA, Sairenji S, Takizawa S, Fujita M, Sasai H. Enantioselective synthesis of tetrahydrocyclopenta[b]indole bearing a chiral quaternary carbon center via Pd(ii)-SPRIX-catalyzed C-H activation. Chemical Communications (Cambridge, England). PMID 28607967 DOI: 10.1039/C7Cc03199H  0.772
2017 Kishi K, Arteaga FA, Takizawa S, Sasai H. Multifunctional catalysis: stereoselective construction of α-methylidene-γ-lactams via an amidation/Rauhut-Currier sequence. Chemical Communications (Cambridge, England). PMID 28589974 DOI: 10.1039/C7Cc02839C  0.409
2017 Sako M, Ichinose K, Takizawa S, Sasai H. Short-step Syntheses of 4-Deoxycarbazomycin B, Sorazolon E, and (+)-Sorazolon E2. Chemistry, An Asian Journal. PMID 28418587 DOI: 10.1002/Asia.201700471  0.402
2016 Sako M, Takeuchi Y, Tsujihara T, Kodera J, Kawano T, Takizawa S, Sasai H. Efficient Enantioselective Synthesis of Oxahelicenes Using Redox/Acid Cooperative Catalysts. Journal of the American Chemical Society. PMID 27574874 DOI: 10.1021/Jacs.6B07424  0.521
2016 Chatupheeraphat A, Liao HH, Mader S, Sako M, Sasai H, Atodiresei I, Rueping M. Asymmetric Brønsted Acid Catalyzed Substitution of Diaryl Methanols with Thiols and Alcohols for the Synthesis of Chiral Thioethers and Ethers. Angewandte Chemie (International Ed. in English). PMID 26952288 DOI: 10.1002/Anie.201511179  0.488
2016 Kumagai N, Kanai M, Sasai H. A Career in Catalysis: Masakatsu Shibasaki Acs Catalysis. 6: 4699-4709. DOI: 10.1021/Acscatal.6B01227  0.469
2016 Chatupheeraphat A, Liao H, Mader S, Sako M, Sasai H, Atodiresei I, Rueping M. Asymmetrische Brønsted-Säure-katalysierte Substitution von Diarylmethanolen mit Thiolen und Alkoholen zur Synthese von chiralen Thioethern und Ethern Angewandte Chemie. 128: 4882-4887. DOI: 10.1002/Ange.201511179  0.421
2015 Takizawa S, Kishi K, Abozeid MA, Murai K, Fujioka H, Sasai H. Enantioselective organocatalytic oxidation of ketimine. Organic & Biomolecular Chemistry. PMID 26587584 DOI: 10.1039/C5Ob02042E  0.753
2015 Takizawa S, Kishi K, Yoshida Y, Mader S, Arteaga FA, Lee S, Hoshino M, Rueping M, Fujita M, Sasai H. Phosphine-Catalyzed β,γ-Umpolung Domino Reaction of Allenic Esters: Facile Synthesis of Tetrahydrobenzofuranones Bearing a Chiral Tetrasubstituted Stereogenic Carbon Center. Angewandte Chemie (International Ed. in English). PMID 26537173 DOI: 10.1002/Anie.201508022  0.516
2015 Suzuki T, Ismiyarto, Ishizaka Y, Zhou DY, Asano K, Sasai H. One-Pot Catalysis Using a Chiral Iridium Complex/Brønsted Base: Catalytic Asymmetric Synthesis of Catalponol. Organic Letters. 17: 5176-9. PMID 26496409 DOI: 10.1021/Acs.Orglett.5B02480  0.522
2015 Yoshida Y, Sako M, Kishi K, Sasai H, Hatakeyama S, Takizawa S. An enantioselective organocatalyzed aza-Morita-Baylis-Hillman reaction of isatin-derived ketimines with acrolein. Organic & Biomolecular Chemistry. PMID 26214279 DOI: 10.1039/C5Ob00874C  0.476
2015 Shigenobu M, Takenaka K, Sasai H. Palladium-Catalyzed Direct CH Arylation of Isoxazoles at the 5-Position. Angewandte Chemie (International Ed. in English). PMID 26130462 DOI: 10.1002/Anie.201504552  0.507
2015 Takenaka K, Lin X, Takizawa S, Sasai H. Structural Features and Asymmetric Environment of i-Pr-SPRIX Ligand. Chirality. 27: 532-7. PMID 26096770 DOI: 10.1002/Chir.22467  0.411
2015 Vinoth P, Vivekanand T, Suryavanshi PA, Menéndez JC, Sasai H, Sridharan V. Palladium(II)-catalyzed intramolecular carboxypalladation-olefin insertion cascade: direct access to indeno[1,2-b]furan-2-ones. Organic & Biomolecular Chemistry. 13: 5175-81. PMID 25849414 DOI: 10.1039/C5Ob00458F  0.493
2015 Takizawa S, Gröger H, Sasai H. Vanadium in asymmetric synthesis: emerging concepts in catalyst design and applications. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 8992-7. PMID 25809123 DOI: 10.1002/Chem.201406444  0.418
2015 Fan L, Takizawa S, Takeuchi Y, Takenaka K, Sasai H. Pd-catalyzed enantioselective intramolecular α-arylation of α-substituted cyclic ketones: facile synthesis of functionalized chiral spirobicycles. Organic & Biomolecular Chemistry. 13: 4837-40. PMID 25806855 DOI: 10.1039/C5Ob00382B  0.474
2015 Abozeid MA, Takizawa S, Sasai H. Pd(II)-catalyzed diastereoselective and enantioselective domino cyclization/cycloaddition reactions of alkenyl oximes for polycyclic heterocycles with four chiral stereogenic centers Tetrahedron Letters. 56: 4316-4319. DOI: 10.1016/J.Tetlet.2015.05.070  0.534
2015 Sako M, Takizawa S, Yoshida Y, Sasai H. Enantioselective and aerobic oxidative coupling of 2-naphthol derivatives using chiral dinuclear vanadium(V) complex in water Tetrahedron Asymmetry. DOI: 10.1016/J.Tetasy.2015.05.002  0.4
2014 Takizawa S, Arteaga FA, Kishi K, Hirata S, Sasai H. Facile regio- and stereoselective metal-free synthesis of all-carbon tetrasubstituted alkenes bearing a C(sp3)-F unit via dehydroxyfluorination of Morita-Baylis-Hillman (MBH) adducts. Organic Letters. 16: 4162-5. PMID 25089369 DOI: 10.1021/Ol501855M  0.431
2014 Takizawa S, Hirata S, Murai K, Fujioka H, Sasai H. C3-Symmetric chiral trisimidazoline-catalyzed Friedel-Crafts (FC)-type reaction. Organic & Biomolecular Chemistry. 12: 5827-30. PMID 24971875 DOI: 10.1039/C4Ob00925H  0.511
2014 Takenaka K, Mohanta SC, Sasai H. Palladium enolate umpolung: cyclative diacetoxylation of alkynyl cyclohexadienones promoted by a Pd/SPRIX catalyst. Angewandte Chemie (International Ed. in English). 53: 4675-9. PMID 24677411 DOI: 10.1002/Anie.201311172  0.497
2014 Takizawa S, Sasai H. Enantioselective acid-base organocatalyzed domino reactions based on aza-Morita-Baylis-Hillman process Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry. 72: 781-796. DOI: 10.5059/Yukigoseikyokaishi.72.781  0.378
2014 Takenaka K, Sako M, Takatani S, Sasai H. Enantioselective construction of C2-symmetric spiro skeleton through intramolecular copper-catalyzed N-arylation Arkivoc. 2015: 52-63. DOI: 10.3998/Ark.5550190.P008.802  0.504
2014 Takizawa S, Kodera J, Yoshida Y, Sako M, Breukers S, Enders D, Sasai H. Enantioselective oxidative-coupling of polycyclic phenols Tetrahedron. 70: 1786-1793. DOI: 10.1016/J.Tet.2014.01.017  0.41
2014 Takizawa S, Arteaga FA, Yoshida Y, Suzuki M, Sasai H. Enantioselective organocatalyzed formal [4+2] cycloaddition of ketimines with allenoates: Easy access to a tetrahydropyridine framework with a chiral tetrasubstituted stereogenic carbon center Asian Journal of Organic Chemistry. 3: 412-415. DOI: 10.1002/Ajoc.201300244  0.554
2013 Takenaka K, Dhage YD, Sasai H. Enantioselective Pd(II)-Pd(IV) catalysis utilizing a SPRIX ligand: efficient construction of chiral 3-oxy-tetrahydrofurans. Chemical Communications (Cambridge, England). 49: 11224-6. PMID 24154537 DOI: 10.1039/C3Cc44797A  0.381
2013 Takizawa S, Rémond E, Arteaga FA, Yoshida Y, Sridharan V, Bayardon J, Jugé S, Sasai H. P-chirogenic organocatalysts: application to the aza-Morita-Baylis-Hillman (aza-MBH) reaction of ketimines. Chemical Communications (Cambridge, England). 49: 8392-4. PMID 23939137 DOI: 10.1039/C3Cc44549F  0.438
2013 Takizawa S, Arteaga FA, Yoshida Y, Suzuki M, Sasai H. Organocatalyzed formal [2 + 2] cycloaddition of ketimines with allenoates: facile access to azetidines with a chiral tetrasubstituted carbon stereogenic center. Organic Letters. 15: 4142-5. PMID 23926881 DOI: 10.1021/Ol401817Q  0.541
2013 Sridharan V, Fan L, Takizawa S, Suzuki T, Sasai H. Pd(II)-SDP-catalyzed enantioselective 5-exo-dig cyclization of γ-alkynoic acids: application to the synthesis of functionalized dihydofuran-2(3H)-ones containing a chiral quaternary carbon center. Organic & Biomolecular Chemistry. 11: 5936-43. PMID 23903490 DOI: 10.1039/C3Ob41103F  0.523
2013 Kusakabe T, Takahashi T, Shen R, Ikeda A, Dhage YD, Kanno Y, Inouye Y, Sasai H, Mochida T, Kato K. Carbonylation of propargyl carbamates with palladium(II) bisoxazoline catalysts: efficient synthesis of 5-methoxy-3(2H)-furanones. Angewandte Chemie (International Ed. in English). 52: 7845-9. PMID 23788484 DOI: 10.1002/Anie.201303684  0.465
2013 Gabr RK, Hatakeyama T, Takenaka K, Takizawa S, Okada Y, Nakamura M, Sasai H. DFT study of a 5-endo-trig-type cyclization of 3-alkenoic acids by using Pd-spiro-bis(isoxazoline) as catalyst: importance of the rigid spiro framework for both selectivity and reactivity. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 9518-25. PMID 23749627 DOI: 10.1002/Chem.201203189  0.487
2013 Rémond E, Bayardon J, Takizawa S, Rousselin Y, Sasai H, Jugé S. o-(Hydroxyalkyl)phenyl P-chirogenic phosphines as functional chiral Lewis bases. Organic Letters. 15: 1870-3. PMID 23577952 DOI: 10.1021/Ol400515E  0.363
2013 Takizawa S, Arteaga Arteaga F, Yoshida Y, Kodera J, Nagata Y, Sasai H. Vanadium-catalyzed enantioselective Friedel-Crafts-type reactions. Dalton Transactions (Cambridge, England : 2003). 42: 11787-90. PMID 23103937 DOI: 10.1039/C2Dt32202A  0.435
2013 Suzuki T, Ishizaka Y, Ghozati K, Zhou DY, Asano K, Sasai H. Enantioselective multicatalytic synthesis of α-benzyl-β- hydroxyindan-1-ones Synthesis (Germany). 45: 2134-2136. DOI: 10.1055/S-0033-1338479  0.46
2013 Hirata S, Tanaka K, Matsui K, Arteaga FA, Yoshida Y, Takizawa S, Sasai H. Chiral bifunctional organocatalysts bearing a 1,3-propanediamine unit for the aza-MBH reaction Tetrahedron Asymmetry. 24: 1189-1192. DOI: 10.1016/J.Tetasy.2013.08.005  0.485
2013 Takizawa S, Nguyen TMN, Grossmann A, Suzuki M, Enders D, Sasai H. Facile synthesis of α-methylidene-γ-butyrolactones: Intramolecular Rauhut-Currier reaction promoted by chiral acid-base organocatalysts Tetrahedron. 69: 1202-1209. DOI: 10.1016/J.Tet.2012.11.046  0.463
2012 Takizawa S, Nguyen TM, Grossmann A, Enders D, Sasai H. Enantioselective synthesis of α-alkylidene-γ-butyrolactones: intramolecular Rauhut-Currier reaction promoted by acid/base organocatalysts. Angewandte Chemie (International Ed. in English). 51: 5423-6. PMID 22511309 DOI: 10.1002/Anie.201201542  0.438
2012 Arya K, Rawat DS, Sasai H. Zeolite supported Bronsted-acid ionic liquids: An eco approach for synthesis of spiro[indole-pyrido[3,2-e]thiazine] in water under ultrasonication Green Chemistry. 14: 1956-1963. DOI: 10.1039/C2Gc35168D  0.406
2012 Yoshida Y, Takizawa S, Sasai H. Design and synthesis of spiro bis(1,2,3-triazolium) salts as chiral ionic liquids Tetrahedron Asymmetry. 23: 843-851. DOI: 10.1016/J.Tetasy.2012.06.007  0.471
2012 Arya K, Rawat DS, Dandia A, Sasai H. Brønsted acidic ionic liquids: Green, efficient and reusable catalyst for synthesis of fluorinated spiro [indole-thiazinones/thiazolidinones] as antihistamic agents Journal of Fluorine Chemistry. 137: 117-122. DOI: 10.1016/J.Jfluchem.2012.03.003  0.389
2011 Takizawa S, Kiriyama K, Ieki K, Sasai H. A bifunctional spiro-type organocatalyst with high enantiocontrol: application to the aza-Morita-Baylis-Hillman reactions. Chemical Communications (Cambridge, England). 47: 9227-9. PMID 21769347 DOI: 10.1039/C1Cc12784E  0.428
2011 Takenaka K, Akita M, Tanigaki Y, Takizawa S, Sasai H. Enantioselective cyclization of 4-alkenoic acids via an oxidative allylic C-H esterification. Organic Letters. 13: 3506-9. PMID 21657245 DOI: 10.1021/Ol201314M  0.503
2011 Yoshida Y, Takizawa S, Sasai H. Synthesis of spiro bis(1,2,3-triazolium) salts as chiral ionic liquids Tetrahedron Letters. 52: 6877-6879. DOI: 10.1016/J.Tetlet.2011.09.152  0.439
2011 Takizawa S, Inoue N, Sasai H. An enantioselective organocatalyzed aza-MBH domino process: Application to the facile synthesis of tetrahydropyridines Tetrahedron Letters. 52: 377-380. DOI: 10.1016/J.Tetlet.2010.11.045  0.451
2011 Ramalingan C, Takenaka K, Sasai H. Pd(II)-SPRIX catalyzed enantioselective construction of pyrrolizines/pyrroloindoles employing molecular oxygen as the sole oxidant Tetrahedron. 67: 2889-2894. DOI: 10.1016/J.Tet.2011.02.057  0.423
2011 Takenaka K, Hashimoto S, Takizawa S, Sasai H. Chlorinative cyclization of 1,6-enynes by enantioselective palladium(II)/palladium(IV) catalysis Advanced Synthesis and Catalysis. 353: 1067-1070. DOI: 10.1002/Adsc.201000926  0.527
2010 Takizawa S, Inoue N, Hirata S, Sasai H. Enantioselective synthesis of isoindolines: an organocatalyzed domino process based On the aza-Morita-Baylis-Hillman reaction. Angewandte Chemie (International Ed. in English). 49: 9725-9. PMID 21064062 DOI: 10.1002/Anie.201004547  0.458
2010 Bajracharya GB, Koranne PS, Nadaf RN, Gabr RK, Takenaka K, Takizawa S, Sasai H. Pd-catalyzed 5-endo-trig-type cyclization of β,γ-unsaturated carbonyl compounds: an efficient ring closing reaction to give γ-butenolides and 3-pyrrolin-2-ones. Chemical Communications (Cambridge, England). 46: 9064-6. PMID 20967355 DOI: 10.1039/C0Cc02352C  0.76
2010 Takenaka K, Mohanta SC, Patil ML, Rao CV, Takizawa S, Suzuki T, Sasai H. Enantioselective Wacker-type cyclization of 2-alkenyl-1,3-diketones promoted by Pd-SPRIX catalyst. Organic Letters. 12: 3480-3. PMID 20578687 DOI: 10.1021/Ol1013069  0.459
2010 Takizawa S, Horii A, Sasai H. Acid-base organocatalysts for the aza-Morita-Baylis-Hillman reaction of nitroalkenes Tetrahedron Asymmetry. 21: 891-894. DOI: 10.1016/J.Tetasy.2010.05.027  0.47
2010 Takenaka K, Tanigaki Y, Patil ML, Rao CVL, Takizawa S, Suzuki T, Sasai H. Enantioselective 6-endo-trig Wacker-type cyclization of 2-geranylphenols: Application to a facile synthesis of (-)-cordiachromene Tetrahedron Asymmetry. 21: 767-770. DOI: 10.1016/j.tetasy.2010.04.060  0.308
2010 Takenaka K, Nagano T, Takizawa S, Sasai H. Asymmetric synthesis of chiral spiro bis(isoxazoline) and spiro (isoxazole-isoxazoline) ligands Tetrahedron Asymmetry. 21: 379-381. DOI: 10.1016/J.Tetasy.2010.03.006  0.491
2010 Suzuki T, Ghozati K, Zhou DY, Katoh T, Sasai H. Formal total synthesis of ottelione using iridium-catalyzed oxidative desymmetrization Tetrahedron. 66: 7562-7568. DOI: 10.1016/J.Tet.2010.07.047  0.452
2010 YAMADA K, ARAI T, SASAI H, SHIBASAKI M. ChemInform Abstract: A Catalytic Asymmetric Synthesis of 11-Deoxy-PGF1α Using ALB, a Heterobimetallic Multifunctional Asymmetric Complex. Cheminform. 29: no-no. DOI: 10.1002/chin.199842242  0.37
2010 SASAI H, BOUGAUCHI M, ARAI T, SHIBASAKI M. ChemInform Abstract: Enantioselective Synthesis of α-Hydroxy Phosphonates Using the LaLi3tris(binaphthoxide) Catalyst (LLB), Prepared by an Improved Method. Cheminform. 28: no-no. DOI: 10.1002/chin.199731052  0.332
2010 SASAI H, SUZUKI T, ITOH N, SHIBASAKI M. ChemInform Abstract: Catalytic Asymmetric Synthesis of Propranolol and Metoprolol Using a La-Li-BINOL Complex. Cheminform. 27: no-no. DOI: 10.1002/chin.199604057  0.303
2009 Tsujihara T, Shinohara T, Takenaka K, Takizawa S, Onitsuka K, Hatanaka M, Sasai H. Enantioselective intramolecular oxidative aminocarbonylation of alkenylureas catalyzed by palladium-spiro bis(isoxazoline) complexes. The Journal of Organic Chemistry. 74: 9274-9. PMID 19925006 DOI: 10.1021/Jo901778A  0.545
2009 Suzuki T, Ghozati K, Katoh T, Sasai H. Ir-catalyzed oxidative desymmetrization of meso-diols. Organic Letters. 11: 4286-8. PMID 19736916 DOI: 10.1021/Ol9016436  0.531
2009 Takenaka K, Itoh N, Sasai H. Enantioselective synthesis of C2-symmetric spirobilactams via Pd-catalyzed intramolecular double N-arylation. Organic Letters. 11: 1483-6. PMID 19254000 DOI: 10.1021/ol900016g  0.349
2009 Onitsuka K, Kameyama C, Sasai H. Regio- and enantioselective allylation of indole catalyzed by a planar-chiral cyelopentadienyl-ruthenium complex Chemistry Letters. 38: 444-445. DOI: 10.1246/Cl.2009.444  0.571
2009 Bajracharya GB, Arai MA, Koranne PS, Suzuki T, Takizawa S, Sasai H. Development of chiral spiro ligands for metal-catalyzed asymmetric reactions Bulletin of the Chemical Society of Japan. 82: 285-302. DOI: 10.1246/Bcsj.82.285  0.757
2009 Takizawa S, Rajesh D, Katayama T, Sasai H. One-pot preparation of chiral dinuclear vanadium(V) complex Synlett. 1667-1669. DOI: 10.1055/S-0029-1217191  0.439
2009 Bajracharya GB, Koranne PS, Tsujihara T, Takizawa S, Onitsuka K, Sasai H. Dicationic palladium(II)-spiro bis(isoxazoline) complex for highly enantioselective isotactic copolymerization of CO with styrene derivatives Synlett. 310-314. DOI: 10.1055/S-0028-1087667  0.741
2008 Takizawa S, Katayama T, Sasai H. Dinuclear chiral vanadium catalysts for oxidative coupling of 2-naphthols via a dual activation mechanism. Chemical Communications (Cambridge, England). 4113-22. PMID 18802502 DOI: 10.1039/B806016A  0.386
2008 Patil ML, Sasai H. Recent developments on chiral ionic liquids: design, synthesis, and applications. Chemical Record (New York, N.Y.). 8: 98-108. PMID 18383110 DOI: 10.1002/tcr.20143  0.371
2008 Takizawa S, Katayama T, Kameyama C, Onitsuka K, Suzuki T, Yanagida T, Kawai T, Sasai H. Chiral dinuclear vanadium(v) catalysts for oxidative coupling of 2-naphthols. Chemical Communications (Cambridge, England). 1810-2. PMID 18379701 DOI: 10.1039/B717068H  0.428
2008 Takenaka K, Nakatsuka S, Tsujihara T, Koranne PS, Sasai H. Divergent synthesis of chiral spiro (isoxazole-isoxazoline) hybrid ligands Tetrahedron Asymmetry. 19: 2492-2496. DOI: 10.1016/J.Tetasy.2008.10.019  0.487
2008 Takizawa S, Katayama T, Somei H, Asano Y, Yoshida T, Kameyama C, Rajesh D, Onitsuka K, Suzuki T, Mikami M, Yamataka H, Jayaprakash D, Sasai H. Dual activation in oxidative coupling of 2-naphthols catalyzed by chiral dinuclear vanadium complexes Tetrahedron. 64: 3361-3371. DOI: 10.1016/J.Tet.2008.01.110  0.452
2008 Sasai H, Patil ML. Other Chiral Phase-Transfer Catalysts for Asymmetric Synthesis Asymmetric Phase Transfer Catalysis. 135-159. DOI: 10.1002/9783527622627.ch7  0.305
2007 Miura T, Natsume S, Kanemoto K, Atsumi K, Fushimi H, Sasai H, Arai T, Yoshida T, Ajito K. Novel azalides derived from sixteen-membered macrolides. The Journal of Antibiotics. 60: 407-35. PMID 17721001 DOI: 10.1038/Ja.2007.55  0.412
2007 Takizawa S, Matsui K, Sasai H. Bifunctional organocatalysts for enantioselective aza-Morita-Baylis-Hillman (aza-MBH) reactions Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry. 65: 1089-1098. DOI: 10.5059/Yukigoseikyokaishi.65.1089  0.49
2007 Koranne PS, Tsujihara T, Arai MA, Bajracharya GB, Suzuki T, Onitsuka K, Sasai H. Design and synthesis of chiral hybrid spiro (isoxazole-isoxazoline) ligands Tetrahedron Asymmetry. 18: 919-923. DOI: 10.1016/J.Tetasy.2007.04.010  0.769
2007 Wakita K, Bajracharya GB, Arai MA, Takizawa S, Suzuki T, Sasai H. Enantioselective glyoxylate-ene reaction using a novel spiro bis(isoxazoline) ligand in copper catalysis Tetrahedron Asymmetry. 18: 372-376. DOI: 10.1016/J.Tetasy.2007.02.004  0.765
2007 Patil ML, Rao CVL, Takizawa S, Takenaka K, Onitsuka K, Sasai H. Synthesis of novel spiro imidazolium salts as chiral ionic liquids Tetrahedron. 63: 12702-12711. DOI: 10.1016/J.Tet.2007.10.002  0.435
2007 Takizawa S, Patil ML, Marubayashi K, Sasai H. Development of new methods toward efficient immobilization of chiral catalysts Tetrahedron. 63: 6512-6528. DOI: 10.1016/J.Tet.2007.03.018  0.45
2007 Takizawa S, Yogo J, Tsujihara T, Onitsuka K, Sasai H. Optical resolution of tetra isopropyl-substituted spiro bis(isoxazoline)i-Pr-SPRIX Journal of Organometallic Chemistry. 692: 495-498. DOI: 10.1016/J.Jorganchem.2006.03.048  0.341
2006 Patil ML, Rao CV, Yonezawa K, Takizawa S, Onitsuka K, Sasai H. Design and synthesis of novel chiral spiro ionic liquids. Organic Letters. 8: 227-30. PMID 16408881 DOI: 10.1021/Ol052466Y  0.476
2006 Jayaprakash D, Takizawa S, Arai T, Sasai H. Development of efficient methods for the immobilisation of multicomponent asymmetric catalysts Journal of Experimental Nanoscience. 1: 477-510. DOI: 10.1080/17458080601067690  0.407
2006 Matsui K, Takizawa S, Sasai H. A Brønsted acid and Lewis base organocatalyst for the aza-Morita-Baylis-Hillman reaction Synlett. 761-765. DOI: 10.1055/S-2006-933112  0.429
2006 Matsui K, Tanaka K, Horii A, Takizawa S, Sasai H. Conformational lock in a Brønsted acid-Lewis base organocatalyst for the aza-Morita-Baylis-Hillman reaction Tetrahedron Asymmetry. 17: 578-583. DOI: 10.1016/J.Tetasy.2006.01.007  0.437
2005 Matsui K, Takizawa S, Sasai H. Bifunctional organocatalysts for enantioselective aza-Morita-Baylis-Hillman reaction. Journal of the American Chemical Society. 127: 3680-1. PMID 15771486 DOI: 10.1021/Ja0500254  0.445
2005 Yonezawa K, Patil ML, Sasai H, Takizawa S. Spiro crown ethers bearing (S)-1,1′-spirobiindanes as chiral backbones Heterocycles. 66: 639-644. DOI: 10.3987/Com-05-S(K)59  0.39
2005 Takizawa S, Patil ML, Yonezawa F, Marubayashi K, Tanaka H, Kawai T, Sasai H. Micelle-derived polymer supports for enantioselective catalysts Tetrahedron Letters. 46: 1193-1197. DOI: 10.1016/J.Tetlet.2004.12.051  0.365
2005 Matsui K, Takizawa S, Sasai H. Enantioselective Morita-Baylis-Hillman (MBH) reaction promoted by a heterobimetallic complex with a Lewis base Tetrahedron Letters. 46: 1943-1946. DOI: 10.1016/J.Tetlet.2004.11.089  0.423
2004 Arai MA, Shinohara T, Aral T, Sasai H. Development of the First Spiro Bis(isoxazoline)Ligands (SPRIXs) and Their Applications to Catalytic Enantioselective Reactions Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry. 62: 59-69. DOI: 10.5059/Yukigoseikyokaishi.62.59  0.529
2004 Wakita K, Arai MA, Kato T, Shinohara T, Sasai H. Spiro bis(isoxazole) as a new chiral ligand Heterocycles. 62: 831-838. DOI: 10.3987/Com-03-S(P)60  0.451
2004 Kawase T, Takizawa S, Jayaprakash D, Sasai H. Enantioselective aldol-type reaction using diketene Synthetic Communications. 34: 4487-4492. DOI: 10.1081/Scc-200043192  0.442
2004 Somei H, Asano Y, Yoshida T, Takizawa S, Yamataka H, Sasai H. Dual activation in a homolytic coupling reaction promoted by an enantioselective dinuclear vanadium(IV) catalyst Tetrahedron Letters. 45: 1841-1844. DOI: 10.1016/J.Tetlet.2004.01.007  0.439
2004 Kato T, Marubayashi K, Takizawa S, Sasai H. Development of a novel chiral spiro ligand bearing oxazoline Tetrahedron Asymmetry. 15: 3693-3697. DOI: 10.1016/j.tetasy.2004.09.037  0.334
2003 Takizawa S, Somei H, Jayaprakash D, Sasai H. Metal-bridged polymers as insoluble multicomponent asymmetric catalysts with high enantiocontrol: an approach for the immobilization of catalysts without using any support. Angewandte Chemie (International Ed. in English). 42: 5711-4. PMID 14661202 DOI: 10.1002/Anie.200352354  0.33
2003 Marubayashi K, Takizawa S, Kawakusu T, Arai T, Sasai H. Monolayer-protected Au cluster (MPC)-supported Ti-BINOLate complex. Organic Letters. 5: 4409-12. PMID 14602012 DOI: 10.1021/Ol035706N  0.362
2003 Sekiguti T, Iizuka Y, Takizawa S, Jayaprakash D, Arai T, Sasai H. Polymer-supported bisBINOL ligands for the immobilization of multicomponent asymmetric catalysts. Organic Letters. 5: 2647-50. PMID 12868880 DOI: 10.1021/Ol034797L  0.407
2003 Arai T, Sekiguti T, Otsuki K, Takizawa S, Sasai H. "Catalyst analogue": a concept for constructing multicomponent asymmetric catalysts (MAC) by using a polymer support. Angewandte Chemie (International Ed. in English). 42: 2144-7. PMID 12761743 DOI: 10.1002/Anie.200250536  0.328
2003 Arai MA, Kuraishi M, Arai T, Sasai H. Synthesis of new chiral bis(isoxazoline) ligands containing spiro[5.5]undecane skeleton. Chirality. 15: 101-4. PMID 12467051 DOI: 10.1002/Chir.10164  0.461
2003 Patil ML, Takizawa S, Sasai H. Design and synthesis of novel spiro pyridinium and quinolinium salts Heterocycles. 61: 581-586. DOI: 10.3987/Com-03-S53  0.453
2003 Takizawa S, Honda Y, Arai MA, Kato T, Sasai H. Synthesis of novel chiral spiro bis(pyrazole) ligands Heterocycles. 60: 2551-2556. DOI: 10.3987/Com-03-9874  0.431
2003 Shinohara T, Wakita K, Arai MA, Arai T, Sasai H. Synthesis and character of new bis(isoxazoline) ligands Heterocycles. 59: 587-593. DOI: 10.3987/Com-02-S57  0.466
2003 Jayaprakash D, Kobayashi Y, Arai T, Hu QS, Zheng XF, Pu L, Sasai H. Catalytic asymmetric epoxidation of α,β-unsaturated ketones using polymeric BINOL Journal of Molecular Catalysis a: Chemical. 196: 145-149. DOI: 10.1016/S1381-1169(02)00644-1  0.461
2003 Jayaprakash D, Kobayashi Y, Watanabe S, Arai T, Sasai H. Enantioselective epoxidation of α,β-unsaturated ketones using polymer-supported lanthanoid-BINOL complexes Tetrahedron Asymmetry. 14: 1587-1592. DOI: 10.1016/S0957-4166(03)00282-9  0.456
2003 Muthiah C, Arai MA, Shinohara T, Arai T, Takizawa S, Sasai H. Enantioselective synthesis of α-methylene-γ-butyrolactones using chiral Pd(II)-SPRIX catalyst Tetrahedron Letters. 44: 5201-5204. DOI: 10.1016/S0040-4039(03)01250-4  0.353
2003 Shinohara T, Arai MA, Wakita K, Arai T, Sasai H. The first enantioselective intramolecular aminocarbonylation of alkenes promoted by Pd(II)-spiro bis(isoxazoline) catalyst Tetrahedron Letters. 44: 711-714. DOI: 10.1016/S0040-4039(02)02650-3  0.301
2003 Sasai H, Watanabe S, Suzuki T, Shibasaki M. Catalytic Asymmetric Synthesis of Nitroaldols Using a Lanthanum‐Lithium‐BINOL Complex: (2S,3S)‐2‐Nitro‐5‐Phenyl‐1,3‐Pentanediol Organic Syntheses. 78: 14-14. DOI: 10.1002/0471264180.Os078.02  0.45
2002 Arai T, Sekiguti T, Iizuka Y, Takizawa S, Sakamoto S, Yamaguchi K, Sasai H. A dendrimer-supported heterobimetallic asymmetric catalyst Tetrahedron-Asymmetry. 13: 2083-2087. DOI: 10.1016/S0957-4166(02)00573-6  0.421
2001 Arai MA, Kuraishi M, Arai T, Sasai H. A new asymmetric Wacker-type cyclization and tandem cyclization promoted by Pd(II)-spiro bis(isoxazoline) catalyst. Journal of the American Chemical Society. 123: 2907-8. PMID 11456988 DOI: 10.1021/ja005920w  0.313
2000 Schlemminger I, Saida Y, Gröger H, Maison W, Durot N, Sasai H, Shibasaki M, Martens J. Concept of improved rigidity: how to make enantioselective hydrophosphonylation of cyclic imines catalyzed by chiral heterobimetallic lanthanoid complexes almost perfect Journal of Organic Chemistry. 65: 4818-4825. PMID 10956457 DOI: 10.1021/Jo991882R  0.51
2000 Sasai H, Arai T, Watanabe S, Shibasaki M. Novel heterobimetallic asymmetric catalysis directing toward enzymatic function Catalysis Today. 62: 17-22. DOI: 10.1016/S0920-5861(00)00405-3  0.463
1999 Arai MA, Arai aT, Sasai H. Design and Synthesis of the First Spiro Bis(isoxazoline) Derivatives as Asymmetric Ligands Organic Letters. 1: 1795-1797. DOI: 10.1021/Ol9902881  0.486
1999 Yoshikawa N, Yamada YMA, Das J, Sasai H, Shibasaki M. Direct Catalytic Asymmetric Aldol Reaction Journal of the American Chemical Society. 121: 4168-4178. DOI: 10.1021/Ja990031Y  0.439
1998 Shimizu S, Ohori K, Arai T, Sasai H, Shibasaki M. A Catalytic Asymmetric Synthesis of Tubifolidine. The Journal of Organic Chemistry. 63: 7547-7551. PMID 11672415 DOI: 10.1021/Jo981069G  0.38
1998 Shibasaki M, Sasai H, Arai T, Iida T. Heterobimetallic asymmetric catalysts. Developments and applications Pure and Applied Chemistry. 70: 1027-1034. DOI: 10.1351/Pac199870051027  0.414
1998 Gröger H, Saida Y, Sasai H, Yamaguchi K, Martens J, Shibasaki M. A New and Highly Efficient Asymmetric Route to Cyclic alpha-Amino Phosphonates: The first Catalytic Enantioselective Hydrophosphonylation of Cyclic Imines Catalyzed by Chiral Heterobimetallic Lanthanoid Complexes J. Am. Chem. Soc.. 120: 3089-3103. DOI: 10.1021/Ja973872I  0.513
1998 Morita T, Arai T, Sasai H, Shibasaki M. Utilization of heterobimetallic complexes as Lewis acids Tetrahedron: Asymmetry. 9: 1445-1450. DOI: 10.1016/S0957-4166(98)00124-4  0.319
1997 Göttlich R, Yamakoshi K, Sasai H, Shibasaki M. A New and Selective Metal-Catalyzed Baeyer-Villiger Oxidation Procedure Synlett. 1997: 971-973. DOI: 10.1055/S-1997-966  0.304
1996 Arai T, Bougauchi M, Sasai H, Shibasaki M. Catalytic Asymmetric Synthesis of alpha-Hydroxy Phosphonates Using the Al-Li-BINOL Complex. The Journal of Organic Chemistry. 61: 2926-2927. PMID 11667145 DOI: 10.1021/Jo960180O  0.344
1996 Shibasaki M, Sasai H. Catalytic asymmetric carbon-carbon bond-forming reaction utilizing rare earth metal complexes Pure and Applied Chemistry. 68: 523-530. DOI: 10.1351/Pac199668030523  0.458
1996 Arai T, Yamada YMA, Yamamoto N, Sasai H, Shibasaki M. Self-Assembly of Heterobimetallic Complexes and Reactive Nucleophiles: A General Strategy for the Activation of Asymmetric Reactions Promoted by Heterobimetallic Catalysts Chemistry - a European Journal. 2: 1368-1372. DOI: 10.1002/Chem.19960021107  0.31
1996 Arai T, Sasai H, Aoe K, Okamura K, Date T, Shibasaki M. Ein neuartiger multifunktioneller asymmetrischer Hetero-Dimetall-Katalysator für Michael-Additionen und Tandem-Michael-Aldol-Reaktionen Angewandte Chemie. 108: 103-105. DOI: 10.1002/Ange.19961080123  0.318
1995 Sasai H, Arai S, Tahara Y, Shibasaki M. Catalytic Asymmetric Synthesis of .alpha.-Amino Phosphonates Using Lanthanoid-Potassium-BINOL Complexes The Journal of Organic Chemistry. 60: 6656-6657. DOI: 10.1021/Jo00126A003  0.333
1995 Sasai H, Arai T, Emori E, Shibasaki M. Efficient Synthesis of C10 Chiron by Lewis Acid Catalyzed Rearrangement of (+)-.alpha.-3,4-Epoxycarane Journal of Organic Chemistry. 60: 465-467. DOI: 10.1021/Jo00107A031  0.362
1995 Nukui S, Sodeoka M, Sasai H, Shibasaki M. Regio- and Stereoselective Functionalization of an Optically Active Tetrahydroindolizine Derivative. Catalytic Asymmetric Syntheses of Lentiginosine, 1,2-Diepilentiginosine, and Gephyrotoxin 209D Journal of Organic Chemistry. 60: 398-404. DOI: 10.1021/Jo00107A019  0.354
1994 Sugita K, Shigeno K, Neville CF, Sasai H, Shibasaki M. Synthetic Studies towards Phorbols: Synthesis of B or C Ring Substituted Phorbol Skeletons in the Naturally Occurring Form Synlett. 1994: 325-329. DOI: 10.1055/S-1994-22841  0.365
1994 Sasai H, Arai S, Shibasaki M. Catalytic Aldol Reaction with Sm(HMDS)3 and Its Application for the Introduction of a Carbon-Carbon Triple Bond at C-13 in Prostaglandin Synthesis The Journal of Organic Chemistry. 59: 2661-2664. DOI: 10.1021/Jo00088A068  0.445
1993 Sasai H, Suzuki T, Itoh N, Tanaka K, Date T, Okamura K, Shibasaki M. Catalytic asymmetric nitroaldol reaction using optically active rare earth BINOL complexes: investigation of the catalyst structure Journal of the American Chemical Society. 115: 10372-10373. DOI: 10.1021/ja00075a068  0.304
1993 Sasai H, Itoh N, Suzuki T, Shibasaki M. Catalytic asymmetric nitroaldol reaction: An efficient synthesis of (S) propranolol using the lanthanum binaphthol complex Tetrahedron Letters. 34: 855-858. DOI: 10.1016/0040-4039(93)89031-K  0.373
1992 Shibasaki M, Shigeno K, Ohne K, Yamaguchi T, Sasai H, Sibasaki M. Synthetic Approaches to Phorbols via the Intramolevular Nitrile Oxide Cycloaddition: Stereocontrol of the B-C Ring Junction Heterocycles. 33: 161. DOI: 10.3987/Com-91-S69  0.39
1992 Sasai H, Suzuki T, Arai S, Arai T, Shibasaki M. Basic character of rare earth metal alkoxides. Utilization in catalytic carbon-carbon bond-forming reactions and catalytic asymmetric nitroaldol reactions Journal of the American Chemical Society. 114: 4418-4420. DOI: 10.1021/Ja00037A068  0.384
1991 Satoh S, Sodeoka M, Sasai H, Shibasaki M. Control of ring-junction stereochemistry via radical cyclization. A new construction of trans-hydrindans Journal of Organic Chemistry. 56: 2278-2280. DOI: 10.1021/Jo00007A004  0.319
1990 Sasai H, Kirio Y, Shibasaki M. Zirconium tetra-tert-butoxide, an efficient and convenient basic reagent in organic synthesis. Utilization in cross and intramolecular aldol reactions The Journal of Organic Chemistry. 55: 5306-5308. DOI: 10.1021/Jo00306A003  0.432
1987 Sasai H, Shibasaki M. Total synthesis of punaglandin 4 Tetrahedron Letters. 28: 333-336. DOI: 10.1016/S0040-4039(00)95721-6  0.467
1986 Suami T, Sasai H, Matsuno K, Suzuki N. Synthetic Approaches Toward Antibiotic Tunicamycins. Part 8. Total Synthesis of Tunicamycin. Cheminform. 17. DOI: 10.1002/Chin.198615376  0.325
1985 Sasai H, Matsuno K, Suami T. Synthetic Approach Toward Antibiotic Tunicamycins - VII Synthesis of Tunicamine and Tunicaminyl Uracil Derivative Journal of Carbohydrate Chemistry. 4: 99-112. DOI: 10.1080/07328308508062952  0.498
1985 Sasai H, Matsuno K, Suami T. Synthetic Approach Toward Antibiotic Tunicamycins. Vii. Synthesis Of Tunicamine And Tunicaminyl Uracil Derivative Cheminform. 16. DOI: 10.1002/Chin.198540350  0.348
1984 Sasai H, Suami T, Matsuno K. Synthesis of Tunicaminyl Uracil. Cheminform. 15: 507. DOI: 10.1002/Chin.198440326  0.393
1983 Suami T, Sasai H, Matsuno K. Synthesis Of Methyl Hexaacetyl-Tunicaminyl Uracil Chemistry Letters. 12: 819-822. DOI: 10.1246/Cl.1983.819  0.376
1982 Fukuda Y, Sasai H, Suami T. Synthetic Approach toward Antibiotic Tunicamycins. 3. Methyl 3,4,7,8-Tetra-O-acetyl-10-O-benzyl-2-benzyloxycarbonylamino-2,6-dideoxy-11,12-O-isopropylidene-β-L-dodecodialdo-(12R)-furanose-(12,9)-pyranosides-(1,5) Bulletin of the Chemical Society of Japan. 55: 1574-1578. DOI: 10.1246/Bcsj.55.1574  0.321
1981 Fukuda Y, Kitasato H, Sasai H, Suami T. Synthetic Approach toward Antibiotic Tunicamycins. II. Bulletin of the Chemical Society of Japan. 54: 1830-1834. DOI: 10.1246/Bcsj.54.1830  0.338
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