| Year |
Citation |
Score |
| 2011 |
Yamamoto T, Nair P, Largent-Milnes TM, Jacobsen NE, Davis P, Ma SW, Yamamura HI, Vanderah TW, Porreca F, Lai J, Hruby VJ. Discovery of a potent and efficacious peptide derivative for δ/μ opioid agonist/neurokinin 1 antagonist activity with a 2',6'-dimethyl-L-tyrosine: in vitro, in vivo, and NMR-based structural studies. Journal of Medicinal Chemistry. 54: 2029-38. PMID 21366266 DOI: 10.1021/Jm101023R |
0.832 |
|
| 2010 |
Yamamoto T, Nair P, Jacobsen NE, Kulkarni V, Davis P, Ma SW, Navratilova E, Yamamura HI, Vanderah TW, Porreca F, Lai J, Hruby VJ. Biological and conformational evaluation of bifunctional compounds for opioid receptor agonists and neurokinin 1 receptor antagonists possessing two penicillamines. Journal of Medicinal Chemistry. 53: 5491-501. PMID 20617791 DOI: 10.1021/Jm100157M |
0.845 |
|
| 2010 |
LIAO S, LIN J, SHENDEROVICH MD, HAN Y, HASOHATA K, DAVIS P, QIU W, PORRECA F, YAMAMURA HI, HRUBY VJ. ChemInform Abstract: The Stereochemical Requirements of the Novel δ-Opioid Selective Dipeptide Antagonist TMT-TIC. Cheminform. 29: no-no. DOI: 10.1002/CHIN.199812174 |
0.528 |
|
| 2010 |
HRUBY VJ, DAVIS TP, O'BRIEN DF, PORRECA F, YAMAMURA HI. ChemInform Abstract: Design of Peptides and Peptidomimetics That Are Selective, Stable and Can Cross Membrane Barriers Cheminform. 28: no-no. DOI: 10.1002/CHIN.199740331 |
0.369 |
|
| 2009 |
Yamamoto T, Nair P, Jacobsen NE, Vagner J, Kulkarni V, Davis P, Ma SW, Navratilova E, Yamamura HI, Vanderah TW, Porreca F, Lai J, Hruby VJ. Improving metabolic stability by glycosylation: bifunctional peptide derivatives that are opioid receptor agonists and neurokinin 1 receptor antagonists. Journal of Medicinal Chemistry. 52: 5164-75. PMID 20560643 DOI: 10.1021/Jm900473P |
0.835 |
|
| 2009 |
Yamamoto T, Nair P, Ma SW, Davis P, Yamamura HI, Vanderah TW, Porreca F, Lai J, Hruby VJ. The biological activity and metabolic stability of peptidic bifunctional compounds that are opioid receptor agonists and neurokinin-1 receptor antagonists with a cystine moiety. Bioorganic & Medicinal Chemistry. 17: 7337-43. PMID 19762245 DOI: 10.1016/J.Bmc.2009.08.035 |
0.801 |
|
| 2009 |
Tumati S, Yamamura HI, Vanderah TW, Roeske WR, Varga EV. Sustained morphine treatment augments capsaicin-evoked calcitonin gene-related peptide release from primary sensory neurons in a protein kinase A- and Raf-1-dependent manner. The Journal of Pharmacology and Experimental Therapeutics. 330: 810-7. PMID 19491327 DOI: 10.1124/jpet.109.151704 |
0.609 |
|
| 2009 |
Nair P, Yamamoto T, Kulkarni V, Moye S, Navratilova E, Davis P, Largent T, Ma SW, Yamamura HI, Vanderah T, Lai J, Porreca F, Hruby VJ. Novel bifunctional peptides as opioid agonists and NK-1 antagonists. Advances in Experimental Medicine and Biology. 611: 537-8. PMID 19400302 DOI: 10.1007/978-0-387-73657-0_235 |
0.839 |
|
| 2009 |
Tumati S, Yamamura HI, St John PA, Vanderah TW, Roeske WR, Varga EV. Sustained cannabinoid agonist treatment augments CGRP release in a PKA-dependent manner. Neuroreport. 20: 815-9. PMID 19387418 DOI: 10.1097/WNR.0b013e32832be50b |
0.54 |
|
| 2008 |
Varga EV, Georgieva T, Tumati S, Alves I, Salamon Z, Tollin G, Yamamura HI, Roeske WR. Functional selectivity in cannabinoid signaling. Current Molecular Pharmacology. 1: 273-84. PMID 20021440 DOI: 10.2174/1874-470210801030273 |
0.444 |
|
| 2008 |
Fioravanti B, De Felice M, Stucky CL, Medler KA, Luo MC, Gardell LR, Ibrahim M, Malan TP, Yamamura HI, Ossipov MH, King T, Lai J, Porreca F, Vanderah TW. Constitutive activity at the cannabinoid CB1 receptor is required for behavioral response to noxious chemical stimulation of TRPV1: antinociceptive actions of CB1 inverse agonists. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 28: 11593-602. PMID 18987195 DOI: 10.1523/Jneurosci.3322-08.2008 |
0.758 |
|
| 2008 |
Tumati S, Milnes TL, Yamamura HI, Vanderah TW, Roeske WR, Varga EV. Intrathecal Raf-1-selective siRNA attenuates sustained morphine-mediated thermal hyperalgesia. European Journal of Pharmacology. 601: 207-8. PMID 18976650 DOI: 10.1016/j.ejphar.2008.10.033 |
0.591 |
|
| 2008 |
Yamamoto T, Nair P, Jacobsen NE, Davis P, Ma SW, Navratilova E, Moye S, Lai J, Yamamura HI, Vanderah TW, Porreca F, Hruby VJ. The importance of micelle-bound states for the bioactivities of bifunctional peptide derivatives for delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists. Journal of Medicinal Chemistry. 51: 6334-47. PMID 18821747 DOI: 10.1021/Jm800389V |
0.835 |
|
| 2008 |
Yue X, Tumati S, Navratilova E, Strop D, St John PA, Vanderah TW, Roeske WR, Yamamura HI, Varga EV. Sustained morphine treatment augments basal CGRP release from cultured primary sensory neurons in a Raf-1 dependent manner. European Journal of Pharmacology. 584: 272-7. PMID 18328477 DOI: 10.1016/J.Ejphar.2008.02.013 |
0.731 |
|
| 2008 |
Yamamoto T, Nair P, Vagner J, Largent-Milnes T, Davis P, Ma SW, Navratilova E, Moye S, Tumati S, Lai J, Yamamura HI, Vanderah TW, Porreca F, Hruby VJ. A structure-activity relationship study and combinatorial synthetic approach of C-terminal modified bifunctional peptides that are delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists. Journal of Medicinal Chemistry. 51: 1369-76. PMID 18266313 DOI: 10.1021/Jm070332F |
0.844 |
|
| 2008 |
Georgieva T, Devanathan S, Stropova D, Park CK, Salamon Z, Tollin G, Hruby VJ, Roeske WR, Yamamura HI, Varga E. Unique agonist-bound cannabinoid CB1 receptor conformations indicate agonist specificity in signaling. European Journal of Pharmacology. 581: 19-29. PMID 18162180 DOI: 10.1016/J.Ejphar.2007.11.053 |
0.473 |
|
| 2008 |
Hruby VJ, Porreca F, Yamamura HI, Tollin G, Agnes RS, Lee YS, Cai M, Alves I, Cowell S, Varga E, Davis P, Salamon Z, Roeske W, Vanderah T, Lai J. New paradigms and tools in drug design for pain and addiction Drug Addiction: From Basic Research to Therapy. 477-494. DOI: 10.1007/978-0-387-76678-2_28 |
0.432 |
|
| 2007 |
Yamamoto T, Nair P, Davis P, Ma SW, Navratilova E, Moye S, Tumati S, Lai J, Vanderah TW, Yamamura HI, Porreca F, Hruby VJ. Design, synthesis, and biological evaluation of novel bifunctional C-terminal-modified peptides for delta/mu opioid receptor agonists and neurokinin-1 receptor antagonists. Journal of Medicinal Chemistry. 50: 2779-86. PMID 17516639 DOI: 10.1021/Jm061369N |
0.856 |
|
| 2007 |
Nissan HP, Lu J, Booth NL, Yamamura HI, Farnsworth NR, Wang ZJ. A red clover (Trifolium pratense) phase II clinical extract possesses opiate activity. Journal of Ethnopharmacology. 112: 207-10. PMID 17350196 DOI: 10.1016/j.jep.2007.02.006 |
0.448 |
|
| 2007 |
Navratilova E, Waite S, Stropova D, Eaton MC, Alves ID, Hruby VJ, Roeske WR, Yamamura HI, Varga EV. Quantitative evaluation of human delta opioid receptor desensitization using the operational model of drug action. Molecular Pharmacology. 71: 1416-26. PMID 17322005 DOI: 10.1124/Mol.106.030023 |
0.742 |
|
| 2006 |
Cai M, Varga EV, Stankova M, Mayorov A, Perry JW, Yamamura HI, Trivedi D, Hruby VJ. Cell signaling and trafficking of human melanocortin receptors in real time using two-photon fluorescence and confocal laser microscopy: differentiation of agonists and antagonists. Chemical Biology & Drug Design. 68: 183-93. PMID 17105482 DOI: 10.1111/J.1747-0285.2006.00432.X |
0.443 |
|
| 2006 |
Hruby VJ, Porreca F, Yamamura HI, Tollin G, Agnes RS, Lee YS, Cai M, Alves I, Cowell S, Varga E, Davis P, Salamon Z, Roeske W, Vanderah T, Lai J. New paradigms and tools in drug design for pain and addiction. The Aaps Journal. 8: E450-60. PMID 17025262 DOI: 10.1208/Aapsj080353 |
0.758 |
|
| 2006 |
Yue X, Varga EV, Stropova D, Vanderah TW, Yamamura HI, Roeske WR. Chronic morphine-mediated adenylyl cyclase superactivation is attenuated by the Raf-1 inhibitor, GW5074. European Journal of Pharmacology. 540: 57-9. PMID 16750187 DOI: 10.1016/j.ejphar.2006.04.033 |
0.656 |
|
| 2006 |
Oki T, Maruyama S, Takagi Y, Yamamura HI, Yamada S. Characterization of muscarinic receptor binding and inhibition of salivation after oral administration of tolterodine in mice. European Journal of Pharmacology. 529: 157-63. PMID 16316647 DOI: 10.1016/j.ejphar.2005.11.004 |
0.411 |
|
| 2005 |
Navratilova E, Eaton MC, Stropova D, Varga EV, Vanderah TW, Roeske WR, Yamamura HI. Morphine promotes phosphorylation of the human delta-opioid receptor at serine 363. European Journal of Pharmacology. 519: 212-4. PMID 16135360 DOI: 10.1016/J.Ejphar.2005.07.024 |
0.778 |
|
| 2005 |
Handl HL, Vagner J, Yamamura HI, Hruby VJ, Gillies RJ. Development of a lanthanide-based assay for detection of receptor-ligand interactions at the delta-opioid receptor. Analytical Biochemistry. 343: 299-307. PMID 16004955 DOI: 10.1016/J.Ab.2005.05.040 |
0.462 |
|
| 2005 |
Dhanasekaran M, Palian MM, Alves I, Yeomans L, Keyari CM, Davis P, Bilsky EJ, Egleton RD, Yamamura HI, Jacobsen NE, Tollin G, Hruby VJ, Porreca F, Polt R. Glycopeptides related to beta-endorphin adopt helical amphipathic conformations in the presence of lipid bilayers. Journal of the American Chemical Society. 127: 5435-48. PMID 15826181 DOI: 10.1021/Ja0432158 |
0.455 |
|
| 2005 |
Varga EV, Hosohata K, Borys D, Navratilova E, Nylen A, Vanderah TW, Porreca F, Roeske WR, Yamamura HI. Antinociception depends on the presence of G protein gamma2-subunits in brain. European Journal of Pharmacology. 508: 93-8. PMID 15680258 DOI: 10.1016/J.Ejphar.2004.11.062 |
0.776 |
|
| 2005 |
Gu X, Ying J, Min B, Cain JP, Davis P, Willey P, Navratilova E, Yamamura HI, Porreca F, Hruby VJ. Parallel synthesis and biological evaluation of different sizes of bicyclo[2,3]-Leu-enkephalin analogues. Biopolymers. 80: 151-63. PMID 15660379 DOI: 10.1002/Bip.20208 |
0.691 |
|
| 2005 |
Egleton RD, Bilsky EJ, Tollin G, Dhanasekaran M, Lowery J, Alves I, Davis P, Porreca F, Yamamura HI, Yeomans L, Keyari CM, Polt R. Biousian glycopeptides penetrate the blood-brain barrier Tetrahedron Asymmetry. 16: 65-75. DOI: 10.1016/J.Tetasy.2004.11.038 |
0.528 |
|
| 2004 |
Varga EV, Navratilova E, Stropova D, Jambrosic J, Roeske WR, Yamamura HI. Agonist-specific regulation of the delta-opioid receptor. Life Sciences. 76: 599-612. PMID 15567186 DOI: 10.1016/J.Lfs.2004.07.020 |
0.732 |
|
| 2004 |
Gu X, Ying J, Agnes RS, Navratilova E, Davis P, Stahl G, Porreca F, Yamamura HI, Hruby VJ. Novel design of bicyclic beta-turn dipeptides on solid-phase supports and synthesis of [3.3.0]-Bicyclo([2,3])-leu-enkephalin analogues. Organic Letters. 6: 3285-8. PMID 15355033 DOI: 10.1021/Ol0488183 |
0.714 |
|
| 2004 |
Alves ID, Ciano KA, Boguslavski V, Varga E, Salamon Z, Yamamura HI, Hruby VJ, Tollin G. Selectivity, cooperativity, and reciprocity in the interactions between the delta-opioid receptor, its ligands, and G-proteins. The Journal of Biological Chemistry. 279: 44673-82. PMID 15317820 DOI: 10.1074/Jbc.M404713200 |
0.422 |
|
| 2004 |
Handl HL, Vagner J, Yamamura HI, Hruby VJ, Gillies RJ. Lanthanide-based time-resolved fluorescence of in cyto ligand-receptor interactions. Analytical Biochemistry. 330: 242-50. PMID 15203329 DOI: 10.1016/J.Ab.2004.04.012 |
0.373 |
|
| 2004 |
Cai M, Stankova M, Pond SJ, Mayorov AV, Perry JW, Yamamura HI, Trivedi D, Hruby VJ. Real time differentiation of G-protein coupled receptor (GPCR) agonist and antagonist by two photon fluorescence laser microscopy. Journal of the American Chemical Society. 126: 7160-1. PMID 15186137 DOI: 10.1021/Ja049473M |
0.478 |
|
| 2004 |
Elmagbari NO, Egleton RD, Palian MM, Lowery JJ, Schmid WR, Davis P, Navratilova E, Dhanasekaran M, Keyari CM, Yamamura HI, Porreca F, Hruby VJ, Polt R, Bilsky EJ. Antinociceptive structure-activity studies with enkephalin-based opioid glycopeptides. The Journal of Pharmacology and Experimental Therapeutics. 311: 290-7. PMID 15166257 DOI: 10.1124/Jpet.104.069393 |
0.745 |
|
| 2004 |
Navratilova E, Varga EV, Stropova D, Jambrosic JC, Roeske WR, Yamamura HI. Mutation S363A in the human delta-opioid receptor selectively reduces down-regulation by a peptide agonist. European Journal of Pharmacology. 485: 341-3. PMID 14757159 DOI: 10.1016/J.Ejphar.2003.11.067 |
0.73 |
|
| 2004 |
Tóth G, Keresztes A, Tömböly C, Péter A, Fülöp F, Tourwé D, Navratilova E, Varga É, Roeske WR, Yamamura HI, Szucs M, Borsodi A. New endomorphin analogs with mu-agonist and delta-antagonist properties Pure and Applied Chemistry. 76: 951-957. DOI: 10.1351/Pac200476050951 |
0.764 |
|
| 2004 |
Tóth G, Keresztes A, Tömböly C, Péter A, Fülöp F, Tourwé D, Navratilova E, Varga E, Roeske WR, Yamamura HI, Szucs M, Borsodi A. New endomorphin analogs with μ-agonist and δ-antagonist properties Pure and Applied Chemistry. 76: 951-957. |
0.648 |
|
| 2003 |
Varga EV, Yamamura HI, Rubenzik MK, Stropova D, Navratilova E, Roeske WR. Molecular mechanisms of excitatory signaling upon chronic opioid agonist treatment. Life Sciences. 74: 299-311. PMID 14607258 DOI: 10.1016/J.Lfs.2003.09.017 |
0.831 |
|
| 2003 |
Alves ID, Salamon Z, Varga E, Yamamura HI, Tollin G, Hruby VJ. Direct observation of G-protein binding to the human delta-opioid receptor using plasmon-waveguide resonance spectroscopy. The Journal of Biological Chemistry. 278: 48890-7. PMID 14522991 DOI: 10.1074/Jbc.M306866200 |
0.478 |
|
| 2003 |
Varga EV, Rubenzik MK, Stropova D, Sugiyama M, Grife V, Hruby VJ, Rice KC, Roeske WR, Yamamura HI. Converging protein kinase pathways mediate adenylyl cyclase superactivation upon chronic delta-opioid agonist treatment. The Journal of Pharmacology and Experimental Therapeutics. 306: 109-15. PMID 12660310 DOI: 10.1124/Jpet.103.049643 |
0.812 |
|
| 2003 |
Hosohata K, Varga EV, Alfaro-Lopez J, Tang X, Vanderah TW, Porreca F, Hruby VJ, Roeske WR, Yamamura HI. (2S,3R) beta-methyl-2',6'-dimethyltyrosine-L-tetrahydroisoquinoline-3-carboxylic acid [(2S,3R)TMT-L-Tic-OH] is a potent, selective delta-opioid receptor antagonist in mouse brain. The Journal of Pharmacology and Experimental Therapeutics. 304: 683-8. PMID 12538822 DOI: 10.1124/Jpet.102.042929 |
0.676 |
|
| 2003 |
Okura T, Varga EV, Hosohata Y, Navratilova E, Cowell SM, Rice K, Nagase H, Hruby VJ, Roeske WR, Yamamura HI. Agonist-specific down-regulation of the human delta-opioid receptor. European Journal of Pharmacology. 459: 9-16. PMID 12505529 DOI: 10.1016/S0014-2999(02)02823-6 |
0.755 |
|
| 2002 |
Varga EV, Rubenzik M, Grife V, Sugiyama M, Stropova D, Roeske WR, Yamamura HI. Involvement of Raf-1 in chronic delta-opioid receptor agonist-mediated adenylyl cyclase superactivation. European Journal of Pharmacology. 451: 101-2. PMID 12223234 DOI: 10.1016/S0014-2999(02)02220-3 |
0.834 |
|
| 2001 |
Stamer WD, Golightly SF, Hosohata Y, Ryan EP, Porter AC, Varga E, Noecker RJ, Felder CC, Yamamura HI. Cannabinoid CB(1) receptor expression, activation and detection of endogenous ligand in trabecular meshwork and ciliary process tissues. European Journal of Pharmacology. 431: 277-86. PMID 11730719 DOI: 10.1016/S0014-2999(01)01438-8 |
0.429 |
|
| 2001 |
Rubenzik M, Varga E, Stropova D, Roeske WR, Yamamura HI. Expression of alpha-transducin in Chinese hamster ovary cells stably transfected with the human delta-opioid receptor attenuates chronic opioid agonist-induced adenylyl cyclase superactivation. Molecular Pharmacology. 60: 1076-82. PMID 11641436 DOI: 10.1124/Mol.60.5.1076 |
0.797 |
|
| 2001 |
Hosohata Y, Varga EV, Stropova D, Li X, Knapp RJ, Hruby VJ, Rice KC, Nagase H, Roeske WR, Yamamura HI. Mutation W284L of the human delta opioid receptor reveals agonist specific receptor conformations for G protein activation. Life Sciences. 68: 2233-42. PMID 11358332 DOI: 10.1016/S0024-3205(01)01011-6 |
0.485 |
|
| 2001 |
Liao S, Shenderovich M, Kövér KE, Zhang Z, Hosohata K, Davis P, Porreca F, Yamamura HI, Hurby VJ. Synthesis, biology, NMR and conformation studies of the topographically constrained delta-opioid selective peptide analogs of [beta-iPrPhe(3)]deltorphin I. The Journal of Peptide Research : Official Journal of the American Peptide Society. 57: 257-76. PMID 11328484 DOI: 10.1046/J.1397-002X.2000.00000.X |
0.583 |
|
| 2001 |
Lipkowski AW, Misicka A, Hosohata K, Davis P, Yamamura HI, Porreca F, Hruby VJ. Biological properties of Phe(o)-opioid peptide analogues. Life Sciences. 68: 969-72. PMID 11213367 DOI: 10.1016/S0024-3205(00)00993-0 |
0.611 |
|
| 2000 |
Salamon Z, Cowell S, Varga E, Yamamura HI, Hruby VJ, Tollin G. Plasmon resonance studies of agonist/antagonist binding to the human delta-opioid receptor: new structural insights into receptor-ligand interactions. Biophysical Journal. 79: 2463-74. PMID 11053123 DOI: 10.1016/S0006-3495(00)76489-7 |
0.484 |
|
| 2000 |
Egleton RD, Mitchell SA, Huber JD, Janders J, Stropova D, Polt R, Yamamura HI, Hruby VJ, Davis TP. Improved bioavailability to the brain of glycosylated Met-enkephalin analogs. Brain Research. 881: 37-46. PMID 11033091 DOI: 10.1016/S0006-8993(00)02794-3 |
0.47 |
|
| 2000 |
Bilsky EJ, Egleton RD, Mitchell SA, Palian MM, Davis P, Huber JD, Jones H, Yamamura HI, Janders J, Davis TP, Porreca F, Hruby VJ, Polt R. Enkephalin glycopeptide analogues produce analgesia with reduced dependence liability. Journal of Medicinal Chemistry. 43: 2586-90. PMID 10891118 DOI: 10.1021/Jm000077Y |
0.554 |
|
| 2000 |
Witt KA, Slate CA, Egleton RD, Huber JD, Yamamura HI, Hruby VJ, Davis TP. Assessment of stereoselectivity of trimethylphenylalanine analogues of delta-opioid [D-Pen(2),D-Pen(5)]-enkephalin. Journal of Neurochemistry. 75: 424-35. PMID 10854288 DOI: 10.1046/J.1471-4159.2000.0750424.X |
0.392 |
|
| 2000 |
Hosohata K, Logan JK, Varga E, Burkey TH, Vanderah TW, Porreca F, Hruby VJ, Roeske WR, Yamamura HI. The role of the G protein gamma(2) subunit in opioid antinociception in mice. European Journal of Pharmacology. 392: R9-R11. PMID 10762674 DOI: 10.1016/S0014-2999(00)00132-1 |
0.632 |
|
| 2000 |
Bonner GG, Davis P, Stropova D, Edsall S, Yamamura HI, Porreca F, Hruby VJ. Opiate aromatic pharmacophore structure-activity relationships in CTAP analogues determined by topographical bias, two-dimensional NMR, and biological activity assays. Journal of Medicinal Chemistry. 43: 569-80. PMID 10691683 DOI: 10.1021/Jm9900218 |
0.55 |
|
| 2000 |
Hosohata Y, Vanderah TW, Burkey TH, Ossipov MH, Kovelowski CJ, Sora I, Uhl GR, Zhang X, Rice KC, Roeske WR, Hruby VJ, Yamamura HI, Lai J, Porreca F. delta-Opioid receptor agonists produce antinociception and [35S]GTPgammaS binding in mu receptor knockout mice. European Journal of Pharmacology. 388: 241-8. PMID 10675732 DOI: 10.1016/S0014-2999(99)00897-3 |
0.789 |
|
| 2000 |
Okura T, Cowell SM, Varga E, Burkey TH, Roeske WR, Hruby VJ, Yamamura HI. Differential down-regulation of the human delta-opioid receptor by SNC80 and [D-Pen(2),D-Pen(5)]enkephalin. European Journal of Pharmacology. 387: R11-3. PMID 10650167 DOI: 10.1016/S0014-2999(99)00761-X |
0.519 |
|
| 2000 |
Varga EV, Stropova D, Kim T, Wang M, Roeske WR, Yamamura HI. Coupling of human delta-opioid receptor to retinal rod transducin in Chinese hamster ovary cells. The Journal of Pharmacology and Experimental Therapeutics. 292: 209-14. PMID 10604950 |
0.32 |
|
| 1999 |
LeVan TD, Babin EA, Yamamura HI, Bloom JW. Pharmacological characterization of glucocorticoid receptors in primary human bronchial epithelial cells. Biochemical Pharmacology. 57: 1003-9. PMID 10796070 DOI: 10.1016/S0006-2952(99)00008-8 |
0.472 |
|
| 1999 |
Alfaro-Lopez J, Okayama T, Hosohata K, Davis P, Porreca F, Yamamura HI, Hruby VJ. Exploring the structure-activity relationships of [1-(4-tert-butyl-3'-hydroxy)benzhydryl-4-benzylpiperazine] (SL-3111), a high-affinity and selective delta-opioid receptor nonpeptide agonist ligand. Journal of Medicinal Chemistry. 42: 5359-68. PMID 10639279 DOI: 10.1021/Jm990337F |
0.576 |
|
| 1999 |
Hosohata K, Burkey TH, Alfaro-Lopez J, Hruby VJ, Roeske WR, Yamamura HI. (2S,3R)TMT-L-Tic-OH is a potent inverse agonist at the human delta-opioid receptor. European Journal of Pharmacology. 380: R9-10. PMID 10513562 DOI: 10.1016/S0014-2999(99)00516-6 |
0.454 |
|
| 1999 |
Lipkowski AW, Misicka A, Davis P, Stropova D, Janders J, Lachwa M, Porreca F, Yamamura HI, Hruby VJ. Biological activity of fragments and analogues of the potent dimeric opioid peptide, biphalin. Bioorganic & Medicinal Chemistry Letters. 9: 2763-6. PMID 10509931 DOI: 10.1016/S0960-894X(99)00464-3 |
0.591 |
|
| 1999 |
Quock RM, Burkey TH, Varga E, Hosohata Y, Hosohata K, Cowell SM, Slate CA, Ehlert FJ, Roeske WR, Yamamura HI. The delta-opioid receptor: molecular pharmacology, signal transduction, and the determination of drug efficacy. Pharmacological Reviews. 51: 503-32. PMID 10471416 |
0.339 |
|
| 1999 |
Bartosz-Bechowski H, Davis P, Slaninova J, Malatynska E, Stropova D, Porreca F, Yamamura HI, Hruby VJ. Cyclic enkephalin analogs that are hybrids of DPDPE-related peptides and metenkephalin-Arg-Gly-Leu: prohormone analogs that retain good potency and selectivity for delta opioid receptors. The Journal of Peptide Research : Official Journal of the American Peptide Society. 53: 329-36. PMID 10231722 DOI: 10.1034/J.1399-3011.1999.00033.X |
0.649 |
|
| 1999 |
Varga EV, Stropova D, Rubenzik M, Waite S, Roeske WR, Yamamura HI. Phosphorylation of adenylyl cyclase VI upon chronic delta-opioid receptor stimulation. European Journal of Pharmacology. 364: R1-3. PMID 9932732 DOI: 10.1016/S0014-2999(98)00847-4 |
0.814 |
|
| 1998 |
Li G, Haq W, Xiang L, Lou BS, Hughes R, De Leon IA, Davis P, Gillespie TJ, Romanowski M, Zhu X, Misicka A, Lipkowski AW, Porreca F, Davis TP, Yamamura HI, et al. Modifications of the 4,4'-residues and SAR studies of Biphalin, a highly potent opioid receptor active peptide. Bioorganic & Medicinal Chemistry Letters. 8: 555-60. PMID 9871617 DOI: 10.1016/S0960-894X(98)00065-1 |
0.642 |
|
| 1998 |
Malatynska E, Waite S, Wei HB, Knapp RJ, Yamamura HI, Roeske WR. Structural correlates for down-regulation of m1 and m2 muscarinic receptor subtypes. Brain Research Bulletin. 47: 285-90. PMID 9865862 DOI: 10.1016/S0361-9230(98)00110-5 |
0.452 |
|
| 1998 |
Liao S, Alfaro-Lopez J, Shenderovich MD, Hosohata K, Lin J, Li X, Stropova D, Davis P, Jernigan KA, Porreca F, Yamamura HI, Hruby VJ. De novo design, synthesis, and biological activities of high-affinity and selective non-peptide agonists of the delta-opioid receptor. Journal of Medicinal Chemistry. 41: 4767-76. PMID 9822547 DOI: 10.1021/Jm980374R |
0.652 |
|
| 1998 |
Varga EV, Stropova D, Rubenzik M, Wang M, Landsman RS, Roeske WR, Yamamura HI. Identification of adenylyl cyclase isoenzymes in CHO and B82 cells. European Journal of Pharmacology. 348: R1-2. PMID 9652350 DOI: 10.1016/S0014-2999(98)00258-1 |
0.76 |
|
| 1998 |
Hosohata K, Burkey TH, Alfaro-Lopez J, Varga E, Hruby VJ, Roeske WR, Yamamura HI. Endomorphin-1 and endomorphin-2 are partial agonists at the human mu-opioid receptor. European Journal of Pharmacology. 346: 111-4. PMID 9617760 DOI: 10.1016/S0014-2999(98)00117-4 |
0.553 |
|
| 1998 |
Burkey TH, Ehlert FJ, Hosohata Y, Quock RM, Cowell S, Hosohata K, Varga E, Stropova D, Li X, Slate C, Nagase H, Porreca F, Hruby VJ, Roeske WR, Yamamura HI. The efficacy of delta-opioid receptor-selective drugs. Life Sciences. 62: 1531-6. PMID 9585131 DOI: 10.1016/S0024-3205(98)00102-7 |
0.562 |
|
| 1998 |
Slaninova J, Appleyard SM, Misicka A, Lipkowski AW, Knapp RJ, Weber SJ, Davis TP, Yamamura HI, Hruby VJ. [125I-Tyr1]biphalin binding to opioid receptors of rat brain and NG108-15 cell membranes. Life Sciences. 62: PL199-204. PMID 9570343 DOI: 10.1016/S0024-3205(98)00058-7 |
0.511 |
|
| 1998 |
Landsman RS, Makriyannis A, Deng H, Consroe P, Roeske WR, Yamamura HI. AM630 is an inverse agonist at the human cannabinoid CB1 receptor. Life Sciences. 62: PL109-13. PMID 9496703 DOI: 10.1016/S0024-3205(97)01187-9 |
0.463 |
|
| 1998 |
Olczak J, Kaczmarek K, Maszczyńska I, Lisowski M, Stropova D, Hruby VJ, Yamamura HI, Lipkowski AW, Zabrocki J. Consequences of cis-amide bond simulation in opioid peptides International Journal of Peptide Research and Therapeutics. 5: 437-440. DOI: 10.1007/Bf02443502 |
0.42 |
|
| 1997 |
Hruby VJ, Bartosz-Bechowski H, Davis P, Slaninova J, Zalewska T, Stropova D, Porreca F, Yamamura HI. Cyclic enkephalin analogues with exceptional potency and selectivity for delta-opioid receptors. Journal of Medicinal Chemistry. 40: 3957-62. PMID 9397176 DOI: 10.1021/Jm9704762 |
0.595 |
|
| 1997 |
Burkey TH, Quock RM, Consroe P, Ehlert FJ, Hosohata Y, Roeske WR, Yamamura HI. Relative efficacies of cannabinoid CB1 receptor agonists in the mouse brain. European Journal of Pharmacology. 336: 295-8. PMID 9384246 DOI: 10.1016/S0014-2999(97)01255-7 |
0.428 |
|
| 1997 |
Landsman RS, Burkey TH, Consroe P, Roeske WR, Yamamura HI. SR141716A is an inverse agonist at the human cannabinoid CB1 receptor. European Journal of Pharmacology. 334: R1-2. PMID 9346339 DOI: 10.1016/S0014-2999(97)01160-6 |
0.443 |
|
| 1997 |
Haaseth RC, Zalewska T, Davis P, Yamamura HI, Porreca F, Hruby VJ. Para-substituted phenylalanine-4 analogues of [L-Ala3]DPDPE: highly selective delta opioid receptor ligands. The Journal of Peptide Research : Official Journal of the American Peptide Society. 50: 171-7. PMID 9309580 DOI: 10.1111/J.1399-3011.1997.Tb01182.X |
0.644 |
|
| 1997 |
Katsura Y, Zhang X, Homma K, Rice KC, Calderon SN, Rothman RB, Yamamura HI, Davis P, Flippen-Anderson JL, Xu H, Becketts K, Foltz EJ, Porreca F. Probes for narcotic receptor-mediated phenomena. 25. Synthesis and evaluation of N-alkyl-substituted (alpha-piperazinylbenzyl)benzamides as novel, highly selective delta opioid receptor agonists. Journal of Medicinal Chemistry. 40: 2936-47. PMID 9288176 DOI: 10.1021/Jm970106D |
0.623 |
|
| 1997 |
Hosohata K, Quock RM, Hosohata Y, Burkey TH, Makriyannis A, Consroe P, Roeske WR, Yamamura HI. AM630 is a competitive cannabinoid receptor antagonist in the guinea pig brain. Life Sciences. 61: PL115-8. PMID 9284087 DOI: 10.1016/S0024-3205(97)00596-1 |
0.458 |
|
| 1997 |
Misicka A, Cavagnero S, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Synthesis and biological properties of beta-MePhe3 analogues of deltorphin I and dermenkephalin: influence of biased chi 1 Phe3 residues on peptide recognition for delta-opioid receptors. The Journal of Peptide Research : Official Journal of the American Peptide Society. 50: 48-54. PMID 9273887 DOI: 10.1111/J.1399-3011.1997.Tb00619.X |
0.601 |
|
| 1997 |
Quock RM, Hosohata Y, Knapp RJ, Burkey TH, Hosohata K, Zhang X, Rice KC, Nagase H, Hruby VJ, Porreca F, Roeske WR, Yamamura HI. Relative efficacies of delta-opioid receptor agonists at the cloned human delta-opioid receptor. European Journal of Pharmacology. 326: 101-4. PMID 9178661 DOI: 10.1016/S0014-2999(97)83488-7 |
0.629 |
|
| 1997 |
Patel D, McKinley BD, Davis TP, Porreca F, Yamamura HI, Hruby VJ. Peptide targeting and delivery across the blood-brain barrier utilizing synthetic triglyceride esters: design, synthesis, and bioactivity. Bioconjugate Chemistry. 8: 434-41. PMID 9177851 DOI: 10.1021/Bc970027G |
0.486 |
|
| 1997 |
Burkey TH, Quock RM, Consroe P, Roeske WR, Yamamura HI. delta 9-Tetrahydrocannabinol is a partial agonist of cannabinoid receptors in mouse brain. European Journal of Pharmacology. 323: R3-4. PMID 9128853 DOI: 10.1016/S0014-2999(97)00146-5 |
0.416 |
|
| 1997 |
Bonner GG, Davis P, Stropova D, Ferguson R, Yamamura HI, Porreca F, Hruby VJ. Opioid peptides: simultaneous delta agonism and mu antagonism in somatostatin analogues. Peptides. 18: 93-100. PMID 9114458 DOI: 10.1016/S0196-9781(96)00242-2 |
0.685 |
|
| 1997 |
Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Structure-activity relationship of biphalin. The synthesis and biological activities of new analogues with modifications in positions 3 and 4. Life Sciences. 60: 1263-9. PMID 9096243 DOI: 10.1016/S0024-3205(97)00069-6 |
0.652 |
|
| 1997 |
Hosohata Y, Quock RM, Hosohata K, Makriyannis A, Consroe P, Roeske WR, Yamamura HI. AM630 antagonism of cannabinoid-stimulated [35S]GTP gamma S binding in the mouse brain. European Journal of Pharmacology. 321: R1-3. PMID 9083796 DOI: 10.1016/S0014-2999(97)00047-2 |
0.44 |
|
| 1997 |
Liao S, Lin J, Shenderovich MD, Han Y, Hasohata K, Davis P, Qiu W, Porreca F, Yamamura HI, Hruby VJ. The stereochemical requirements of the novel δ-opioid selective dipeptide antagonist TMT-Tic Bioorganic & Medicinal Chemistry Letters. 7: 3049-3052. DOI: 10.1016/S0960-894X(97)10145-7 |
0.574 |
|
| 1997 |
Liao S, Lin J, Shenderovich MD, Han Y, Hasohata K, Davis P, Qiu W, Porreca F, Yamamura HI, Hruby VJ. The stereochemical requirements of the novel δ-opioid selective dipeptide antagonist TMT-Tic Bioorganic and Medicinal Chemistry Letters. 7: 3049-3052. |
0.346 |
|
| 1996 |
Millard SL, Bloom JW, Yamamura HI. Heterogeneity of tachykinin receptors in the rabbit lung. Neurochemical Research. 21: 277-83. PMID 9182253 DOI: 10.1007/BF02529145 |
0.397 |
|
| 1996 |
Varga EV, Li X, Stropova D, Zalewska T, Landsman RS, Knapp RJ, Malatynska E, Kawai K, Mizusura A, Nagase H, Calderon SN, Rice K, Hruby VJ, Roeske WR, Yamamura HI. The third extracellular loop of the human delta-opioid receptor determines the selectivity of delta-opioid agonists. Molecular Pharmacology. 50: 1619-24. PMID 8967985 |
0.454 |
|
| 1996 |
Qian X, Liao S, Stropova D, Yamamura HI, Hruby VJ. Novel scaffolds for non-peptide mimetics of delta opioid receptor agonists based on peptide leads. Regulatory Peptides. 65: 79-82. PMID 8876039 DOI: 10.1016/0167-0115(96)00075-4 |
0.457 |
|
| 1996 |
Boteju LW, Nikiforovich GV, Haskell-Luevano C, Fang SN, Zalewska T, Stropova D, Yamamura HI, Hruby VJ. The use of topographical constraints in receptor mapping: investigation of the topographical requirements of the tryptophan 30 residue for receptor binding of Asp-Tyr-D-Phe-Gly-Trp-(N-Me)Nle-Asp-Phe-NH2 (SNF 9007), a cholecystokinin (26-33) analogue that binds to both CCK-B and delta-opioid receptors. Journal of Medicinal Chemistry. 39: 4120-4. PMID 8831778 DOI: 10.1021/Jm960078J |
0.532 |
|
| 1996 |
Malatynska E, Wang Y, Knapp RJ, Waite S, Calderon S, Rice K, Hruby VJ, Yamamura HI, Roeske WR. Human delta opioid receptor: functional studies on stably transfected Chinese hamster ovary cells after acute and chronic treatment with the selective nonpeptidic agonist SNC-80. The Journal of Pharmacology and Experimental Therapeutics. 278: 1083-9. PMID 8819489 |
0.445 |
|
| 1996 |
Misicka A, Maszczynska I, Lipkowski AW, Stropova D, Yamamura HI, Hruby VJ. Synthesis and biological properties of gamma-glutamyl-dermorphin, a prodrug. Life Sciences. 58: 905-11. PMID 8786696 DOI: 10.1016/0024-3205(96)00033-1 |
0.387 |
|
| 1996 |
Vanderah TW, Bernstein RN, Yamamura HI, Hruby VJ, Porreca F. Enhancement of morphine antinociception by a CCKB antagonist in mice is mediated via opioid delta receptors. The Journal of Pharmacology and Experimental Therapeutics. 278: 212-9. PMID 8764354 |
0.618 |
|
| 1996 |
Li X, Varga EV, Stropova D, Zalewska T, Malatynska E, Knapp RJ, Roeske WR, Yamamura HI. delta-Opioid receptor: the third extracellular loop determines naltrindole selectivity. European Journal of Pharmacology. 300: R1-2. PMID 8741185 DOI: 10.1016/0014-2999(96)00098-2 |
0.529 |
|
| 1996 |
Edsall SA, Knapp RJ, Vanderah TW, Roeske WR, Consroe P, Yamamura HI. Antisense oligodeoxynucleotide treatment to the brain cannabinoid receptor inhibits antinociception. Neuroreport. 7: 593-6. PMID 8730837 DOI: 10.1097/00001756-199601310-00052 |
0.667 |
|
| 1996 |
Lung FD, Meyer JP, Lou BS, Xiang L, Li G, Davis P, DeLeon IA, Yamamura HI, Porreca F, Hruby VJ. Effects of modifications of residues in position 3 of dynorphin A(1-11)-NH2 on kappa receptor selectivity and potency. Journal of Medicinal Chemistry. 39: 2456-60. PMID 8691442 DOI: 10.1021/jm950655o |
0.586 |
|
| 1996 |
Lung FD, Collins N, Stropova D, Davis P, Yamamura HI, Porreca F, Hruby VJ. Design, synthesis, and biological activities of cyclic lactam peptide analogues of dynorphine A(1-11)-NH2. Journal of Medicinal Chemistry. 39: 1136-41. PMID 8676350 DOI: 10.1021/Jm950369C |
0.644 |
|
| 1996 |
Knapp RJ, Santoro G, De Leon IA, Lee KB, Edsall SA, Waite S, Malatynska E, Varga E, Calderon SN, Rice KC, Rothman RB, Porreca F, Roeske WR, Yamamura HI. Structure-activity relationships for SNC80 and related compounds at cloned human delta and mu opioid receptors. The Journal of Pharmacology and Experimental Therapeutics. 277: 1284-91. PMID 8667189 |
0.492 |
|
| 1996 |
Qian X, Shenderovich MD, Kover KE, Davis P, Horvath R, Zalewska T, Yamamura HI, Porreca F, Hruby VJ. Probing the stereochemical requirements for receptor recognition of δ opioid agonists through topographic modifications in position 1 Journal of the American Chemical Society. 118: 7280-7290. DOI: 10.1021/Ja954241W |
0.61 |
|
| 1995 |
Knapp RJ, Landsman R, Waite S, Malatynska E, Varga E, Haq W, Hruby VJ, Roeske WR, Nagase H, Yamamura HI. Properties of TAN-67, a nonpeptidic delta-opioid receptor agonist, at cloned human delta- and mu-opioid receptors. European Journal of Pharmacology. 291: 129-34. PMID 8566162 DOI: 10.1016/0922-4106(95)90134-5 |
0.563 |
|
| 1995 |
Lung FD, Meyer JP, Li G, Lou BS, Stropova D, Davis P, Yamamura HI, Porreca F, Hruby VJ. Highly kappa receptor-selective dynorphin A analogues with modifications in position 3 of dynorphin A(1-11)-NH2. Journal of Medicinal Chemistry. 38: 585-6. PMID 7861405 DOI: 10.1021/Jm00004A002 |
0.591 |
|
| 1995 |
Slaninova J, Knapp RJ, Weber SJ, Davis TP, Fang SN, Hruby VJ, Yamamura HI. [125I]SNF 8702: a selective radioligand for CCKB receptors. Peptides. 16: 221-4. PMID 7784252 DOI: 10.1016/0196-9781(94)00168-5 |
0.445 |
|
| 1995 |
Knapp RJ, Malatynska E, Collins N, Fang L, Wang JY, Hruby VJ, Roeske WR, Yamamura HI. Molecular biology and pharmacology of cloned opioid receptors. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 9: 516-25. PMID 7737460 DOI: 10.1096/Fasebj.9.7.7737460 |
0.542 |
|
| 1995 |
Malatynska E, Knapp RJ, Stropova D, Varga E, Yamamura HI. The role of the Val353 residue in antagonist binding to rat CCK-B receptors. Neuroreport. 6: 1325-9. PMID 7669996 DOI: 10.1097/00001756-199506090-00024 |
0.455 |
|
| 1995 |
Meyer JP, Davis P, Lee KB, Porreca F, Yamamura HI, Hruby VJ. Synthesis using a Fmoc-based strategy and biological activities of some reduced peptide bond pseudopeptide analogues of dynorphin A1. Journal of Medicinal Chemistry. 38: 3462-8. PMID 7658433 DOI: 10.1021/Jm00018A006 |
0.595 |
|
| 1995 |
Hruby VJ, Yamamura HI, Porreca F. Molecular organization of receptors. Efficacy, agonists, and antagonists. Annals of the New York Academy of Sciences. 757: 7-22. PMID 7611710 DOI: 10.1111/J.1749-6632.1995.Tb17461.X |
0.579 |
|
| 1995 |
Malatynska E, De Leon I, Allen D, Yamamura HI. Effects of amitriptyline on GABA-stimulated 36CI- uptake in relation to a behavioral model of depression. Brain Research Bulletin. 37: 53-9. PMID 7606479 DOI: 10.1016/0361-9230(94)00257-6 |
0.316 |
|
| 1995 |
Malatynska E, Wang Y, Knapp RJ, Santoro G, Li X, Waite S, Roeske WR, Yamamura HI. Human delta opioid receptor: a stable cell line for functional studies of opioids. Neuroreport. 6: 613-6. PMID 7605911 |
0.417 |
|
| 1995 |
Misicka A, Lipkowski AW, Slaninova J, Davis P, Yamamura HI, Porreca F, Hruby VJ. The synthesis and opioid receptor binding affinities of analogues of dermorphin and its N-terminal tetrapeptide fragment with dibasic acids in position 2. Life Sciences. 57: 1633-40. PMID 7475903 DOI: 10.1016/0024-3205(95)02142-6 |
0.597 |
|
| 1995 |
Li X, Knapp RJ, Stropova D, Varga E, Wang Y, Malatynska E, Calderont S, Ricet K, Rothman R, Porreca F, Hruby VJ, Roeske WR, Yamamura HI. Trp284 of the Human δ Opioid Receptor is Required for SNC121 Binding but Not Binding of pCl-DPDPE, Deltorphin II or Naltrindole Analgesia. 1: 539-542. DOI: 10.3727/107156995819563302 |
0.556 |
|
| 1995 |
Hruby VJ, Davis T, Polt R, Porreca F, O’Brien D, Yamamura H, Bartosz H, Szabo L, Gillespie T, Williams S, Misicka A, Lipkowski A, Qian X, Li G, Patel D, et al. DESIGN AND SYNTHESIS OF PEPTIDE LIGANDS WITH UNIQUE BIOCHEMICAL AND BIOLOGICAL PROFILES AT OPIOID RECEPTORS THAT CROSS THE BLOOD BRAIN BARRIER Analgesia. 1: 469-472. DOI: 10.3727/107156995819562961 |
0.533 |
|
| 1995 |
Santoro G, Knapp R, Malatinska E, Varga E, Li X, Lee K, Edsall S, Stropova D, Leon ID, Wang Y, Waite S, Roeske WR, Yamamura HI. Cloning, expression and pharmacological characterization of a human delta opioid receptor Behavioural Pharmacology. 6: 136. DOI: 10.1097/00008877-199505001-00162 |
0.487 |
|
| 1995 |
Malatynska E, Wang Y, Knapp RJ, Santoro G, Li X, Waite S, Roeske WR, Yamamura HI. Human δ opioid receptor: A stable cell line for functional studies of opioids Neuroreport. 6: 613-616. DOI: 10.1097/00001756-199503000-00007 |
0.513 |
|
| 1995 |
Misicka A, Lipkowski AW, Stropova D, Davis P, Porreca F, Yamamura HI, Hruby VJ. Amino acids with amphiphilic side chains: Deltorphin analogues with Phe3 replaced by all β-hydroxyphenylalanine diastereoisomers Letters in Peptide Science. 2: 203-205. DOI: 10.1007/Bf00119153 |
0.495 |
|
| 1995 |
Lipkowski AW, Misicka A, Porreca F, Davis P, Yamamura HI, Stropova D, Hruby VJ. Benzomorphan alkaloids: Natural peptidomimetics of opioid peptide pharmacophores Letters in Peptide Science. 2: 177-181. DOI: 10.1007/Bf00119147 |
0.539 |
|
| 1994 |
Bartosz-Bechowski H, Davis P, Zalewska T, Slaninova J, Porreca F, Yamamura HI, Hruby VJ. Cyclic enkephalin analogs with exceptional potency at peripheral delta opioid receptors. Journal of Medicinal Chemistry. 37: 146-50. PMID 8289188 DOI: 10.1021/Jm00027A018 |
0.639 |
|
| 1994 |
Misicka A, Lipkowski AW, Horvath R, Davis P, Yamamura HI, Porreca F, Hruby VJ. Design of cyclic deltorphins and dermenkephalins with a disulfide bridge leads to analogues with high selectivity for delta-opioid receptors. Journal of Medicinal Chemistry. 37: 141-5. PMID 8289187 DOI: 10.1021/Jm00027A017 |
0.617 |
|
| 1994 |
Haaseth RC, Horan PJ, Bilsky EJ, Davis P, Zalewska T, Slaninova J, Yamamura HI, Weber SJ, Davis TP, Porreca F. [L-Ala3]DPDPE: a new enkephalin analog with a unique opioid receptor activity profile. Further evidence of delta-opioid receptor multiplicity. Journal of Medicinal Chemistry. 37: 1572-7. PMID 8201592 DOI: 10.1021/Jm00037A007 |
0.632 |
|
| 1994 |
Knapp RJ, Malatynska E, Hashimoto S, Fang S, Hunt M, Wamsley JK, Peterson P, Zalewska T, Hruby VJ, Yamamura HI. [3H]SNF8702 autoradiography of CCK-B receptors in guinea pig brain and studies with a cloned rat CCK-B receptor. Annals of the New York Academy of Sciences. 713: 380-3. PMID 8185194 DOI: 10.1111/J.1749-6632.1994.Tb44099.X |
0.412 |
|
| 1994 |
Fang L, Knapp RJ, Horvath R, Matsunaga TO, Haaseth RC, Hruby VJ, Porreca F, Yamamura HI. Characterization of [3H]naltrindole binding to delta opioid receptors in mouse brain and mouse vas deferens: evidence for delta opioid receptor heterogeneity. The Journal of Pharmacology and Experimental Therapeutics. 268: 836-46. PMID 8113996 |
0.438 |
|
| 1994 |
Rao RK, Levenson S, Fang SN, Hruby VJ, Yamamura HI, Porreca F. Characterization of SNF 9007, a novel cholecystokinin/opoid ligand in mouse ileum in vitro: evidence for involvement of cholecystokininA and cholecystokininB receptors in regulation of ion transport. The Journal of Pharmacology and Experimental Therapeutics. 268: 1003-9. PMID 8113956 |
0.347 |
|
| 1994 |
Polt R, Porreca F, Szabò LZ, Bilsky EJ, Davis P, Abbruscato TJ, Davis TP, Harvath R, Yamamura HI, Hruby VJ. Glycopeptide enkephalin analogues produce analgesia in mice: evidence for penetration of the blood-brain barrier. Proceedings of the National Academy of Sciences of the United States of America. 91: 7114-8. PMID 8041755 DOI: 10.1073/Pnas.91.15.7114 |
0.573 |
|
| 1994 |
Qian X, Kövér KE, Shenderovich MD, Lou BS, Misicka A, Zalewska T, Horváth R, Davis P, Bilsky EJ, Porreca F, Yamamura HI, Hruby VJ. Newly discovered stereochemical requirements in the side-chain conformation of δ opioid agonists for recognizing opioid δ receptors Journal of Medicinal Chemistry. 37: 1746-1757. PMID 8021915 DOI: 10.1021/JM00038A004 |
0.612 |
|
| 1994 |
Ehlert FJ, Roeske WR, Yamamura HI. Muscarinic receptors and novel strategies for the treatment of age-related brain disorders. Life Sciences. 55: 2135-45. PMID 7997072 DOI: 10.1016/0024-3205(94)00394-7 |
0.439 |
|
| 1994 |
Wild KD, Porreca F, Yamamura HI, Raffa RB. Differentiation of receptor subtypes by thermodynamic analysis: application to opioid delta receptors. Proceedings of the National Academy of Sciences of the United States of America. 91: 12018-21. PMID 7991576 DOI: 10.1073/pnas.91.25.12018 |
0.636 |
|
| 1994 |
Meyer JP, Collins N, Lung FD, Davis P, Zalewska T, Porreca F, Yamamura HI, Hruby VJ. Design, synthesis, and biological properties of highly potent cyclic dynorphin A analogues. Analogues cyclized between positions 5 and 11. Journal of Medicinal Chemistry. 37: 3910-7. PMID 7966152 DOI: 10.1021/Jm00049A010 |
0.557 |
|
| 1994 |
Sora I, Richman J, Santoro G, Wei HB, Wang Y, Vanderah T, Horvath R, Nguyen M, Waite S, Roeske WR, Yamamura HI. The Cloning and Expression of a Human Creatine Transporter Biochemical and Biophysical Research Communications. 204: 419-427. PMID 7945388 DOI: 10.1006/bbrc.1994.2475 |
0.52 |
|
| 1994 |
Knapp RJ, Malatynska E, Peterson P, Zalewska T, Fang S, Hruby VJ, Smith TL, Yamamura HI. [N-methylnorleucine-(28,31)]cholecystokinin-(26-33) (SNF 8702) activity at a cloned rat CCKB receptor. European Journal of Pharmacology. 269: 133-8. PMID 7851490 DOI: 10.1016/0922-4106(94)90079-5 |
0.49 |
|
| 1994 |
Wei HB, Yamamura HI, Roeske WR. Down-regulation and desensitization of the muscarinic M1 and M2 receptors in transfected fibroblast B82 cells. European Journal of Pharmacology. 268: 381-91. PMID 7805762 DOI: 10.1016/0922-4106(94)90063-9 |
0.419 |
|
| 1994 |
Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Delta opioid receptor selective ligands; DPLPE-deltorphin chimeric peptide analogues. International Journal of Peptide and Protein Research. 44: 80-4. PMID 7718035 DOI: 10.1111/J.1399-3011.1994.Tb00407.X |
0.623 |
|
| 1994 |
Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Delta opioid receptor selective ligands; DPLPE-deltorphin chimeric peptide analogues. International Journal of Peptide and Protein Research. 44: 607. PMID 7705984 |
0.406 |
|
| 1994 |
Vanderah TW, Lai J, Yamamura HI, Porreca F. Antisense oligodeoxynucleotide to the CCKB receptor produces naltrindole- and [Leu5]enkephalin antiserum-sensitive enhancement of morphine antinociception. Neuroreport. 5: 2601-5. PMID 7696612 DOI: 10.1097/00001756-199412000-00049 |
0.792 |
|
| 1994 |
Rao RK, Levenson S, Fang SN, Hruby VJ, Yamamura HI, Porreca F. Role of substance P in the regulation of ion transport by CCKA and CCKB receptors in mouse ileum. Annals of the New York Academy of Sciences. 713: 420-1. PMID 7514373 DOI: 10.1111/J.1749-6632.1994.Tb44113.X |
0.491 |
|
| 1994 |
Malatynska E, Knapp R, Fang L, Li X, Wang Y, Santoro G, Leon ID, Waite S, Roeske W, Yamamura H. Cloning, expression and partial characterization of a human delta opioid receptor Regulatory Peptides. 54: 173-174. DOI: 10.1016/0167-0115(94)90446-4 |
0.483 |
|
| 1994 |
Hruby VJ, Collins N, Lung FD, Meyer JP, Davis TP, Yamamura HI, Porreca F. Design of peptides and peptidomimetics for delta and kappa opioid receptor subtypes Regulatory Peptides. 54: 123-124. DOI: 10.1016/0167-0115(94)90420-0 |
0.617 |
|
| 1994 |
Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Structure-activity relationships of analogues of higly potent opioid peptide, biphalin Regulatory Peptides. 53: S131-S132. DOI: 10.1016/0167-0115(94)90276-3 |
0.495 |
|
| 1994 |
Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Topographic model of delta opioid selective ligands; DPLPE-deltorphin hybrid analogues Regulatory Peptides. 53: S129-S130. DOI: 10.1016/0167-0115(94)90275-5 |
0.608 |
|
| 1994 |
Hruby VJ, Misicka A, Lipkowski AW, Haaseth R, Bartosz H, Qian X, Collins N, Meyer JP, Szabo L, Polt R, Porreca F, Davis T, Yamamura HI. New opioid compounds in analgesia Regulatory Peptides. 53: S71-S72. DOI: 10.1016/0167-0115(94)90246-1 |
0.659 |
|
| 1993 |
Wild KD, Horan PJ, Misicka A, Lipkowski A, Haaseth RC, Matsunaga TO, Hruby VJ, Toth G, Borsodi A, Yamamura HI. Pseudoirreversible binding characteristics of [D-Ala2,Glu4]deltorphin and its Cys4 substituted derivative to delta-opioid receptors. European Journal of Pharmacology. 246: 25-31. PMID 8394818 DOI: 10.1016/0922-4106(93)90005-T |
0.49 |
|
| 1993 |
Horan PJ, Mattia A, Bilsky EJ, Weber S, Davis TP, Yamamura HI, Malatynska E, Appleyard SM, Slaninova J, Misicka A. Antinociceptive profile of biphalin, a dimeric enkephalin analog. The Journal of Pharmacology and Experimental Therapeutics. 265: 1446-54. PMID 8389867 |
0.343 |
|
| 1993 |
Horan PJ, Wild KD, Misicka A, Lipkowski A, Haaseth RC, Hruby VJ, Weber SJ, Davis TP, Yamamura HI, Porreca F. Agonist and antagonist profiles of [D-Ala2,Glu4]deltorphin and its [Cys4]- and [Ser4]-substituted derivatives: further evidence of opioid delta receptor multiplicity. The Journal of Pharmacology and Experimental Therapeutics. 265: 896-902. PMID 8388462 |
0.403 |
|
| 1993 |
Henderson AK, Roeske WR, Smith TL, Yamamura HI. Desensitization of neurokinin A receptors expressed by B82 fibroblasts. European Journal of Pharmacology. 245: 75-8. PMID 8386670 DOI: 10.1016/0922-4106(93)90172-6 |
0.424 |
|
| 1993 |
Horan PJ, Wild KD, Kazmierski WM, Ferguson R, Hruby VJ, Weber SJ, Davis TP, Fang L, Knapp RJ, Yamamura HI. Unexpected antinociceptive potency of cyclic [D-Tca1]CTAP: potential for a novel mechanism of action. European Journal of Pharmacology. 233: 53-62. PMID 8386089 DOI: 10.1016/0014-2999(93)90348-L |
0.503 |
|
| 1993 |
Parola AL, Yamamura HI, Laird HE. Peripheral-type benzodiazepine receptors. Life Sciences. 52: 1329-42. PMID 8385255 DOI: 10.1016/0024-3205(93)90168-3 |
0.466 |
|
| 1993 |
Wild KD, Fang L, McNutt RW, Chang KJ, Toth G, Borsodi A, Yamamura HI, Porreca F. Binding of BW 373U86, a non-peptidic delta opioid receptor agonist, is not regulated by guanine nucleotides and sodium. European Journal of Pharmacology. 246: 289-92. PMID 8223952 DOI: 10.1016/0922-4106(93)90044-A |
0.643 |
|
| 1993 |
Kawasaki AM, Knapp RJ, Kramer TH, Walton A, Wire WS, Hashimoto S, Yamamura HI, Porreca F, Burks TF, Hruby VJ. Design and synthesis of highly potent and selective cyclic dynorphin A analogs. 2. New analogs. Journal of Medicinal Chemistry. 36: 750-7. PMID 8096246 DOI: 10.1021/Jm00058A012 |
0.672 |
|
| 1993 |
Fujiwara Y, Tomita H, Hikiji M, Kashihara K, Otsuki S, Ohnuki T, Hamagishi Y, Oki T, Sora I, Roeske WR, Yamamura HI. Characterization of a cloned rat serotonin 5-HT1A receptor expressed in the HeLa cell line Life Sciences. 52: 949-958. PMID 8095315 DOI: 10.1016/0024-3205(93)90530-G |
0.458 |
|
| 1993 |
Kawasaki AM, Knapp RJ, Walton A, Wire WS, Zalewska T, Yamamura HI, Porreca F, Burks TF, Hruby VJ. Syntheses, opioid binding affinities, and potencies of dynorphin A analogues substituted in positions, 1, 6, 7, 8 and 10. International Journal of Peptide and Protein Research. 42: 411-9. PMID 7906258 DOI: 10.1111/J.1399-3011.1993.Tb00148.X |
0.618 |
|
| 1993 |
Witt-Enderby PA, Yamamura HI, Halonen M, Palmer JD, Bloom JW. Chronic exposure to a beta 2-adrenoceptor agonist increases the airway response to methacholine. European Journal of Pharmacology. 241: 121-3. PMID 7901034 DOI: 10.1016/0014-2999(93)90942-B |
0.31 |
|
| 1993 |
Boteju LW, Zalewska T, Yamamura HI, Hruby VJ. Tryptophan-norleucine 1,5-disubstituted tetrazoles as cis peptide bond mimics: Investigation of the bioactive conformation of a potent and selective peptide for the cholecystokinin-B receptor Bioorganic and Medicinal Chemistry Letters. 3: 2011-2016. DOI: 10.1016/S0960-894X(01)81005-2 |
0.39 |
|
| 1993 |
Hristova-Kazmierski MK, Horan P, Davis P, Yamamura HI, Kramer T, Horvath R, Kazmierski WM, Porreca F, Hruby VJ. A new approach to enhance bioavailability of biologically active peptides: conjugation of a δ opioid agonist to β-cyclodextrin Bioorganic and Medicinal Chemistry Letters. 3: 831-834. DOI: 10.1016/S0960-894X(00)80675-7 |
0.588 |
|
| 1993 |
Kovacs I, Yamamura H, Waite S, Roeske W. Pharmacological comparison of the cloned rat and human M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line Life Sciences. 52: 577. DOI: 10.1016/0024-3205(93)90371-9 |
0.349 |
|
| 1992 |
Lai J, Nunan L, Waite SL, Ma SW, Bloom JW, Roeske WR, Yamamura HI. Chimeric M1/M2 muscarinic receptors: correlation of ligand selectivity and functional coupling with structural modifications. The Journal of Pharmacology and Experimental Therapeutics. 262: 173-80. PMID 1625198 |
0.303 |
|
| 1992 |
Mahesh VK, Nunan LM, Halonen M, Yamamura HI, Palmer JD, Bloom JW. A minority of muscarinic receptors mediate rabbit tracheal smooth muscle contraction. American Journal of Respiratory Cell and Molecular Biology. 6: 279-86. PMID 1540392 DOI: 10.1165/Ajrcmb/6.3.279 |
0.451 |
|
| 1992 |
Kazmierski WM, Ferguson RD, Knapp RJ, Lui GK, Yamamura HI, Hruby VJ. Reduced peptide bond cyclic somatostatin based opioid octapeptides. Synthesis, conformational properties and pharmacological characterization. International Journal of Peptide and Protein Research. 39: 401-14. PMID 1358847 DOI: 10.1111/J.1399-3011.1992.Tb01444.X |
0.494 |
|
| 1992 |
Knapp RJ, Yamamura HI. Delta opioid receptor radioligands. Biochemical Pharmacology. 44: 1687-95. PMID 1333204 DOI: 10.1016/0006-2952(92)90060-V |
0.522 |
|
| 1992 |
Fang L, Knapp RJ, Matsunaga T, Weber SJ, Davis T, Hruby VJ, Yamamura HI. Synthesis of [D-Ala2,4'-125I-Phe3,Glu4]deltorphin and characterization of its delta opioid receptor binding properties. Life Sciences. 51: PL189-93. PMID 1331636 DOI: 10.1016/0024-3205(92)90628-3 |
0.566 |
|
| 1992 |
Misicka A, Lipkowski AW, Horvath R, Davis P, Kramer TH, Yamamura HI, Hruby VJ. Topographical requirements for delta opioid ligands: common structural features of dermenkephalin and deltorphin. Life Sciences. 51: 1025-32. PMID 1326067 DOI: 10.1016/0024-3205(92)90501-F |
0.455 |
|
| 1992 |
Kashihara K, Varga EV, Waite SL, Roeske WR, Yamamura HI. Cloning of the rat M3, M4 and M5 muscarinic acetylcholine receptor genes by the polymerase chain reaction (PCR) and the pharmacological characterization of the expressed genes. Life Sciences. 51: 955-71. PMID 1325587 DOI: 10.1016/0024-3205(92)90403-C |
0.32 |
|
| 1992 |
Toth G, Russell KC, Landis G, Kramer TH, Fang L, Knapp R, Davis P, Burks TF, Yamamura HI, Hruby VJ. Ring substituted and other conformationally constrained tyrosine analogues of [D-Pen2,D-Pen5]enkephalin with delta opioid receptor selectivity. Journal of Medicinal Chemistry. 35: 2384-91. PMID 1320122 DOI: 10.1021/Jm00091A006 |
0.535 |
|
| 1992 |
Yamamura MS, Horvath R, Toth G, Otvos F, Malatynska E, Knapp RJ, Porreca F, Hruby VJ, Yamamura HI. Characterization of [3H]naltrindole binding to delta opioid receptors in rat brain. Life Sciences. 50: PL119-24. PMID 1313133 DOI: 10.1016/0024-3205(92)90464-Z |
0.649 |
|
| 1992 |
Henderson AK, Yamamura HI, Maggi CA, Buck SH, Van Giersbergen PL, Roeske WR. Demonstration of a neurokinin A receptor subtype in transfected fibroblasts. European Journal of Pharmacology. 225: 175-8. PMID 1312943 DOI: 10.1016/0922-4106(92)90099-H |
0.48 |
|
| 1992 |
Horan P, Taylor J, Yamamura HI, Porreca F. Extremely long-lasting antagonistic actions of nor-binaltorphimine (nor-BNI) in the mouse tail-flick test. The Journal of Pharmacology and Experimental Therapeutics. 260: 1237-43. PMID 1312164 |
0.335 |
|
| 1992 |
Wei HB, Roeske WR, Lai J, Wanibuchi F, Hidaka K, Usuda S, Yamamura HI. Pharmacological characterization of a novel muscarinic partial agonist, YM796, in transfected cells expressing the m1 or m2 muscarinic receptor gene. Life Sciences. 50: 355-63. PMID 1310135 DOI: 10.1016/0024-3205(92)90437-T |
0.634 |
|
| 1992 |
Misicka A, Nikiforovich G, Lipkowski AW, Horvath R, Davis P, Kramer TH, Yamamura HI, Hruby VJ. Topographical requirements for delta opioid ligands: The synthesis and biological properties of a cyclic analogue of deltorphin I Bioorganic and Medicinal Chemistry Letters. 2: 547-552. DOI: 10.1016/S0960-894X(01)81195-1 |
0.532 |
|
| 1992 |
Lai J, Roeske W, Yamamura HI. Structure-function correlation of muscarinic acetylfholine receptors European Neuropsychopharmacology. 2: 227-228. DOI: 10.1016/0924-977X(92)90078-M |
0.574 |
|
| 1991 |
Malatynska E, Dilsaver SC, Knapp RJ, Giroux ML, Ikeda M, Yamamura HI. The interaction of a benzodiazepine receptor antagonist (Ro15-1788) with GABA and GABA receptor antagonists at the GABA(A) receptor chloride-ionophore complex. Neurochemistry International. 18: 405-10. PMID 20504718 DOI: 10.1016/0197-0186(91)90173-B |
0.539 |
|
| 1991 |
Davis TP, Gillespie TJ, Shook J, Kramer TH, Hoyer G, Hawkins K, Davis P, Yamamura HI, Burks TF. Changes in opioid receptor selectivity following processing of peptide E: effect on gut motility. Gastroenterology. 100: 1603-15. PMID 1850373 DOI: 10.1016/0016-5085(91)90659-9 |
0.454 |
|
| 1991 |
van Giersbergen PL, Shatzer SA, Henderson AK, Lai J, Nakanishi S, Yamamura HI, Buck SH. Characterization of a tachykinin peptide NK2 receptor transfected into murine fibroblast B82 cells. Proceedings of the National Academy of Sciences of the United States of America. 88: 1661-5. PMID 1848006 DOI: 10.1073/Pnas.88.5.1661 |
0.441 |
|
| 1991 |
Lai J, Smith TL, Mei L, Ikeda M, Fujiwara Y, Gomez J, Halonen M, Roeske WR, Yamamura HI. The molecular properties of the M1 muscarinic receptor and its regulation of cytosolic calcium in a eukaryotic gene expression system. Advances in Experimental Medicine and Biology. 287: 313-30. PMID 1759615 DOI: 10.1007/978-1-4684-5907-4_26 |
0.689 |
|
| 1991 |
Mei L, Lai J, Yamamura HI, Roeske WR. Pharmacologic comparison of selected agonists for the M1 muscarinic receptor in transfected murine fibroblast cells (B82). The Journal of Pharmacology and Experimental Therapeutics. 256: 689-94. PMID 1704434 |
0.352 |
|
| 1991 |
Slaninova J, Knapp RJ, Wu JJ, Fang SN, Kramer T, Burks TF, Hruby VJ, Yamamura HI. Opioid receptor binding properties of analgesic analogues of cholecystokinin octapeptide. European Journal of Pharmacology. 200: 195-8. PMID 1663041 DOI: 10.1016/0014-2999(91)90688-M |
0.55 |
|
| 1991 |
Misicka A, Lipkowski AW, Fang L, Knapp RJ, Davis P, Kramer T, Burks TF, Yamamura HI, Carr DB, Hruby VJ. Topographical requirements for delta opioid ligands: presence of a carboxyl group in position 4 is not critical for deltorphin high delta receptor affinity and analgesic activity. Biochemical and Biophysical Research Communications. 180: 1290-7. PMID 1659410 DOI: 10.1016/S0006-291X(05)81335-X |
0.49 |
|
| 1991 |
Cavagnero S, Misicka A, Knapp RJ, Davis P, Fang L, Burks TF, Yamamura HI, Hruby VJ. Delta opioid receptor-selective ligands: [D-Pen2,D-Pen5]enkephalin-dermenkephalin chimeric peptides. Life Sciences. 49: 495-503. PMID 1650414 DOI: 10.1016/0024-3205(91)90066-K |
0.479 |
|
| 1991 |
Henderson AK, Yamamura HI, Maggi CA, Roeske WR, Smith TL. Neurokinin A receptors are coupled to calcium mobilization in transfected fibroblasts. European Journal of Pharmacology. 206: 251-3. PMID 1649764 DOI: 10.1016/S0922-4106(05)80026-4 |
0.352 |
|
| 1991 |
Hruby VJ, Toth G, Gehrig CA, Kao LF, Knapp R, Lui GK, Yamamura HI, Kramer TH, Davis P, Burks TF. Topographically designed analogues of [D-Pen,D-Pen5]enkephalin. Journal of Medicinal Chemistry. 34: 1823-30. PMID 1648137 DOI: 10.1021/Jm00110A010 |
0.47 |
|
| 1991 |
Parola AL, Yamamura HI. Pharmacological and molecular basis for reclassifying peripheral-type benzodiazepine receptors as τ (tau) receptors European Neuropsychopharmacology. 1: 289-294. DOI: 10.1016/0924-977X(91)90533-Z |
0.322 |
|
| 1991 |
Tomita H, Hikiji M, Fujiwara Y, Kashihara K, Akiyama K, Otsuki S, Yamamura HI. Expression of dopamine D2 receptor and kainate receptor mRNAs in the phencyclidine treated rat brain Neuroscience Research Supplements. 16: 15. DOI: 10.1016/0921-8696(91)90680-L |
0.412 |
|
| 1990 |
Hruby VJ, Fang SA, Knapp R, Kazmierski W, Lui GK, Yamamura HI. Cholecystokinin analogues with high affinity and selectivity for brain membrane receptors. International Journal of Peptide and Protein Research. 35: 566-73. PMID 2401597 DOI: 10.1111/J.1399-3011.1990.Tb00263.X |
0.429 |
|
| 1990 |
Mei L, Roeske WR, Izutsu KT, Yamamura HI. Characterization of muscarinic acetylcholine receptors in human labial salivary glands. European Journal of Pharmacology. 176: 367-70. PMID 2328757 DOI: 10.1016/0014-2999(90)90032-2 |
0.45 |
|
| 1990 |
Fujiwara Y, Nelson DL, Kashihara K, Varga E, Roeske WR, Yamamura HI. The cloning and sequence analysis of the rat serotonin-1A receptor gene. Life Sciences. 47: PL127-32. PMID 2273937 DOI: 10.1016/0024-3205(90)90445-W |
0.388 |
|
| 1990 |
Knapp RJ, Vaughn LK, Fang SN, Bogert CL, Yamamura MS, Hruby VJ, Yamamura HI. A new, highly selective CCK-B receptor radioligand ([3H][N-methyl-Nle28,31]CCK26-33): evidence for CCK-B receptor heterogeneity. The Journal of Pharmacology and Experimental Therapeutics. 255: 1278-86. PMID 2262906 |
0.338 |
|
| 1990 |
Lai J, Bloom JW, Yamamura HI, Roeske WR. Amplification of the rat M2 muscarinic receptor gene by the polymerase chain reaction: functional expression of the M2 muscarinic receptor. Life Sciences. 47: 1001-13. PMID 2172674 DOI: 10.1016/0024-3205(90)90472-4 |
0.651 |
|
| 1990 |
Gomez J, Bloom JW, Yamamura HI, Halonen M. Characterization of receptors for platelet-activating factor in guinea pig lung membranes. American Journal of Respiratory Cell and Molecular Biology. 3: 259-64. PMID 2167700 DOI: 10.1165/Ajrcmb/3.3.259 |
0.387 |
|
| 1990 |
Knapp RJ, Yamamura HI. [3H][D-Pen2, D-Pen5]enkephalin binding to delta opioid receptors on intact neuroblastoma-glioma (NG 108-15) hybrid cells. Life Sciences. 46: 1457-63. PMID 2161068 DOI: 10.1016/0024-3205(90)90462-Z |
0.515 |
|
| 1990 |
Vaughn LK, Wire WS, Davis P, Shimohigashi Y, Toth G, Knapp RJ, Hruby VJ, Burks TF, Yamamura HI. Differentiation between rat brain and mouse vas deferens delta opioid receptors. European Journal of Pharmacology. 177: 99-101. PMID 2160370 DOI: 10.1016/0014-2999(90)90556-L |
0.53 |
|
| 1990 |
Toth G, Kramer TH, Knapp R, Lui G, Davis P, Burks TF, Yamamura HI, Hruby VJ. [D-Pen2,D-Pen5]enkephalin analogues with increased affinity and selectivity for delta opioid receptors. Journal of Medicinal Chemistry. 33: 249-53. PMID 2153205 DOI: 10.1021/Jm00163A041 |
0.504 |
|
| 1990 |
Kawasaki AM, Knapp RJ, Kramer TH, Wire WS, Vasquez OS, Yamamura HI, Burks TF, Hruby VJ. Design and synthesis of highly potent and selective cyclic dynorphin A analogues. Journal of Medicinal Chemistry. 33: 1874-9. PMID 1972964 DOI: 10.1021/Jm00169A007 |
0.536 |
|
| 1990 |
Gehlert DR, Yamamura HI. Light Microscopic Localization of Drug and Neurotransmitter Receptors in the Brain Methods in Neurosciences. 3: 425-440. DOI: 10.1016/B978-0-12-185255-9.50029-8 |
0.409 |
|
| 1990 |
Henderson AK, Lai J, Buck SH, Fujiwara Y, Singh G, Yamamura MS, Nakanishi S, Roeske WR, Yamamura HI. Accelerated communication a cloned NK2 receptor mediates phosphatidylinositol hydrolysis in a transfected murine fibrolast Life Sciences. 47: PL7-PL12. DOI: 10.1016/0024-3205(90)90329-P |
0.66 |
|
| 1990 |
Roeske WR, Lai J, Mei L, Bloom JW, Yamamura HI. Pharmacologic comparison of the cloned M1 and M2 muscarinic receptors of the rat expressed in murine fibroblast cells European Journal of Pharmacology. 183: 1618. DOI: 10.1016/0014-2999(90)91905-Q |
0.655 |
|
| 1990 |
Hruby VJ, Kazmierski W, Pelton JT, Yamamura HI, Burks TF. Conversion of somatostatin to an opioid peptide: design using a conformational template and topographical constraints European Journal of Pharmacology. 183: 54. DOI: 10.1016/0014-2999(90)91304-T |
0.391 |
|
| 1989 |
Mei L, Lai J, Yamamura HI, Roeske WR. The relationship between agonist states of the M1 muscarinic receptor and the hydrolysis of inositol lipids in transfected murine fibroblast cells (B82) expressing different receptor densities. The Journal of Pharmacology and Experimental Therapeutics. 251: 90-7. PMID 2795474 |
0.336 |
|
| 1989 |
Palfreyman MG, Dudley MW, Cheng HC, Mir AK, Yamada S, Roeske WR, Obata T, Yamamura HI. Lactamimides: a novel chemical class of calcium antagonists with diltiazem-like properties. Biochemical Pharmacology. 38: 2459-65. PMID 2757648 DOI: 10.1016/0006-2952(89)90089-0 |
0.332 |
|
| 1989 |
Wang JX, Roeske WR, Hawkins KN, Gehlert DR, Yamamura HI. Quantitative autoradiography of M2 muscarinic receptors in the rat brain identified by using a selective radioligand [3H]AF-DX 116. Brain Research. 477: 322-6. PMID 2702492 DOI: 10.1016/0006-8993(89)91421-2 |
0.413 |
|
| 1989 |
Ikeda M, Weber KH, Bechtel WD, Malatynska E, Yamamura HI. Relative efficacies of 1,4-diazepines on GABA-stimulated chloride influx in rat brain vesicles. Life Sciences. 45: 349-58. PMID 2569655 DOI: 10.1016/0024-3205(89)90145-8 |
0.497 |
|
| 1989 |
Hawkins KN, Knapp RJ, Lui GK, Gulya K, Kazmierski W, Wan YP, Pelton JT, Hruby VJ, Yamamura HI. [3H]-[H-D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2] ([3H]CTOP), a potent and highly selective peptide for mu opioid receptors in rat brain. The Journal of Pharmacology and Experimental Therapeutics. 248: 73-80. PMID 2563293 |
0.41 |
|
| 1989 |
Ikeda M, Knapp RJ, Malatynska E, Yamamura HI. Amoxapine inhibition of GABA-stimulated chloride conductance: investigations of potential sites of activity. Life Sciences. 45: 1903-10. PMID 2557507 DOI: 10.1016/0024-3205(89)90544-4 |
0.567 |
|
| 1989 |
Mei L, Roeske WR, Yamamura HI. The coupling of muscarinic receptors to hydrolysis of inositol lipids in human neuroblastoma SH-SY5Y cells. Brain Research. 504: 7-14. PMID 2557126 DOI: 10.1016/0006-8993(89)91591-6 |
0.537 |
|
| 1989 |
Vaughn LK, Knapp RJ, Toth G, Wan YP, Hruby VJ, Yamamura HI. A high affinity, highly selective ligand for the delta opioid receptor: [3H]-[D-Pen2, pCl-Phe4, d-Pen5]enkephalin. Life Sciences. 45: 1001-8. PMID 2552241 DOI: 10.1016/0024-3205(89)90154-9 |
0.509 |
|
| 1989 |
Fujiwara Y, Bloom JW, Mantione CR, Yamamura HI. Identification of B2 bradykinin binding sites in the guinea pig nasal turbinate. Peptides. 10: 701-3. PMID 2550915 DOI: 10.1016/0196-9781(89)90163-0 |
0.377 |
|
| 1989 |
Malatynska E, Knapp R, Ikeda M, Yamamura HI. Beta-carboline interactions at the BZ-GABA receptor chloride-ionophore complex in the rat cerebral cortex. Brain Research Bulletin. 22: 845-8. PMID 2548678 DOI: 10.1016/0361-9230(89)90028-2 |
0.589 |
|
| 1989 |
Knapp RJ, Kazmierski W, Hruby VJ, Yamamura HI. Structural characteristics of two highly selective opioid peptides. Bioessays : News and Reviews in Molecular, Cellular and Developmental Biology. 10: 58-61. PMID 2541696 DOI: 10.1002/Bies.950100206 |
0.534 |
|
| 1989 |
Landis G, Lui G, Shook JE, Yamamura HI, Burks TF, Hruby VJ. Synthesis of highly mu and delta opioid receptor selective peptides containing a photoaffinity group. Journal of Medicinal Chemistry. 32: 638-43. PMID 2537426 DOI: 10.1021/Jm00123A023 |
0.527 |
|
| 1989 |
Mei L, Lai J, Roeske WR, Fraser CM, Venter JC, Yamamura HI. Pharmacological characterization of the M1 muscarinic receptors expressed in murine fibroblast B82 cells. The Journal of Pharmacology and Experimental Therapeutics. 248: 661-70. PMID 2537406 |
0.322 |
|
| 1989 |
Mei L, Roeske WR, Yamamura HI. Molecular pharmacology of muscarinic receptor heterogeneity. Life Sciences. 45: 1831-51. PMID 2513460 DOI: 10.1016/0024-3205(89)90537-7 |
0.438 |
|
| 1988 |
Yamada S, Yamazawa T, Harada Y, Yamamura HI, Nakayama K. Muscarinic receptor subtype in porcine coronary artery. European Journal of Pharmacology. 150: 373-6. PMID 3416915 DOI: 10.1016/0014-2999(88)90021-0 |
0.308 |
|
| 1988 |
Mei L, Yamamura HI, Roeske WR. Muscarinic receptor-mediated hydrolysis of phosphatidylinositols in human neuroblastoma (SH-SY5Y) cells is sensitive to pertussis toxin. Brain Research. 447: 360-3. PMID 3390705 DOI: 10.1016/0006-8993(88)91140-7 |
0.528 |
|
| 1988 |
Lai J, Mei L, Roeske WR, Chung FZ, Yamamura HI, Venter JC. The cloned murine M1 muscarinic receptor is associated with the hydrolysis of phosphatidylinositols in transfected murine B82 cells. Life Sciences. 42: 2489-502. PMID 3374268 DOI: 10.1016/0024-3205(88)90348-7 |
0.393 |
|
| 1988 |
Wang JX, Roeske WR, Wang W, Yamamura HI. Himbacine recognizes a high affinity subtype of M2 muscarinic cholinergic receptors in the rat cerebral cortex. Brain Research. 446: 155-8. PMID 3370478 DOI: 10.1016/0006-8993(88)91306-6 |
0.436 |
|
| 1988 |
Serra M, Mei L, Roeske WR, Lui GK, Watson M, Yamamura HI. The intact human neuroblastoma cell (SH-SY5Y) exhibits high-affinity [3H]pirenzepine binding associated with hydrolysis of phosphatidylinositols. Journal of Neurochemistry. 50: 1513-21. PMID 3361307 DOI: 10.1111/J.1471-4159.1988.Tb03038.X |
0.396 |
|
| 1988 |
Malatynska E, Serra M, Ikeda M, Biggio G, Yamamura HI. Modulation of GABA-stimulated chloride influx by beta-carbolines in rat brain membrane vesicles. Brain Research. 443: 395-7. PMID 3359279 DOI: 10.1016/0006-8993(88)91640-X |
0.504 |
|
| 1988 |
Bloom JW, Halonen M, Yamamura HI. Characterization of muscarinic cholinergic receptor subtypes in human peripheral lung. The Journal of Pharmacology and Experimental Therapeutics. 244: 625-32. PMID 3346839 |
0.301 |
|
| 1988 |
Bloom JW, Baumgartener-Folkerts C, Palmer JD, Yamamura HI, Halonen M. A muscarinic receptor subtype modulates vagally stimulated bronchial contraction. Journal of Applied Physiology (Bethesda, Md. : 1985). 65: 2144-50. PMID 3209557 DOI: 10.1152/Jappl.1988.65.5.2144 |
0.332 |
|
| 1988 |
Wang JX, Yamamura HI, Wang W, Roeske WR. Irreversible inhibition by tyrosine-directed alkylating reagents of muscarinic cholinergic receptors in membranes from rat forebrain and heart. Biochemical Pharmacology. 37: 3787-90. PMID 3178894 DOI: 10.1016/0006-2952(88)90418-2 |
0.361 |
|
| 1988 |
Berzetei IP, Fong A, Yamamura HI, Duckles SP. Characterization of kappa opioid receptors in the rabbit ear artery. European Journal of Pharmacology. 151: 449-55. PMID 2905660 DOI: 10.1016/0014-2999(88)90542-0 |
0.512 |
|
| 1988 |
Kazmierski W, Wire WS, Lui GK, Knapp RJ, Shook JE, Burks TF, Yamamura HI, Hruby VJ. Design and synthesis of somatostatin analogues with topographical properties that lead to highly potent and specific mu opioid receptor antagonists with greatly reduced binding at somatostatin receptors. Journal of Medicinal Chemistry. 31: 2170-7. PMID 2903246 DOI: 10.1021/Jm00119A019 |
0.557 |
|
| 1988 |
Hawkins KN, Knapp RJ, Gehlert DR, Lui GK, Yamamura MS, Roeske LC, Hruby VJ, Yamamura HI. Quantitative autoradiography of [3H]CTOP binding to mu opioid receptors in rat brain. Life Sciences. 42: 2541-51. PMID 2898716 DOI: 10.1016/0024-3205(88)90322-0 |
0.479 |
|
| 1988 |
Obata T, Yamamura HI, Malatynska E, Ikeda M, Laird H, Palmer CJ, Casida JE. Modulation of gamma-aminobutyric acid-stimulated chloride influx by bicycloorthocarboxylates, bicyclophosphorus esters, polychlorocycloalkanes and other cage convulsants. The Journal of Pharmacology and Experimental Therapeutics. 244: 802-6. PMID 2855243 |
0.501 |
|
| 1988 |
Sugg EE, Serra M, Shook JE, Yamamura HI, Burks TF, Korc M, Hruby VJ. Cholecystokinic activity of N alpha-hydroxysulfonyl-[Nle28,31]CCK26-33 analogues modified at the C-terminal residue. International Journal of Peptide and Protein Research. 31: 514-9. PMID 2457563 DOI: 10.1111/J.1399-3011.1988.Tb00910.X |
0.317 |
|
| 1988 |
Malatynska E, Knapp RJ, Ikeda M, Yamamura HI. Antidepressants and seizure-interactions at the GABA-receptor chloride-ionophore complex. Life Sciences. 43: 303-7. PMID 2456440 DOI: 10.1016/0024-3205(88)90107-5 |
0.529 |
|
| 1988 |
Dudley MW, Wiech NL, Miller FP, Carr AA, Cheng HC, Roebel LE, Doherty NS, Yamamura HI, Ursillo RC, Palfreyman MG. Pharmacological effects of MDL 11,939: A selective, centrally acting antagonist of 5-HT2 receptors Drug Development Research. 13: 29-43. DOI: 10.1002/DDR.430130104 |
0.368 |
|
| 1987 |
Yamada S, Gehlert DR, Hawkins KN, Nakayama K, Roeske WR, Yamamura HI. Autoradiographic localization of nicotinic receptor binding in rat brain using [3H]methylcarbamylcholine, a novel radioligand. Life Sciences. 41: 2851-61. PMID 3695812 DOI: 10.1016/0024-3205(87)90432-2 |
0.408 |
|
| 1987 |
Smith TL, Yamamura HI. Competitive inhibition of phosphoinositide hydrolysis by the muscarinic receptor antagonist AF-DX 116 is of low affinity in mouse cerebral cortex. Brain Research. 420: 362-4. PMID 3676767 DOI: 10.1016/0006-8993(87)91257-1 |
0.428 |
|
| 1987 |
Wang JX, Yamamura HI, Wang W, Roeske WR. Differential regulation of M2 muscarinic receptors by guanine nucleotides in rat cerebral cortical and cardiac membranes. European Journal of Pharmacology. 139: 357-8. PMID 3666011 DOI: 10.1016/0014-2999(87)90595-4 |
0.335 |
|
| 1987 |
Wang JX, Roeske WR, Gulya K, Wang W, Yamamura HI. [3H]AF-DX 116 labels subsets of muscarinic cholinergic receptors in rat brain and heart. Life Sciences. 41: 1751-60. PMID 3657382 DOI: 10.1016/0024-3205(87)90604-7 |
0.369 |
|
| 1987 |
Lemcke PK, Sugg E, Malarchik M, Lui G, Serra M, Yamamura HI, Hruby VJ, Shook JE, Burks TF. N-terminal cyclization of a nonsulfated CCK analogue exhibits opioid antagonist activity in vitro. Proceedings of the Western Pharmacology Society. 30: 223-6. PMID 3628282 |
0.322 |
|
| 1987 |
Bloom JW, Halonen M, Seaver NA, Yamamura HI. Heterogeneity of the M1 muscarinic receptor subtype between peripheral lung and cerebral cortex demonstrated by the selective antagonist AF-DX 116. Life Sciences. 41: 491-6. PMID 3600190 DOI: 10.1016/0024-3205(87)90226-8 |
0.386 |
|
| 1987 |
Duckles SP, Yamamura HI, Lee V. AF-DX 116 discriminates between muscarinic M2 receptors of the heart and vasculature. Life Sciences. 40: 1507-11. PMID 3561162 DOI: 10.1016/0024-3205(87)90383-3 |
0.38 |
|
| 1987 |
Bloom JW, Yamamura HI, Baumgartener C, Halonen M. A muscarinic receptor with high affinity for pirenzepine mediates vagally induced bronchoconstriction. European Journal of Pharmacology. 133: 21-7. PMID 3556389 DOI: 10.1016/0014-2999(87)90201-9 |
0.386 |
|
| 1987 |
Earle ME, Concas A, Wamsley JK, Yamamura HI. Temperature dependence and GABA modulation of [3H]triazolam binding in the rat brain. Life Sciences. 41: 397-403. PMID 3037225 DOI: 10.1016/0024-3205(87)90214-1 |
0.319 |
|
| 1987 |
Hawkins KN, Morelli M, Gulya K, Chang KJ, Yamamura HI. Autoradiographic localization of [3H] [MePhe3,D-Pro4]morphiceptin ([3H]PL017) to mu opioid receptors in rat brain. European Journal of Pharmacology. 133: 351-2. PMID 3030778 DOI: 10.1016/0014-2999(87)90033-1 |
0.365 |
|
| 1987 |
Nelson DL, Monroe PJ, Lambert G, Yamamura HI. [3H]spiroxatrine labels a serotonin1A-like site in the rat hippocampus. Life Sciences. 41: 1567-76. PMID 2957559 DOI: 10.1016/0024-3205(87)90723-5 |
0.344 |
|
| 1987 |
Berzetei IP, Yamamura HI, Duckles SP. Characterization of rabbit ear artery opioid receptors using a delta-selective agonist and antagonist. European Journal of Pharmacology. 139: 61-6. PMID 2820755 DOI: 10.1016/0014-2999(87)90497-3 |
0.506 |
|
| 1987 |
Fox DA, Ayres EA, Wire WS, Lui G, Yamamura HI, Burks TF. Kentsin: tetrapeptide from hamster embryos produces naloxone-sensitive effects without binding to opioid receptors. Peptides. 8: 613-8. PMID 2819832 DOI: 10.1016/0196-9781(87)90034-9 |
0.507 |
|
| 1986 |
Brinton RE, Gehlert DR, Wamsley JK, Wan YP, Yamamura HI. Vasopressin metabolite, AVP4-9, binding sites in brain: distribution distinct from that of parent peptide. Life Sciences. 38: 443-52. PMID 3945171 DOI: 10.1016/0024-3205(86)90069-X |
0.323 |
|
| 1986 |
Hynes MR, Banner W, Yamamura HI, Duckles SP. Characterization of muscarinic receptors of the rabbit ear artery smooth muscle and endothelium. The Journal of Pharmacology and Experimental Therapeutics. 238: 100-5. PMID 3755169 |
0.329 |
|
| 1986 |
Clark JA, Itzhak Y, Hruby VJ, Yamamura HI, Pasternak GW. [D-Pen2,D-Pen5]enkephalin (DPDPE): a delta-selective enkephalin with low affinity for mu 1 opiate binding sites. European Journal of Pharmacology. 128: 303-4. PMID 3025000 DOI: 10.1016/0014-2999(86)90784-3 |
0.566 |
|
| 1986 |
Serra M, Smith TL, Yamamura HI. Phorbol esters alter muscarinic receptor binding and inhibit polyphosphoinositide breakdown in human neuroblastoma (SH-SY5Y) cells. Biochemical and Biophysical Research Communications. 140: 160-6. PMID 3022714 DOI: 10.1016/0006-291X(86)91071-5 |
0.399 |
|
| 1986 |
Gulya K, Gehlert DR, Wamsley JK, Mosberg H, Hruby VJ, Yamamura HI. Light microscopic autoradiographic localization of delta opioid receptors in the rat brain using a highly selective bis-penicillamine cyclic enkephalin analog. The Journal of Pharmacology and Experimental Therapeutics. 238: 720-6. PMID 3016247 |
0.417 |
|
| 1986 |
Yamada S, Yamamura HI, Roeske WR. Effects of chemical sympathectomy with 6-hydroxydopamine on alpha- and beta-adrenoceptors and muscarinic cholinoceptors in rat kidney. European Journal of Pharmacology. 121: 345-53. PMID 3009209 DOI: 10.1016/0014-2999(86)90255-4 |
0.32 |
|
| 1986 |
Akiyama K, Vickroy TW, Watson M, Roeske WR, Reisine TD, Smith TL, Yamamura HI. Muscarinic cholinergic ligand binding to intact mouse pituitary tumor cells (AtT-20/D16-16) coupling with two biochemical effectors: adenylate cyclase and phosphatidylinositol turnover. The Journal of Pharmacology and Experimental Therapeutics. 236: 653-61. PMID 3005550 |
0.303 |
|
| 1986 |
Gulya K, Lui GK, Pelton JT, Kazmierski W, Hruby VJ, Yamamura HI. H-D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2: a potent and selective antagonist opioid receptors. Nida Research Monograph. 75: 209-12. PMID 2893264 |
0.462 |
|
| 1986 |
Pelton JT, Kazmierski W, Gulya K, Yamamura HI, Hruby VJ. Design and synthesis of conformationally constrained somatostatin analogues with high potency and specificity for mu opioid receptors. Journal of Medicinal Chemistry. 29: 2370-5. PMID 2878079 DOI: 10.1021/Jm00161A037 |
0.481 |
|
| 1986 |
Gulya K, Pelton JT, Hruby VJ, Yamamura HI. Cyclic somatostatin octapeptide analogues with high affinity and selectivity toward mu opioid receptors. Life Sciences. 38: 2221-9. PMID 2872570 DOI: 10.1016/0024-3205(86)90574-6 |
0.554 |
|
| 1986 |
Obata T, Yamamura HI. The effect of benzodiazepines and beta-carbolines on GABA-stimulated chloride influx by membrane vesicles from the rat cerebral cortex. Biochemical and Biophysical Research Communications. 141: 1-6. PMID 2432889 DOI: 10.1016/S0006-291X(86)80325-4 |
0.303 |
|
| 1985 |
Gehlert DR, Dawson TM, Yamamura HI, Wamsley JK. Quantitative autoradiography of [3H]forskolin binding sites in the rat brain. Brain Research. 361: 351-60. PMID 4084804 DOI: 10.1016/0006-8993(85)91305-8 |
0.55 |
|
| 1985 |
Brinton RE, Wamsley JK, Gehlert D, Wan YP, Yamamura HI. Vasopressin metabolite peptide (AVP-(4-9)) binding sites in rat kidney: distribution distinct from vasopressin binding sites. European Journal of Pharmacology. 108: 321-2. PMID 3987807 DOI: 10.1016/0014-2999(85)90457-1 |
0.312 |
|
| 1985 |
Vickroy TW, Roeske WR, Gehlert DR, Wamsley JK, Yamamura HI. Quantitative light microscopic autoradiography of [3H]hemicholinium-3 binding sites in the rat central nervous system: a novel biochemical marker for mapping the distribution of cholinergic nerve terminals. Brain Research. 329: 368-73. PMID 3978459 DOI: 10.1016/0006-8993(85)90553-0 |
0.313 |
|
| 1985 |
Dawson TM, Gehlert DR, Yamamura HI, Barnett A, Wamsley JK. D-1 dopamine receptors in the rat brain: autoradiographic localization using [3H]SCH 23390. European Journal of Pharmacology. 108: 323-5. PMID 3886408 DOI: 10.1016/0014-2999(85)90458-3 |
0.538 |
|
| 1985 |
Watson M, Vickroy TW, Roeske WR, Yamamura HI. Functional and biochemical basis for multiple muscarinic acetylcholine receptors. Progress in Neuro-Psychopharmacology & Biological Psychiatry. 9: 569-74. PMID 3841401 DOI: 10.1016/0278-5846(85)90018-1 |
0.406 |
|
| 1985 |
Vickroy TW, Watson M, Leventer SM, Roeske WR, Hanin I, Yamamura HI. Regional differences in ethylcholine mustard aziridinium ion (AF64A)-induced deficits in presynaptic cholinergic markers for the rat central nervous system. The Journal of Pharmacology and Experimental Therapeutics. 235: 577-82. PMID 3841155 |
0.303 |
|
| 1985 |
Watson M, Vickroy TW, Fibiger HC, Roeske WR, Yamamura HI. Effects of bilateral ibotenate-induced lesions of the nucleus basalis magnocellularis upon selective cholinergic biochemical markers in the rat anterior cerebral cortex. Brain Research. 346: 387-91. PMID 3840399 DOI: 10.1016/0006-8993(85)90876-5 |
0.364 |
|
| 1985 |
Smith TL, Yamamura HI. Carbachol stimulation of phosphatidic acid synthesis: competitive inhibition by pirenzepine in synaptosomes from rat cerebral cortex. Biochemical and Biophysical Research Communications. 130: 282-5. PMID 3839668 DOI: 10.1016/0006-291X(85)90414-0 |
0.317 |
|
| 1985 |
Yamamura HI, Vickroy TW, Gehlert DR, Wamsley JK, Roeske WR. Autoradiographic localization of muscarinic agonist binding sites in the rat central nervous system with (+)-cis-[3H]methyldioxolane. Brain Research. 325: 340-4. PMID 3838491 DOI: 10.1016/0006-8993(85)90336-1 |
0.399 |
|
| 1985 |
Lawrence LJ, Palmer CJ, Gee KW, Wang X, Yamamura HI, Casida JE. t-[3H]butylbicycloorthobenzoate: new radioligand probe for the gamma-aminobutyric acid-regulated chloride ionophore. Journal of Neurochemistry. 45: 798-804. PMID 2993514 DOI: 10.1111/J.1471-4159.1985.Tb04063.X |
0.368 |
|
| 1985 |
Gulya K, Gehlert DR, Wamsley JK, Mosberg HI, Hruby VJ, Duckles SP, Yamamura HI. Autoradiographic localization of delta opioid receptors in the rat brain using a highly selective bis-penicillamine cyclic enkephalin analog. European Journal of Pharmacology. 111: 285-6. PMID 2990955 DOI: 10.1016/0014-2999(85)90770-8 |
0.506 |
|
| 1985 |
Gehlert DR, Yamamura HI, Wamsley JK. gamma-Aminobutyric acidB receptors in the rat brain: quantitative autoradiographic localization using [3H](-)-baclofen. Neuroscience Letters. 56: 183-8. PMID 2989740 DOI: 10.1016/0304-3940(85)90126-0 |
0.382 |
|
| 1985 |
Akiyama K, Gee KW, Mosberg HI, Hruby VJ, Yamamura HI. Characterization of [3H][2-D-penicillamine, 5-D-penicillamine]-enkephalin binding to delta opiate receptors in the rat brain and neuroblastoma--glioma hybrid cell line (NG 108-15). Proceedings of the National Academy of Sciences of the United States of America. 82: 2543-7. PMID 2986120 DOI: 10.1073/Pnas.82.8.2543 |
0.427 |
|
| 1985 |
Gehlert DR, Yamamura HI, Wamsley JK. Autoradiographic localization of "peripheral-type" benzodiazepine binding sites in the rat brain, heart and kidney. Naunyn-Schmiedeberg's Archives of Pharmacology. 328: 454-60. PMID 2986017 DOI: 10.1007/BF00692915 |
0.345 |
|
| 1985 |
Wamsley JK, Golden JS, Yamamura HI, Barnett A. Autoradiographic demonstration of the selectivity of two 1-N-trifluoroethyl benzodiazepines for the BZD-1 receptors in the rat brain. Pharmacology, Biochemistry, and Behavior. 23: 973-8. PMID 2867566 DOI: 10.1016/0091-3057(85)90103-0 |
0.476 |
|
| 1985 |
Pelton JT, Gulya K, Hruby VJ, Duckles S, Yamamura HI. Somatostatin analogs with affinity for opiate receptors in rat brain binding assay. Peptides. 6: 159-63. PMID 2864680 DOI: 10.1016/0196-9781(85)90026-9 |
0.524 |
|
| 1985 |
Gulya K, Wamsley JK, Gehlert D, Pelton JT, Duckles SP, Hruby VJ, Yamamura HI. Light microscopic autoradiographic localization of somatostatin receptors in the rat brain. The Journal of Pharmacology and Experimental Therapeutics. 235: 254-8. PMID 2864434 |
0.307 |
|
| 1985 |
Pelton JT, Gulya K, Hruby VJ, Duckles SP, Yamamura HI. Conformationally restricted analogs of somatostatin with high mu-opiate receptor specificity. Proceedings of the National Academy of Sciences of the United States of America. 82: 236-9. PMID 2857488 DOI: 10.1073/Pnas.82.1.236 |
0.497 |
|
| 1985 |
Darman PS, Landis GC, Smits JR, Hirning LD, Gulya K, Yamamura HI, Burks TF, Hruby VJ. Conformationally restricted cyclic analogues of substance P: insight into the receptor binding process. Biochemical and Biophysical Research Communications. 127: 656-62. PMID 2579658 DOI: 10.1016/S0006-291X(85)80211-4 |
0.394 |
|
| 1985 |
Lee HR, Watson M, Yamamura HI, Roeske WR. Decreased [3H]nitrendipine binding in the brainstem of deoxycorticosterone-NaCl hypertensive rats. Life Sciences. 37: 971-7. PMID 2412086 DOI: 10.1016/0024-3205(85)90534-X |
0.348 |
|
| 1985 |
Yamamura HI, Akiyama K, Gee KW. Tritium (D-pen2,D-pen5)enkephalin, a highly selective radioligand for the identification and characterization of the delta opioid receptor Federation Proceedings. 44. |
0.362 |
|
| 1984 |
Wilkes BC, Hruby VJ, Yamamura HI, Akiyama K, Castrucci AM, Hadley ME, Andrews JR, Wan YP. Synthesis of tritium labeled Ac-[Nle4, D-Phe7]-alpha-MSH4-11-NH2: a superpotent melanotropin with prolonged biological activity. Life Sciences. 34: 977-84. PMID 6608041 DOI: 10.1016/0024-3205(84)90302-3 |
0.353 |
|
| 1984 |
Yamamura HI, Watson M, Wamsley JK, Johnson PC, Roeske WR. Light microscopic autoradiographic localization of [3H]pirenzepine and [3H](-)quinuclidinyl benzilate binding in human stellate ganglia. Life Sciences. 35: 753-7. PMID 6547993 DOI: 10.1016/0024-3205(84)90344-8 |
0.359 |
|
| 1984 |
Wamsley JK, Gehlert DR, Roeske WR, Yamamura HI. Muscarinic antagonist binding site heterogeneity as evidenced by autoradiography after direct labeling with [3H]-QNB and [3H]-pirenzepine. Life Sciences. 34: 1395-402. PMID 6546776 DOI: 10.1016/0024-3205(84)90012-2 |
0.358 |
|
| 1984 |
Akiyama K, Watson M, Roeske WR, Yamamura HI. High-affinity [3H]pirenzepine binding to putative M1 muscarinic sites in the neuroblastoma x glioma hybrid cell line (NG 108-15). Biochemical and Biophysical Research Communications. 119: 289-97. PMID 6546688 DOI: 10.1016/0006-291X(84)91650-4 |
0.377 |
|
| 1984 |
Watson M, Roeske WR, Johnson PC, Yamamura HI. [3H]Pirenzepine identifies putative M1 muscarinic receptors in human stellate ganglia. Brain Research. 290: 179-82. PMID 6546354 DOI: 10.1016/0006-8993(84)90751-0 |
0.328 |
|
| 1984 |
Gehlert DR, Dawson TM, Yamamura HI, Wamsley JK. Localization of [3H]forskolin binding sites in the rat brain using quantitative autoradiography. European Journal of Pharmacology. 106: 223-5. PMID 6543336 DOI: 10.1016/0014-2999(84)90707-6 |
0.493 |
|
| 1984 |
Vickroy TW, Roeske WR, Yamamura HI. Sodium-dependent high-affinity binding of [3H]hemicholinium-3 in the rat brain: a potentially selective marker for presynaptic cholinergic sites. Life Sciences. 35: 2335-43. PMID 6503616 DOI: 10.1016/0024-3205(84)90525-3 |
0.354 |
|
| 1984 |
Vickroy TW, Watson M, Yamamura HI, Roeske WR. Agonist binding to multiple muscarinic receptors. Federation Proceedings. 43: 2785-90. PMID 6383872 |
0.34 |
|
| 1984 |
Ehlert FJ, Yamamura HI. A comparison of the effects of cinnarizine and related compounds on [3H]nitrendipine binding in the brain, heart and ileum. Life Sciences. 34: 2347-55. PMID 6328164 DOI: 10.1016/0024-3205(84)90421-1 |
0.314 |
|
| 1984 |
Buck SH, Maurin Y, Burks TF, Yamamura HI. High-affinity 3H-substance P binding to longitudinal muscle membranes of the guinea pig small intestine. Life Sciences. 34: 497-507. PMID 6319946 DOI: 10.1016/0024-3205(84)90506-X |
0.323 |
|
| 1984 |
Vickroy TW, Watson M, Yamamura HI, Roeske WR. Differential regulation of putative M1/M2 muscarinic receptors: implications for different receptor-effector coupling mechanisms. Advances in Experimental Medicine and Biology. 175: 99-114. PMID 6208760 DOI: 10.1007/978-1-4684-4805-4_8 |
0.439 |
|
| 1984 |
Gehlert DR, Yamamura HI, Wamsley JK. Use of autoradiographic techniques for the localization of neurotransmitter receptors in brain and periphery: recent applications. Advances in Experimental Medicine and Biology. 175: 255-70. PMID 6208759 DOI: 10.1007/978-1-4684-4805-4_20 |
0.385 |
|
| 1984 |
Brinton RE, Gee KW, Wamsley JK, Davis TP, Yamamura HI. Regional distribution of putative vasopressin receptors in rat brain and pituitary by quantitative autoradiography. Proceedings of the National Academy of Sciences of the United States of America. 81: 7248-52. PMID 6095279 DOI: 10.1073/Pnas.81.22.7248 |
0.36 |
|
| 1984 |
Lawrence LJ, Gee KW, Yamamura HI. Benzodiazepine anticonvulsant action: gamma-aminobutyric acid-dependent modulation of the chloride ionophore. Biochemical and Biophysical Research Communications. 123: 1130-7. PMID 6091648 DOI: 10.1016/S0006-291X(84)80250-8 |
0.443 |
|
| 1984 |
Gee KW, Yamamura SH, Roeske WR, Yamamura HI. Benzodiazepine receptor heterogeneity: possible molecular basis and functional significance. Federation Proceedings. 43: 2767-72. PMID 6090222 |
0.34 |
|
| 1984 |
Brinton RE, Wamsley JK, Gee KW, Wan YP, Yamamura HI. [3H]oxytocin binding sites in the rat brain demonstrated by quantitative light microscopic autoradiography. European Journal of Pharmacology. 102: 365-7. PMID 6090165 DOI: 10.1016/0014-2999(84)90270-X |
0.318 |
|
| 1984 |
Lee HR, Roeske WR, Yamamura HI. High affinity specific [3H](+)PN 200-110 binding to dihydropyridine receptors associated with calcium channels in rat cerebral cortex and heart. Life Sciences. 35: 721-32. PMID 6088927 DOI: 10.1016/0024-3205(84)90340-0 |
0.366 |
|
| 1984 |
ROESKE W, LEE H, YAMAMURA H. High affinity specific [3H](+)PN 200-110 binding to a dihydropyridine receptor calcium channel complex in rat heart and cerebral cortex Journal of Molecular and Cellular Cardiology. 16: 31-31. DOI: 10.1016/S0022-2828(84)80123-6 |
0.357 |
|
| 1983 |
Ehlert FJ, Roeske WR, Yamamura HI. A simple and rapid radio-receptor assay for the estimation of acetylcholine. Life Sciences. 31: 347-54. PMID 7144444 DOI: 10.1016/0024-3205(82)90414-3 |
0.366 |
|
| 1983 |
Schoemaker H, Lee HR, Roeske WR, Yamamura HI. In vivo identification of calcium antagonist binding sites using [3H]nitrendipine European Journal of Pharmacology. 88: 275-276. PMID 6852115 DOI: 10.1016/0014-2999(83)90019-5 |
0.32 |
|
| 1983 |
Yamamura HI, Wamsley JK, Deshmukh P, Roeske WR. Differential light microscopic autoradiographic localization of muscarinic cholinergic receptors in the brainstem and spinal cord of the rat using [3H]pirenzepine European Journal of Pharmacology. 91: 147-149. PMID 6688587 DOI: 10.1016/0014-2999(83)90379-5 |
0.325 |
|
| 1983 |
Watson M, Yamamura HI, Roeske WR. A unique regulatory profile and regional distribution of [3H]pirenzepine binding in the rat provide evidence for distinct M1 and M2 muscarinic receptor subtypes Life Sciences. 32: 3001-3011. PMID 6688111 DOI: 10.1016/0024-3205(83)90652-5 |
0.412 |
|
| 1983 |
Deshmukh PP, Yamamura HI, Woods L, Nelson DL. Computer-assisted autoradiographic localization of subtypes of serotonin1 receptors in rat brain. Brain Research. 288: 338-43. PMID 6661625 DOI: 10.1016/0006-8993(83)90114-2 |
0.41 |
|
| 1983 |
Erman RD, Yamamura HI, Roeske WR. The ontogeny of specific binding sites for the calcium channel antagonist, nitrendipine, in mouse heart and brain. Brain Research. 278: 327-31. PMID 6640324 DOI: 10.1016/0006-8993(83)90265-2 |
0.345 |
|
| 1983 |
Vickroy TW, Yamamura HI, Roeske WR. Differential regulation of high-affinity agonist binding to muscarinic sites in the rat heart, cerebellum, and cerebral cortex. Biochemical and Biophysical Research Communications. 116: 284-90. PMID 6639662 DOI: 10.1016/0006-291X(83)90412-6 |
0.397 |
|
| 1983 |
Mosberg HI, Hurst R, Hruby VJ, Gee K, Akiyama K, Yamamura HI, Galligan JJ, Burks TF. Cyclic penicillamine containing enkephalin analogs display profound delta receptor selectivities. Life Sciences. 33: 447-50. PMID 6319901 DOI: 10.1016/0024-3205(83)90538-6 |
0.6 |
|
| 1983 |
Gehlert DR, Yamamura HI, Wamsley JK. Autoradiographic localization of 'peripheral' benzodiazepine binding sites in the rat brain and kidney using [3H]RO5-4864. European Journal of Pharmacology. 95: 329-30. PMID 6317419 DOI: 10.1016/0014-2999(83)90658-1 |
0.322 |
|
| 1983 |
Wamsley JK, Gee KW, Yamamura HI. Comparison of the distribution of convulsant/barbiturate and benzodiazepine receptors using light microscopic autoradiography. Life Sciences. 33: 2321-9. PMID 6316061 DOI: 10.1016/0024-3205(83)90266-7 |
0.437 |
|
| 1983 |
Gee KW, Yamamura HI. Photoaffinity labeling of benzodiazepine receptors in rat brain with flunitrazepam alters the affinity of benzodiazepine receptor agonist but not antagonist binding. Journal of Neurochemistry. 41: 1407-13. PMID 6311986 DOI: 10.1111/J.1471-4159.1983.Tb00839.X |
0.435 |
|
| 1983 |
Ehlert FJ, Roeske WR, Gee KW, Yamamura HI. An allosteric model for benzodiazepine receptor function Biochemical Pharmacology. 32: 2375-2383. PMID 6311215 DOI: 10.1016/0006-2952(83)90679-2 |
0.502 |
|
| 1983 |
Mosberg HI, Hurst R, Hruby VJ, Gee K, Yamamura HI, Galligan JJ, Burks TF. Bis-penicillamine enkephalins possess highly improved specificity toward delta opioid receptors. Proceedings of the National Academy of Sciences of the United States of America. 80: 5871-4. PMID 6310598 DOI: 10.1073/Pnas.80.19.5871 |
0.647 |
|
| 1983 |
Mosberg HI, Hurst R, Hruby VJ, Galligan JJ, Burks TF, Gee K, Yamamura HI. Conformationally constrained cyclic enkephalin analogs with pronounced delta opioid receptor agonist selectivity. Life Sciences. 32: 2565-9. PMID 6304440 DOI: 10.1016/0024-3205(83)90239-4 |
0.663 |
|
| 1983 |
Gee KW, Brinton RE, Yamamura HI. PK 8165 and PK 9084, two quinoline derivatives with anxiolytic properties, antagonize the anticonvulsant effects of diazepam Brain Research. 264: 168-172. PMID 6303496 DOI: 10.1016/0006-8993(83)91138-1 |
0.487 |
|
| 1983 |
Yamamura HI, Gee KW, Brinton RE, Davis TP, Hadley M, Wamsley JK. Light microscopic autoradiographic visualization of [3H]-arginine vasopressin binding sites in rat brain. Life Sciences. 32: 1919-24. PMID 6300592 DOI: 10.1016/0024-3205(83)90072-3 |
0.366 |
|
| 1983 |
Gee KW, Brinton RE, Yamamura HI. CL 218872 antagonism of diazepam induced loss of righting reflex: Evidence for partial agonistic activity at the benzodiazepine receptor Life Sciences. 32: 1037-1040. PMID 6298552 DOI: 10.1016/0024-3205(83)90936-0 |
0.474 |
|
| 1983 |
Hynes MR, Culling AJ, Galligan JJ, Burks TF, Schoemaker H, Yamamura HI, Davis TP. Processing of beta-endorphin in the dog intestine: regional specificity. Proceedings of the Western Pharmacology Society. 26: 95-9. PMID 6193534 |
0.405 |
|
| 1983 |
Gee KW, Yamamura HI. Selective anxiolytics: are the actions related to partial "agonist" activity or a preferential affinity for benzodiazepine receptor subtypes? Advances in Biochemical Psychopharmacology. 38: 1-9. PMID 6142598 |
0.409 |
|
| 1983 |
Yamanaka K, Yamamura HI, Roeske WR. Regulation of (-)epinephrine high affinity state of (β-adrenoceptors in the rat heart left ventricles Japanese Journal of Pharmacology. 33: 58. DOI: 10.1016/S0021-5198(19)60250-7 |
0.305 |
|
| 1983 |
Brinton RE, Gee KW, Yamamura HI. CL 218872, PK 8165 and PK 9084: Selective anxiolytics that may act as partial agonist at the benzodiazepine receptor Federation Proceedings. 42. |
0.38 |
|
| 1982 |
Ehlert FJ, Roeske WR, Itoga E, Yamamura HI. The binding of [3H]nitrendipine to receptors for calcium channel antagonists in the heart, cerebral cortex, and ileum of rats Life Sciences. 30: 2191-2202. PMID 7109844 DOI: 10.1016/0024-3205(82)90293-4 |
0.362 |
|
| 1982 |
Ehlert FJ, Itoga E, Roeske WR, Yamamura HI. The interaction of [3H]nitrendipine with receptors for calcium antagonists in the cerebral cortex and heart of rats Biochemical and Biophysical Research Communications. 104: 937-943. PMID 7073736 DOI: 10.1016/0006-291X(82)91339-0 |
0.369 |
|
| 1982 |
Barritt D, Yamamura HI, Roeske WR. Muscarinic receptor binding in the mouse heart: the selective modulatory effect of fluoride ion on agonist binding Life Sciences. 30: 875-877. PMID 7070200 DOI: 10.1016/0024-3205(82)90602-6 |
0.399 |
|
| 1982 |
Watson M, Roeske WR, Yamamura HI. [3H] pirenzepine selectively identifies a high affinity population of muscarinic cholinergic receptors in the rat cerebral cortex Life Sciences. 31: 2019-2023. PMID 6897437 DOI: 10.1016/0024-3205(82)90041-8 |
0.404 |
|
| 1982 |
Gee KW, Yamamura HI. Regional heterogeneity of benzodiazepine receptors at 37°C: An in vitro study in various regions of the rat brain Life Sciences. 31: 1939-1945. PMID 6294423 DOI: 10.1016/0024-3205(82)90032-7 |
0.453 |
|
| 1982 |
Yamamura HI, Schoemaker H, Boles RG, Roeske WR. Diltiazem enhancement of [3H]nitrendipine binding to calcium channel associated drug receptor sites in rat brain synaptosomes Biochemical and Biophysical Research Communications. 108: 640-646. PMID 6293498 DOI: 10.1016/0006-291X(82)90877-4 |
0.394 |
|
| 1982 |
Yamada S, Yamamura HI, Roeske WR. Characterization of postsynaptic β-adrenergic receptors and presynaptic muscarinic cholinergic receptors in the rat spleen Life Sciences. 31: 1161-1170. PMID 6292605 DOI: 10.1016/0024-3205(82)90091-1 |
0.403 |
|
| 1982 |
Schoemaker H, Morelli M, Deshmukh P, Yamamura HI. [3H]Ro5-4864 benzodiazepine binding in the kainate lesioned striatum and Huntington's diseased basal ganglia Brain Research. 248: 396-401. PMID 6291702 DOI: 10.1016/0006-8993(82)90602-3 |
0.352 |
|
| 1982 |
Gee KW, Yamamura HI. Differentiation of benzodiazepine receptor agonist and antagonist: Sparing of [3H]benzodiazepine antagonist binding following the photolabelling of benzodiazepine receptors European Journal of Pharmacology. 82: 239-241. PMID 6290239 DOI: 10.1016/0014-2999(82)90521-0 |
0.511 |
|
| 1982 |
Yamada S, Yamamura HI, Roeske WR. An increase in cardiac alpha1-adrenoceptors following chronic clonidine treatment Naunyn-Schmiedeberg's Archives of Pharmacology. 320: 115-118. PMID 6289138 DOI: 10.1007/BF00506311 |
0.304 |
|
| 1982 |
Gee KW, Ehlert FJ, Yamamura HI. The influence of temperature and gamma-aminobutyric acid on benzodiazepine receptor subtypes in the hippocampus of the rat Biochemical and Biophysical Research Communications. 106: 1134-1140. PMID 6288041 DOI: 10.1016/0006-291X(82)91230-X |
0.41 |
|
| 1982 |
Morelli M, Gee KW, Yamamura HI. The effect of GABA on in vitro binding of two novel non-benzodiazepines, PK 8165 and CGS 8216, to benzodiazepine receptors in the rat brain Life Sciences. 31: 77-81. PMID 6287150 DOI: 10.1016/0024-3205(82)90403-9 |
0.414 |
|
| 1982 |
Gee KW, Yamamura HI. A novel pyrazoloquinoline that interacts with brain benzodiazepine receptors: Characterization of some in vitro and in vivo properties of CGS 9896 Life Sciences. 30: 2245-2252. PMID 6287145 DOI: 10.1016/0024-3205(82)90251-X |
0.411 |
|
| 1982 |
Mosberg HI, Hurst R, Hruby VJ, Galligan JJ, Burks TF, Gee K, Yamamura HI. [D-Pen2, L-Cys5]enkephalinamide and[D-Pen2, D-Cys5] enkephalinamide, conformationally constrained cyclic enkephalinamide analogs with delta receptor specificity. Biochemical and Biophysical Research Communications. 106: 506-12. PMID 6285922 DOI: 10.1016/0006-291X(82)91139-1 |
0.605 |
|
| 1982 |
Ehlert FJ, Ragan P, Chen A, Roeske WR, Yamamura HI. Modulation of benzodiazepine receptor binding: insight into pharmacological efficacy. European Journal of Pharmacology. 78: 249-53. PMID 6281035 DOI: 10.1016/0014-2999(82)90246-1 |
0.378 |
|
| 1982 |
Davis TP, Schoemaker H, Chen A, Yamamura HI. I. High performance liquid chromatography of pharmacologically active amines and peptides in biological materials Life Sciences. 30: 971-987. PMID 6280002 DOI: 10.1016/0024-3205(82)90515-X |
0.31 |
|
| 1982 |
Yamamura HI, Mimaki T, Yamamura SH, Horst WD, Morelli M, Bautz G, O'Brien RA. [3H]CL 218,872, a novel triazolopyridazine which labels the benzodiazepine receptors in rat brain. European Journal of Pharmacology. 77: 351-4. PMID 6277678 DOI: 10.1016/0014-2999(82)90143-1 |
0.433 |
|
| 1982 |
Schoemaker H, Davis TP, Pedigo NW, Chen A, Berens ES, Ragan P, Ling NC, Yamamura HI. Identification of beta-endorphin-6(16-17) as the principal metabolite of des-tyrosin-gamma-endorphin (DTgammaE) in vitro and assessment of its activity in neurotransmitter receptor binding assays. European Journal of Pharmacology. 81: 459-68. PMID 6126374 DOI: 10.1016/0014-2999(82)90111-X |
0.41 |
|
| 1982 |
Gee KW, Morelli M, Yamamura HI. The effect of temperature on CL 218872 and propyl beta-carboline-3-carboxylate inhibition of [3H]-flunitrazepam binding in rat brain Biochemical and Biophysical Research Communications. 105: 1532-1537. PMID 6125147 DOI: 10.1016/0006-291X(82)90962-7 |
0.406 |
|
| 1982 |
Gee KW, Horst WD, O'Brien R, Yamamura HI. High affinity inhibition of [3H]-Flunitrazepam binding to brain benzodiazepine receptors by CGS 9896, a novel pyrazoloquinoline Biochemical and Biophysical Research Communications. 105: 457-461. PMID 6124246 DOI: 10.1016/0006-291X(82)91456-5 |
0.374 |
|
| 1982 |
Yamamura HI, Mimaki T, Morelli M, Yamamura SH, Horst WD, Bautz G, O'brien R. A novel triazolopyridazine, [3H]CL 218,872 which labels the benzodiazepine receptor in rat brain Protides of the Biological Fluids. 29: 487-492. DOI: 10.1016/B978-0-08-027988-6.50114-2 |
0.448 |
|
| 1982 |
Ehlert FJ, Roeske WR, Yamamura HI. Muscarinic cholinergic receptor heterogeneity Trends in Neurosciences. 5: 336-339. DOI: 10.1016/0166-2236(82)90199-0 |
0.48 |
|
| 1981 |
Pedigo NW, Yamamura HI, Nelson DL. Discrimination of multiple [3H]5-hydroxytryptamine binding sites by the neuroleptic spiperone in rat brain Journal of Neurochemistry. 36: 220-226. PMID 7463047 DOI: 10.1111/j.1471-4159.1981.tb02397.x |
0.32 |
|
| 1981 |
Ehlert FJ, Roeske WR, Yamamura HI. Dopaminergic regulation of muscarinic receptor binding in the corpus striatum Proceedings of the Western Pharmacology Society. 93-95. PMID 7255494 |
0.317 |
|
| 1981 |
Ehlert FJ, Roeske WR, Yamamura HI. Striatal muscarinic receptors: regulation by dopaminergic agonists. Life Sciences. 28: 2441-8. PMID 7253832 DOI: 10.1016/0024-3205(81)90512-9 |
0.377 |
|
| 1981 |
Overstreet DH, Driscoll P, Martin JR, Yamamura HI. Brain muscarinic cholinergic receptor binding in Roman high- and low-avoidance rats Psychopharmacology. 72: 143-145. PMID 6782603 DOI: 10.1007/BF00431647 |
0.423 |
|
| 1981 |
Pedigo NW, Schoemaker H, Morelli M, McDougal JN, Malick JB, Burks TF, Yamamura HI. Benzodiazepine receptor binding in young, mature and senescent rat brain and kidney Neurobiology of Aging. 2: 83-88. PMID 6272144 DOI: 10.1016/0197-4580(81)90003-8 |
0.424 |
|
| 1981 |
Ehlert FJ, Roeske WR, Yamamura HI. Multiple benzodiazepine receptors and their regulation by γ-aminobutyric Life Sciences. 29: 235-248. PMID 6270491 DOI: 10.1016/0024-3205(81)90239-3 |
0.398 |
|
| 1981 |
Schoemaker H, Bliss M, Yamamura HI. Specific high-affinity saturable binding of [3H] Ro5-4864 To benzodiazepine binding sites in the rat cerebral cortex European Journal of Pharmacology. 71: 173-175. PMID 6263650 DOI: 10.1016/0014-2999(81)90405-2 |
0.322 |
|
| 1981 |
Lippa AS, Critchett DJ, Ehlert F, Yamamura HI, Enna SJ, Bartus RT. Age-related alterations in neurotransmitter receptors: an electrophysiological and biochemical analysis. Neurobiology of Aging. 2: 3-8. PMID 6115325 DOI: 10.1016/0197-4580(81)90052-X |
0.528 |
|
| 1981 |
Ehlert FJ, Roeske WR, Braestrup C, Yamamura SH, Yamamura HI. gamma-Aminobutyric acid regulation of the benzodiazepine receptor: biochemical evidence for pharmacologically different effects of benzodiazepines and propyl beta-carboline-3-carboxylate. European Journal of Pharmacology. 70: 593-5. PMID 6113152 DOI: 10.1016/0014-2999(81)90375-7 |
0.376 |
|
| 1981 |
Regan JW, Yamamura HI, Yamada S, Roeske WR. High affinity renal [3H]flunitrazepam binding: Characterization, localization, and alteration in hypertension Life Sciences. 28: 991-998. PMID 6111733 DOI: 10.1016/0024-3205(81)90744-X |
0.306 |
|
| 1981 |
Yamamura HI, Ehlert F, Mimaki T. Benzodiazepine receptor binding studies in rat brain using two novel nonbenzodiazepines Neuroendocrinology Letters. 3: 67. |
0.315 |
|
| 1980 |
Smit MH, Ehlert FJ, Yamamura S, Roeske WR, Yamamura HI. Differential regulation of muscarinic agonist binding sites following chronic cholinesterase inhibition. European Journal of Pharmacology. 66: 379-80. PMID 7418725 DOI: 10.1016/0014-2999(80)90471-9 |
0.355 |
|
| 1980 |
Schallert T, Overstreet DH, Yamamura HI. Muscarinic receptor binding and behavioral effects of atropoine following chronic catecholamine depletion or acetylcholinesterase inhibition in rats. Pharmacology, Biochemistry, and Behavior. 13: 187-92. PMID 7413689 DOI: 10.1016/0091-3057(80)90071-4 |
0.4 |
|
| 1980 |
Ehlert FJ, Dumont Y, Roeske WR, Yamamura HI. Muscarinic receptor binding in rat brain using the agonist, [3H]cis methyldioxolane Life Sciences. 26: 961-967. PMID 7392777 DOI: 10.1016/0024-3205(80)90117-4 |
0.388 |
|
| 1980 |
Ehlert FJ, Yamamura HI, Triggle DJ, Roeske WR. The influence of guanyl-5'-yl imidodiphosphate and sodium chloride on the binding of the muscarinic agonist, [3H] cis methyldioxolane. European Journal of Pharmacology. 61: 317-8. PMID 7363942 DOI: 10.1016/0014-2999(80)90135-1 |
0.356 |
|
| 1980 |
Ehlert FJ, Roeske WR, Rosenberger LB, Yamamura HI. The influence of guanyl-5'-yl imidodiphosphate and sodium on muscarinic receptor binding in the rat brain and longitudinal muscle of the rat ileum. Life Sciences. 26: 245-52. PMID 7360006 DOI: 10.1016/0024-3205(80)90300-8 |
0.427 |
|
| 1980 |
Ehlert FJ, Roeske WR, Yamamura HI. Regulation of muscarinic receptor binding by guanine nucleotides and N-ethylmaleimide Journal of Supramolecular and Cellular Biochemistry. 14: 149-162. PMID 7230804 DOI: 10.1002/Jss.400140204 |
0.361 |
|
| 1980 |
Mimaki T, Deshmukh PP, Yamamura HI. Decreased benzodiazepine receptor density in rat cerebellum following neurotoxic doses of phenytoin Journal of Neurochemistry. 35: 1473-1475. PMID 6255101 DOI: 10.1111/J.1471-4159.1980.Tb09029.X |
0.36 |
|
| 1980 |
Johnson RW, Reisine T, Spotnitz S, Wiech N, Ursillo R, Yamamura HI. Effects of desipramine and yohimbine on alpha 2- and beta-adrenoreceptor sensitivity. European Journal of Pharmacology. 67: 123-7. PMID 6252022 DOI: 10.1016/0014-2999(80)90019-9 |
0.329 |
|
| 1980 |
Olsen RW, Reisine TD, Yamamura HI. Neurotransmitter receptors - biochemistry and alterations in neuropsychiatric disorders Life Sciences. 27: 801-808. PMID 6251327 DOI: 10.1016/0024-3205(80)90073-9 |
0.364 |
|
| 1980 |
Rosenberger LB, Yamamura HI, Roeske WR. The regulation of cardiac muscarinic cholinergic receptors by isoproterenol. European Journal of Pharmacology. 65: 129-30. PMID 6249619 DOI: 10.1016/0014-2999(80)90223-X |
0.362 |
|
| 1980 |
Yamada S, Yamamura HI, Roeske WR. The regulation of cardiac α1-adrenergic receptors by guanine nucleotides and by muscarinic cholinergic agonists European Journal of Pharmacology. 63: 239-241. PMID 6247169 DOI: 10.1016/0014-2999(80)90455-0 |
0.395 |
|
| 1980 |
Reisine TD, U'Prichard DC, Wiech NL, Ursillo RC, Yamamura HI. Effects of combined administration of amphetamine and iprindole on brain adrenergic receptors. Brain Research. 188: 587-92. PMID 6245760 DOI: 10.1016/0006-8993(80)90060-8 |
0.428 |
|
| 1980 |
U'Prichard DC, Reisine TD, Yamamura S, Mason ST, Fibiger HC, Ehlert F, Yamamura HI. Differential supersensitivity of beta-receptor subtypes in rat cortex and cerebellum after central noradrenergic denervation. Life Sciences. 26: 355-64. PMID 6245317 DOI: 10.1016/0024-3205(80)90151-4 |
0.346 |
|
| 1980 |
Reisine TD, Overstreet D, Gale K, Rossor M, Iversen L, Yamamura HI. Benzodiazepine receptors: the effect of GABA on their characteristics in human brain and their alteration in Huntington's disease. Brain Research. 199: 79-88. PMID 6105905 DOI: 10.1016/0006-8993(80)90231-0 |
0.447 |
|
| 1980 |
Martin AR, Kim SH, Yamamura HI, Horn AS. Conformationally restricted phenothiazine neuroleptics. 1. 3-(Dimethylamino)-1,2,3,4-tetrahydroazepino[3,2,1-kl]phenothiazine. Journal of Medicinal Chemistry. 23: 938-41. PMID 6105219 DOI: 10.1021/JM00182A022 |
0.331 |
|
| 1980 |
Regan JW, Roeske WR, Yamamura HI. 3H-flunitrazepam binding to bovine retina and the effect of GABA thereon Neuropharmacology. 19: 413-414. PMID 6104311 DOI: 10.1016/0028-3908(80)90195-1 |
0.402 |
|
| 1980 |
Chen FM, Yamamura HI, Roeske WR. Ontogeny of mammalian myocardial beta-adrenergic receptors. European Journal of Pharmacology. 58: 255-64. PMID 228943 DOI: 10.1016/0014-2999(79)90474-6 |
0.364 |
|
| 1980 |
Speth RC, Wastek GJ, Reisine TD, Yamamura HI. Benzodiazepine receptors: effect of tissue preincubation at 37 degrees C. Neuroscience Letters. 13: 243-7. PMID 43491 DOI: 10.1016/0304-3940(79)91501-5 |
0.411 |
|
| 1980 |
Regan JW, Roeske WR, Yamamura HI. The effect of GABA on the binding of 3H-flunitrazepam in mouse brains during development Brain Research Bulletin. 5: 857-860. DOI: 10.1016/0361-9230(80)90144-6 |
0.329 |
|
| 1980 |
Yamamura HI, Reisine TD, Beaumont K. Huntington's disease: Alterations in GABA and benzodiazepine receptors in the human brain Brain Research Bulletin. 5: 773-775. DOI: 10.1016/0361-9230(80)90128-8 |
0.428 |
|
| 1979 |
Johnson RW, Yamamura HI. Photoaffinity labeling of the benzodiazepine receptor in bovine cerebral cortex Life Sciences. 25: 1613-1620. PMID 522618 DOI: 10.1016/0024-3205(79)90445-4 |
0.409 |
|
| 1979 |
Speth RC, Bresolin N, Yamamura HI. Acute diazepam administration produces rapid increases in brain benzodiazepine receptor density European Journal of Pharmacology. 59: 159-160. PMID 510397 DOI: 10.1016/0014-2999(79)90041-4 |
0.391 |
|
| 1979 |
Speth RC, Yamamura HI. On the ability of choline and its analogues to interact with muscarinic cholinergic receptors in the rat brain European Journal of Pharmacology. 58: 197-201. PMID 499350 DOI: 10.1016/0014-2999(79)90012-8 |
0.439 |
|
| 1979 |
Rosenberger LB, Roeske WR, Yamamura HI. The regulation of muscarinic cholinergic receptors by guanine nucleotides in cardiac tissue. European Journal of Pharmacology. 56: 179-80. PMID 467508 DOI: 10.1016/0014-2999(79)90451-5 |
0.35 |
|
| 1979 |
Reisine TD, Nagy JI, Fibiger HC, Yamamura HI. Localization of dopamine receptors in rat brain. Brain Research. 169: 209-14. PMID 455093 DOI: 10.1016/0006-8993(79)90391-3 |
0.362 |
|
| 1979 |
Reisine TD, Nagy JI, Beaumont K, Fibiger HC, Yamamura HI. The localization of receptor binding sites in the substantia nigra and striatum of the rat. Brain Research. 177: 241-52. PMID 227532 DOI: 10.1016/0006-8993(79)90775-3 |
0.367 |
|
| 1979 |
Reisine TD, Azari J, Johnson PC, Barbeau A, Huxtable R, Yamamura HI. Brain neurotransmitter receptors in Friedreich's ataxia. The Canadian Journal of Neurological Sciences. Le Journal Canadien Des Sciences Neurologiques. 6: 259-62. PMID 226258 DOI: 10.1017/S0317167100119754 |
0.41 |
|
| 1979 |
Reisine TD, Rossor M, Spokes E, Iversen LL, Yamamura HI. Alterations in brain opiate receptors in Parkinson's disease. Brain Research. 173: 378-82. PMID 226215 DOI: 10.1016/0006-8993(79)90642-5 |
0.372 |
|
| 1979 |
Beaumont K, Maurin Y, Reisine TD, Fields JZ, Spokes E, Bird ED, Yamamura HI. Huntington's disease and its animal model: alterations in kainic acid binding. Life Sciences. 24: 809-16. PMID 156298 DOI: 10.1016/0024-3205(79)90365-5 |
0.349 |
|
| 1979 |
Overstreet DH, Yamamura HI. Receptor alterations and drug tolerance Life Sciences. 25: 1865-1877. PMID 43446 DOI: 10.1016/0024-3205(79)90607-6 |
0.426 |
|
| 1979 |
Pedigo NW, Schallert T, Overstreet DH, Ling NC, Ragan P, Reisine TD, Yamamura HI. Inhibition of in vivo 3H-spiperone binding by the proposed antipsychotic Des-Tyr1-gamma-endorphin. European Journal of Pharmacology. 60: 359-64. PMID 43261 DOI: 10.1016/0014-2999(79)90242-5 |
0.333 |
|
| 1979 |
Speth RC, Yamamura HI. Benzodiazepine receptors: alterations in mutant mouse cerebellum. European Journal of Pharmacology. 54: 397-9. PMID 35356 DOI: 10.1016/0014-2999(79)90071-2 |
0.306 |
|
| 1979 |
Speth RC, Wastek GJ, Yamamura HI. Benzodiazepine receptors: temperature dependence of [3H]flunitrazepam binding. Life Sciences. 24: 351-7. PMID 34765 DOI: 10.1016/0024-3205(79)90331-X |
0.38 |
|
| 1978 |
Fields JZ, Reisine TD, Yamamura HI. Biochemical demonstration of dopaminergic receptors in rat and human brain using [3H]spiroperidol. Brain Research. 136: 578-84. PMID 922503 DOI: 10.1016/0006-8993(77)90084-1 |
0.402 |
|
| 1978 |
Pedigo NW, Reisine TD, Fields JZ, Yamamura HI. 3H-spiroperidol binding to two receptor sites in both the corpus striatum and frontal cortex of rat brain European Journal of Pharmacology. 50: 451-453. PMID 699968 DOI: 10.1016/0014-2999(78)90154-1 |
0.398 |
|
| 1978 |
Kobayashi RM, Palkovits M, Hruska RE, Rothschild R, Yamamura HI. Regional distribution of muscarinic cholinergic receptors in rat brain. Brain Research. 154: 13-23. PMID 698807 DOI: 10.1016/0006-8993(78)91047-8 |
0.418 |
|
| 1978 |
Fields JZ, Reisine TD, Yamamura HI. Loss of striatal dopaminergic receptors after intrastriatal kainic acid injection. Life Sciences. 23: 569-73. PMID 692281 DOI: 10.1016/0024-3205(78)90036-X |
0.382 |
|
| 1978 |
Hruska RE, Schwarcz R, Coyle JT, Yamamura HI. Alterations of muscarinic cholinergic receptors in the rat striatum after kainic acid injections. Brain Research. 152: 620-5. PMID 687979 DOI: 10.1016/0006-8993(78)91120-4 |
0.368 |
|
| 1978 |
Roeske WR, Yamamura HI. Maturation of mammalian myocardial muscarinic cholinergic receptors Life Sciences. 23: 127-132. PMID 682873 DOI: 10.1016/0024-3205(78)90260-6 |
0.403 |
|
| 1978 |
Hruska RE, White R, Azari J, Yamamura HI. Muscarinic cholinergic receptors in mammalian retina Brain Research. 148: 493-498. PMID 656944 DOI: 10.1016/0006-8993(78)90736-9 |
0.416 |
|
| 1978 |
Reisine TD, Yamamura HI, Bird ED, Spokes E, Enna SJ. Pre- and postsynaptic neurochemical alterations in Alzheimer's disease. Brain Research. 159: 477-81. PMID 215272 DOI: 10.1016/0006-8993(78)90562-0 |
0.435 |
|
| 1978 |
Beaumont K, Chilton WS, Yamamura HI, Enna SJ. Muscimol binding in rat brain: association with synaptic GABA receptors. Brain Research. 148: 153-62. PMID 207386 DOI: 10.1016/0006-8993(78)90385-2 |
0.529 |
|
| 1978 |
Wastek GJ, Yamamura HI. Biochemical characterization of the muscarinic cholinergic receptor in human brain: Alterations in Huntington's disease Molecular Pharmacology. 14: 768-780. PMID 152407 |
0.349 |
|
| 1978 |
Wastek GJ, Speth RC, Reisine TD, Yamamura HI. The effect of gamma-aminobutyric acid on 3H-flunitrazepam binding in rat brain. European Journal of Pharmacology. 50: 445-7. PMID 29760 DOI: 10.1016/0014-2999(78)90152-8 |
0.325 |
|
| 1978 |
Speth RC, Wastek GJ, Johnson PC, Yamamura HI. Benzodiazepine binding in human brain: characterization using [3H]flunitrazepam. Life Sciences. 22: 859-66. PMID 25362 DOI: 10.1016/0024-3205(78)90610-0 |
0.347 |
|
| 1977 |
Speth RC, Chen FM, Lindstrom JM, Kobayashi RM, Yamamura HI. Nicotinic cholinergic receptors in rat brain identified by [125I]Naja naja siamensis alpha-toxin binding. Brain Research. 131: 350-5. PMID 890462 DOI: 10.1016/0006-8993(77)90527-3 |
0.373 |
|
| 1977 |
Yaksh TL, Yamamura HI. Depression by morphine of the resting and evoked release of [3H]-acetylcholine from the cat caudate nucleus in vivo Neuropharmacology. 16: 227-233. PMID 859683 DOI: 10.1016/0028-3908(77)90099-5 |
0.318 |
|
| 1977 |
Arregui A, Bennett JP, Bird ED, Yamamura HI, Iversen LL, Snyder SH. Huntington's chorea: selective depletion of activity of angiotensin coverting enzyme in the corpus striatum. Annals of Neurology. 2: 294-8. PMID 214022 DOI: 10.1002/ana.410020406 |
0.399 |
|
| 1977 |
Reisine TD, Fields JZ, Yamamura HI. Neurotransmitter receptor alterations in Parkinson's disease. Life Sciences. 21: 335-43. PMID 197361 DOI: 10.1016/0024-3205(77)90514-8 |
0.435 |
|
| 1977 |
Reisine TD, Fields JZ, Stern LZ, Johnson PC, Bird ED, Yamamura HI. Alterations in dopaminergic receptors in Huntington's disease. Life Sciences. 21: 1123-8. PMID 144230 DOI: 10.1016/0024-3205(77)90111-4 |
0.442 |
|
| 1977 |
Enna SJ, Stern LZ, Wastek GJ, Yamamura HI. Cerebrospinal fluid gamma-aminobutyric acid variations in neurological disorders. Archives of Neurology. 34: 683-5. PMID 143928 DOI: 10.1001/Archneur.1977.00500230053008 |
0.455 |
|
| 1977 |
Wastek GJ, Stern LZ, Johnson PC, Yamamura HI. Huntington's disease: regional alteration in muscarinic cholinergic receptor binding in human brain. Life Sciences. 19: 1033-9. PMID 136582 DOI: 10.1016/0024-3205(76)90295-2 |
0.412 |
|
| 1977 |
Snyder SH, Yamamura HI. Antidepressants and the muscarinic acetylcholine receptor. Archives of General Psychiatry. 34: 236-9. PMID 14603 DOI: 10.1001/archpsyc.1977.01770140126014 |
0.555 |
|
| 1977 |
Enna SJ, Bennett JP, Bylund DB, Creese I, Burt DR, Charness ME, Yamamura HI, Simantov R, Snyder SH. Neurotransmitter receptor binding: regional distribution in human brain. Journal of Neurochemistry. 28: 233-6. PMID 13155 DOI: 10.1111/j.1471-4159.1977.tb07733.x |
0.73 |
|
| 1977 |
Hruska RE, Yamamura HI. Biochemical characterization of muscarinic cholinergic receptors in mammalian retina Pharmacologist. 19. |
0.301 |
|
| 1976 |
Yamamura HI, Manian AA, Snyder SH. Muscarinic cholinergic receptor binding: influence of pimozide and chlorpromazine metabolites. Life Sciences. 18: 685-91. PMID 1263751 DOI: 10.1016/0024-3205(76)90179-X |
0.536 |
|
| 1976 |
Enna SJ, Yamamura HI, Snyder SH. Development of muscarinic cholinergic and GABA receptor binding in chick embryo brain. Brain Research. 101: 177-83. PMID 1244218 DOI: 10.1016/0006-8993(76)91001-5 |
0.622 |
|
| 1976 |
Yamamura HI, Wastek G, Chang KJ, Snyder SH. Cholinergic receptors in the mammalian central nervous system. Proceedings of the Western Pharmacology Society. 19: 13-8. PMID 995977 |
0.316 |
|
| 1976 |
Kuhar MJ, Yamamura HI. Localization of cholinergic muscarinic receptors in rat brain by light microscopic radioautography Brain Research. 110: 229-243. PMID 938940 DOI: 10.1016/0006-8993(76)90399-1 |
0.569 |
|
| 1976 |
Enna SJ, Bird ED, Bennett JP, Bylund DB, Yamamura HI, Iversen LL, Snyder SH. Huntington's chorea. Changes in neurotransmitter receptors in the brain. The New England Journal of Medicine. 294: 1305-9. PMID 4733 DOI: 10.1056/NEJM197606102942402 |
0.643 |
|
| 1976 |
Speth R, Yamamura HI, Dettbarn WD. Prolonged cholinesterase inhibition and central muscarinic receptor activity Trans.Amer.Soc.Neurochem.. 7. |
0.323 |
|
| 1975 |
Kuhar MJ, DeHaven RN, Yamamura HI, Rommel-Spacher H, Simon JR. Further evidence for cholinergic habenulo-interpeduncular neurons: Pharmacologic and functional characteristics Brain Research. 97: 265-275. PMID 1175046 DOI: 10.1016/0006-8993(75)90449-7 |
0.49 |
|
| 1975 |
Yaksh TL, Yamamura HI. Blockade by morphine of acetylcholine release from the caudate nucleus in the mid-pontine pretrigeminal cat Brain Research. 83: 520-524. PMID 1111819 DOI: 10.1016/0006-8993(75)90847-1 |
0.33 |
|
| 1975 |
Snyder SH, Chang KJ, Kuhar MJ, Yamamura HI. Biochemical indentification of the mammalian muscarinic cholinergic receptor. Federation Proceedings. 34: 1915-21. PMID 808430 |
0.537 |
|
| 1975 |
Guarnieri M, Krell LS, McKhann GM, Pasternak GW, Yamamura HI. The effects of cell isolation techniques on neuronal membrane receptors. Brain Research. 93: 337-42. PMID 169956 DOI: 10.1016/0006-8993(75)90355-8 |
0.525 |
|
| 1975 |
Yamamura HI, Snyder SH. Tricyclic antidepressants and the central cholinergic muscarinic receptor Pharmacologist. 17. |
0.327 |
|
| 1974 |
Snyder SH, Banerjee SP, Yamamura HI, Greenberg D. Drugs, neurotransmitters, and schizophrenia. Science (New York, N.Y.). 184: 1243-53. PMID 17784215 DOI: 10.1126/science.184.4143.1243 |
0.332 |
|
| 1974 |
Yamamura HI, Snyder SH. Postsynaptic localization of muscarinic cholinergic receptor binding in rat hippocampus. Brain Research. 78: 320-6. PMID 4853717 DOI: 10.1016/0006-8993(74)90556-3 |
0.516 |
|
| 1974 |
Mulder AH, Yamamura HI, Kuhar MJ, Snyder SH. Release of acetylcholine from hippocampal slices by potassium depolarization: dependence on high affinity choline uptake. Brain Research. 70: 372-6. PMID 4825681 DOI: 10.1016/0006-8993(74)90329-1 |
0.528 |
|
| 1974 |
Yamamura HI, Kuhar MJ, Snyder SH. In vivo identification of muscarinic cholinergic receptor binding in rat brain. Brain Research. 80: 170-6. PMID 4421615 DOI: 10.1016/0006-8993(74)90738-0 |
0.63 |
|
| 1974 |
Snyder S, Greenberg D, Yamamura HI. Antischizophrenic Drugs and Brain Cholinergic Receptors: Affinity for Muscarinic Sites Predicts Extrapyramidal Effects Archives of General Psychiatry. 31: 58-61. PMID 4152054 DOI: 10.1001/archpsyc.1974.01760130040006 |
0.51 |
|
| 1974 |
Yamamura HI, Snyder SH. Muscarinic cholinergic binding in rat brain. Proceedings of the National Academy of Sciences of the United States of America. 71: 1725-9. PMID 4151898 DOI: 10.1073/pnas.71.5.1725 |
0.5 |
|
| 1974 |
Yamamura HI, Kuhar MJ, Greenberg D, Snyder SH. Muscarinic cholinergic receptor binding: regional distribution in monkey brain Brain Research. 66: 541-546. DOI: 10.1016/0006-8993(74)90069-9 |
0.621 |
|
| 1974 |
Yamamura HI, Kuhar MJ, Snyder SH. Identification in vivo of muscarinic cholinergic receptor binding in rat brain Pharmacologist. 16. |
0.306 |
|
| 1974 |
Yamamura HI, Kuhar MJ, Snyder SH. Muscarinic cholinergic receptor binding in mammalian central and peripheral nervous system: demonstration in vitro and in vivo Trans.Amer.Soc.Neurochem.. 5. |
0.337 |
|
| 1974 |
Yamamura HI, Broomfield CA, Snyder SH. Muscarinic cholinergic receptor binding in mammalian central and peripheral nervous system with (3H) quinuclidinyl benzilate Federation Proceedings. 33. |
0.329 |
|
| 1973 |
Yamamura HI, Snyder SH. High affinity transport of choline into synaptosomes of rat brain. Journal of Neurochemistry. 21: 1355-74. PMID 4771436 DOI: 10.1111/j.1471-4159.1973.tb06022.x |
0.448 |
|
| 1973 |
Yamamura HI, Reichard DW, Gardner TL, Morrisett JD, Broomfield CA. Guinea pig brain acetylcholinesterase: partial purification by affinity chromatography. Biochimica Et Biophysica Acta. 302: 305-15. PMID 4699242 DOI: 10.1016/0005-2744(73)90159-9 |
0.312 |
|
| 1972 |
Yamamura HI, Snyder SH. Choline: high-affinity uptake by rat brain synaptosomes. Science (New York, N.Y.). 178: 626-8. PMID 5086398 DOI: 10.1126/science.178.4061.626 |
0.424 |
|
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