Emmanuel A. Theodorakis - Publications

Affiliations: 
1995- University of California, San Diego, La Jolla, CA 
Area:
Synthetic, Medicinal, Bioorganic and Biological Chemistry, Methods and Strategies in Natural Products Chemistry
Website:
https://profiles.ucsd.edu/emmanuel.theodorakis

98 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2019 Braddock AA, Theodorakis EA. Marine Spirotetronates: Biosynthetic Edifices That Inspire Drug Discovery. Marine Drugs. 17. PMID 31010150 DOI: 10.3390/Md17040232  0.302
2019 Chantarasriwong O, Milcarek AT, Morales TH, Settle AL, Rezende CO, Althufairi BD, Theodoraki MA, Alpaugh ML, Theodorakis EA. Synthesis, structure-activity relationship and in vitro pharmacodynamics of A-ring modified caged xanthones in a preclinical model of inflammatory breast cancer. European Journal of Medicinal Chemistry. 168: 405-413. PMID 30831408 DOI: 10.1016/J.Ejmech.2019.02.047  0.354
2016 Ke H, Morrisey JM, Qu S, Chantarasriwong O, Mather MW, Theodorakis EA, Vaidya AB. Caged Garcinia xanthones: a novel chemical scaffold with potent antimalarial activity. Antimicrobial Agents and Chemotherapy. PMID 27799215 DOI: 10.1128/Aac.01220-16  0.345
2015 Lacoske MH, Xu J, Mansour N, Gao C, Theodorakis EA. Synthetic Strategies Toward the Decalin Motif of Maklamicin and Related Spirotetronates. Organic Chemistry Frontiers : An International Journal of Organic Chemistry / Royal Society of Chemistry. 2: 388-393. PMID 26257916 DOI: 10.1039/C4Qo00332B  0.46
2015 Nicolaou KC, Shah AA, Korman H, Khan T, Shi L, Worawalai W, Theodorakis EA. Total Synthesis and Structural Revision of Antibiotic CJ-16,264. Angewandte Chemie (International Ed. in English). PMID 26096055 DOI: 10.1002/Anie.201504337  0.818
2015 Kocsis LS, Elbel KM, Hardigree BA, Brummond KM, Haidekker MA, Theodorakis EA. Cyclopenta[b]naphthalene cyanoacrylate dyes: synthesis and evaluation as fluorescent molecular rotors. Organic & Biomolecular Chemistry. 13: 2965-73. PMID 25614187 DOI: 10.1039/C4Ob02563F  0.34
2014 Caro-Diaz EJ, Aung A, Xu J, Varghese S, Theodorakis EA. Fusarisetins: Structure-function studies on a novel class of cell migration inhibitors. Organic Chemistry Frontiers : An International Journal of Organic Chemistry / Royal Society of Chemistry. 1: 135-139. PMID 24910777 DOI: 10.1039/C3Qo00067B  0.78
2013 Trzoss L, Xu J, Lacoske MH, Theodorakis EA. Synthesis of the tetracyclic core of Illicium sesquiterpenes using an organocatalyzed asymmetric Robinson annulation. Beilstein Journal of Organic Chemistry. 9: 1135-40. PMID 23843905 DOI: 10.3762/Bjoc.9.126  0.817
2013 Saitman A, Theodorakis EA. Synthesis of a highly functionalized core of verrillin. Organic Letters. 15: 2410-3. PMID 23627293 DOI: 10.1021/Ol400872H  0.83
2013 Saitman A, Sullivan SD, Theodorakis EA. A strategy toward the synthesis of C13-oxidized cembrenolides. Tetrahedron Letters. 54: 1612-1615. PMID 23626379 DOI: 10.1016/J.Tetlet.2013.01.085  0.784
2013 Elbel KM, Guizzunti G, Theodoraki MA, Xu J, Batova A, Dakanali M, Theodorakis EA. A-ring oxygenation modulates the chemistry and bioactivity of caged Garcinia xanthones. Organic & Biomolecular Chemistry. 11: 3341-8. PMID 23563530 DOI: 10.1039/C3Ob40395E  0.407
2013 Trzoss L, Xu J, Lacoske MH, Mobley WC, Theodorakis EA. Illicium sesquiterpenes: divergent synthetic strategy and neurotrophic activity studies. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 6398-408. PMID 23526661 DOI: 10.1002/Chem.201300198  0.819
2012 Xu J, Caro-Diaz EJ, Lacoske MH, Hung CI, Jamora C, Theodorakis EA. Fusarisetin A: Scalable Total Synthesis and Related Studies. Chemical Science (Royal Society of Chemistry : 2010). 3: 3378-3386. PMID 23227303 DOI: 10.1039/C2Sc21308G  0.827
2012 Martínez-Montero S, Fernández S, Sanghvi YS, Theodorakis EA, Detorio MA, McBrayer TR, Whitaker T, Schinazi RF, Gotor V, Ferrero M. Synthesis, evaluation of anti-HIV-1 and anti-HCV activity of novel 2',3'-dideoxy-2',2'-difluoro-4'-azanucleosides. Bioorganic & Medicinal Chemistry. 20: 6885-93. PMID 23085031 DOI: 10.1016/J.Bmc.2012.09.026  0.323
2012 Xu J, Caro-Diaz EJ, Batova A, Sullivan SD, Theodorakis EA. Formal synthesis of (-)-englerin A and cytotoxicity studies of truncated englerins. Chemistry, An Asian Journal. 7: 1052-60. PMID 22415793 DOI: 10.1002/Asia.201101021  0.822
2012 Xu J, Caro-Diaz EJ, Trzoss L, Theodorakis EA. Nature-inspired total synthesis of (-)-fusarisetin A. Journal of the American Chemical Society. 134: 5072-5. PMID 22390338 DOI: 10.1021/Ja300807E  0.831
2011 Saitman A, Rulliere P, Sullivan SD, Theodorakis EA. Total synthesis of norcembrenolide B and scabrolide D. Organic Letters. 13: 5854-7. PMID 21973225 DOI: 10.1021/Ol202476J  0.802
2011 Fischer D, Nguyen TX, Trzoss L, Dakanali M, Theodorakis EA. Intramolecular Cyclization Strategies Toward the Synthesis of Zoanthamine Alkaloids. Tetrahedron Letters. 52: 4920-4923. PMID 21857757 DOI: 10.1016/J.Tetlet.2011.07.054  0.824
2011 Trzoss L, Xu J, Lacoske MH, Mobley WC, Theodorakis EA. Enantioselective synthesis of (-)-jiadifenin, a potent neurotrophic modulator. Organic Letters. 13: 4554-7. PMID 21812392 DOI: 10.1021/Ol201742J  0.826
2011 Ling T, Xu J, Smith R, Ali A, Cantrell CL, Theodorakis EA. Synthesis of (-)-callicarpenal, a potent arthropod-repellent. Tetrahedron. 67: 3023-3029. PMID 21643472 DOI: 10.1016/J.Tet.2011.02.078  0.64
2011 Nguyen TX, Dakanali M, Trzoss L, Theodorakis EA. Enantioselective synthesis of the ABC ring motif of norzoanthamine based on asymmetric Robinson annulation reactions. Organic Letters. 13: 3308-11. PMID 21615125 DOI: 10.1021/Ol200966Z  0.835
2011 Xu J, Trzoss L, Chang WK, Theodorakis EA. Enantioselective total synthesis of (-)-jiadifenolide. Angewandte Chemie (International Ed. in English). 50: 3672-6. PMID 21400650 DOI: 10.1002/Anie.201100313  0.823
2010 Sutharsan J, Lichlyter D, Wright NE, Dakanali M, Haidekker MA, Theodorakis EA. Molecular rotors: Synthesis and evaluation as viscosity sensors. Tetrahedron. 66: 2582-2588. PMID 20694175 DOI: 10.1016/J.Tet.2010.01.093  0.306
2010 Xu J, Caro-Diaz EJ, Theodorakis EA. Enantioselective formal synthesis of (-)-englerin A via a Rh-catalyzed [4 + 3] cycloaddition reaction. Organic Letters. 12: 3708-11. PMID 20669919 DOI: 10.1021/Ol1015652  0.836
2010 Guizzunti G, Brady TP, Fischer D, Malhotra V, Theodorakis EA. Chemical biology studies on norrisolide. Bioorganic & Medicinal Chemistry. 18: 2115-22. PMID 20189813 DOI: 10.1016/J.Bmc.2010.02.007  0.751
2010 Xu J, Caro-Diaz EJE, Theodorakis EA. ChemInform Abstract: Enantioselective Formal Synthesis of (-)-Englerin A (V) via a Rh-Catalyzed [4 + 3] Cycloaddition Reaction. Cheminform. 41: no-no. DOI: 10.1002/chin.201051188  0.329
2009 Pongkittiphan V, Theodorakis EA, Chavasiri W. Hexachloroethane: a highly efficient reagent for the synthesis of chlorosilanes from hydrosilanes. Tetrahedron Letters. 50: 5080-5082. PMID 20360997 DOI: 10.1016/J.Tetlet.2009.05.087  0.436
2009 Chantarasriwong O, Cho WC, Batova A, Chavasiri W, Moore C, Rheingold AL, Theodorakis EA. Evaluation of the pharmacophoric motif of the caged Garcinia xanthones. Organic & Biomolecular Chemistry. 7: 4886-94. PMID 19907779 DOI: 10.1039/B913496D  0.411
2009 Díaz-Rodríguez A, Sanghvi YS, Fernández S, Schinazi RF, Theodorakis EA, Ferrero M, Gotor V. Synthesis and anti-HIV activity of conformationally restricted bicyclic hexahydroisobenzofuran nucleoside analogs. Organic & Biomolecular Chemistry. 7: 1415-23. PMID 19300828 DOI: 10.1039/B818707J  0.343
2007 Fischer D, Theodorakis EA, Haidekker MA. Synthesis and use of an in-solution ratiometric fluorescent viscosity sensor. Nature Protocols. 2: 227-36. PMID 17401358 DOI: 10.1038/Nprot.2006.455  0.526
2007 Traves PG, Hortelano S, Zeini M, Chao TH, Lam T, Neuteboom ST, Theodorakis EA, Palladino MA, Castrillo A, Bosca L. Selective activation of liver X receptors by acanthoic acid-related diterpenes. Molecular Pharmacology. 71: 1545-53. PMID 17329499 DOI: 10.1124/Mol.106.031906  0.567
2007 Batova A, Lam T, Wascholowski V, Yu AL, Giannis A, Theodorakis EA. Synthesis and evaluation of caged Garcinia xanthones. Organic & Biomolecular Chemistry. 5: 494-500. PMID 17252132 DOI: 10.1039/B612903J  0.654
2007 Guizzunti G, Brady TP, Malhotra V, Theodorakis EA. Trifunctional norrisolide probes for the study of Golgi vesiculation. Bioorganic & Medicinal Chemistry Letters. 17: 320-5. PMID 17110104 DOI: 10.1016/J.Bmcl.2006.10.101  0.696
2007 Fischer D, Theodorakis EA. Studies on the synthesis of Schisandraceae natural products: Exploring a cyclopropylcarbinol ring expansion strategy European Journal of Organic Chemistry. 4193-4196. DOI: 10.1002/Ejoc.200700336  0.617
2006 Haidekker MA, Akers WJ, Fischer D, Theodorakis EA. Optical fiber-based fluorescent viscosity sensor. Optics Letters. 31: 2529-31. PMID 16902608 DOI: 10.1364/Ol.31.002529  0.478
2006 Guizzunti G, Brady TP, Malhotra V, Theodorakis EA. Chemical analysis of norrisolide-induced Golgi vesiculation. Journal of the American Chemical Society. 128: 4190-1. PMID 16568969 DOI: 10.1021/Ja058259A  0.701
2006 Alexander MD, Burkart MD, Leonard MS, Portonovo P, Liang B, Ding X, Joullié MM, Gulledge BM, Aggen JB, Chamberlin AR, Sandler J, Fenical W, Cui J, Gharpure SJ, Polosukhin A, ... ... Theodorakis EA, et al. A central strategy for converting natural products into fluorescent probes. Chembiochem : a European Journal of Chemical Biology. 7: 409-16. PMID 16432909 DOI: 10.1002/Cbic.200500466  0.756
2006 Haidekker MA, Brady TP, Lichlyter D, Theodorakis EA. A ratiometric fluorescent viscosity sensor. Journal of the American Chemical Society. 128: 398-9. PMID 16402812 DOI: 10.1021/Ja056370A  0.669
2006 Sorensen EJ, Theodorakis EA. Nature-inspired approaches to chemical synthesis Tetrahedron. 62: 5169. DOI: 10.1016/J.Tet.2006.02.084  0.6
2005 Haidekker MA, Brady TP, Lichlyter D, Theodorakis EA. Effects of solvent polarity and solvent viscosity on the fluorescent properties of molecular rotors and related probes. Bioorganic Chemistry. 33: 415-25. PMID 16182338 DOI: 10.1016/J.Bioorg.2005.07.005  0.671
2005 Brady TP, Kim SH, Wen K, Kim C, Theodorakis EA. Norrisolide: total synthesis and related studies. Chemistry (Weinheim An Der Bergstrasse, Germany). 11: 7175-90. PMID 16163770 DOI: 10.1002/Chem.200500513  0.777
2005 Chao TH, Lam T, Vong BG, Través PG, Hortelano S, Chowdhury C, Bahjat FR, Lloyd GK, Moldawer LL, Boscá L, Palladino MA, Theodorakis EA. A new family of synthetic diterpenes that regulates cytokine synthesis by inhibiting IkappaBalpha phosphorylation. Chembiochem : a European Journal of Chemical Biology. 6: 133-44. PMID 15540220 DOI: 10.1002/Cbic.200400089  0.781
2005 Haidekker MA, Akers W, Lichlyter D, Brady TP, Theodorakis EA. Sensing of flow and shear stress using fluorescent molecular rotors Sensor Letters. 3: 42-48. DOI: 10.1166/Sl.2005.003  0.663
2005 Rivas F, Ghosh S, Theodorakis EA. Synthetic studies toward the zoanthamine alkaloids: Synthesis of the fully functionalized BC ring motif Tetrahedron Letters. 46: 5281-5284. DOI: 10.1016/J.Tetlet.2005.06.037  0.811
2005 Brady TP, Kim SH, Wen K, Kim C, Theodorakis EA. Cover Picture: Norrisolide: Total Synthesis and Related Studies (Chem. Eur. J. 24/2005) Chemistry - a European Journal. 11: 7135-7135. DOI: 10.1002/Chem.200590075  0.731
2004 Brady TP, Wallace EK, Kim SH, Guizzunti G, Malhotra V, Theodorakis EA. Fragmentation of Golgi membranes by norrisolide and designed analogues. Bioorganic & Medicinal Chemistry Letters. 14: 5035-9. PMID 15380194 DOI: 10.1016/J.Bmcl.2004.08.003  0.696
2004 Vong BG, Kim SH, Abraham S, Theodorakis EA. Stereoselective total synthesis of (-)-borrelidin. Angewandte Chemie (International Ed. in English). 43: 3947-51. PMID 15274222 DOI: 10.1002/Anie.200460203  0.831
2004 Tisdale EJ, Slobodov I, Theodorakis EA. Unified synthesis of caged Garcinia natural products based on a site-selective Claisen/Diels-Alder/Claisen rearrangement. Proceedings of the National Academy of Sciences of the United States of America. 101: 12030-5. PMID 15210986 DOI: 10.1073/Pnas.0401932101  0.782
2004 Haidekker MA, Brady TP, Chalian SH, Akers W, Lichlyter D, Theodorakis EA. Hydrophilic molecular rotor derivatives-synthesis and characterization. Bioorganic Chemistry. 32: 274-89. PMID 15210341 DOI: 10.1016/J.Bioorg.2004.04.002  0.702
2004 Oka N, Sanghvi YS, Theodorakis EA. 3,3(')-Oxybis(dimethoxytrityl chloride) (O-DMTCl): synthesis and applications of a novel bifunctional protecting group. Bioorganic & Medicinal Chemistry Letters. 14: 3241-4. PMID 15149683 DOI: 10.1016/J.Bmcl.2004.03.097  0.356
2004 Ghosh S, Rivas F, Fischer D, González MA, Theodorakis EA. Stereoselective synthesis of the ABC ring system of norzoanthamine. Organic Letters. 6: 941-4. PMID 15012070 DOI: 10.1021/Ol036492C  0.836
2004 Brady TP, Kim SH, Wen K, Theodorakis EA. Stereoselective total synthesis of (+)-norrisolide. Angewandte Chemie (International Ed. in English). 43: 739-42. PMID 14755708 DOI: 10.1002/Anie.200352868  0.774
2004 Kim C, Brady T, Kim SH, Theodorakis EA. Synthesis of fused tetrahydrofuran-γ-lactone motifs via one-pot ring expansion of cyclopropane rings Synthetic Communications. 34: 1951-1965. DOI: 10.1081/Scc-120037907  0.759
2004 Oka N, Sanghvi YS, Theodorakis EA. 1,2-Ethylene-3,3-bis(4′,4″-dimethoxytrityl chloride) (E-DMT): Synthesis and applications of a novel protecting reagent Synlett. 823-826. DOI: 10.1055/S-2004-820033  0.409
2004 Theodorakis EA, Ling T, Rueden EJ, Poupon E, Kim SH. Chapter 4 Quinone sesquiterpenes: A challenge for the development of a new synthetic methodology Strategies and Tactics in Organic Synthesis. 5: 111-131. DOI: 10.1016/S1874-6004(04)80027-3  0.691
2004 González MA, Ghosh S, Rivas F, Fischer D, Theodorakis EA. Synthesis of (+)- and (-)-isocarvone Tetrahedron Letters. 45: 5039-5041. DOI: 10.1016/J.Tetlet.2004.04.181  0.816
2003 Tisdale EJ, Slobodov I, Theodorakis EA. Biomimetic total synthesis of forbesione and desoxymorellin utilizing a tandem Claisen/Diels--Alder/Claisen rearrangement. Organic & Biomolecular Chemistry. 1: 4418-22. PMID 14727628 DOI: 10.1039/B311833A  0.784
2003 Chow S, Wen K, Sanghvi YS, Theodorakis EA. MDPSCL2: a new protecting group for chemoselective synthesis of 2'-O-alkylated guanosines. Nucleosides, Nucleotides & Nucleic Acids. 22: 583-7. PMID 14565233 DOI: 10.1081/Ncn-120021959  0.398
2003 Lam T, Ling T, Chowdhury C, Chao TH, Bahjat FR, Lloyd GK, Moldawer LL, Palladino MA, Theodorakis EA. Synthesis of a novel family of diterpenes and their evaluation as anti-inflammatory agents. Bioorganic & Medicinal Chemistry Letters. 13: 3217-21. PMID 12951096 DOI: 10.1016/S0960-894X(03)00669-3  0.793
2003 Vong BG, Abraham S, Xiang AX, Theodorakis EA. Synthetic studies on borrelidin: enantioselective synthesis of the C1-C12 fragment. Organic Letters. 5: 1617-20. PMID 12735735 DOI: 10.1021/Ol034243I  0.802
2003 Chow S, Wen K, Sanghvi YS, Theodorakis EA. Novel synthesis of 2'-O-methylguanosine. Bioorganic & Medicinal Chemistry Letters. 13: 1631-4. PMID 12729629 DOI: 10.1016/S0960-894X(03)00291-9  0.321
2003 Tisdale EJ, Li H, Vong BG, Kim SH, Theodorakis EA. Regioselective synthesis of the tricyclic core of lateriflorone. Organic Letters. 5: 1491-4. PMID 12713306 DOI: 10.1021/Ol034276Y  0.823
2003 Tisdale EJ, Kochman DA, Theodorakis EA. Total synthesis of atroviridin Tetrahedron Letters. 44: 3281-3284. DOI: 10.1016/S0040-4039(03)00629-4  0.792
2003 Tisdale EJ, Vong BG, Li H, Kim SH, Chowdhury C, Theodorakis EA. Total synthesis of seco-lateriflorone Tetrahedron. 59: 6873-6887. DOI: 10.1016/S0040-4020(03)00862-7  0.821
2003 Lee NJ, Ju SS, Cho WJ, Kim SH, Kang KT, Brady T, Theodorakis EA. Synthesis and biological activity of medium molecular weight polymers of camptothecin European Polymer Journal. 39: 367-374. DOI: 10.1016/S0014-3057(02)00219-7  0.684
2003 Lee NJ, Ju SS, Cho WJ, Kim SH, Kang KT, Brady T, Theodorakis EA. Synthesis and antitumour activity of medium molecular weight phthalimide polymers of camptothecin Polymer International. 52: 1339-1345. DOI: 10.1002/Pi.1138  0.678
2002 Wen K, Chow S, Sanghvi YS, Theodorakis EA. Synthesis of 2'-O-methoxyethylguanosine using a novel silicon-based protecting group. The Journal of Organic Chemistry. 67: 7887-9. PMID 12398522 DOI: 10.1021/Jo025970E  0.398
2002 Ling T, Poupon E, Rueden EJ, Kim SH, Theodorakis EA. Unified synthesis of quinone sesquiterpenes based on a radical decarboxylation and quinone addition reaction. Journal of the American Chemical Society. 124: 12261-7. PMID 12371868 DOI: 10.1021/Ja027517Q  0.689
2002 Haidekker MA, Brady T, Wen K, Okada C, Stevens HY, Snell JM, Frangos JA, Theodorakis EA. Phospholipid-bound molecular rotors: synthesis and characterization. Bioorganic & Medicinal Chemistry. 10: 3627-36. PMID 12213479 DOI: 10.1016/S0968-0896(02)00240-7  0.681
2002 Haidekker MA, Tsai AG, Brady T, Stevens HY, Frangos JA, Theodorakis E, Intaglietta M. A novel approach to blood plasma viscosity measurement using fluorescent molecular rotors. American Journal of Physiology. Heart and Circulatory Physiology. 282: H1609-14. PMID 11959622 DOI: 10.1152/Ajpheart.00712.2001  0.676
2002 Tisdale EJ, Chowdhury C, Vong BG, Li H, Theodorakis EA. Regioselective synthesis of the bridged tricyclic core of Garcinia natural products via intramolecular aryl acrylate cycloadditions. Organic Letters. 4: 909-12. PMID 11893183 DOI: 10.1021/Ol017278W  0.816
2002 Ling T, Poupon E, Rueden EJ, Theodorakis EA. Synthesis of (-)-ilimaquinone via a radical decarboxylation and quinone addition reaction. Organic Letters. 4: 819-22. PMID 11869136 DOI: 10.1021/Ol025501Z  0.654
2002 Ling T, Rivas F, Theodorakis EA. Stereoselective synthesis of the fully functionalized core fragment of terpentecin Tetrahedron Letters. 43: 9019-9022. DOI: 10.1016/S0040-4039(02)02314-6  0.811
2001 Ling T, Chowdhury C, Kramer BA, Vong BG, Palladino MA, Theodorakis EA. Enantioselective synthesis of the antiinflammatory agent (-)-acanthoic acid. The Journal of Organic Chemistry. 66: 8843-53. PMID 11749614 DOI: 10.1021/Jo0159035  0.834
2001 Haidekker MA, Ling T, Anglo M, Stevens HY, Frangos JA, Theodorakis EA. New fluorescent probes for the measurement of cell membrane viscosity. Chemistry & Biology. 8: 123-31. PMID 11251287 DOI: 10.1016/S1074-5521(00)90061-9  0.524
2001 Lee N, Kang N, Cho W, Kim S, Kang K, Theodorakis EA. Synthesis and biological activity of medium range molecular weight polymers containingexo-3,6-epoxy-1,2,3,6-tetrahydrophthalimidocaproic acid Polymer International. 50: 1010-1015. DOI: 10.1002/Pi.736  0.305
2000 Drouet KE, Theodorakis EA. Stereoselective total synthesis of reveromycin B and C19-epi-reveromycin B. Chemistry (Weinheim An Der Bergstrasse, Germany). 6: 1987-2001. PMID 10894398 DOI: 10.1002/1521-3765(20000602)6:11<1987::Aid-Chem1987>3.0.Co;2-U  0.493
2000 Ling T, Kramer BA, Palladino MA, Theodorakis EA. Stereoselective synthesis of (-)-acanthoic acid. Organic Letters. 2: 2073-6. PMID 10891233 DOI: 10.1021/Ol0060578  0.696
2000 Drouet KE, Ling T, Tran HV, Theodorakis EA. Enantioselective synthesis of the [6,6] spiroketal core of reveromycin A. Organic Letters. 2: 207-10. PMID 10814283 DOI: 10.1021/Ol991290V  0.655
2000 Drouet KE, Tran HV, Theodorakis EA. Efficient synthesis of the C1-C8 fragment of reveromycins Synthetic Communications. 30: 3617-3628. DOI: 10.1080/00397910008087279  0.403
1999 Ling T, Xiang AX, Theodorakis EA. Enantioselective Total Synthesis of Avarol and Avarone. Angewandte Chemie (International Ed. in English). 38: 3089-3091. PMID 10540432 DOI: 10.1002/(Sici)1521-3773(19991018)38:20<3089::Aid-Anie3089>3.0.Co;2-W  0.819
1999 Blom P, Xiang AX, Kao D, Theodorakis EA. Design, synthesis, and evaluation of N-aroyloxy-2-thiopyridones as DNA photocleaving reagents. Bioorganic & Medicinal Chemistry. 7: 727-36. PMID 10400326 DOI: 10.1016/S0968-0896(98)00211-9  0.737
1999 Kim C, Hoang R, Theodorakis EA. Synthetic studies on norrisolide: Enantioselective synthesis of the norrisane side chain Organic Letters. 1: 1295-1297. DOI: 10.1021/Ol9909785  0.413
1999 Drouet KE, Theodorakis EA. Enantioselective total synthesis of reveromycin B Journal of the American Chemical Society. 121: 456-457. DOI: 10.1021/Ja983429N  0.425
1999 Ling T, Xiang AX, Theodorakis EA. Enantioselektive Totalsynthese von Avarol und Avaron Angewandte Chemie. 111: 3277-3279. DOI: 10.1002/(Sici)1521-3757(19991018)111:20<3277::Aid-Ange3277>3.0.Co;2-M  0.741
1998 Xiang AX, Watson DA, Ling T, Theodorakis EA. Total Synthesis of Clerocidin via a Novel, Enantioselective Homoallenylboration Methodology. The Journal of Organic Chemistry. 63: 6774-6775. PMID 11672290 DOI: 10.1021/Jo981331L  0.807
1996 Liu C, Smith BM, Ajito K, Komatsu H, Gomez-Paloma L, Li T, Theodorakis EA, Nicolaou KC, Vogt PK. Sequence-selective carbohydrate-DNA interaction: dimeric and monomeric forms of the calicheamicin oligosaccharide interfere with transcription factor function. Proceedings of the National Academy of Sciences of the United States of America. 93: 940-4. PMID 8570664 DOI: 10.1073/Pnas.93.2.940  0.488
1996 Nicolaou KC, Theodorakis EA, Claiborne CF. Chemistry and biology of selected natural products Pure and Applied Chemistry. 68: 2129-2136. DOI: 10.1351/Pac199668112129  0.568
1995 Gawley RE, Rein KS, Jeglitsch G, Adams DJ, Theodorakis EA, Tiebes J, Nicolaou KC, Baden DG. The relationship of brevetoxin 'length' and A-ring functionality to binding and activity in neuronal sodium channels. Chemistry & Biology. 2: 533-41. PMID 9383457 DOI: 10.1016/1074-5521(95)90187-6  0.491
1995 Nicolaou KC, Sato M, Theodorakis EA, Miller ND. Conversion of thionoesters and thionolactones to ethers; a general and efficient radical desulfurisation Journal of the Chemical Society, Chemical Communications. 1583-1585. DOI: 10.1039/C39950001583  0.552
1995 Nicolaou KC, Rutjes FPJT, Theodorakis EA, Tiebes J, Sato M, Untersteller E. Total synthesis of brevetoxin B. 3. Final strategy and completion Journal of the American Chemical Society. 117: 10252-10263. DOI: 10.1021/Ja00146A010  0.618
1995 Nicolaou KC, Theodorakis EA, Rutjes FPJT, Sato M, Tiebes J, Xiao XY, Hwang CK, Duggan ME, Yang Z, Couladouros EA, Sato F, Shin J, He HM, Bleckman T. Total synthesis of brevetoxin B. 2. Second generation strategies and construction of the dioxepane region [DEFG] Journal of the American Chemical Society. 117: 10239-10251. DOI: 10.1021/Ja00146A009  0.681
1995 Nicolaou KC, Hwang CK, Duggan ME, Nugiel DA, Abe Y, Bal Reddy K, DeFrees SA, Reddy DR, Awartani RA, Conley SR, Rutjes FPJT, Theodorakis EA. Total synthesis of brevetoxin B. 1. First generation strategies and new approaches to oxepane systems Journal of the American Chemical Society. 117: 10227-10238. DOI: 10.1021/Ja00146A008  0.614
1995 Nicolaou KC, Rutjes FPJT, Theodorakis EA, Tiebes J, Sato M, Untersteller E. Total synthesis of brevetoxin B. 2. Completion Journal of the American Chemical Society. 117: 1173-1174. DOI: 10.1021/Ja00108A052  0.569
1995 Nicolaou KC, Theodorakis EA, Rutjes FPJT, Tiebes J, Sato M, Untersteller E, Xiao XY. Total synthesis of brevetoxin B. 1. CDEFG framework Journal of the American Chemical Society. 117: 1171-1172. DOI: 10.1021/Ja00108A051  0.569
1994 Nicolaou KC, Pitsinos EN, Theodorakis EA, Saimoto H, Wrasidlo W. Synthetic calicheamicin mimics with novel initiation mechanisms: DNA cleavage, cytotoxicity, and apoptosis. Chemistry & Biology. 1: 57-66. PMID 9383371 DOI: 10.1016/1074-5521(94)90041-8  0.527
1994 Nicolaou KC, Tiebes J, Theodorakis EA, Rutjes FPJT, Koide K, Sato M, Untersteller E. Total Synthesis of Truncated Brevetoxin B [AFGHIJK] Journal of the American Chemical Society. 116: 9371-9372. DOI: 10.1021/Ja00099A081  0.674
1991 Theodorakis E, Royer J, Husson HP. Asymmetric Synthesis XXIII.1 A 100% CIS Diastereoselectivity in the Synthesis of Enantiomerically Pure 2,6-Dialkylpiperidines Synthetic Communications. 21: 521-529. DOI: 10.1080/00397919108016778  0.431
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