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Sandip B. Bharate - Publications

Affiliations: 
2011- CSIR-IIIM (Academy of Scientific and Innovative Research) 
Area:
Pharmaceutical chemistry, medicinal chemistry
Website:
https://sites.google.com/site/bharatesb/
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273 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Sharma M, Sharma A, Thakur S, Nuthakki VK, Jamwal A, Nandi U, Jadhav HR, Bharate SB. Discovery of blood-brain barrier permeable and orally bioavailable caffeine-based amide derivatives as acetylcholinesterase inhibitors. Bioorganic Chemistry. 139: 106719. PMID 37473478 DOI: 10.1016/j.bioorg.2023.106719  0.815
2023 Bhurta D, Hossain MM, Bhardwaj M, Showket F, Nandi U, Dar MJ, Bharate SB. Orally bioavailable styryl derivative of rohitukine-N-oxide inhibits CDK9/T1 and the growth of pancreatic cancer cells. European Journal of Medicinal Chemistry. 258: 115533. PMID 37302342 DOI: 10.1016/j.ejmech.2023.115533  0.822
2023 Abdullaha M, Banoo R, Nuthakki VK, Sharma M, Kaur S, Thakur S, Kumar A, Jadhav HR, Bharate SB. Methoxy-naphthyl-Linked -Benzyl Pyridinium Styryls as Dual Cholinesterase Inhibitors: Design, Synthesis, Biological Evaluation, and Structure-Activity Relationship. Acs Omega. 8: 17591-17608. PMID 37251153 DOI: 10.1021/acsomega.2c08167  0.811
2023 Sharma A, Bharate SB. Synthesis and Biological Evaluation of Coumarin Triazoles as Dual Inhibitors of Cholinesterases and β-Secretase. Acs Omega. 8: 11161-11176. PMID 37008108 DOI: 10.1021/acsomega.2c07993  0.621
2023 Nuthakki VK, Choudhary S, Reddy CN, Bhatt S, Jamwal A, Jotshi A, Raghuvanshi R, Sharma A, Thakur S, Jadhav HR, Bharate SS, Nandi U, Kumar A, Bharate SB. Design, Synthesis, and Pharmacological Evaluation of Embelin-Aryl/alkyl Amine Hybrids as Orally Bioavailable Blood-Brain Barrier Permeable Multitargeted Agents with Therapeutic Potential in Alzheimer's Disease: Discovery of SB-1448. Acs Chemical Neuroscience. 14: 1193-1219. PMID 36812360 DOI: 10.1021/acschemneuro.3c00030  0.812
2022 Bhurta D, Bharate SB. Discovery of Pongol, the Furanoflavonoid, as an Inhibitor of CDK7/Cyclin H/MAT1 and Its Preliminary Structure-Activity Relationship. Acs Omega. 8: 1291-1300. PMID 36643464 DOI: 10.1021/acsomega.2c06733  0.812
2022 Raghuvanshi R, Jamwal A, Nandi U, Bharate SB. Multitargeted C9-substituted ester and ether derivatives of berberrubine for Alzheimer's disease: Design, synthesis, biological evaluation, metabolic stability, and pharmacokinetics. Drug Development Research. PMID 36461610 DOI: 10.1002/ddr.22017  0.824
2022 Ntemafack A, Qayum A, Dhiman SK, Guefack MF, Thapa S, Wamba BEN, Kuete V, Singh SK, Bharate SB, Hassan QP, Gandhi SG. Antimicrobial and Cytotoxic Potential of Helminthosporin from Rumex abyssiniscus Jacq. Discovered as a Novel Source of Syringic Acid and Bis(2-ethyloctyl) Phthalate. Current Microbiology. 80: 7. PMID 36445554 DOI: 10.1007/s00284-022-03101-2  0.404
2022 Malik S, Mintoo MJ, Reddy CN, Kumar R, Kotwal P, Bharate SB, Nandi U, Mondhe DM, Shukla SK. In vitro and in vivo anticancer potential and molecular targets of the new colchicine analog IIIM-067. Journal of Integrative Medicine. PMID 36253285 DOI: 10.1016/j.joim.2022.09.006  0.369
2022 Sharma M, Sharma A, Nuthakki VK, Bhatt S, Nandi U, Bharate SB. Design, synthesis, and structure-activity relationship of caffeine-based triazoles as dual AChE and BACE-1 inhibitors. Drug Development Research. PMID 36161804 DOI: 10.1002/ddr.21998  0.823
2022 Jain SK, Pathania AS, Parshad R, Raina C, Ali A, Gupta AP, Kushwaha M, Aravinda S, Bhushan S, Bharate SB, Vishwakarma RA. Correction: Chrysomycins A-C, antileukemic naphthocoumarins from . Rsc Advances. 12: 23680-23682. PMID 36125971 DOI: 10.1039/d2ra90078e  0.756
2022 Banoo R, Nuthakki VK, Abdullaha M, Sharma M, Bharate SB. Blood-brain barrier permeable benzylpiperidin-4-yl-linked benzylamino benzamides as dual cholinesterase inhibitors. Drug Development Research. PMID 36112736 DOI: 10.1002/ddr.21997  0.802
2022 Nazir LA, Shahid NH, Amit K, Umar SA, Rajni S, Bharate S, Sangwan PL, Tasduq SA. Synthesis and anti-melanoma effect of 3-O-prenyl glycyrrhetinic acid against B16F10 cells induction of endoplasmic reticulum stress-mediated autophagy through ERK/AKT signaling pathway. Frontiers in Oncology. 12: 890299. PMID 35982963 DOI: 10.3389/fonc.2022.890299  0.341
2022 Sharma A, Nuthakki VK, Gairola S, Singh B, Bharate SB. A Coumarin-donepezil Hybrid as a Blood-brain Barrier Permeable Dual Cholinesterase Inhibitor: Isolation, Synthetic Modifications and Biological Evaluation of Natural Coumarins. Chemmedchem. PMID 35892288 DOI: 10.1002/cmdc.202200300  0.815
2022 Shah K, Maradana MR, Joaquina Delàs M, Metidji A, Graelmann F, Llorian M, Chakravarty P, Li Y, Tolaini M, Shapiro M, Kelly G, Cheshire C, Bhurta D, Bharate SB, Stockinger B. Cell-intrinsic Aryl Hydrocarbon Receptor signalling is required for the resolution of injury-induced colonic stem cells. Nature Communications. 13: 1827. PMID 35383166 DOI: 10.1038/s41467-022-29098-7  0.771
2022 Ntemafack A, Ahmed S, Kumar A, Chouhan R, Kapoor N, Bharate SB, Hassan QP, Gandhi SG. Plant growth promoting potential of butyl isobutyl phthalate and Streptomyces sp. from Rumex dentatus on rice. Applied Microbiology and Biotechnology. 106: 2603-2617. PMID 35262787 DOI: 10.1007/s00253-022-11862-w  0.299
2022 Bhurta D, Bharate SB. Styryl Group, a Friend or Foe in Medicinal Chemistry. Chemmedchem. 17: e202100706. PMID 35166041 DOI: 10.1002/cmdc.202100706  0.791
2021 Nuthakki VK, Mudududdla R, Bharate SB. Role of basic aminoalkyl chains in the lead optimization of Indoloquinoline alkaloids. European Journal of Medicinal Chemistry. 227: 113938. PMID 34710743 DOI: 10.1016/j.ejmech.2021.113938  0.79
2021 Bhurta D, Bharate SB. Analyzing the scaffold diversity of cyclin-dependent kinase inhibitors and revisiting the clinical and preclinical pipeline. Medicinal Research Reviews. PMID 34605036 DOI: 10.1002/med.21856  0.79
2021 Girme A, Saste G, Pawar S, Ghule C, Mirgal A, Patel S, Tiwari A, Ghoshal S, Bharate SB, Bharate SS, Reddy DS, Vishwakarma RA, Hingorani L. Quantitative Determination and Characterization of a Kashmir Saffron ( L.)-Based Botanical Supplement Using Single-Laboratory Validation Study by HPLC-PDA with LC-MS/MS and HPTLC Investigations. Acs Omega. 6: 23460-23474. PMID 34549144 DOI: 10.1021/acsomega.1c03470  0.489
2021 Abdullaha M, Ali M, Kour D, Mudududdla R, Khajuria P, Kumar A, Bharate SB. Tetramethoxystilbene Inhibits NLRP3 Inflammasome Assembly via Blocking the Oligomerization of Apoptosis-Associated Speck-like Protein Containing Caspase Recruitment Domain: and Evaluation. Acs Pharmacology & Translational Science. 4: 1437-1448. PMID 34423275 DOI: 10.1021/acsptsci.1c00126  0.747
2021 Raghuvanshi R, Nuthakki VK, Singh L, Singh B, Bharate SS, Bhatti R, Bharate SB. Identification of plant-based multitargeted leads for Alzheimer's disease: In-vitro and in-vivo validation of Woodfordia fruticosa (L.) Kurz. Phytomedicine : International Journal of Phytotherapy and Phytopharmacology. 91: 153659. PMID 34332286 DOI: 10.1016/j.phymed.2021.153659  0.769
2021 Mintoo M, Khan S, Wani A, Malik S, Bhurta D, Bharate S, Malik F, Mondhe D. A rohitukine derivative IIIM-290 induces p53 dependent mitochondrial apoptosis in acute lymphoblastic leukemia cells. Molecular Carcinogenesis. PMID 34324743 DOI: 10.1002/mc.23332  0.799
2021 Prabhakara C, Godbole R, Sil P, Jahnavi S, Gulzar SE, van Zanten TS, Sheth D, Subhash N, Chandra A, Shivaraj A, Panikulam P, U I, Nuthakki VK, Puthiyapurayil TP, Ahmed R, ... ... Bharate SB, et al. Strategies to target SARS-CoV-2 entry and infection using dual mechanisms of inhibition by acidification inhibitors. Plos Pathogens. 17: e1009706. PMID 34252168 DOI: 10.1371/journal.ppat.1009706  0.781
2021 Prabhakara C, Godbole R, Sil P, Jahnavi S, Gulzar SE, van Zanten TS, Sheth D, Subhash N, Chandra A, Shivaraj A, Panikulam P, U I, Nuthakki VK, Puthiyapurayil TP, Ahmed R, ... ... Bharate SB, et al. Strategies to target SARS-CoV-2 entry and infection using dual mechanisms of inhibition by acidification inhibitors. Plos Pathogens. 17: e1009706. PMID 34252168 DOI: 10.1371/journal.ppat.1009706  0.781
2021 Ali M, Gupta M, Wani A, Sharma A, Abdullaha M, Kour D, Choudhary S, Bharate SB, Singh G, Kumar A. IIIM-941, a Stilbene Derivative Inhibits NLRP3 Inflammasome Activation by Inducing Autophagy. Frontiers in Pharmacology. 12: 695712. PMID 34248643 DOI: 10.3389/fphar.2021.695712  0.612
2021 Ali M, Gupta M, Wani A, Sharma A, Abdullaha M, Kour D, Choudhary S, Bharate SB, Singh G, Kumar A. IIIM-941, a Stilbene Derivative Inhibits NLRP3 Inflammasome Activation by Inducing Autophagy. Frontiers in Pharmacology. 12: 695712. PMID 34248643 DOI: 10.3389/fphar.2021.695712  0.612
2021 Gupta M, Wani A, Ahsan AU, Ali M, Chibber P, Singh S, Digra SK, Datt M, Bharate S, Vishwakarma RA, Singh G, Kumar A. Safranal inhibits NLRP3 inflammasome activation by preventing ASC oligomerization. Toxicology and Applied Pharmacology. 115582. PMID 34019860 DOI: 10.1016/j.taap.2021.115582  0.506
2021 Gupta M, Wani A, Ahsan AU, Ali M, Chibber P, Singh S, Digra SK, Datt M, Bharate S, Vishwakarma RA, Singh G, Kumar A. Safranal inhibits NLRP3 inflammasome activation by preventing ASC oligomerization. Toxicology and Applied Pharmacology. 115582. PMID 34019860 DOI: 10.1016/j.taap.2021.115582  0.506
2021 Raghuvanshi R, Bharate SB. Recent Developments in the Use of Kinase Inhibitors for Management of Viral Infections. Journal of Medicinal Chemistry. PMID 33539089 DOI: 10.1021/acs.jmedchem.0c01467  0.785
2021 Raghuvanshi R, Bharate SB. Recent Developments in the Use of Kinase Inhibitors for Management of Viral Infections. Journal of Medicinal Chemistry. PMID 33539089 DOI: 10.1021/acs.jmedchem.0c01467  0.308
2021 Nuthakki VK, Yadav Bheemanaboina RR, Bharate SB. Identification of aplysinopsin as a blood-brain barrier permeable scaffold for anti-cholinesterase and anti-BACE-1 activity. Bioorganic Chemistry. 107: 104568. PMID 33418314 DOI: 10.1016/j.bioorg.2020.104568  0.781
2021 Nuthakki VK, Yadav Bheemanaboina RR, Bharate SB. Identification of aplysinopsin as a blood-brain barrier permeable scaffold for anti-cholinesterase and anti-BACE-1 activity. Bioorganic Chemistry. 107: 104568. PMID 33418314 DOI: 10.1016/j.bioorg.2020.104568  0.42
2021 Wani A, Al Rihani SB, Sharma A, Weadick B, Govindarajan R, Khan SU, Sharma PR, Dogra A, Nandi U, Reddy CN, Bharate SS, Singh G, Bharate SB, Vishwakarma RA, Kaddoumi A, et al. Crocetin promotes clearance of amyloid-β by inducing autophagy via the STK11/LKB1-mediated AMPK pathway. Autophagy. PMID 33404280 DOI: 10.1080/15548627.2021.1872187  0.658
2020 Mahajan S, Slathia N, Nuthakki VK, Bharate SB, Kapoor KK. Malononitrile-activated synthesis and anti-cholinesterase activity of styrylquinoxalin-2(1)-ones. Rsc Advances. 10: 15966-15975. PMID 35493659 DOI: 10.1039/d0ra02816a  0.762
2020 Mahajan S, Slathia N, Nuthakki VK, Bharate SB, Kapoor KK. Malononitrile-activated synthesis and anti-cholinesterase activity of styrylquinoxalin-2(1)-ones. Rsc Advances. 10: 15966-15975. PMID 35493659 DOI: 10.1039/d0ra02816a  0.762
2020 Sharma V, Sharma A, Bharate SB. Natural Products in Mitigation of SARS CoV Infections. Current Medicinal Chemistry. PMID 33109028 DOI: 10.2174/0929867327666201027153940  0.551
2020 Sharma V, Sharma A, Bharate SB. Natural Products in Mitigation of SARS CoV Infections. Current Medicinal Chemistry. PMID 33109028 DOI: 10.2174/0929867327666201027153940  0.273
2020 Dheer D, Behera C, Singh D, Abdullaha M, Chashoo G, Bharate SB, Gupta PN, Shankar R. Design, synthesis and comparative analysis of triphenyl-1,2,3-triazoles as anti-proliferative agents. European Journal of Medicinal Chemistry. 207: 112813. PMID 32947093 DOI: 10.1016/j.ejmech.2020.112813  0.386
2020 Abdullaha M, Nuthakki VK, Bharate SB. Discovery of methoxy-naphthyl linked N-(1-benzylpiperidine) benzamide as a blood-brain permeable dual inhibitor of acetylcholinesterase and butyrylcholinesterase. European Journal of Medicinal Chemistry. 207: 112761. PMID 32942070 DOI: 10.1016/j.ejmech.2020.112761  0.771
2020 Abdullaha M, Nuthakki VK, Bharate SB. Discovery of methoxy-naphthyl linked N-(1-benzylpiperidine) benzamide as a blood-brain permeable dual inhibitor of acetylcholinesterase and butyrylcholinesterase. European Journal of Medicinal Chemistry. 207: 112761. PMID 32942070 DOI: 10.1016/j.ejmech.2020.112761  0.391
2020 Bharate SB. Modulation of Kinases by Small Molecules for Therapeutic Management of Various Diseases - Part II. Current Topics in Medicinal Chemistry. 20: 1521. PMID 32830621 DOI: 10.2174/156802662017200624114631  0.236
2020 Bharate SB. Modulation of Kinases by Small Molecules for Therapeutic Management of Various Diseases - Part II. Current Topics in Medicinal Chemistry. 20: 1521. PMID 32830621 DOI: 10.2174/156802662017200624114631  0.236
2020 Bharate SB. Modulation of Kinases by Small Molecules for Therapeutic Management of Various Diseases - Part I. Current Topics in Medicinal Chemistry. 20: 1057-1058. PMID 32495727 DOI: 10.2174/156802662012200504090532  0.24
2020 Bharate SB. Modulation of Kinases by Small Molecules for Therapeutic Management of Various Diseases - Part I. Current Topics in Medicinal Chemistry. 20: 1057-1058. PMID 32495727 DOI: 10.2174/156802662012200504090532  0.24
2020 Raghuvanshi R, Bharate SB. Preclinical and Clinical Studies on Bryostatins, A Class of Marine-Derived Protein Kinase C Modulators: A Mini-Review. Current Topics in Medicinal Chemistry. 20: 1124-1135. PMID 32209043 DOI: 10.2174/1568026620666200325110444  0.803
2020 Raghuvanshi R, Bharate SB. Preclinical and Clinical Studies on Bryostatins, A Class of Marine-Derived Protein Kinase C Modulators: A Mini-Review. Current Topics in Medicinal Chemistry. 20: 1124-1135. PMID 32209043 DOI: 10.2174/1568026620666200325110444  0.369
2020 Kumar V, Bharate SS, Bhurta D, Gupta M, Gandhi SG, Singh D, Jaglan S, Kumar A, Vishwakarma RA, Bharate SB. Evaluation of rohitukine-enriched fraction of Dysoxylum binectariferum Hook.f. (leaves) as anti-arthritic phytopharmaceutical candidate: Chemical standardization, in-vivo validation, formulation development and oral pharmacokinetics. Journal of Ethnopharmacology. 112758. PMID 32165175 DOI: 10.1016/J.Jep.2020.112758  0.767
2020 Augustin N, Nuthakki VK, Abdullaha M, Hassan QP, Gandhi SG, Bharate SB. Discovery of Helminthosporin, an Anthraquinone Isolated from Jacq as a Dual Cholinesterase Inhibitor. Acs Omega. 5: 1616-1624. PMID 32010836 DOI: 10.1021/acsomega.9b03693  0.78
2020 Reddy CN, Bharate SB, Vishwakarma RA, Bharate SS. Chemical analysis of saffron by HPLC based crocetin estimation. Journal of Pharmaceutical and Biomedical Analysis. 181: 113094. PMID 31927167 DOI: 10.1016/J.Jpba.2020.113094  0.488
2020 Bharate SB. Meet Our Editorial Board Member Current Medicinal Chemistry. 27: 4153-4154. DOI: 10.2174/092986732725200619124856  0.182
2019 Abdullaha M, Ali M, Kour D, Kumar A, Bharate SB. Discovery of benzo[cd]indol-2-one and benzylidene-thiazolidine-2,4-dione as new classes of NLRP3 inflammasome inhibitors via ER-β structure based virtual screening. Bioorganic Chemistry. 95: 103500. PMID 31869665 DOI: 10.1016/j.bioorg.2019.103500  0.357
2019 Kumar V, Mintoo MJ, Mondhe DM, Bharate SB, Vishwakarma RA, Bharate SS. Binary and ternary solid dispersions of an anticancer preclinical lead, IIIM-290: In vitro and in vivo studies. International Journal of Pharmaceutics. 118683. PMID 31513869 DOI: 10.1016/J.Ijpharm.2019.118683  0.525
2019 Bharate SB, Chao CK, Thompson CM. Comparison of the reactivation rates of acetylcholinesterase modified by structurally different organophosphates using novel pyridinium oximes. Environmental Toxicology and Pharmacology. 71: 103218. PMID 31302432 DOI: 10.1016/J.Etap.2019.103218  0.703
2019 Derf A, Sharma A, Bharate SB, Chaudhuri B. Corrigendum to "Aegeline, a natural product from the plant Aegle marmelos, mimics the yeast SNARE protein Sec22p in suppressing α-synuclein and Bax toxicity in yeast" [Bioorg. Med. Chem. Lett. 29 (2019) 454-460]. Bioorganic & Medicinal Chemistry Letters. PMID 31281017 DOI: 10.1016/j.bmcl.2019.06.053  0.54
2019 Sonawane VR, Siddique MUM, Gatchie L, Williams IS, Bharate SB, Jayaprakash V, Sinha BN, Chaudhuri B. Corrigendum to "CYP enzymes, expressed within live human suspension cells, are superior to widely-used microsomal enzymes in identifying potent CYP1A1/CYP1B1 inhibitors: Identification of quinazolinones as CYP1A1/CYP1B1 inhibitors that efficiently reverse B[a]P toxicity and cisplatin resistance" [Eur. J. Pharm. Sci. 131 (2019) 177-194]. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. 104960. PMID 31230886 DOI: 10.1016/j.ejps.2019.104960  0.346
2019 Nuthakki VK, Mudududdla R, Sharma A, Kumar A, Bharate SB. Synthesis and biological evaluation of indoloquinoline alkaloid cryptolepine and its bromo-derivative as dual cholinesterase inhibitors. Bioorganic Chemistry. 90: 103062. PMID 31220673 DOI: 10.1016/j.bioorg.2019.103062  0.826
2019 Syed SH, Dar MI, Nargotra A, Mahajan P, Tiwari H, Jan S, Sandey J, Jain SK, Bharate S. Rottlerin is a pan phosphodiesterase inhibitor and can induce neurodifferentiation in IMR-32 human neuroblastoma cells. European Journal of Pharmacology. 172448. PMID 31202802 DOI: 10.1016/j.ejphar.2019.172448  0.826
2019 Nuthakki VK, Sharma A, Kumar A, Bharate SB. Identification of embelin, a 3-undecyl-1,4-benzoquinone from Embelia ribes as a multitargeted anti-Alzheimer agent. Drug Development Research. PMID 31050027 DOI: 10.1002/ddr.21544  0.817
2019 Bharate SB, Kumar V, Bharate SS, Singh B, Singh G, Singh A, Gupta M, Singh D, Kumar A, Singh S, Vishwakarma RA. Discovery and preclinical development of IIIM-160, a Bergenia ciliata-based anti-inflammatory and anti-arthritic botanical drug candidate. Journal of Integrative Medicine. PMID 30898582 DOI: 10.1016/J.Joim.2019.03.001  0.493
2019 Abdullaha M, Mohammed S, Ali M, Kumar A, Vishwakarma RA, Bharate SB. Discovery of Quinazolin-4(3H)-ones as NLRP3 Inflammasome Inhibitors: Computational Design, Metal-free Synthesis and In-vitro Biological Evaluation. The Journal of Organic Chemistry. PMID 30896160 DOI: 10.1021/Acs.Joc.9B00138  0.79
2019 Abdullaha M, Mohammed S, Ali M, Kumar A, Vishwakarma RA, Bharate SB. Discovery of Quinazolin-4(3H)-ones as NLRP3 Inflammasome Inhibitors: Computational Design, Metal-free Synthesis and In-vitro Biological Evaluation. The Journal of Organic Chemistry. PMID 30896160 DOI: 10.1021/Acs.Joc.9B00138  0.79
2019 Wani A, Gupta M, Ahmad M, Shah AM, Ahsan AU, Hassan Qazi PH, Malik F, Singh G, Sharma PR, Kaddoumi A, Bharate SB, Vishwakarma RA, Kumar A. Alborixin clears amyloid-β by inducing autophagy through PTEN-mediated inhibition of the AKT pathway. Autophagy. PMID 30894052 DOI: 10.1080/15548627.2019.1596476  0.536
2019 Wani A, Gupta M, Ahmad M, Shah AM, Ahsan AU, Hassan Qazi PH, Malik F, Singh G, Sharma PR, Kaddoumi A, Bharate SB, Vishwakarma RA, Kumar A. Alborixin clears amyloid-β by inducing autophagy through PTEN-mediated inhibition of the AKT pathway. Autophagy. PMID 30894052 DOI: 10.1080/15548627.2019.1596476  0.536
2019 Sonawane VR, Siddique MUM, Gatchie L, Williams IS, Bharate SB, Jayaprakash V, Sinha BN, Chaudhuri B. CYP enzymes, expressed within live human suspension cells, are superior to widely-used microsomal enzymes in identifying potent CYP1A1/CYP1B1 inhibitors: Identification of quinazolinones as CYP1A1/CYP1B1 inhibitors that efficiently reverse B[a]P toxicity and cisplatin resistance. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. PMID 30776468 DOI: 10.1016/j.ejps.2019.02.016  0.407
2019 Sonawane VR, Siddique MUM, Gatchie L, Williams IS, Bharate SB, Jayaprakash V, Sinha BN, Chaudhuri B. CYP enzymes, expressed within live human suspension cells, are superior to widely-used microsomal enzymes in identifying potent CYP1A1/CYP1B1 inhibitors: Identification of quinazolinones as CYP1A1/CYP1B1 inhibitors that efficiently reverse B[a]P toxicity and cisplatin resistance. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. PMID 30776468 DOI: 10.1016/j.ejps.2019.02.016  0.407
2019 Rajani P, Aiswarya H, Vasanthakumari MM, Jain SK, Bharate SB, Rajasekaran C, Ravikanth G, Uma Shaanker R. Inhibition of the collar rot fungus, Sclerotium rolfsii Sacc. by an endophytic fungus Alternaria sp.: implications for biocontrol Plant Physiology Reports. 24: 521-532. DOI: 10.1007/s40502-019-00484-6  0.739
2018 Bharate SS, Kumar V, Singh G, Singh A, Gupta M, Singh D, Kumar A, Vishwakarma RA, Bharate SB. Preclinical Development of -Based Botanical Lead IIIM-141 for Alzheimer's Disease: Chemical Standardization, Efficacy, Formulation Development, Pharmacokinetics, and Safety Pharmacology. Acs Omega. 3: 9572-9585. PMID 31459089 DOI: 10.1021/acsomega.8b00841  0.52
2018 Derf A, Mudududdla R, Akintade D, Williams IS, Abdullaha M, Chaudhuri B, Bharate SB. Nonantioxidant Tetramethoxystilbene Abrogates α-Synuclein-Induced Yeast Cell Death but Not That Triggered by the Bax or βA4 Peptide. Acs Omega. 3: 9513-9532. PMID 31459084 DOI: 10.1021/acsomega.8b01154  0.744
2018 Williams IS, Gatchie L, Bharate SB, Chaudhuri B. Biotransformation, Using Recombinant CYP450-Expressing Baker's Yeast Cells, Identifies a Novel CYP2D6.10 Variant Which Is a Superior Metabolizer of Codeine to Morphine Than the Wild-Type Enzyme. Acs Omega. 3: 8903-8912. PMID 31459022 DOI: 10.1021/acsomega.8b00809  0.322
2018 Sharma R, Williams IS, Gatchie L, Sonawane VR, Chaudhuri B, Bharate SB. Khellinoflavanone, a Semisynthetic Derivative of Khellin, Overcomes Benzo[]pyrene Toxicity in Human Normal and Cancer Cells That Express CYP1A1. Acs Omega. 3: 8553-8566. PMID 31458985 DOI: 10.1021/acsomega.8b01088  0.631
2018 Derf A, Verekar SA, Jain SK, Deshmukh SK, Bharate SB, Chaudhuri B. Radicicol rescues yeast cell death triggered by expression of human α-synuclein and its A53T mutant, but not by human βA4 peptide and proapoptotic protein bax. Bioorganic Chemistry. 85: 152-158. PMID 30612081 DOI: 10.1016/j.bioorg.2018.12.033  0.791
2018 Derf A, Verekar SA, Jain SK, Deshmukh SK, Bharate SB, Chaudhuri B. Radicicol rescues yeast cell death triggered by expression of human α-synuclein and its A53T mutant, but not by human βA4 peptide and proapoptotic protein bax. Bioorganic Chemistry. 85: 152-158. PMID 30612081 DOI: 10.1016/j.bioorg.2018.12.033  0.791
2018 Kumar V, Bhurta D, Sharma A, Kumar P, Bharate SB, Vishwakarma RA, Bharate SS. Impurity profiling of anticancer preclinical candidate, IIIM-290. Journal of Pharmaceutical and Biomedical Analysis. 166: 1-5. PMID 30590350 DOI: 10.1016/J.Jpba.2018.12.027  0.787
2018 Kumar V, Bhurta D, Sharma A, Kumar P, Bharate SB, Vishwakarma RA, Bharate SS. Impurity profiling of anticancer preclinical candidate, IIIM-290. Journal of Pharmaceutical and Biomedical Analysis. 166: 1-5. PMID 30590350 DOI: 10.1016/J.Jpba.2018.12.027  0.787
2018 Derf A, Sharma A, Bharate SB, Chaudhuri B. Aegeline, a natural product from the plant Aegle marmelos, mimics the yeast SNARE protein Sec22p in suppressing α-synuclein and Bax toxicity in yeast. Bioorganic & Medicinal Chemistry Letters. PMID 30579794 DOI: 10.1016/j.bmcl.2018.12.028  0.596
2018 Derf A, Sharma A, Bharate SB, Chaudhuri B. Aegeline, a natural product from the plant Aegle marmelos, mimics the yeast SNARE protein Sec22p in suppressing α-synuclein and Bax toxicity in yeast. Bioorganic & Medicinal Chemistry Letters. PMID 30579794 DOI: 10.1016/j.bmcl.2018.12.028  0.596
2018 Derf A, Mudududdla R, Bharate SB, Chaudhuri B. Inhibitors of Aβ42-induced endoplasmic reticular unfolded protein response (UPR), in yeast, also rescue yeast cells from Aβ42-mediated apoptosis. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. PMID 30502452 DOI: 10.1016/j.ejps.2018.11.029  0.752
2018 Derf A, Mudududdla R, Bharate SB, Chaudhuri B. Inhibitors of Aβ42-induced endoplasmic reticular unfolded protein response (UPR), in yeast, also rescue yeast cells from Aβ42-mediated apoptosis. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. PMID 30502452 DOI: 10.1016/j.ejps.2018.11.029  0.752
2018 Sharma R, Williams IS, Gatchie L, Sonawane VR, Chaudhuri B, Bharate SB. Furanoflavones pongapin and lanceolatin B blocks the cell cycle and induce senescence in CYP1A1-overexpressing breast cancer cells. Bioorganic & Medicinal Chemistry. PMID 30448188 DOI: 10.1016/j.bmc.2018.11.013  0.581
2018 Sharma R, Williams IS, Gatchie L, Sonawane VR, Chaudhuri B, Bharate SB. Furanoflavones pongapin and lanceolatin B blocks the cell cycle and induce senescence in CYP1A1-overexpressing breast cancer cells. Bioorganic & Medicinal Chemistry. PMID 30448188 DOI: 10.1016/j.bmc.2018.11.013  0.581
2018 Bharate SB, Mudududdla R, Mohanakrishnan D, Bharate SS, Vishwakarma RA, Sahal D. Orally Effective Aminoalkyl 10H-Indolo-[3,2-b]quinoline-11-carboxamide Kills the Malaria Parasite by Inhibiting Host Hemoglobin Uptake. Chemmedchem. PMID 30358112 DOI: 10.1002/Cmdc.201800579  0.789
2018 Bharate SB, Mudududdla R, Mohanakrishnan D, Bharate SS, Vishwakarma RA, Sahal D. Orally Effective Aminoalkyl 10H-Indolo-[3,2-b]quinoline-11-carboxamide Kills the Malaria Parasite by Inhibiting Host Hemoglobin Uptake. Chemmedchem. PMID 30358112 DOI: 10.1002/Cmdc.201800579  0.789
2018 Joshi P, Sonawane VR, Williams IS, McCann GJP, Gatchie L, Sharma R, Satti N, Chaudhuri B, Bharate SB. Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy screening of a natural product repository. Medchemcomm. 9: 371-382. PMID 30108931 DOI: 10.1039/c7md00388a  0.725
2018 Joshi P, Sonawane VR, Williams IS, McCann GJP, Gatchie L, Sharma R, Satti N, Chaudhuri B, Bharate SB. Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy screening of a natural product repository. Medchemcomm. 9: 371-382. PMID 30108931 DOI: 10.1039/c7md00388a  0.725
2018 Kumar V, Bharate SB, Vishwakarma RA, Bharate SS. Selection of a Water-Soluble Salt Form of a Preclinical Candidate, IIIM-290: Multiwell-Plate Salt Screening and Characterization. Acs Omega. 3: 8365-8377. PMID 30087943 DOI: 10.1021/acsomega.8b00801  0.553
2018 Kumar V, Bharate SB, Vishwakarma RA, Bharate SS. Selection of a Water-Soluble Salt Form of a Preclinical Candidate, IIIM-290: Multiwell-Plate Salt Screening and Characterization. Acs Omega. 3: 8365-8377. PMID 30087943 DOI: 10.1021/acsomega.8b00801  0.553
2018 Bharate SB, Kumar V, Jain SK, Mintoo MJ, Guru SK, Nuthakki VK, Sharma M, Bharate SS, Gandhi SG, Mondhe DM, Bhushan S, Vishwakarma RA. Discovery and Preclinical Development of IIIM-290, an Orally Active Potent Cyclin-dependent Kinase Inhibitor. Journal of Medicinal Chemistry. PMID 29370702 DOI: 10.1021/Acs.Jmedchem.7B01765  0.819
2018 Bharate SB, Kumar V, Jain SK, Mintoo MJ, Guru SK, Nuthakki VK, Sharma M, Bharate SS, Gandhi SG, Mondhe DM, Bhushan S, Vishwakarma RA. Discovery and Preclinical Development of IIIM-290, an Orally Active Potent Cyclin-dependent Kinase Inhibitor. Journal of Medicinal Chemistry. PMID 29370702 DOI: 10.1021/Acs.Jmedchem.7B01765  0.819
2017 Sharma R, Gatchie L, Williams IS, Jain SK, Vishwakarma RA, Chaudhuri B, Bharate SB. Glycyrrhiza glabra extract and quercetin reverses cisplatin resistance in triple-negative MDA-MB-468 breast cancer cells via inhibition of cytochrome P450 1B1 enzyme. Bioorganic & Medicinal Chemistry Letters. PMID 29150398 DOI: 10.1016/J.Bmcl.2017.11.013  0.812
2017 Sharma R, Gatchie L, Williams IS, Jain SK, Vishwakarma RA, Chaudhuri B, Bharate SB. Glycyrrhiza glabra extract and quercetin reverses cisplatin resistance in triple-negative MDA-MB-468 breast cancer cells via inhibition of cytochrome P450 1B1 enzyme. Bioorganic & Medicinal Chemistry Letters. PMID 29150398 DOI: 10.1016/J.Bmcl.2017.11.013  0.812
2017 Horley NJ, Beresford KJM, Kaduskar S, Joshi P, McCann GJP, Ruparelia KC, Williams IS, Gatchie L, Sonawane VR, Bharate SB, Chaudhuri B. (E)-3-(3,4,5-Trimethoxyphenyl)-1-(pyridin-4-yl)prop-2-en-1-one, a heterocyclic chalcone is a potent and selective CYP1A1 inhibitor and cancer chemopreventive agent. Bioorganic & Medicinal Chemistry Letters. PMID 29138024 DOI: 10.1016/j.bmcl.2017.11.009  0.633
2017 Horley NJ, Beresford KJM, Kaduskar S, Joshi P, McCann GJP, Ruparelia KC, Williams IS, Gatchie L, Sonawane VR, Bharate SB, Chaudhuri B. (E)-3-(3,4,5-Trimethoxyphenyl)-1-(pyridin-4-yl)prop-2-en-1-one, a heterocyclic chalcone is a potent and selective CYP1A1 inhibitor and cancer chemopreventive agent. Bioorganic & Medicinal Chemistry Letters. PMID 29138024 DOI: 10.1016/j.bmcl.2017.11.009  0.633
2017 Singh S, Kalia NP, Joshi P, Kumar A, Sharma PR, Kumar A, Bharate SB, Khan IA. Boeravinone B, A Novel Dual Inhibitor of NorA Bacterial Efflux Pump of Staphylococcus aureus and Human P-Glycoprotein, Reduces the Biofilm Formation and Intracellular Invasion of Bacteria. Frontiers in Microbiology. 8: 1868. PMID 29046665 DOI: 10.3389/fmicb.2017.01868  0.603
2017 Singh S, Kalia NP, Joshi P, Kumar A, Sharma PR, Kumar A, Bharate SB, Khan IA. Boeravinone B, A Novel Dual Inhibitor of NorA Bacterial Efflux Pump of Staphylococcus aureus and Human P-Glycoprotein, Reduces the Biofilm Formation and Intracellular Invasion of Bacteria. Frontiers in Microbiology. 8: 1868. PMID 29046665 DOI: 10.3389/fmicb.2017.01868  0.603
2017 Sharma R, Abdullaha M, Bharate SB. Oxidant-Controlled C-sp2/sp3 - H Cross-dehydrogenative Coupling of N-Heterocycles with Benzylamines. The Journal of Organic Chemistry. PMID 28820259 DOI: 10.1021/acs.joc.7b00856  0.454
2017 Sharma R, Abdullaha M, Bharate SB. Oxidant-Controlled C-sp2/sp3 - H Cross-dehydrogenative Coupling of N-Heterocycles with Benzylamines. The Journal of Organic Chemistry. PMID 28820259 DOI: 10.1021/acs.joc.7b00856  0.454
2017 Williams IS, Chib S, Nuthakki V, Gatchie L, Joshi P, Narkhede N, Vishwakarma RA, Bharate SB, Saran S, Chaudhuri B. Biotransformation of chrysin to baicalein: Selective C6-hydroxylation of 5,7-dihydroxyflavone using whole yeast cells stably expressing human CYP1A1 enzyme. Journal of Agricultural and Food Chemistry. PMID 28782952 DOI: 10.1021/Acs.Jafc.7B02690  0.819
2017 Williams IS, Chib S, Nuthakki V, Gatchie L, Joshi P, Narkhede N, Vishwakarma RA, Bharate SB, Saran S, Chaudhuri B. Biotransformation of chrysin to baicalein: Selective C6-hydroxylation of 5,7-dihydroxyflavone using whole yeast cells stably expressing human CYP1A1 enzyme. Journal of Agricultural and Food Chemistry. PMID 28782952 DOI: 10.1021/Acs.Jafc.7B02690  0.819
2017 Sharma S, Guru SK, Manda S, Kumar A, Mintoo MJ, Prasad VD, Sharma PR, Mondhe DM, Bharate SB, Bhushan S. A marine sponge alkaloid derivative 4-chloro fascaplysin inhibits tumor growth and VEGF mediated angiogenesis by disrupting PI3K/Akt/mTOR signaling cascade. Chemico-Biological Interactions. 275: 47-60. PMID 28756150 DOI: 10.1016/j.cbi.2017.07.017  0.797
2017 Sharma S, Guru SK, Manda S, Kumar A, Mintoo MJ, Prasad VD, Sharma PR, Mondhe DM, Bharate SB, Bhushan S. A marine sponge alkaloid derivative 4-chloro fascaplysin inhibits tumor growth and VEGF mediated angiogenesis by disrupting PI3K/Akt/mTOR signaling cascade. Chemico-Biological Interactions. 275: 47-60. PMID 28756150 DOI: 10.1016/j.cbi.2017.07.017  0.797
2017 Williams IS, Joshi P, Gatchie L, Sharma M, Satti NK, Vishwakarma RA, Chaudhuri B, Bharate SB. Synthesis and biological evaluation of pyrrole-based chalcones as CYP1 enzyme inhibitors, for possible prevention of cancer and overcoming cisplatin resistance. Bioorganic & Medicinal Chemistry Letters. PMID 28711350 DOI: 10.1016/J.Bmcl.2017.07.010  0.786
2017 Williams IS, Joshi P, Gatchie L, Sharma M, Satti NK, Vishwakarma RA, Chaudhuri B, Bharate SB. Synthesis and biological evaluation of pyrrole-based chalcones as CYP1 enzyme inhibitors, for possible prevention of cancer and overcoming cisplatin resistance. Bioorganic & Medicinal Chemistry Letters. PMID 28711350 DOI: 10.1016/J.Bmcl.2017.07.010  0.786
2017 Joshi P, Vishwakarma RA, Bharate SB. Natural alkaloids as P-gp inhibitors for multidrug resistance reversal in cancer. European Journal of Medicinal Chemistry. 138: 273-292. PMID 28675836 DOI: 10.1016/J.Ejmech.2017.06.047  0.684
2017 Joshi P, Vishwakarma RA, Bharate SB. Natural alkaloids as P-gp inhibitors for multidrug resistance reversal in cancer. European Journal of Medicinal Chemistry. 138: 273-292. PMID 28675836 DOI: 10.1016/J.Ejmech.2017.06.047  0.684
2017 Joshi P, McCann GJP, Sonawane V, Vishwakarma RA, Chaudhuri B, Bharate SB. Identification of Potent and Selective CYP1A1 Inhibitors via Combined Ligand and Structure Based Virtual Screening and their In-vitro Validation in Sacchrosomes and Live human cells. Journal of Chemical Information and Modeling. PMID 28489395 DOI: 10.1021/Acs.Jcim.7B00095  0.716
2017 Joshi P, McCann GJP, Sonawane V, Vishwakarma RA, Chaudhuri B, Bharate SB. Identification of Potent and Selective CYP1A1 Inhibitors via Combined Ligand and Structure Based Virtual Screening and their In-vitro Validation in Sacchrosomes and Live human cells. Journal of Chemical Information and Modeling. PMID 28489395 DOI: 10.1021/Acs.Jcim.7B00095  0.716
2017 Batarseh YS, Bharate SS, Kumar V, Kumar A, Vishwakarma RA, Bharate SB, Kaddoumi A. Crocus sativus extract tighten the blood-brain barrier, reduces amyloid-β load and related toxicity in 5XFAD mice. Acs Chemical Neuroscience. PMID 28471166 DOI: 10.1021/Acschemneuro.7B00101  0.496
2017 Batarseh YS, Bharate SS, Kumar V, Kumar A, Vishwakarma RA, Bharate SB, Kaddoumi A. Crocus sativus extract tighten the blood-brain barrier, reduces amyloid-β load and related toxicity in 5XFAD mice. Acs Chemical Neuroscience. PMID 28471166 DOI: 10.1021/Acschemneuro.7B00101  0.496
2017 Mohd Siddique MU, McCann GJ, Sonawane VR, Horley N, Gatchie L, Joshi P, Bharate SB, Jayaprakash V, Sinha BN, Chaudhuri B. Quinazoline derivatives as selective CYP1B1 inhibitors. European Journal of Medicinal Chemistry. 130: 320-327. PMID 28259840 DOI: 10.1016/j.ejmech.2017.02.032  0.659
2017 Mohd Siddique MU, McCann GJ, Sonawane VR, Horley N, Gatchie L, Joshi P, Bharate SB, Jayaprakash V, Sinha BN, Chaudhuri B. Quinazoline derivatives as selective CYP1B1 inhibitors. European Journal of Medicinal Chemistry. 130: 320-327. PMID 28259840 DOI: 10.1016/j.ejmech.2017.02.032  0.659
2017 Horley NJ, Beresford KJ, Chawla T, McCann GJ, Ruparelia KC, Gatchie L, Sonawane VR, Williams IS, Tan HL, Joshi P, Bharate SS, Kumar V, Bharate SB, Chaudhuri B. Discovery and characterization of novel CYP1B1 inhibitors based on heterocyclic chalcones: Overcoming cisplatin resistance in CYP1B1-overexpressing lines. European Journal of Medicinal Chemistry. 129: 159-174. PMID 28222316 DOI: 10.1016/j.ejmech.2017.02.016  0.656
2017 Horley NJ, Beresford KJ, Chawla T, McCann GJ, Ruparelia KC, Gatchie L, Sonawane VR, Williams IS, Tan HL, Joshi P, Bharate SS, Kumar V, Bharate SB, Chaudhuri B. Discovery and characterization of novel CYP1B1 inhibitors based on heterocyclic chalcones: Overcoming cisplatin resistance in CYP1B1-overexpressing lines. European Journal of Medicinal Chemistry. 129: 159-174. PMID 28222316 DOI: 10.1016/j.ejmech.2017.02.016  0.656
2017 Kumar V, Gupta M, Gandhi SG, Bharate SS, Kumar A, Vishwakarma RA, Bharate SB. Anti-inflammatory chromone alkaloids and glycoside from Dysoxylum binectariferum Tetrahedron Letters. 58: 3974-3978. DOI: 10.1016/J.Tetlet.2017.09.005  0.56
2017 Sharma R, Abdullaha M, Bharate SB. Metal-Free Ionic-Liquid-Mediated Synthesis of Benzimidazoles and Quinazolin-4(3H )-ones from Benzylamines Asian Journal of Organic Chemistry. 6: 1370-1374. DOI: 10.1002/AJOC.201700214  0.25
2016 Joshi P, Gupta M, Vishwakarma RA, Kumar A, Bharate SB. (Z)-2-(3-Chlorobenzylidene)-3,4-dihydro-N-(2-methoxyethyl)-3-oxo-2H-benzo[b][1,4]oxazine-6-carboxamide as GSK-3β inhibitor: Identification by virtual screening, and its validation in enzyme and cell-based assay. Chemical Biology & Drug Design. PMID 27896926 DOI: 10.1111/Cbdd.12913  0.688
2016 Joshi P, Gupta M, Vishwakarma RA, Kumar A, Bharate SB. (Z)-2-(3-Chlorobenzylidene)-3,4-dihydro-N-(2-methoxyethyl)-3-oxo-2H-benzo[b][1,4]oxazine-6-carboxamide as GSK-3β inhibitor: Identification by virtual screening, and its validation in enzyme and cell-based assay. Chemical Biology & Drug Design. PMID 27896926 DOI: 10.1111/Cbdd.12913  0.688
2016 Mohd Siddique MU, McCann GJ, Sonawane V, Horley N, Williams IS, Joshi P, Bharate SB, Jayaprakash V, Sinha BN, Chaudhuri B. Biphenyl urea derivatives as selective CYP1B1 inhibitors. Organic & Biomolecular Chemistry. 14: 8931-8936. PMID 27714268 DOI: 10.1039/c6ob01506a  0.657
2016 Mohd Siddique MU, McCann GJ, Sonawane V, Horley N, Williams IS, Joshi P, Bharate SB, Jayaprakash V, Sinha BN, Chaudhuri B. Biphenyl urea derivatives as selective CYP1B1 inhibitors. Organic & Biomolecular Chemistry. 14: 8931-8936. PMID 27714268 DOI: 10.1039/c6ob01506a  0.657
2016 Padala AK, Wani A, Vishwakarma RA, Kumar A, Bharate SB. Functional induction of P-glycoprotein efflux pump by phenyl benzenesulfonamides: Synthesis and biological evaluation of T0901317 analogs. European Journal of Medicinal Chemistry. 122: 744-755. PMID 27497733 DOI: 10.1016/J.Ejmech.2016.07.005  0.561
2016 Padala AK, Wani A, Vishwakarma RA, Kumar A, Bharate SB. Functional induction of P-glycoprotein efflux pump by phenyl benzenesulfonamides: Synthesis and biological evaluation of T0901317 analogs. European Journal of Medicinal Chemistry. 122: 744-755. PMID 27497733 DOI: 10.1016/J.Ejmech.2016.07.005  0.561
2016 Yadav RR, Guru SK, Joshi P, Mahajan G, Mintoo MJ, Kumar V, Bharate SS, Mondhe DM, Vishwakarma RA, Bhushan S, Bharate SB. 6-Aryl substituted 4-(4-cyanomethyl) phenylamino quinazolines as a new class of isoform-selective PI3K-alpha inhibitors. European Journal of Medicinal Chemistry. 122: 731-743. PMID 27479483 DOI: 10.1016/J.Ejmech.2016.07.006  0.813
2016 Yadav RR, Guru SK, Joshi P, Mahajan G, Mintoo MJ, Kumar V, Bharate SS, Mondhe DM, Vishwakarma RA, Bhushan S, Bharate SB. 6-Aryl substituted 4-(4-cyanomethyl) phenylamino quinazolines as a new class of isoform-selective PI3K-alpha inhibitors. European Journal of Medicinal Chemistry. 122: 731-743. PMID 27479483 DOI: 10.1016/J.Ejmech.2016.07.006  0.813
2016 Mahajan P, Gnana Oli R, Jachak SM, Bharate SB, Chaudhuri B. Antioxidant and antiproliferative activity of indigocarpan, a pterocarpan from Indigofera aspalathoides. The Journal of Pharmacy and Pharmacology. PMID 27464528 DOI: 10.1111/jphp.12609  0.28
2016 Mahajan P, Gnana Oli R, Jachak SM, Bharate SB, Chaudhuri B. Antioxidant and antiproliferative activity of indigocarpan, a pterocarpan from Indigofera aspalathoides. The Journal of Pharmacy and Pharmacology. PMID 27464528 DOI: 10.1111/jphp.12609  0.28
2016 Kumar A, Singh B, Mahajan G, Sharma PR, Bharate SB, Mintoo MJ, Mondhe DM. A novel colchicine-based microtubule inhibitor exhibits potent antitumor activity by inducing mitochondrial mediated apoptosis in MIA PaCa-2 pancreatic cancer cells. Tumour Biology : the Journal of the International Society For Oncodevelopmental Biology and Medicine. PMID 27449046 DOI: 10.1007/S13277-016-5160-5  0.522
2016 Kumar A, Singh B, Mahajan G, Sharma PR, Bharate SB, Mintoo MJ, Mondhe DM. A novel colchicine-based microtubule inhibitor exhibits potent antitumor activity by inducing mitochondrial mediated apoptosis in MIA PaCa-2 pancreatic cancer cells. Tumour Biology : the Journal of the International Society For Oncodevelopmental Biology and Medicine. PMID 27449046 DOI: 10.1007/S13277-016-5160-5  0.522
2016 Kumar V, Guru SK, Jain SK, Joshi P, Gandhi SG, Bharate SB, Bhushan S, Bharate SS, Vishwakarma RA. A chromatography-free isolation of rohitukine from leaves of Dysoxylum binectariferum: Evaluation for in vitro cytotoxicity, Cdk inhibition and physicochemical properties. Bioorganic & Medicinal Chemistry Letters. PMID 27363938 DOI: 10.1016/J.Bmcl.2016.06.046  0.82
2016 Kumar V, Guru SK, Jain SK, Joshi P, Gandhi SG, Bharate SB, Bhushan S, Bharate SS, Vishwakarma RA. A chromatography-free isolation of rohitukine from leaves of Dysoxylum binectariferum: Evaluation for in vitro cytotoxicity, Cdk inhibition and physicochemical properties. Bioorganic & Medicinal Chemistry Letters. PMID 27363938 DOI: 10.1016/J.Bmcl.2016.06.046  0.82
2016 Bharate SB, Singh B, Kachler S, Oliveira A, Kumar V, Bharate SS, Vishwakarma RA, Klotz KN, Gutiérrez-de-Terán H. Discovery of 7-(prolinol-N-yl)-2-phenylamino-thiazolo[5,4-d]pyrimidines as novel non-nucleoside partial agonists for the A2A adenosine receptor: Prediction from molecular modeling. Journal of Medicinal Chemistry. PMID 27227326 DOI: 10.1021/Acs.Jmedchem.6B00552  0.605
2016 Bharate SB, Singh B, Kachler S, Oliveira A, Kumar V, Bharate SS, Vishwakarma RA, Klotz KN, Gutiérrez-de-Terán H. Discovery of 7-(prolinol-N-yl)-2-phenylamino-thiazolo[5,4-d]pyrimidines as novel non-nucleoside partial agonists for the A2A adenosine receptor: Prediction from molecular modeling. Journal of Medicinal Chemistry. PMID 27227326 DOI: 10.1021/Acs.Jmedchem.6B00552  0.605
2016 Hussain A, Qazi AK, Mupparapu N, Guru SK, Kumar A, Sharma PR, Singh SK, Singh P, Dar MJ, Bharate SB, Zargar MA, Ahmed QN, Bhushan S, Vishwakarma RA, Hamid A. Modulation of glycolysis and lipogenesis by novel PI3K selective molecule represses tumor angiogenesis and decreases colorectal cancer growth. Cancer Letters. PMID 26921131 DOI: 10.1016/J.Canlet.2016.02.030  0.517
2016 Hussain A, Qazi AK, Mupparapu N, Guru SK, Kumar A, Sharma PR, Singh SK, Singh P, Dar MJ, Bharate SB, Zargar MA, Ahmed QN, Bhushan S, Vishwakarma RA, Hamid A. Modulation of glycolysis and lipogenesis by novel PI3K selective molecule represses tumor angiogenesis and decreases colorectal cancer growth. Cancer Letters. PMID 26921131 DOI: 10.1016/J.Canlet.2016.02.030  0.517
2016 Kumar A, Singh B, Sharma PR, Bharate SB, Saxena AK, Mondhe DM. A novel microtubule depolymerizing colchicine analogue triggers apoptosis and autophagy in HCT-116 colon cancer cells. Cell Biochemistry and Function. 34: 69-81. PMID 26919061 DOI: 10.1002/Cbf.3166  0.547
2016 Kumar A, Singh B, Sharma PR, Bharate SB, Saxena AK, Mondhe DM. A novel microtubule depolymerizing colchicine analogue triggers apoptosis and autophagy in HCT-116 colon cancer cells. Cell Biochemistry and Function. 34: 69-81. PMID 26919061 DOI: 10.1002/Cbf.3166  0.547
2016 Hussain A, Qazi AK, Mupparapu N, Kumar A, Mintoo MJ, Mahajan G, Sharma PR, Singh SK, Bharate SB, Zargar MA, Ahmed QN, Mondhe DM, Vishwakarma RA, Hamid A. A novel PI3K axis selective molecule exhibits potent tumor inhibition in colorectal carcinogenesis. Molecular Carcinogenesis. PMID 26764221 DOI: 10.1002/Mc.22457  0.567
2016 Hussain A, Qazi AK, Mupparapu N, Kumar A, Mintoo MJ, Mahajan G, Sharma PR, Singh SK, Bharate SB, Zargar MA, Ahmed QN, Mondhe DM, Vishwakarma RA, Hamid A. A novel PI3K axis selective molecule exhibits potent tumor inhibition in colorectal carcinogenesis. Molecular Carcinogenesis. PMID 26764221 DOI: 10.1002/Mc.22457  0.567
2016 Manda S, Wani A, Bharate SS, Vishwakarma RA, Kumar A, Bharate SB. Design, synthesis and P-gp induction activity of aryl phosphonate esters: identification of tetraethyl-2-phenylethene-1,1-diyldiphosphonate as an orally bioavailable P-gp inducer Medchemcomm. 7: 1910-1915. DOI: 10.1039/C6Md00300A  0.551
2016 Sharma R, Vishwakarma RA, Bharate SB. Bimetallic Cu–Mn‐Catalyzed Synthesis of 2‐Arylquinazolin‐4(3H)‐ones: Aqueous Ammonia as Source of a Ring Nitrogen Atom European Journal of Organic Chemistry. 2016: 5227-5233. DOI: 10.1002/Ejoc.201601024  0.505
2016 Sharma R, Vishwakarma RA, Bharate SB. Ligand-Free Copper-Manganese Spinel Oxide-Catalyzed Tandem One-Pot C-H Amidation andN-Arylation of Benzylamines: A Facile Access to 2-Arylquinazolin-4(3H)-ones Advanced Synthesis & Catalysis. 358: 3027-3033. DOI: 10.1002/Adsc.201600549  0.496
2015 Sharma R, Patel N, Vishwakarma RA, Bharatam PV, Bharate SB. Metal-free oxidative cyclization of acetophenones with diamines: a facile access to phenylpyridines. Chemical Communications (Cambridge, England). PMID 26593387 DOI: 10.1039/C5Cc08498A  0.584
2015 Sharma R, Patel N, Vishwakarma RA, Bharatam PV, Bharate SB. Metal-free oxidative cyclization of acetophenones with diamines: a facile access to phenylpyridines. Chemical Communications (Cambridge, England). PMID 26593387 DOI: 10.1039/C5Cc08498A  0.584
2015 Manda S, Sharma S, Wani A, Joshi P, Kumar V, Guru SK, Bharate SS, Bhushan S, Vishwakarma RA, Kumar A, Bharate SB. Discovery of a marine-derived bis-indole alkaloid fascaplysin, as a new class of potent P-glycoprotein inducer and establishment of its structure-activity relationship. European Journal of Medicinal Chemistry. 107: 1-11. PMID 26560048 DOI: 10.1016/J.Ejmech.2015.10.049  0.808
2015 Manda S, Sharma S, Wani A, Joshi P, Kumar V, Guru SK, Bharate SS, Bhushan S, Vishwakarma RA, Kumar A, Bharate SB. Discovery of a marine-derived bis-indole alkaloid fascaplysin, as a new class of potent P-glycoprotein inducer and establishment of its structure-activity relationship. European Journal of Medicinal Chemistry. 107: 1-11. PMID 26560048 DOI: 10.1016/J.Ejmech.2015.10.049  0.808
2015 Sharma R, Vishwakarma RA, Bharate SB. An efficient transformation of furano-hydroxychalcones to furanoflavones via base mediated intramolecular tandem O-arylation and C-O bond cleavage: a new approach for the synthesis of furanoflavones. Organic & Biomolecular Chemistry. PMID 26426474 DOI: 10.1039/C5Ob01802A  0.621
2015 Sharma R, Vishwakarma RA, Bharate SB. An efficient transformation of furano-hydroxychalcones to furanoflavones via base mediated intramolecular tandem O-arylation and C-O bond cleavage: a new approach for the synthesis of furanoflavones. Organic & Biomolecular Chemistry. PMID 26426474 DOI: 10.1039/C5Ob01802A  0.621
2015 Singh B, Jain SK, Bharate SB, Kushwaha M, Gupta AP, Vishwakarma RA. Simultaneous Quantification of Five Bioactive Flavonoids in High Altitude Plant Actinocarya tibetica by LC-ESI-MS/MS. Journal of Aoac International. 98: 907-12. PMID 26268971 DOI: 10.5740/Jaoacint.14-270  0.769
2015 Singh B, Jain SK, Bharate SB, Kushwaha M, Gupta AP, Vishwakarma RA. Simultaneous Quantification of Five Bioactive Flavonoids in High Altitude Plant Actinocarya tibetica by LC-ESI-MS/MS. Journal of Aoac International. 98: 907-12. PMID 26268971 DOI: 10.5740/Jaoacint.14-270  0.769
2015 Bharate JB, Abbat S, Bharatam PV, Vishwakarma RA, Bharate SB. CuBr catalyzed aerobic oxidative coupling of 2-aminopyridines with cinnamaldehydes: direct access to 3-formyl-2-phenyl-imidazo[1,2-a]pyridines. Organic & Biomolecular Chemistry. 13: 7790-4. PMID 26103156 DOI: 10.1039/C5Ob00776C  0.502
2015 Bharate JB, Abbat S, Bharatam PV, Vishwakarma RA, Bharate SB. CuBr catalyzed aerobic oxidative coupling of 2-aminopyridines with cinnamaldehydes: direct access to 3-formyl-2-phenyl-imidazo[1,2-a]pyridines. Organic & Biomolecular Chemistry. 13: 7790-4. PMID 26103156 DOI: 10.1039/C5Ob00776C  0.502
2015 Mohammed S, Vishwakarma RA, Bharate SB. Iodine Catalyzed Oxidative Synthesis of Quinazolin-4(3H)-ones and Pyrazolo[4,3-d]pyrimidin-7(6H)-ones via Amination of sp3 C-H Bond Journal of Organic Chemistry. 80: 6915-6921. PMID 26067767 DOI: 10.1021/Acs.Joc.5B00989  0.51
2015 Mohammed S, Vishwakarma RA, Bharate SB. Iodine Catalyzed Oxidative Synthesis of Quinazolin-4(3H)-ones and Pyrazolo[4,3-d]pyrimidin-7(6H)-ones via Amination of sp3 C-H Bond Journal of Organic Chemistry. 80: 6915-6921. PMID 26067767 DOI: 10.1021/Acs.Joc.5B00989  0.51
2015 Yadav RR, Sharma S, Joshi P, Wani A, Vishwakarma RA, Kumar A, Bharate SB. Meridianin derivatives as potent Dyrk1A inhibitors and neuroprotective agents. Bioorganic & Medicinal Chemistry Letters. 25: 2948-52. PMID 26048785 DOI: 10.1016/J.Bmcl.2015.05.034  0.825
2015 Yadav RR, Sharma S, Joshi P, Wani A, Vishwakarma RA, Kumar A, Bharate SB. Meridianin derivatives as potent Dyrk1A inhibitors and neuroprotective agents. Bioorganic & Medicinal Chemistry Letters. 25: 2948-52. PMID 26048785 DOI: 10.1016/J.Bmcl.2015.05.034  0.825
2015 Yadav RR, Khan SI, Singh S, Khan IA, Vishwakarma RA, Bharate SB. Synthesis, antimalarial and antitubercular activities of meridianin derivatives. European Journal of Medicinal Chemistry. 98: 160-9. PMID 26005918 DOI: 10.1016/J.Ejmech.2015.05.020  0.765
2015 Yadav RR, Khan SI, Singh S, Khan IA, Vishwakarma RA, Bharate SB. Synthesis, antimalarial and antitubercular activities of meridianin derivatives. European Journal of Medicinal Chemistry. 98: 160-9. PMID 26005918 DOI: 10.1016/J.Ejmech.2015.05.020  0.765
2015 Mahale S, Bharate SB, Manda S, Joshi P, Jenkins PR, Vishwakarma RA, Chaudhuri B. Antitumour potential of BPT: a dual inhibitor of cdk4 and tubulin polymerization. Cell Death & Disease. 6: e1743. PMID 25950473 DOI: 10.1038/Cddis.2015.96  0.716
2015 Singh B, Kumar A, Joshi P, Guru SK, Kumar S, Wani ZA, Mahajan G, Hussain A, Qazi AK, Kumar A, Bharate SS, Gupta BD, Sharma PR, Hamid A, Saxena AK, ... ... Bharate SB, et al. Colchicine derivatives with potent anticancer activity and reduced P-glycoprotein induction liability. Organic & Biomolecular Chemistry. 13: 5674-89. PMID 25895604 DOI: 10.1039/C5Ob00406C  0.745
2015 Singh B, Kumar A, Joshi P, Guru SK, Kumar S, Wani ZA, Mahajan G, Hussain A, Qazi AK, Kumar A, Bharate SS, Gupta BD, Sharma PR, Hamid A, Saxena AK, ... ... Bharate SB, et al. Colchicine derivatives with potent anticancer activity and reduced P-glycoprotein induction liability. Organic & Biomolecular Chemistry. 13: 5674-89. PMID 25895604 DOI: 10.1039/C5Ob00406C  0.745
2015 Bharate JB, Batarseh YS, Wani A, Sharma S, Vishwakarma RA, Kaddoumi A, Kumar A, Bharate SB. Synthesis and P-glycoprotein induction activity of colupulone analogs. Organic & Biomolecular Chemistry. 13: 5488-96. PMID 25875530 DOI: 10.1039/C5Ob00554J  0.553
2015 Bharate JB, Batarseh YS, Wani A, Sharma S, Vishwakarma RA, Kaddoumi A, Kumar A, Bharate SB. Synthesis and P-glycoprotein induction activity of colupulone analogs. Organic & Biomolecular Chemistry. 13: 5488-96. PMID 25875530 DOI: 10.1039/C5Ob00554J  0.553
2015 Bharate JB, Singh S, Wani A, Sharma S, Joshi P, Khan IA, Kumar A, Vishwakarma RA, Bharate SB. Discovery of 4-acetyl-3-(4-fluorophenyl)-1-(p-tolyl)-5-methylpyrrole as a dual inhibitor of human P-glycoprotein and Staphylococcus aureus Nor A efflux pump. Organic & Biomolecular Chemistry. 13: 5424-31. PMID 25865846 DOI: 10.1039/C5Ob00246J  0.702
2015 Bharate JB, Singh S, Wani A, Sharma S, Joshi P, Khan IA, Kumar A, Vishwakarma RA, Bharate SB. Discovery of 4-acetyl-3-(4-fluorophenyl)-1-(p-tolyl)-5-methylpyrrole as a dual inhibitor of human P-glycoprotein and Staphylococcus aureus Nor A efflux pump. Organic & Biomolecular Chemistry. 13: 5424-31. PMID 25865846 DOI: 10.1039/C5Ob00246J  0.702
2015 Bharate JB, Abbat S, Sharma R, Bharatam PV, Vishwakarma RA, Bharate SB. Cobalt(II) catalyzed C(sp)-H bond functionalization of alkynes with phenyl hydrazines: facile access to diaryl 1,2-diketones. Organic & Biomolecular Chemistry. 13: 5235-42. PMID 25856782 DOI: 10.1039/C5Ob00419E  0.61
2015 Bharate JB, Abbat S, Sharma R, Bharatam PV, Vishwakarma RA, Bharate SB. Cobalt(II) catalyzed C(sp)-H bond functionalization of alkynes with phenyl hydrazines: facile access to diaryl 1,2-diketones. Organic & Biomolecular Chemistry. 13: 5235-42. PMID 25856782 DOI: 10.1039/C5Ob00419E  0.61
2015 Mudududdla R, Guru SK, Wani A, Sharma S, Joshi P, Vishwakarma RA, Kumar A, Bhushan S, Bharate SB. 3-(Benzo[d][1,3]dioxol-5-ylamino)-N-(4-fluorophenyl)thiophene-2-carboxamide overcomes cancer chemoresistance via inhibition of angiogenesis and P-glycoprotein efflux pump activity. Organic & Biomolecular Chemistry. 13: 4296-309. PMID 25758415 DOI: 10.1039/C5Ob00233H  0.832
2015 Mudududdla R, Guru SK, Wani A, Sharma S, Joshi P, Vishwakarma RA, Kumar A, Bhushan S, Bharate SB. 3-(Benzo[d][1,3]dioxol-5-ylamino)-N-(4-fluorophenyl)thiophene-2-carboxamide overcomes cancer chemoresistance via inhibition of angiogenesis and P-glycoprotein efflux pump activity. Organic & Biomolecular Chemistry. 13: 4296-309. PMID 25758415 DOI: 10.1039/C5Ob00233H  0.832
2015 Kumar S, Guru SK, Pathania AS, Manda S, Kumar A, Bharate SB, Vishwakarma RA, Malik F, Bhushan S. Fascaplysin induces caspase mediated crosstalk between apoptosis and autophagy through the inhibition of PI3K/AKT/mTOR signaling cascade in human leukemia HL-60 cells. Journal of Cellular Biochemistry. 116: 985-97. PMID 25561006 DOI: 10.1002/Jcb.25053  0.791
2015 Kumar S, Guru SK, Pathania AS, Manda S, Kumar A, Bharate SB, Vishwakarma RA, Malik F, Bhushan S. Fascaplysin induces caspase mediated crosstalk between apoptosis and autophagy through the inhibition of PI3K/AKT/mTOR signaling cascade in human leukemia HL-60 cells. Journal of Cellular Biochemistry. 116: 985-97. PMID 25561006 DOI: 10.1002/Jcb.25053  0.791
2015 Bharate JB, Vishwakarma RA, Bharate SB. Metal-free domino one-pot protocols for quinoline synthesis Rsc Advances. 5: 42020-42053. DOI: 10.1039/C5Ra07798B  0.476
2015 Mohammed S, Vishwakarma RA, Bharate SB. Metal-free DBU promoted regioselective synthesis of isoxazoles and isoxazolines Rsc Advances. 5: 3470-3473. DOI: 10.1039/C4Ra14694H  0.503
2015 Sharma R, Guru SK, Jain SK, Pathania AS, Vishwakarma RA, Bhushan S, Bharate SB. 3-(2,6-Dichloro-benzyloxy)-11-oxo-olean-12-ene-29-oic acid, a semisynthetic derivative of glycyrrhetic acid: synthesis, antiproliferative, apoptotic and anti-angiogenesis activity Medchemcomm. 6: 564-575. DOI: 10.1039/C4Md00344F  0.817
2015 Sharma R, Abbat S, Mudududdla R, Vishwakarma RA, Bharatam PV, Bharate SB. ortho-Quinone methides: TFA-mediated generation in water and trapping with lactams and styrenes Tetrahedron Letters. 56: 4057-4059. DOI: 10.1016/J.Tetlet.2015.04.072  0.769
2015 Mohammed S, Vishwakarma RA, Bharate SB. ChemInform Abstract: Iodine Catalyzed Oxidative Synthesis of Quinazolin-4(3H)-ones and Pyrazolo[4,3-d]pyrimidin-7(6H)-ones via Amination of sp3C-H Bond. Cheminform. 46: no-no. DOI: 10.1002/CHIN.201545180  0.263
2015 Sharma R, Abbat S, Mudududdla R, Vishwakarma RA, Bharatam PV, Bharate SB. ChemInform Abstract: ortho-Quinone Methides: TFA-Mediated Generation in Water and Trapping with Lactams and Styrenes. Cheminform. 46: no-no. DOI: 10.1002/CHIN.201542194  0.704
2015 Bharate JB, Vishwakarma RA, Bharate SB. ChemInform Abstract: Metal-Free Domino One-Pot Protocols for Quinoline Synthesis Cheminform. 46: no-no. DOI: 10.1002/CHIN.201529285  0.232
2015 Mohammed S, Vishwakarma RA, Bharate SB. ChemInform Abstract: Metal-Free DBU Promoted Regioselective Synthesis of Isoxazoles and Isoxazolines. Cheminform. 46: no-no. DOI: 10.1002/CHIN.201524144  0.235
2014 Kumar S, Guru SK, Pathania AS, Mupparapu N, Kumar A, Malik F, Bharate SB, Naveed Ahmed Q, Vishwakarma RA, Bhushan S. A novel quinazolinone derivative induces cytochrome c interdependent apoptosis and autophagy in human leukemia MOLT-4 cells. Toxicology Reports. 1: 1013-1025. PMID 28962314 DOI: 10.1016/J.Toxrep.2014.07.018  0.541
2014 Kumar S, Guru SK, Pathania AS, Mupparapu N, Kumar A, Malik F, Bharate SB, Naveed Ahmed Q, Vishwakarma RA, Bhushan S. A novel quinazolinone derivative induces cytochrome c interdependent apoptosis and autophagy in human leukemia MOLT-4 cells. Toxicology Reports. 1: 1013-1025. PMID 28962314 DOI: 10.1016/J.Toxrep.2014.07.018  0.541
2014 Bharate JB, Vishwakarma RA, Bharate SB, Kushwaha M, Gupta AP. Quantification of the Polyisoprenylated Benzophenones Garcinol and Isogarcinol Using Multiple Reaction Monitoring LC/Electrospray Ionization-MS/MS Analysis of Ultrasound-Assisted Extracts of Garcinia indica Fruits. Journal of Aoac International. 97: 1317-22. PMID 25902981 DOI: 10.5740/Jaoacint.13-137  0.481
2014 Mahale S, Bharate SB, Manda S, Joshi P, Bharate SS, Jenkins PR, Vishwakarma RA, Chaudhuri B. Biphenyl-4-carboxylic acid [2-(1H-indol-3-yl)-ethyl]-methylamide (CA224), a nonplanar analogue of fascaplysin, inhibits Cdk4 and tubulin polymerization: evaluation of in vitro and in vivo anticancer activity. Journal of Medicinal Chemistry. 57: 9658-72. PMID 25368960 DOI: 10.1021/Jm5014743  0.819
2014 Mahale S, Bharate SB, Manda S, Joshi P, Bharate SS, Jenkins PR, Vishwakarma RA, Chaudhuri B. Biphenyl-4-carboxylic acid [2-(1H-indol-3-yl)-ethyl]-methylamide (CA224), a nonplanar analogue of fascaplysin, inhibits Cdk4 and tubulin polymerization: evaluation of in vitro and in vivo anticancer activity. Journal of Medicinal Chemistry. 57: 9658-72. PMID 25368960 DOI: 10.1021/Jm5014743  0.819
2014 Bharate SS, Bharate SB. Non-enzymatic browning in citrus juice: chemical markers, their detection and ways to improve product quality. Journal of Food Science and Technology. 51: 2271-88. PMID 25328169 DOI: 10.1007/s13197-012-0718-8  0.272
2014 Bharate SS, Bharate SB. Non-enzymatic browning in citrus juice: chemical markers, their detection and ways to improve product quality. Journal of Food Science and Technology. 51: 2271-88. PMID 25328169 DOI: 10.1007/s13197-012-0718-8  0.272
2014 Bharate JB, Bharate SB, Vishwakarma RA. Metal-free, ionic liquid-mediated synthesis of functionalized quinolines. Acs Combinatorial Science. 16: 624-30. PMID 25314670 DOI: 10.1021/Co500047W  0.512
2014 Singh B, Guru SK, Sharma R, Bharate SS, Khan IA, Bhushan S, Bharate SB, Vishwakarma RA. Synthesis and anti-proliferative activities of new derivatives of embelin. Bioorganic & Medicinal Chemistry Letters. 24: 4865-70. PMID 25240254 DOI: 10.1016/J.Bmcl.2014.08.052  0.666
2014 Singh B, Guru SK, Sharma R, Bharate SS, Khan IA, Bhushan S, Bharate SB, Vishwakarma RA. Synthesis and anti-proliferative activities of new derivatives of embelin. Bioorganic & Medicinal Chemistry Letters. 24: 4865-70. PMID 25240254 DOI: 10.1016/J.Bmcl.2014.08.052  0.666
2014 Mudududdla R, Sharma R, Abbat S, Bharatam PV, Vishwakarma RA, Bharate SB. Synthesis of 2-phenylnaphthalenes from styryl-2-methoxybenzenes. Chemical Communications (Cambridge, England). 50: 12076-9. PMID 25163506 DOI: 10.1039/C4Cc05151C  0.789
2014 Mudududdla R, Sharma R, Abbat S, Bharatam PV, Vishwakarma RA, Bharate SB. Synthesis of 2-phenylnaphthalenes from styryl-2-methoxybenzenes. Chemical Communications (Cambridge, England). 50: 12076-9. PMID 25163506 DOI: 10.1039/C4Cc05151C  0.789
2014 Jain SK, Singh S, Khajuria A, Guru SK, Joshi P, Meena S, Nadkarni JR, Singh A, Bharate SS, Bhushan S, Bharate SB, Vishwakarma RA. Pyrano-isochromanones as IL-6 inhibitors: synthesis, in vitro and in vivo antiarthritic activity. Journal of Medicinal Chemistry. 57: 7085-97. PMID 25111439 DOI: 10.1021/Jm500901E  0.813
2014 Jain SK, Singh S, Khajuria A, Guru SK, Joshi P, Meena S, Nadkarni JR, Singh A, Bharate SS, Bhushan S, Bharate SB, Vishwakarma RA. Pyrano-isochromanones as IL-6 inhibitors: synthesis, in vitro and in vivo antiarthritic activity. Journal of Medicinal Chemistry. 57: 7085-97. PMID 25111439 DOI: 10.1021/Jm500901E  0.813
2014 Jain SK, Aravinda Kumar KA, Bharate SB, Vishwakarma RA. Facile access to amides and hydroxamic acids directly from nitroarenes. Organic & Biomolecular Chemistry. 12: 6465-9. PMID 25019340 DOI: 10.1039/C4Ob01155D  0.776
2014 Jain SK, Aravinda Kumar KA, Bharate SB, Vishwakarma RA. Facile access to amides and hydroxamic acids directly from nitroarenes. Organic & Biomolecular Chemistry. 12: 6465-9. PMID 25019340 DOI: 10.1039/C4Ob01155D  0.776
2014 Bharate JB, Wani A, Sharma S, Reja SI, Kumar M, Vishwakarma RA, Kumar A, Bharate SB. Synthesis, and the antioxidant, neuroprotective and P-glycoprotein induction activity of 4-arylquinoline-2-carboxylates. Organic & Biomolecular Chemistry. 12: 6267-77. PMID 25007760 DOI: 10.1039/C4Ob00488D  0.596
2014 Bharate JB, Wani A, Sharma S, Reja SI, Kumar M, Vishwakarma RA, Kumar A, Bharate SB. Synthesis, and the antioxidant, neuroprotective and P-glycoprotein induction activity of 4-arylquinoline-2-carboxylates. Organic & Biomolecular Chemistry. 12: 6267-77. PMID 25007760 DOI: 10.1039/C4Ob00488D  0.596
2014 Manda S, Khan SI, Jain SK, Mohammed S, Tekwani BL, Khan IA, Vishwakarma RA, Bharate SB. Synthesis, antileishmanial and antitrypanosomal activities of N-substituted tetrahydro-β-carbolines. Bioorganic & Medicinal Chemistry Letters. 24: 3247-50. PMID 24980054 DOI: 10.1016/J.Bmcl.2014.06.030  0.816
2014 Manda S, Khan SI, Jain SK, Mohammed S, Tekwani BL, Khan IA, Vishwakarma RA, Bharate SB. Synthesis, antileishmanial and antitrypanosomal activities of N-substituted tetrahydro-β-carbolines. Bioorganic & Medicinal Chemistry Letters. 24: 3247-50. PMID 24980054 DOI: 10.1016/J.Bmcl.2014.06.030  0.816
2014 Jain SK, Meena S, Gupta AP, Kushwaha M, Uma Shaanker R, Jaglan S, Bharate SB, Vishwakarma RA. Dysoxylum binectariferum bark as a new source of anticancer drug camptothecin: bioactivity-guided isolation and LCMS-based quantification. Bioorganic & Medicinal Chemistry Letters. 24: 3146-9. PMID 24878199 DOI: 10.1016/J.Bmcl.2014.05.001  0.787
2014 Jain SK, Meena S, Gupta AP, Kushwaha M, Uma Shaanker R, Jaglan S, Bharate SB, Vishwakarma RA. Dysoxylum binectariferum bark as a new source of anticancer drug camptothecin: bioactivity-guided isolation and LCMS-based quantification. Bioorganic & Medicinal Chemistry Letters. 24: 3146-9. PMID 24878199 DOI: 10.1016/J.Bmcl.2014.05.001  0.787
2014 Joshi P, Singh S, Wani A, Sharma S, Jain SK, Singh B, Gupta BD, Satti NK, Koul S, Khan IA, Kumar A, Bharate SB, Vishwakarma RA. Osthol and curcumin as inhibitors of human Pgp and multidrug efflux pumps of Staphylococcus aureus: Reversing the resistance against frontline antibacterial drugs Medchemcomm. 5: 1540-1547. DOI: 10.1039/C4Md00196F  0.8
2014 Mudududdla R, Sharma R, Guru SK, Kushwaha M, Gupta AP, Bharate SS, Aravinda S, Kant R, Bhushan S, Vishwakarma RA, Bharate SB. Trifluoroacetic acid catalyzed thiophenylmethylation and thioalkylmethylation of lactams and phenols via domino three-component reaction in water Rsc Advances. 4: 14081-14088. DOI: 10.1039/C3Ra47874B  0.792
2014 Bahl A, Joshi P, Bharate SB, Chopra H. Pharmacophore modeling and 3D-QSAR studies of leucettines as potent Dyrk2 inhibitors Medicinal Chemistry Research. 23: 1925-1933. DOI: 10.1007/s00044-013-0767-1  0.601
2013 Singh B, Guru SK, Kour S, Jain SK, Sharma R, Sharma PR, Singh SK, Bhushan S, Bharate SB, Vishwakarma RA. Synthesis, antiproliferative and apoptosis-inducing activity of thiazolo[5,4-d]pyrimidines. European Journal of Medicinal Chemistry. 70: 864-74. PMID 24262379 DOI: 10.1016/J.Ejmech.2013.10.039  0.81
2013 Singh B, Guru SK, Kour S, Jain SK, Sharma R, Sharma PR, Singh SK, Bhushan S, Bharate SB, Vishwakarma RA. Synthesis, antiproliferative and apoptosis-inducing activity of thiazolo[5,4-d]pyrimidines. European Journal of Medicinal Chemistry. 70: 864-74. PMID 24262379 DOI: 10.1016/J.Ejmech.2013.10.039  0.81
2013 Jain SK, Pathania AS, Meena S, Sharma R, Sharma A, Singh B, Gupta BD, Bhushan S, Bharate SB, Vishwakarma RA. Semisynthesis of mallotus B from rottlerin: evaluation of cytotoxicity and apoptosis-inducing activity. Journal of Natural Products. 76: 1724-30. PMID 24041234 DOI: 10.1021/Np400433G  0.81
2013 Jain SK, Pathania AS, Meena S, Sharma R, Sharma A, Singh B, Gupta BD, Bhushan S, Bharate SB, Vishwakarma RA. Semisynthesis of mallotus B from rottlerin: evaluation of cytotoxicity and apoptosis-inducing activity. Journal of Natural Products. 76: 1724-30. PMID 24041234 DOI: 10.1021/Np400433G  0.81
2013 Singh B, Vishwakarma RA, Bharate SB. QSAR and pharmacophore modeling of natural and synthetic antimalarial prodiginines. Current Computer-Aided Drug Design. 9: 350-9. PMID 24010933 DOI: 10.2174/15734099113099990020  0.617
2013 Singh B, Vishwakarma RA, Bharate SB. QSAR and pharmacophore modeling of natural and synthetic antimalarial prodiginines. Current Computer-Aided Drug Design. 9: 350-9. PMID 24010933 DOI: 10.2174/15734099113099990020  0.617
2013 Singh B, Sidiq T, Joshi P, Jain SK, Lawaniya Y, Kichlu S, Khajuria A, Vishwakarma RA, Bharate SB. Anti-inflammatory and immunomodulatory flavones from Actinocarya tibetica Benth. Natural Product Research. 27: 2227-30. PMID 23768253 DOI: 10.1080/14786419.2013.805334  0.794
2013 Singh B, Sidiq T, Joshi P, Jain SK, Lawaniya Y, Kichlu S, Khajuria A, Vishwakarma RA, Bharate SB. Anti-inflammatory and immunomodulatory flavones from Actinocarya tibetica Benth. Natural Product Research. 27: 2227-30. PMID 23768253 DOI: 10.1080/14786419.2013.805334  0.794
2013 Bharate SB, Sawant SD, Singh PP, Vishwakarma RA. Kinase inhibitors of marine origin. Chemical Reviews. 113: 6761-815. PMID 23679846 DOI: 10.1021/Cr300410V  0.5
2013 Bharate SB, Sawant SD, Singh PP, Vishwakarma RA. Kinase inhibitors of marine origin. Chemical Reviews. 113: 6761-815. PMID 23679846 DOI: 10.1021/Cr300410V  0.5
2013 Bharate SB, Bharate JB, Khan SI, Tekwani BL, Jacob MR, Mudududdla R, Yadav RR, Singh B, Sharma PR, Maity S, Singh B, Khan IA, Vishwakarma RA. Discovery of 3,3'-diindolylmethanes as potent antileishmanial agents. European Journal of Medicinal Chemistry. 63: 435-43. PMID 23517732 DOI: 10.1016/J.Ejmech.2013.02.024  0.817
2013 Bharate SB, Bharate JB, Khan SI, Tekwani BL, Jacob MR, Mudududdla R, Yadav RR, Singh B, Sharma PR, Maity S, Singh B, Khan IA, Vishwakarma RA. Discovery of 3,3'-diindolylmethanes as potent antileishmanial agents. European Journal of Medicinal Chemistry. 63: 435-43. PMID 23517732 DOI: 10.1016/J.Ejmech.2013.02.024  0.817
2013 Bahl A, Joshi P, Bharate S, Chopra H. Pharmacophore Based 3D-QSAR Modeling and Molecular Docking of Leucettines as Potent Dyrk1A Inhibitors Letters in Drug Design & Discovery. 10: 719-726. DOI: 10.2174/15701808113100890024  0.583
2013 Bharate JB, Vishwakarma RA, Bharate SB, Thite TB, Kushwaha M, Gupta AP. Quantification and Validation of Two Isomeric Anticancer Compounds, Garcinol and Isogarcinol, in Ultrasound- Assisted Extracts of Garcinia indica Fruits Using High- Performance Thin-Layer Chromatography Jpc-Journal of Planar Chromatography-Modern Tlc. 26: 480-485. DOI: 10.1556/Jpc.26.2013.6.4  0.508
2013 Bharate JB, Vishwakarma RA, Bharate SB, Kushwaha M, Gupta AP. Quantification Of Anticancer Polyisoprenylated Benzophenones Garcinol And Isogarcinol Using Multiple Reaction Monitoring Lc-Esi-Ms-Ms In Ultra-Sound Assisted Extracts Of Garcinia Indica Fruits Journal of Liquid Chromatography & Related Technologies. 150527103729000. DOI: 10.1080/10826076.2013.873872  0.48
2013 Bharate JB, Sharma R, Aravinda S, Gupta VK, Singh B, Bharate SB, Vishwakarma RA. Montmorillonite clay catalyzed synthesis of functionalized pyrroles through domino four-component coupling of amines, aldehydes, 1,3-dicarbonyl compounds and nitroalkanes Rsc Advances. 3: 21736-21742. DOI: 10.1039/C3Ra43324B  0.514
2013 Jain SK, Pathania AS, Parshad R, Raina C, Ali A, Gupta AP, Kushwaha M, Aravinda S, Bhushan S, Bharate SB, Vishwakarma RA. Chrysomycins A-C, antileukemic naphthocoumarins from Streptomyces sporoverrucosus Rsc Advances. 3: 21046-21053. DOI: 10.1039/C3Ra42884B  0.807
2013 Bharate JB, Guru SK, Jain SK, Meena S, Singh PP, Bhushan S, Singh B, Bharate SB, Vishwakarma RA. Cu–Mn spinel oxide catalyzed synthesis of imidazo[1,2-a]pyridines through domino three-component coupling and 5-exo-dig cyclization in water Rsc Advances. 3: 20869-20876. DOI: 10.1039/C3Ra42046A  0.77
2013 Bharate SB, Yadav RR, Khan SI, Tekwani BL, Jacob MR, Khan IA, Vishwakarma RA. Meridianin G and its analogs as antimalarial agents Medchemcomm. 4: 1042-1048. DOI: 10.1039/C3Md00097D  0.756
2013 Jain SK, Meena S, Qazi AK, Hussain A, Bhola SK, Kshirsagar R, Pari K, Khajuria A, Hamid A, Shaanker RU, Bharate SB, Vishwakarma RA. Isolation and biological evaluation of chromone alkaloid dysoline, a new regioisomer of rohitukine from Dysoxylum binectariferum Tetrahedron Letters. 54: 7140-7143. DOI: 10.1016/J.Tetlet.2013.10.096  0.792
2013 Singh B, Parshad R, Khajuria R, Guru SK, Pathania AS, Sharma R, Chib R, Aravinda S, Gupta VK, Khan IA, Bhushan S, Bharate SB, Vishwakarma RA. Saccharonol B, a new cytotoxic methylated isocoumarin from Saccharomonospora azurea Tetrahedron Letters. 54: 6695-6699. DOI: 10.1016/J.Tetlet.2013.09.060  0.641
2013 Bharate SB, Padala AK, Dar BA, Yadav RR, Singh B, Vishwakarma RA. Montmorillonite clay Cu(II) catalyzed domino one-pot multicomponent synthesis of 3,5-disubstituted isoxazoles Tetrahedron Letters. 54: 3558-3561. DOI: 10.1016/J.Tetlet.2013.04.102  0.713
2013 Bharate SB, Mudududdla R, Sharma R, Vishwakarma RA. The first method for C-devinylation of aromatic systems Tetrahedron Letters. 54: 2913-2915. DOI: 10.1016/J.Tetlet.2013.03.064  0.764
2013 Bharate SB, Padala AK, Dar BA, Yadav RR, Singh B, Vishwakarma RA. ChemInform Abstract: Montmorillonite Clay Cu(II) Catalyzed Domino One-Pot Multicomponent Synthesis of 3,5-Disubstituted Isoxazoles. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201341143  0.634
2013 Bharate SB, Sawant SD, Singh PP, Vishwakarma RA. ChemInform Abstract: Kinase Inhibitors of Marine Origin Cheminform. 44: no-no. DOI: 10.1002/CHIN.201340271  0.285
2013 Bharate SB, Mudududdla R, Sharma R, Vishwakarma RA. ChemInform Abstract: The First Method for C-Devinylation of Aromatic Systems. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201337051  0.706
2013 Mohammed S, Padala AK, Dar BA, Singh B, Sreedhar B, Vishwakarma RA, Bharate SB. ChemInform Abstract: Recyclable Clay-Supported Cu(II)-Catalyzed Tandem One-Pot Synthesis of 1-Aryl-1,2,3-triazoles. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201309139  0.24
2013 Yadav RR, Vishwakarma RA, Bharate SB. ChemInform Abstract: Catalyst-Free ipso-Nitration of Aryl Boronic Acids Using Bismuth Nitrate. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201304040  0.636
2012 Mudududdla R, Jain SK, Bharate JB, Gupta AP, Singh B, Vishwakarma RA, Bharate SB. ortho-Amidoalkylation of phenols via tandem one-pot approach involving oxazine intermediate. The Journal of Organic Chemistry. 77: 8821-7. PMID 22970791 DOI: 10.1021/Jo3017132  0.775
2012 Bharate SB, Yadav RR, Vishwakarma RA. QSAR and Pharmacophore Study of Dyrk1A Inhibitory Meridianin Analogs as Potential Agents for Treatment of Neurodegenerative Diseases Medicinal Chemistry. 9: 152-161. PMID 22920091 DOI: 10.2174/157340613804488459  0.751
2012 Bharate SB, Yadav RR, Vishwakarma RA. QSAR and Pharmacophore Study of Dyrk1A Inhibitory Meridianin Analogs as Potential Agents for Treatment of Neurodegenerative Diseases Medicinal Chemistry. 9: 152-161. PMID 22920091 DOI: 10.2174/157340613804488459  0.751
2012 Bharate SS, Bharate SB. Modulation of thermoreceptor TRPM8 by cooling compounds. Acs Chemical Neuroscience. 3: 248-67. PMID 22860192 DOI: 10.1021/cn300006u  0.357
2012 Bharate SS, Bharate SB. Modulation of thermoreceptor TRPM8 by cooling compounds. Acs Chemical Neuroscience. 3: 248-67. PMID 22860192 DOI: 10.1021/cn300006u  0.357
2012 Bharate SB, Mudududdla R, Bharate JB, Battini N, Battula S, Yadav RR, Singh B, Vishwakarma RA. Tandem one-pot synthesis of flavans by recyclable silica-HClO4 catalyzed Knoevenagel condensation and [4 + 2]-Diels-Alder cycloaddition. Organic & Biomolecular Chemistry. 10: 5143-50. PMID 22648274 DOI: 10.1039/C2Ob25376C  0.789
2012 Jain SK, Bharate SB, Vishwakarma RA. Cyclin-dependent kinase inhibition by flavoalkaloids. Mini-Reviews in Medicinal Chemistry. 12: 632-649. PMID 22512551 DOI: 10.2174/138955712800626683  0.564
2012 Bharate SB, Yadav RR, Battula S, Vishwakarma RA. Meridianins: Marine-Derived Potent Kinase Inhibitors Mini-Reviews in Medicinal Chemistry. 12: 618-631. PMID 22512550 DOI: 10.2174/138955712800626728  0.775
2012 Bharate SB, Manda S, Mupparapu N, Battini N, Vishwakarma RA. Chemistry and biology of fascaplysin, a potent marine-derived CDK-4 inhibitor. Mini-Reviews in Medicinal Chemistry. 12: 650-664. PMID 22512549 DOI: 10.2174/138955712800626719  0.601
2012 Singh B, Nadkarni JR, Vishwakarma RA, Bharate SB, Nivsarkar M, Anandjiwala S. The hydroalcoholic extract of Cassia alata (Linn.) leaves and its major compound rhein exhibits antiallergic activity via mast cell stabilization and lipoxygenase inhibition. Journal of Ethnopharmacology. 141: 469-73. PMID 22449441 DOI: 10.1016/J.Jep.2012.03.012  0.617
2012 Bharate SB, Singh B, Vishwakarma RA. Modulation of k-Ras signaling by natural products. Current Medicinal Chemistry. 19: 2273-2291. PMID 22414109 DOI: 10.2174/092986712800229050  0.585
2012 Chauthe SK, Bharate SB, Periyasamy G, Khanna A, Bhutani KK, Mishra PD, Singh IP. One pot synthesis and anticancer activity of dimeric phloroglucinols. Bioorganic & Medicinal Chemistry Letters. 22: 2251-6. PMID 22342146 DOI: 10.1016/j.bmcl.2012.01.089  0.82
2012 Bharate SB, Mupparapu N, Manda S, Bharate JB, Mudududdla R, Yadav RR, Vishwakarma RA. Efficient synthesis of 2,3-dihydroquinazolin-4(1H)-ones using heterogeneous solid acid catalysts: unexpected formation of 2,3-dihydro-2-(4-(tetrahydro-2H-pyran-2-yloxy)butyl)-quinazolin-4(1H)-one Arkivoc. 2012: 308-318. DOI: 10.3998/Ark.5550190.0013.826  0.786
2012 Jain SK, Meena S, Singh B, Bharate JB, Joshi P, Singh VP, Vishwakarma RA, Bharate SB. KF/alumina catalyzed regioselective benzylation and benzoylation using solvent-free grind-stone chemistry Rsc Advances. 2: 8929. DOI: 10.1039/C2Ra21154H  0.781
2012 Bharate SB, Manda S, Joshi P, Singh B, Vishwakarma RA. Total synthesis and anti-cholinesterase activity of marine-derived bis-indole alkaloid fascaplysin Medchemcomm. 3: 1098. DOI: 10.1039/C2Md20076G  0.747
2012 Yadav RR, Vishwakarma RA, Bharate SB. Catalyst-free ipso-nitration of aryl boronic acids using bismuth nitrate☆ Tetrahedron Letters. 53: 5958-5960. DOI: 10.1016/J.Tetlet.2012.08.121  0.714
2012 Yadav RR, Battini N, Mudududdla R, Bharate JB, Muparappu N, Bharate SB, Vishwakarma RA. Deformylation of indole and azaindole-3-carboxaldehydes using anthranilamide and solid acid heterogeneous catalyst via quinazolinone intermediate Tetrahedron Letters. 53: 2222-2225. DOI: 10.1016/J.Tetlet.2012.02.079  0.772
2012 Mohammed S, Padala AK, Dar BA, Singh B, Sreedhar B, Vishwakarma RA, Bharate SB. Recyclable clay supported Cu (II) catalyzed tandem one-pot synthesis of 1-aryl-1,2,3-triazoles ☆ Tetrahedron. 68: 8156-8162. DOI: 10.1016/J.Tet.2012.07.080  0.482
2012 Bharate SB, Singh B, Bharate JB, Jain SK, Meena S, Vishwakarma RA. QSAR and pharmacophore modeling of N-acetyl-2-aminobenzothiazole class of phosphoinositide-3-kinase-α inhibitors Medicinal Chemistry Research. 22: 890-899. DOI: 10.1007/S00044-012-0081-3  0.803
2012 Yadav RR, Battini N, Mudududdla R, Bharate JB, Muparappu N, Bharate SB, Vishwakarma RA. ChemInform Abstract: Deformylation of Indole and Azaindole-3-carboxaldehydes Using Anthranilamide and Solid Acid Heterogeneous Catalyst via Quinazolinone Intermediate. Cheminform. 43: no-no. DOI: 10.1002/CHIN.201232119  0.765
2011 Bharate SB, Singh IP. Quantitative structure-activity relationship study of phloroglucinol-terpene adducts as anti-leishmanial agents. Bioorganic & Medicinal Chemistry Letters. 21: 4310-5. PMID 21665468 DOI: 10.1016/j.bmcl.2011.05.053  0.604
2011 Bharate SB, Singh IP. Quantitative structure-activity relationship study of phloroglucinol-terpene adducts as anti-leishmanial agents. Bioorganic & Medicinal Chemistry Letters. 21: 4310-5. PMID 21665468 DOI: 10.1016/j.bmcl.2011.05.053  0.355
2011 Bharate SS, Bharate SB, Bajaj AN. ChemInform Abstract: Interactions and Incompatibilities of Pharmaceutical Excipients with Active Pharmaceutical Ingredients Cheminform. 42: no-no. DOI: 10.1002/CHIN.201147271  0.258
2010 Bharate SB, Thompson CM. Antimicrobial, antimalarial, and antileishmanial activities of mono- and bis-quaternary pyridinium compounds. Chemical Biology & Drug Design. 76: 546-51. PMID 21040494 DOI: 10.1111/J.1747-0285.2010.01035.X  0.581
2010 Jacobson SM, Birkholz DA, McNamara ML, Bharate SB, George KM. Subacute developmental exposure of zebrafish to the organophosphate pesticide metabolite, chlorpyrifos-oxon, results in defects in Rohon-Beard sensory neuron development. Aquatic Toxicology (Amsterdam, Netherlands). 100: 101-11. PMID 20701988 DOI: 10.1016/J.Aquatox.2010.07.015  0.257
2010 Jacobson SM, Birkholz DA, McNamara ML, Bharate SB, George KM. Subacute developmental exposure of zebrafish to the organophosphate pesticide metabolite, chlorpyrifos-oxon, results in defects in Rohon-Beard sensory neuron development. Aquatic Toxicology (Amsterdam, Netherlands). 100: 101-11. PMID 20701988 DOI: 10.1016/J.Aquatox.2010.07.015  0.257
2010 Bharate SB, Prins JM, George KM, Thompson CM. Thionate versus Oxon: comparison of stability, uptake, and cell toxicity of ((14)CH(3)O)(2)-labeled methyl parathion and methyl paraoxon with SH-SY5Y cells. Journal of Agricultural and Food Chemistry. 58: 8460-6. PMID 20590114 DOI: 10.1021/Jf100976V  0.508
2010 Singh IP, Sidana J, Bharate SB, Foley WJ. Phloroglucinol compounds of natural origin: synthetic aspects. Natural Product Reports. 27: 393-416. PMID 20179878 DOI: 10.1039/B914364P  0.59
2010 Chauthe SK, Bharate SB, Sabde S, Mitra D, Bhutani KK, Singh IP. Biomimetic synthesis and anti-HIV activity of dimeric phloroglucinols. Bioorganic & Medicinal Chemistry. 18: 2029-36. PMID 20137956 DOI: 10.1016/j.bmc.2010.01.023  0.792
2010 Bharate SB, Guo L, Reeves TE, Cerasoli DM, Thompson CM. Bisquaternary pyridinium oximes: Comparison of in vitro reactivation potency of compounds bearing aliphatic linkers and heteroaromatic linkers for paraoxon-inhibited electric eel and recombinant human acetylcholinesterase. Bioorganic & Medicinal Chemistry. 18: 787-94. PMID 20005727 DOI: 10.1016/J.Bmc.2009.11.052  0.696
2009 Bharate SB, Guo L, Reeves TE, Cerasoli DM, Thompson CM. New series of monoquaternary pyridinium oximes: Synthesis and reactivation potency for paraoxon-inhibited electric eel and recombinant human acetylcholinesterase. Bioorganic & Medicinal Chemistry Letters. 19: 5101-4. PMID 19640713 DOI: 10.1016/J.Bmcl.2009.07.035  0.693
2009 Bharate SB, Nemmani KVS, Vishwakarma RA. Progress in the discovery and development of small-molecule modulators of G-protein-coupled receptor 40 (GPR40/FFA1/FFAR1): an emerging target for type 2 diabetes. Expert Opinion On Therapeutic Patents. 19: 237-264. PMID 19441920 DOI: 10.1517/13543770802665717  0.498
2008 Bharate SB, Rodge A, Joshi RK, Kaur J, Srinivasan S, Kumar SS, Kulkarni-Almeida A, Balachandran S, Balakrishnan A, Vishwakarma RA. Discovery of diacylphloroglucinols as a new class of GPR40 (FFAR1) agonists. Bioorganic & Medicinal Chemistry Letters. 18: 6357-61. PMID 18993064 DOI: 10.1016/J.Bmcl.2008.10.085  0.538
2008 Bharate SB, Mahajan TR, Gole YR, Nambiar M, Matan TT, Kulkarni-Almeida A, Balachandran S, Junjappa H, Balakrishnan A, Vishwakarma RA. Synthesis and evaluation of pyrazolo[3,4-b]pyridines and its structural analogues as TNF-alpha and IL-6 inhibitors. Bioorganic & Medicinal Chemistry. 16: 7167-76. PMID 18625560 DOI: 10.1016/J.Bmc.2008.06.042  0.654
2007 Bharate SB, Khan SI, Tekwani BL, Jacob M, Khan IA, Singh IP. S-Euglobals: biomimetic synthesis, antileishmanial, antimalarial, and antimicrobial activities. Bioorganic & Medicinal Chemistry. 16: 1328-36. PMID 17976995 DOI: 10.1016/J.Bmc.2007.10.055  0.63
2007 Bharate SB, Khan SI, Yunus NA, Chauthe SK, Jacob MR, Tekwani BL, Khan IA, Singh IP. Antiprotozoal and antimicrobial activities of O-alkylated and formylated acylphloroglucinols. Bioorganic & Medicinal Chemistry. 15: 87-96. PMID 17070063 DOI: 10.1016/J.Bmc.2006.10.006  0.813
2007 Bharate SB, Khan SI, Yunus NA, Chauthe SK, Jacob MR, Tekwani BL, Khan IA, Singh IP. Antiprotozoal and antimicrobial activities of O-alkylated and formylated acylphloroglucinols. Bioorganic & Medicinal Chemistry. 15: 87-96. PMID 17070063 DOI: 10.1016/J.Bmc.2006.10.006  0.813
2006 Pal Singh I, Bharate SB. Phloroglucinol compounds of natural origin. Natural Product Reports. 23: 558-91. PMID 16874390 DOI: 10.1039/b600518g  0.324
2006 Bharate SB, Singh IP. A two-step biomimetic synthesis of antimalarial robustadials A and B Tetrahedron Letters. 47: 7021-7024. DOI: 10.1016/J.TETLET.2006.07.113  0.27
2005 Bharate SB, Bhutani KK, Khan SI, Tekwani BL, Jacob MR, Khan IA, Singh IP. Biomimetic synthesis, antimicrobial, antileishmanial and antimalarial activities of euglobals and their analogues. Bioorganic & Medicinal Chemistry. 14: 1750-60. PMID 16274995 DOI: 10.1016/J.Bmc.2005.10.027  0.606
2005 Bharate SB, Bhutani KK, Khan SI, Tekwani BL, Jacob MR, Khan IA, Singh IP. Biomimetic synthesis, antimicrobial, antileishmanial and antimalarial activities of euglobals and their analogues. Bioorganic & Medicinal Chemistry. 14: 1750-60. PMID 16274995 DOI: 10.1016/J.Bmc.2005.10.027  0.606
2005 Bharate SB, Chauthe SK, Bhutani KK, Singh IP. An Efficient Two-Step Synthesis of Jensenone Isolated from Eucalyptus jensenii. Synthesis of Analogues and Evaluation as Antioxidants Australian Journal of Chemistry. 58: 551. DOI: 10.1071/CH05061  0.363
2005 Bharate SB, Chauthe SK, Bhutani KK, Singh IP. An Efficient Two-Step Synthesis of Jensenone Isolated from Eucalyptus jensenii. Synthesis of Analogues and Evaluation as Antioxidants. Cheminform. 36. DOI: 10.1002/CHIN.200549194  0.299
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