| Year |
Citation |
Score |
| 2014 |
Lee H, Park KD, Torregrosa R, Yang XF, Dustrude ET, Wang Y, Wilson SM, Barbosa C, Xiao Y, Cummins TR, Khanna R, Kohn H. Substituted N-(biphenyl-4'-yl)methyl (R)-2-acetamido-3-methoxypropionamides: potent anticonvulsants that affect frequency (use) dependence and slow inactivation of sodium channels. Journal of Medicinal Chemistry. 57: 6165-82. PMID 25004277 DOI: 10.1021/Jm500707R |
0.406 |
|
| 2013 |
Lee H, Gold AS, Yang XF, Khanna R, Kohn H. Benzyloxybenzylammonium chlorides: Simple amine salts that display anticonvulsant activity. Bioorganic & Medicinal Chemistry. 21: 7655-62. PMID 24238903 DOI: 10.1016/J.Bmc.2013.10.031 |
0.328 |
|
| 2013 |
Park KD, Yang XF, Lee H, Dustrude ET, Wang Y, Khanna R, Kohn H. Discovery of lacosamide affinity bait agents that exhibit potent voltage-gated sodium channel blocking properties. Acs Chemical Neuroscience. 4: 463-74. PMID 23509982 DOI: 10.1021/Cn300188H |
0.363 |
|
| 2012 |
King AM, Yang XF, Wang Y, Dustrude ET, Barbosa C, Due MR, Piekarz AD, Wilson SM, White FA, Salomé C, Cummins TR, Khanna R, Kohn H. Identification of the benzyloxyphenyl pharmacophore: a structural unit that promotes sodium channel slow inactivation. Acs Chemical Neuroscience. 3: 1037-49. PMID 23259039 DOI: 10.1021/Cn300129D |
0.601 |
|
| 2012 |
Baruah PK, Dinsmore J, King AM, Salomé C, De Ryck M, Kaminski R, Provins L, Kohn H. Synthesis, anticonvulsant activity, and neuropathic pain-attenuating activity of N-benzyl 2-amino-2-(hetero)aromatic acetamides. Bioorganic & Medicinal Chemistry. 20: 3551-64. PMID 22546207 DOI: 10.1016/J.Bmc.2012.04.002 |
0.635 |
|
| 2011 |
King AM, De Ryck M, Kaminski R, Valade A, Stables JP, Kohn H. Defining the structural parameters that confer anticonvulsant activity by the site-by-site modification of (R)-N'-benzyl 2-amino-3-methylbutanamide. Journal of Medicinal Chemistry. 54: 6432-42. PMID 21861466 DOI: 10.1021/Jm200760A |
0.665 |
|
| 2011 |
King AM, Salomé C, Salomé-Grosjean E, De Ryck M, Kaminski R, Valade A, Stables JP, Kohn H. Primary amino acid derivatives: substitution of the 4'-N'-benzylamide site in (R)-N'-benzyl 2-amino-3-methylbutanamide, (R)-N'-benzyl 2-amino-3,3-dimethylbutanamide, and (R)-N'-benzyl 2-amino-3-methoxypropionamide provides potent anticonvulsants with pain-attenuating properties. Journal of Medicinal Chemistry. 54: 6417-31. PMID 21861463 DOI: 10.1021/Jm200759T |
0.659 |
|
| 2011 |
Wang Y, Wilson SM, Brittain JM, Ripsch MS, Salomé C, Park KD, White FA, Khanna R, Kohn H. Merging Structural Motifs of Functionalized Amino Acids and α-Aminoamides Results in Novel Anticonvulsant Compounds with Significant Effects on Slow and Fast Inactivation of Voltage-gated Sodium Channels and in the Treatment of Neuropathic Pain. Acs Chemical Neuroscience. 2: 317-322. PMID 21765969 DOI: 10.1021/Cn200024Z |
0.35 |
|
| 2011 |
Park KD, Kim D, Reamtong O, Eyers C, Gaskell SJ, Liu R, Kohn H. Identification of a lacosamide binding protein using an affinity bait and chemical reporter strategy: 14-3-3 ζ. Journal of the American Chemical Society. 133: 11320-30. PMID 21692503 DOI: 10.1021/Ja2034156 |
0.35 |
|
| 2011 |
King AM, Salomé C, Dinsmore J, Salomé-Grosjean E, De Ryck M, Kaminski R, Valade A, Kohn H. Primary amino acid derivatives: compounds with anticonvulsant and neuropathic pain protection activities. Journal of Medicinal Chemistry. 54: 4815-30. PMID 21639114 DOI: 10.1021/Jm2004305 |
0.665 |
|
| 2011 |
Wang Y, Park KD, Salome C, Wilson SM, Stables JP, Liu R, Khanna R, Kohn H. Development and characterization of novel derivatives of the antiepileptic drug lacosamide that exhibit far greater enhancement in slow inactivation of voltage-gated sodium channels. Acs Chemical Neuroscience. 2: 90-106. PMID 21532923 DOI: 10.1021/Cn100089B |
0.368 |
|
| 2010 |
Morieux P, Salomé C, Park KD, Stables JP, Kohn H. The structure-activity relationship of the 3-oxy site in the anticonvulsant (R)-N-benzyl 2-acetamido-3-methoxypropionamide. Journal of Medicinal Chemistry. 53: 5716-26. PMID 20614888 DOI: 10.1021/Jm100508M |
0.77 |
|
| 2010 |
Park KD, Stables JP, Liu R, Kohn H. Proteomic searches comparing two (R)-lacosamide affinity baits: An electrophilic arylisothiocyanate and a photoactivated arylazide group. Organic & Biomolecular Chemistry. 8: 2803-13. PMID 20405068 DOI: 10.1039/C000987C |
0.371 |
|
| 2010 |
Salomé C, Salomé-Grosjean E, Stables JP, Kohn H. Merging the structural motifs of functionalized amino acids and alpha-aminoamides: compounds with significant anticonvulsant activities. Journal of Medicinal Chemistry. 53: 3756-71. PMID 20394379 DOI: 10.1021/Jm100185C |
0.366 |
|
| 2010 |
Salomé C, Salomé-Grosjean E, Park KD, Morieux P, Swendiman R, DeMarco E, Stables JP, Kohn H. Synthesis and anticonvulsant activities of (R)-N-(4'-substituted)benzyl 2-acetamido-3-methoxypropionamides. Journal of Medicinal Chemistry. 53: 1288-305. PMID 20041718 DOI: 10.1021/Jm901563P |
0.78 |
|
| 2009 |
Park KD, Morieux P, Salomé C, Cotten SW, Reamtong O, Eyers C, Gaskell SJ, Stables JP, Liu R, Kohn H. Lacosamide isothiocyanate-based agents: novel agents to target and identify lacosamide receptors. Journal of Medicinal Chemistry. 52: 6897-911. PMID 19795888 DOI: 10.1021/Jm9012054 |
0.762 |
|
| 2009 |
Lee SH, Kohn H. Nucleophilic activation of a tetra-substituted mitomycin cyclic bis-disulfide. Chemical & Pharmaceutical Bulletin. 57: 149-57. PMID 19182404 DOI: 10.1248/Cpb.57.149 |
0.404 |
|
| 2009 |
LEGALL P, SAWHNEY KN, CONLEY JD, KOHN H. Synthesis of functionalized non-natural amino acid derivatives via amidoalkylation transformations International Journal of Peptide and Protein Research. 32: 279-291. DOI: 10.1111/J.1399-3011.1988.Tb01262.X |
0.309 |
|
| 2008 |
Morieux P, Stables JP, Kohn H. Synthesis and anticonvulsant activities of N-benzyl (2R)-2-acetamido-3-oxysubstituted propionamide derivatives. Bioorganic & Medicinal Chemistry. 16: 8968-75. PMID 18789868 DOI: 10.1016/J.Bmc.2008.08.055 |
0.778 |
|
| 2005 |
Kohn H, Widger W. The molecular basis for the mode of action of bicyclomycin. Current Drug Targets. Infectious Disorders. 5: 273-95. PMID 16181146 DOI: 10.2174/1568005054880136 |
0.301 |
|
| 2005 |
Brogan AP, Widger WR, Bensadek D, Riba-Garcia I, Gaskell SJ, Kohn H. Development of a technique to determine bicyclomycin-rho binding and stoichiometry by isothermal titration calorimetry and mass spectrometry. Journal of the American Chemical Society. 127: 2741-51. PMID 15725032 DOI: 10.1021/Ja046441Q |
0.658 |
|
| 2005 |
Brogan AP, Verghese J, Widger WR, Kohn H. Bismuth-dithiol inhibition of the Escherichia coli rho transcription termination factor. Journal of Inorganic Biochemistry. 99: 841-51. PMID 15708806 DOI: 10.1016/J.Jinorgbio.2004.12.019 |
0.68 |
|
| 2005 |
Lee SH, Kohn H. 7-N,7'-N'-(1",2"-Dithianyl-3",6"-dimethylenyl)bismitomycin C: synthesis and nucleophilic activation of a dimeric mitomycin. Organic & Biomolecular Chemistry. 3: 471-82. PMID 15678185 DOI: 10.1039/B414806A |
0.391 |
|
| 2005 |
Skordalakes E, Brogan AP, Park BS, Kohn H, Berger JM. Structural mechanism of inhibition of the Rho transcription termination factor by the antibiotic bicyclomycin. Structure (London, England : 1993). 13: 99-109. PMID 15642265 DOI: 10.1016/J.Str.2004.10.013 |
0.675 |
|
| 2005 |
Jin AY, Kohn H, Béguin C, Andurkar SV, Stables JP, Weaver DF. A quantitative structure-activity relationship study for α-substituted acetamido-N-benzylacetamide derivatives - A novel anticonvulsant drug class Canadian Journal of Chemistry. 83: 37-45. DOI: 10.1139/V04-160 |
0.403 |
|
| 2005 |
Lee SH, Brodnick RL, Glish GL, Kohn H. 3,8,11,16-Tetrakis(aminomethyl)-1,2,9,10-tetrathia-cyclohexadecane tetra-trifluoroacetic acid: Synthetic precursor to a novel thio-substituted diamine Tetrahedron. 61: 1749-1754. DOI: 10.1016/J.Tet.2004.12.030 |
0.336 |
|
| 2004 |
Béguin C, LeTiran A, Stables JP, Voyksner RD, Kohn H. N-Substituted amino acid N'-benzylamides: synthesis, anticonvulsant, and metabolic activities. Bioorganic & Medicinal Chemistry. 12: 3079-96. PMID 15142567 DOI: 10.1016/J.Bmc.2004.02.043 |
0.376 |
|
| 2004 |
Kim MG, Bodor ET, Harden TK, Kohn H. C(8)-substituted 1-azabicyclo[3.3.1]non-3-enes: a novel scaffold for muscarinic receptor ligands. Bioorganic & Medicinal Chemistry. 12: 2357-67. PMID 15080933 DOI: 10.1016/J.Bmc.2004.02.016 |
0.332 |
|
| 2003 |
Vedejs E, Naidu BN, Klapars A, Warner DL, Li VS, Na Y, Kohn H. Synthetic enantiopure aziridinomitosenes: preparation, reactivity, and DNA alkylation studies. Journal of the American Chemical Society. 125: 15796-806. PMID 14677970 DOI: 10.1021/Ja030452M |
0.557 |
|
| 2003 |
Béguin C, Andurkar SV, Jin AY, Stables JP, Weaver DF, Kohn H. Functionalized amido ketones: new anticonvulsant agents. Bioorganic & Medicinal Chemistry. 11: 4275-85. PMID 12951158 DOI: 10.1016/S0968-0896(03)00434-6 |
0.345 |
|
| 2003 |
Brogan AP, Widger WR, Kohn H. Bicyclomycin fluorescent probes: synthesis and biochemical, biophysical, and biological properties. The Journal of Organic Chemistry. 68: 5575-87. PMID 12839449 DOI: 10.1021/Jo030020U |
0.673 |
|
| 2003 |
Kim MG, Bodor ET, Wang C, Harden TK, Kohn H. C(8) substituted 1-azabicyclo[3.3.1]non-3-enes and C(8) substituted 1-azabicyclo[3.3.1]nonan-4-ones: novel muscarinic receptor antagonists. Journal of Medicinal Chemistry. 46: 2216-26. PMID 12747793 DOI: 10.1021/Jm020572P |
0.402 |
|
| 2003 |
Lee SH, Kohn H. Phosphine-assisted rearrangement of 4,5-dihydroxy-1,2-dithianes to 4-hydroxy-3-mercaptotetrahydrothiophenes Heterocycles. 60: 47-56. DOI: 10.3987/Com-02-9603 |
0.306 |
|
| 2002 |
LeTiran A, Stables JP, Kohn H. Design and evaluation of affinity labels of functionalized amino acid anticonvulsants. Journal of Medicinal Chemistry. 45: 4762-73. PMID 12361404 DOI: 10.1021/Jm020225F |
0.402 |
|
| 2002 |
Shen M, LeTiran A, Xiao Y, Golbraikh A, Kohn H, Tropsha A. Quantitative structure-activity relationship analysis of functionalized amino acid anticonvulsant agents using k nearest neighbor and simulated annealing PLS methods. Journal of Medicinal Chemistry. 45: 2811-23. PMID 12061883 DOI: 10.1021/Jm010488U |
0.303 |
|
| 2002 |
Na Y, Wang S, Kohn H. 7-N-(mercaptoalkyl)mitomycins: implications of cyclization for drug function. Journal of the American Chemical Society. 124: 4666-77. PMID 11971715 DOI: 10.1021/Ja0124313 |
0.625 |
|
| 2001 |
Na Y, Li VS, Nakanishi Y, Bastow KF, Kohn H. Synthesis, DNA cross-linking activity, and cytotoxicity of dimeric mitomycins. Journal of Medicinal Chemistry. 44: 3453-62. PMID 11585450 DOI: 10.1021/Jm010090Y |
0.516 |
|
| 2001 |
Vincent F, Srinivasan J, Santillán A, Widger WR, Kohn H. C(5)-C(5a)-modified bicyclomycins: synthesis, structure, and biochemical and biological properties. The Journal of Organic Chemistry. 66: 2251-64. PMID 11281764 DOI: 10.1021/Jo0013150 |
0.355 |
|
| 2001 |
Na Y, Kohn H. Quinone-cyclized porfiromycins Heterocycles. 55: 1347-1363. DOI: 10.3987/Com-01-9215 |
0.567 |
|
| 2000 |
Vincent F, Openshaw M, Trautwein M, Gaskell SJ, Kohn H, Widger WR. Rho transcription factor: symmetry and binding of bicyclomycin. Biochemistry. 39: 9077-83. PMID 10924100 DOI: 10.1021/Bi000504+ |
0.317 |
|
| 2000 |
Vincent F, Widger WR, Openshaw M, Gaskell SJ, Kohn H. 5a-formylbicyclomycin: studies on the bicyclomycin-Rho interaction. Biochemistry. 39: 9067-76. PMID 10924099 DOI: 10.1021/Bi000503H |
0.366 |
|
| 2000 |
Wang C, Kohn H. Formation of aromatic rings through enamine annulation Organic Letters. 2: 1773-5. PMID 10880223 DOI: 10.1021/Ol000093P |
0.348 |
|
| 2000 |
Li VS, Reed M, Zheng Y, Kohn H, Tang M. C5 cytosine methylation at CpG sites enhances sequence selectivity of mitomycin C-DNA bonding. Biochemistry. 39: 2612-8. PMID 10704210 DOI: 10.1021/Bi991307H |
0.303 |
|
| 1999 |
Andurkar SV, Stables JP, Kohn H. The anticonvulsant activities of N-benzyl 3-methoxypropionamides. Bioorganic & Medicinal Chemistry. 7: 2381-9. PMID 10632047 DOI: 10.1016/S0968-0896(99)00186-8 |
0.395 |
|
| 1999 |
Wang S, Kohn H. Studies on the mode of action of mitomycin C(7) aminoethylene disulfides (BMS-181174 and KW-2149): reactivity of 7-N-(mercaptoethyl)mitomycin C. Journal of Medicinal Chemistry. 42: 788-90. PMID 10072677 DOI: 10.1021/Jm9806796 |
0.324 |
|
| 1998 |
Riba I, Gaskell SJ, Cho H, Widger WR, Kohn H. Evidence for the location of bicyclomycin binding to the Escherichia coli transcription termination factor Rho. The Journal of Biological Chemistry. 273: 34033-41. PMID 9852059 DOI: 10.1074/Jbc.273.51.34033 |
0.349 |
|
| 1997 |
Huh N, Kogan TP, Kohn H. Synthesis of N-substituted 10-des(carbamoyloxy)-10-azidomitomycins Synthesis. 921-924. DOI: 10.1055/S-1997-1297 |
0.332 |
|
| 1997 |
Cho H, Park HG, Zhang X, Riba I, Gaskell SJ, Widger WR, Kohn H. Design, syntheses, and evaluations of bicyclomycin-based rho inactivators Journal of Organic Chemistry. 62: 5432-5440. DOI: 10.1021/Jo970575N |
0.374 |
|
| 1996 |
Santillán A, Park Hg, Zhang X, Lee OS, Widger WR, Kohn H. Role of the [4.2.2] Bicyclic Unit in Bicyclomycin: Synthesis, Structure, Chemical, Biochemical, and Biological Properties. The Journal of Organic Chemistry. 61: 7756-7763. PMID 11667731 DOI: 10.1021/Jo961003Q |
0.423 |
|
| 1996 |
Park Hg, Zhang X, Widger WR, Kohn H. Role of the C(1) Triol Group in Bicyclomycin: Synthesis and Biochemical and Biological Properties. The Journal of Organic Chemistry. 61: 7750-7755. PMID 11667730 DOI: 10.1021/Jo961002Y |
0.37 |
|
| 1996 |
Choi D, Stables JP, Kohn H. The anticonvulsant activities of functionalized N-benzyl 2-acetamidoacetamides. The importance of the 2-acetamido substituent Bioorganic and Medicinal Chemistry. 4: 2105-2114. PMID 9022975 DOI: 10.1016/S0968-0896(96)00225-8 |
0.389 |
|
| 1996 |
Huh N, Rege AA, Yoo B, Kogan TP, Kohn H. Design, synthesis, and evaluation of mitomycin-tethered phosphorothioate oligodeoxynucleotides Bioconjugate Chemistry. 7: 659-669. PMID 8950485 DOI: 10.1021/Bc960060N |
0.388 |
|
| 1996 |
Magyar A, Zhang X, Kohn H, Widger WR. The antibiotic bicyclomycin affects the secondary RNA binding site of Escherichia coli transcription termination factor Rho Journal of Biological Chemistry. 271: 25369-25374. PMID 8810302 DOI: 10.1074/Jbc.271.41.25369 |
0.325 |
|
| 1996 |
Choi D, Stables JP, Kohn H. Synthesis and anticonvulsant activities of N-benzyl-2-acetamidopropionamide derivatives Journal of Medicinal Chemistry. 39: 1907-1916. PMID 8627614 DOI: 10.1021/Jm9508705 |
0.394 |
|
| 1996 |
Wang S, Kohn H. Mitomycin betaines: Synthesis, structure, and solvolytic reactivity Journal of Organic Chemistry. 61: 9202-9206. DOI: 10.1021/Jo961378B |
0.34 |
|
| 1996 |
Kohn H, Wang S. Studies on the mechanism of activation of C(7) ethylenediamine substituted mitomycins. Relevance to the proposed mode of action of BMY-25067 and KW-2149 Tetrahedron Letters. 37: 2337-2340. DOI: 10.1016/0040-4039(96)00279-1 |
0.358 |
|
| 1995 |
Park Hg, Zhang X, Moon Hs, Zwiefka A, Cox K, Gaskell SJ, Widger WR, Kohn H. Bicyclomycin and Dihydrobicyclomycin Inhibition Kinetics ofEscherichia colirho-Dependent Transcription Termination Factor ATPase Activity Archives of Biochemistry and Biophysics. 323: 447-454. PMID 7487110 DOI: 10.1006/Abbi.1995.0066 |
0.333 |
|
| 1994 |
Kohn H, Sawhney KN, Robertson DW, Leander JD. Anticonvulsant properties of N-substituted alpha,alpha-diamino acid derivatives. Journal of Pharmaceutical Sciences. 83: 689-91. PMID 8071822 DOI: 10.1002/Jps.2600830519 |
0.324 |
|
| 1994 |
Bardel P, Bolanos A, Kohn H. Synthesis and anticonvulsant activities of alpha-acetamido-N-benzylacetamide derivatives containing an electron-deficient alpha-heteroaromatic substituent. Journal of Medicinal Chemistry. 37: 4567-4571. PMID 7799408 DOI: 10.1021/Jm00052A017 |
0.336 |
|
| 1994 |
Zhang Z, Kohn H. The role of the C-1 triol group in bicyclomycin Journal of the Chemical Society, Chemical Communications. 1343-1344. DOI: 10.1039/C39940001343 |
0.368 |
|
| 1994 |
Zhang Z, Kohn H. Chemical, biochemical, and biological studies on select C(1) triol modified bicyclomycins Journal of the American Chemical Society. 116: 9815-9826. DOI: 10.1021/Ja00101A001 |
0.312 |
|
| 1994 |
Park HG, Vela MA, Kohn H. Synthesis and reactivity of bicyclomycin C(3′) amines Journal of the American Chemical Society. 116: 471-478. DOI: 10.1021/Ja00081A006 |
0.396 |
|
| 1992 |
Han I, Russell DJ, Kohn H. Studies on the mechanism of mitomycin C(1) electrophilic transformations: structure-reactivity relationships The Journal of Organic Chemistry. 57: 1799-1807. DOI: 10.1021/Jo00032A037 |
0.32 |
|
| 1992 |
Schiltz P, Kohn H. Sodium dithionite-mediated mitomycin C reductive activation processes Tetrahedron Letters. 33: 4709-4712. DOI: 10.1016/S0040-4039(00)61265-0 |
0.329 |
|
| 1991 |
Hong YP, Kohn H. Studies on the use of chromium dichlorate for the reductive activation of Mitomycin C Journal of the American Chemical Society. 113: 4634-4644. DOI: 10.1021/Ja00012A036 |
0.334 |
|
| 1990 |
Lee C‐, Kohn H. Anticonvulsant Properties of 3-Oxo- and 3-Imino-4-Substituted 1,2,5-Thiadiazolidine 1,1-Dioxides Journal of Pharmaceutical Sciences. 79: 716-718. PMID 2231335 DOI: 10.1002/Jps.2600790813 |
0.344 |
|
| 1990 |
Kohn H, J. Russell D. Development of a Hydrazine-mediated System for the Reductive Activation of Mitomycin C Heterocycles. 31: 223. DOI: 10.3987/Com-89-5270 |
0.348 |
|
| 1990 |
Lee CH, Kohn H. Intra- and intermolecular .alpha.-sulfamidoalkylation reactions The Journal of Organic Chemistry. 55: 6098-6104. DOI: 10.1021/Jo00312A013 |
0.354 |
|
| 1989 |
Sawhney KN, Kohn H. Mitomycin C analogues with a substituted hydrazine at position 7. Synthesis, spectral properties, and biological activity. Journal of Medicinal Chemistry. 32: 248-252. PMID 2909738 DOI: 10.1021/Jm00121A044 |
0.375 |
|
| 1988 |
Kohn H, Conley JD, Leander JD. Marked stereospecificity in a new class of anticonvulsants. Brain Research. 457: 371-5. PMID 3219563 DOI: 10.1016/0006-8993(88)90709-3 |
0.312 |
|
| 1988 |
Kohn H, Abuzar S, Korp JD, Zektzer AS, Martin GE. Structural studies of bicyclomycin Journal of Heterocyclic Chemistry. 25: 1511-1517. DOI: 10.1002/Jhet.5570250548 |
0.326 |
|
| 1987 |
Conley JD, Kohn H. Functionalized DL-amino acid derivatives. Potent new agents for the treatment of epilepsy. Journal of Medicinal Chemistry. 30: 567-574. PMID 3820228 DOI: 10.1021/Jm00386A021 |
0.362 |
|
| 1987 |
Kohn H, Zein N, Lin XQ, Ding JQ, Kadish KM. Mechanistic studies on the mode of reaction of mitomycin C under catalytic and electrochemical reductive conditions Journal of the American Chemical Society. 109: 1833-1840. DOI: 10.1021/Ja00240A038 |
0.327 |
|
| 1985 |
Cortes S, Liao ZK, Watson D, Kohn H. Effect of structural modification of the hydantoin ring on anticonvulsant activity. Journal of Medicinal Chemistry. 28: 601-606. PMID 3989820 DOI: 10.1021/Jm50001A012 |
0.364 |
|
| 1985 |
Liao ZK, Kohn H. Synthesis of spiroimidazolidin-2-ones via intramolecular N-carbamoyliminium ion cyclization reactions Journal of Organic Chemistry. 50: 1884-1888. DOI: 10.1021/Jo00211A020 |
0.326 |
|
| 1985 |
Cortes S, Liao Z, Watson D, Kohn H. Additions and Corrections - Effect of Structural Modification of the Hydantoin Ring on Anticonvulsant Activity Journal of Medicinal Chemistry. 28: 1965-1965. DOI: 10.1021/Jm00150A604 |
0.311 |
|
| 1985 |
Cortes S, Liao Z-, Watson D, Kohn H. Effect Of Structural Modification Of The Hydantoin Ring On Anticonvulsant Activity Cheminform. 16. DOI: 10.1002/Chin.198534214 |
0.311 |
|
| 1985 |
Bean M, Kohn H. Studies on the reaction of mitomycin C with potassium thiobenzoate under reductive conditions The Journal of Organic Chemistry. 50: 293-298. DOI: 10.1002/Chin.198525374 |
0.744 |
|
| 1983 |
Bean M, Kohn H. Studies on the reaction of mitomycin C with potassium ethyl monothiocarbonate under reductive conditions The Journal of Organic Chemistry. 48: 5033-5041. DOI: 10.1002/Chin.198427181 |
0.746 |
|
| 1983 |
Hornemann U, Iguchi K, Keller PJ, Vu HM, Kozlowski JF, Kohn H. Reactions of mitomycin C with potassium ethyl xanthate in neutral aqueous solution The Journal of Organic Chemistry. 48: 5026-5033. DOI: 10.1002/Chin.198427180 |
0.316 |
|
| 1981 |
Kohn H, Bean MB, von Rohrscheidt C, Willcott MR, Warnhoff EW. Participation in the formation of iodo ureas from 3-buten-1-ol derivatives. A reinvestigation1 1 Alfred P. Sloan Fellow, 1977-1981. Camille and Henry Dreyfus Teacher-Scholar Grant Recipient, 1977-1982. Tetrahedron. 37: 3195-3201. DOI: 10.1016/S0040-4020(01)98853-2 |
0.714 |
|
| 1981 |
Flaster H, Kohn H. Syntheses and spectral properties of 2-Thiobiotin and biotin derivatives Journal of Heterocyclic Chemistry. 18: 1425-1436. DOI: 10.1002/Jhet.5570180730 |
0.307 |
|
| 1978 |
Arceneaux JH, Kohn H, Steenberg ML, Buckley JP. Syntheses and pharmacological activity of N-acyl-substituted imidazolidinethiones and thioimidazolines. Journal of Pharmaceutical Sciences. 67: 600-2. PMID 641789 DOI: 10.1002/Jps.2600670506 |
0.368 |
|
| 1978 |
Kohn H, Charumilind P, Gopichand Y. Studies of the reaction of thiocarbonyl-containing compounds with ketenes The Journal of Organic Chemistry. 43: 4961-4965. DOI: 10.1002/Chin.197918249 |
0.315 |
|
| 1977 |
Kohn H, Kohn BA, Steenberg ML, Buckley JP. Syntheses and pharmacological activity of substituted imidazolidinethiones and thioimidazolines Journal of Medicinal Chemistry. 20: 158-160. PMID 833815 DOI: 10.1021/Jm00211A034 |
0.3 |
|
| 1977 |
Kohn H, Arceneaux JH. Thermolysis of N-acyl substituted 2-allylthioimidazolines. Evidence for a [3,3] sigmatropic rearrangement The Journal of Organic Chemistry. 42: 2339-2341. DOI: 10.1002/Chin.197742178 |
0.326 |
|
| 1977 |
Arceneaux JH, Kohn H, Steenberg ML, Buckley JP. Syntheses And Pharmacological Activity Of N-Acyl-Substituted Imidazolidinethiones And Thioimidazolines Cheminform. 8. DOI: 10.1002/Chin.197721214 |
0.371 |
|
| 1977 |
Kohn H, Davis RE. Syntheses and chemistry of N-acyl substituted dihydroimidazo[2,1-b]thiazolium salts Journal of Organic Chemistry. 42: 72-77. DOI: 10.1002/Chin.197720253 |
0.313 |
|
| 1976 |
Breslow R, Kohn H, Siegel B. Methylated cyclodextrin and a cyclodextrin polymer as catalysts in selective anisole chlorination Tetrahedron Letters. 17: 1645-1646. DOI: 10.1016/S0040-4039(00)92912-5 |
0.432 |
|
| 1972 |
Kohn H, Benkovic SJ, Olofson RA. Dependence of mechanism on pH for deuterium-hydrogen exchange in 1-methyltetrazole-5-d. Transition metal ion catalysis of a deprotonation process. Journal of the American Chemical Society. 94: 5759-65. PMID 5053862 DOI: 10.1021/Ja00771A037 |
0.501 |
|
| 1972 |
Kohn H, Olofson RA. 1,4-Dimethyl-1,4-dihydro-1,2,4,5-tetrazine and its N-alkyl salt. Synthesis, structure, and chemistry The Journal of Organic Chemistry. 37: 3504-3509. DOI: 10.1021/jo00795a024 |
0.589 |
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| Show low-probability matches. |
