| Year |
Citation |
Score |
| 2024 |
d'Orchymont F, Narvaez A, Raymond R, Sachdev P, Charil A, Krause S, Vasdev N. In vitro evaluation of PET radiotracers for imaging synaptic density, the acetylcholine transporter, AMPA-tarp-γ8 and muscarinic M4 receptors in Alzheimer's disease. American Journal of Nuclear Medicine and Molecular Imaging. 14: 1-12. PMID 38500748 |
0.35 |
|
| 2024 |
Pees A, Tong J, Birudaraju S, Munot YS, Liang SH, Saturnino Guarino D, Mach R, Mathis CA, Vasdev N. Development of Pyridothiophene Compounds for PET Imaging of α-Synuclein. Chemistry (Weinheim An Der Bergstrasse, Germany). e202303921. PMID 38354298 DOI: 10.1002/chem.202303921 |
0.331 |
|
| 2023 |
Desmond KL, Lindberg A, Garcia A, Tong J, Harkness MB, Dobrota E, Smart K, Uribe C, Meyer JH, Houle S, Strafella AP, Li S, Huang Y, Vasdev N. First-in-Human PET Imaging of [F]SDM-4MP3: A Cautionary Tale. Molecular Imaging. 2023: 8826977. PMID 37719326 DOI: 10.1155/2023/8826977 |
0.434 |
|
| 2023 |
Graham TJA, Lindberg A, Tong J, Stehouwer JS, Vasdev N, Mach RH, Mathis CA. Discovery and Subsequent Characterization of Potent 4R-Tauopathy Positron Emission Tomography Radiotracers. Journal of Medicinal Chemistry. PMID 37487189 DOI: 10.1021/acs.jmedchem.3c00775 |
0.328 |
|
| 2023 |
Smart K, Zheng MQ, Holden D, Felchner Z, Zhang L, Han Y, Ropchan J, Carson RE, Vasdev N, Huang Y. In Vivo Imaging and Kinetic Modeling of Novel Glycogen Synthase Kinase-3 Radiotracers [C]OCM-44 and [F]OCM-50 in Non-Human Primates. Pharmaceuticals (Basel, Switzerland). 16. PMID 37259346 DOI: 10.3390/ph16020194 |
0.349 |
|
| 2023 |
Lindberg A, Chassé M, Varlow C, Pees A, Vasdev N. Strategies for designing novel PET radiotracers to cross the blood brain barrier. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 36815704 DOI: 10.1002/jlcr.4019 |
0.31 |
|
| 2022 |
Boyle AJ, Murrell E, Tong J, Schifani C, Narvaez A, Wuest M, West F, Wuest F, Vasdev N. PET Imaging of Fructose Metabolism in a Rodent Model of Neuroinflammation with 6-[F]fluoro-6-deoxy-D-fructose. Molecules (Basel, Switzerland). 27. PMID 36500626 DOI: 10.3390/molecules27238529 |
0.414 |
|
| 2021 |
Ismailani US, Buchler A, Farber G, Pekošak A, Farber E, MacMullin N, Suuronen EJ, Vasdev N, Beanlands RSB, de Kemp RA, Rotstein BH. Cardiac Sympathetic Positron Emission Tomography Imaging with -[F]Fluorobenzylguanidine is Sensitive to Uptake-1 in Rats. Acs Chemical Neuroscience. 12: 4350-4360. PMID 34714061 DOI: 10.1021/acschemneuro.1c00575 |
0.373 |
|
| 2021 |
Pees A, Vosjan MJWD, Vasdev N, Windhorst AD, Vugts DJ. Fluorine-18 labelled Ruppert-Prakash reagent ([F]MeSiCF) for the synthesis of F-trifluoromethylated compounds. Chemical Communications (Cambridge, England). 57: 5286-5289. PMID 33942818 DOI: 10.1039/d1cc01789f |
0.433 |
|
| 2021 |
Varlow C, Mossine AV, Bernard-Gauthier V, Scott PJH, Vasdev N. Radiofluorination of oxazole-carboxamides for preclinical PET neuroimaging of GSK-3. Journal of Fluorine Chemistry. 245. PMID 33840834 DOI: 10.1016/j.jfluchem.2021.109760 |
0.446 |
|
| 2021 |
Narayanaswami V, Tong J, Schifani C, Bloomfield PM, Dahl K, Vasdev N. Preclinical Evaluation of TSPO and MAO-B PET Radiotracers in an LPS Model of Neuroinflammation. Pet Clinics. 16: 233-247. PMID 33648665 DOI: 10.1016/j.cpet.2020.12.003 |
0.314 |
|
| 2021 |
Zhang L, Hu K, Shao T, Hou L, Zhang S, Ye W, Josephson L, Meyer JH, Zhang MR, Vasdev N, Wang J, Xu H, Wang L, Liang SH. Recent developments on PET radiotracers for TSPO and their applications in neuroimaging. Acta Pharmaceutica Sinica. B. 11: 373-393. PMID 33643818 DOI: 10.1016/J.Apsb.2020.08.006 |
0.375 |
|
| 2020 |
Dahl K, Turner T, Vasdev N. Radiosynthesis of a Bruton's Tyrosine Kinase Inhibitor, [ C]Tolebrutinib, via Palladium-NiXantphos-Mediated Carbonylation. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 32726870 DOI: 10.1002/Jlcr.3872 |
0.37 |
|
| 2020 |
Murrell E, Pham JM, Sowa AR, Brooks AF, Kilbourn MR, Scott PJH, Vasdev N. Classics in Neuroimaging: Development of Positron Emission Tomography Tracers for Imaging the GABAergic Pathway. Acs Chemical Neuroscience. PMID 32578977 DOI: 10.1021/Acschemneuro.0C00343 |
0.342 |
|
| 2020 |
Varlow C, Boileau I, Wey HY, Liang SH, Vasdev N. Classics in Neuroimaging: Imaging the Endocannabinoid Pathway with PET. Acs Chemical Neuroscience. PMID 32559067 DOI: 10.1021/Acschemneuro.0C00305 |
0.374 |
|
| 2020 |
Narayanaswami V, Tong J, Fiorino F, Severino B, Sparaco R, Magli E, Giordano F, Bloomfield PM, Prabhakaran J, Mann JJ, Vasdev N, Dahl K, Kumar JSD. Synthesis, in vitro and in vivo evaluation of C-O-methylated arylpiperazines as potential serotonin 1A (5-HT) receptor antagonist radiotracers. Ejnmmi Radiopharmacy and Chemistry. 5: 13. PMID 32430632 DOI: 10.1186/S41181-020-00096-8 |
0.336 |
|
| 2020 |
Varlow C, Murrell E, Holland JP, Kassenbrock A, Shannon W, Liang SH, Vasdev N, Stephenson NA. Revisiting the Radiosynthesis of [F]FPEB and Preliminary PET Imaging in a Mouse Model of Alzheimer's Disease. Molecules (Basel, Switzerland). 25. PMID 32098347 DOI: 10.3390/Molecules25040982 |
0.512 |
|
| 2019 |
Bernard-Gauthier V, Mossine AV, Knight A, Patnaik D, Zhao W, Cheng C, Krishnan HS, Xuan LL, Chindavong PS, Reis SA, Chen JM, Shao X, Stauff J, Arteaga J, Sherman PS, ... ... Vasdev N, et al. Structural Basis for Achieving GSK-3 Inhibition with High Potency, Selectivity and Brain Exposure for PET Imaging and Drug Discovery. Journal of Medicinal Chemistry. PMID 31535859 DOI: 10.1021/Acs.Jmedchem.9B01030 |
0.374 |
|
| 2019 |
Duffy IR, Boyle AJ, Vasdev N. Improving PET Imaging Acquisition and Analysis With Machine Learning: A Narrative Review With Focus on Alzheimer's Disease and Oncology. Molecular Imaging. 18: 1536012119869070. PMID 31429375 DOI: 10.1177/1536012119869070 |
0.357 |
|
| 2019 |
Dahl K, Garcia A, Stephenson NA, Vasdev N. "In-loop" F-fluorination: A proof-of-concept study. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 31083778 DOI: 10.1002/Jlcr.3751 |
0.534 |
|
| 2019 |
Dahl K, Bernard-Gauthier V, Nag S, Varnäs K, Narayanaswami V, Mahdi Moein M, Arakawa R, Vasdev N, Halldin C. Synthesis and preclinical evaluation of [F]FSL25.1188, a reversible PET radioligand for monoamine oxidase-B. Bioorganic & Medicinal Chemistry Letters. PMID 31060887 DOI: 10.1016/J.Bmcl.2019.04.040 |
0.553 |
|
| 2019 |
Liang SH, Wang L, Stephenson NA, Rotstein BH, Vasdev N. Facile F labeling of non-activated arenes via a spirocyclic iodonium(III) ylide method and its application in the synthesis of the mGluR PET radiopharmaceutical [F]FPEB. Nature Protocols. PMID 30980032 DOI: 10.1038/S41596-019-0149-3 |
0.547 |
|
| 2019 |
Chen Z, Mori W, Deng X, Cheng R, Ogasawara D, Zhang G, Schafroth MA, Dahl K, Fu H, Hatori A, Shao T, Zhang Y, Yamasaki T, Zhang X, Rong J, ... ... Vasdev N, et al. Design, synthesis and evaluation of reversible and irreversible monoacylglycerol lipase positron emission tomography (PET) tracers using a 'tail switching' strategy on a piperazinyl azetidine skeleton. Journal of Medicinal Chemistry. PMID 30829483 DOI: 10.1021/Acs.Jmedchem.8B01778 |
0.468 |
|
| 2019 |
Narayanaswami V, Drake LR, Brooks AF, Meyer JH, Houle S, Kilbourn MR, Scott PJH, Vasdev N. Classics in Neuroimaging: Development of PET Tracers for Imaging Monoamine Oxidases. Acs Chemical Neuroscience. PMID 30789704 DOI: 10.1021/Acschemneuro.9B00081 |
0.358 |
|
| 2018 |
Narayanaswami V, Dahl K, Bernard-Gauthier V, Josephson L, Cumming P, Vasdev N. Emerging PET Radiotracers and Targets for Imaging of Neuroinflammation in Neurodegenerative Diseases: Outlook Beyond TSPO. Molecular Imaging. 17: 1536012118792317. PMID 30203712 DOI: 10.1177/1536012118792317 |
0.354 |
|
| 2018 |
Varlow C, Szames D, Dahl K, Bernard-Gauthier V, Vasdev N. Fluorine-18: an untapped resource in inorganic chemistry. Chemical Communications (Cambridge, England). PMID 30191929 DOI: 10.1039/C8Cc04751K |
0.488 |
|
| 2018 |
Deng X, Rong J, Wang L, Vasdev N, Zhang L, Josephson L, Liang S. Chemistry for Positron Emission Tomography: Recent Advances in 11C-, 18F-, 13N- and 15O-labeling Reactions. Angewandte Chemie (International Ed. in English). PMID 30054961 DOI: 10.1002/Anie.201805501 |
0.469 |
|
| 2018 |
Cheng R, Mori W, Ma L, Alhouayek M, Hatori A, Zhang Y, Ogasawara D, Yuan G, Chen Z, Zhang X, Shi H, Yamasaki T, Xie L, Kumata K, Fujinaga M, ... ... Vasdev N, et al. In vitro and in vivo evaluation ofC-labeled azetidine-carboxylates for imaging monoacylglycerol lipase by PET imaging studies. Journal of Medicinal Chemistry. PMID 29481079 DOI: 10.1021/Acs.Jmedchem.7B01400 |
0.379 |
|
| 2018 |
Krishnan HS, Bernard-Gauthier V, Placzek MS, Dahl K, Narayanaswami V, Livni E, Chen Z, Yang J, Collier TL, Ran C, Hooker JM, Liang SH, Vasdev N. A metal protein-attenuating compound for PET neuroimaging: Synthesis and preclinical evaluation of [11C]PBT2. Molecular Pharmaceutics. PMID 29298483 DOI: 10.1021/Acs.Molpharmaceut.7B00936 |
0.377 |
|
| 2017 |
Collier TL, Liang SH, Mann JJ, Vasdev N, Kumar JSD. Microfluidic radiosynthesis of [F]FEMPT, a high affinity PET radiotracer for imaging serotonin receptors. Beilstein Journal of Organic Chemistry. 13: 2922-2927. PMID 29564020 DOI: 10.3762/Bjoc.13.285 |
0.468 |
|
| 2017 |
Bernard-Gauthier V, Lepage M, Waengler B, Bailey JA, Liang SH, Perrin D, Vasdev N, Schirrmacher R. Recent advances in fluorine-18 radiochemistry: Focus on B-18F, Si-18F, Al-18F and C-18F radiofluorination via spirocyclic iodonium ylides. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 29284673 DOI: 10.2967/Jnumed.117.197095 |
0.539 |
|
| 2017 |
Cumming P, Burgher B, Patkar O, Breakspear M, Vasdev N, Thomas P, Liu GJ, Banati R. Sifting through the surfeit of neuroinflammation tracers. Journal of Cerebral Blood Flow and Metabolism : Official Journal of the International Society of Cerebral Blood Flow and Metabolism. 271678X17748786. PMID 29256293 DOI: 10.1177/0271678X17748786 |
0.372 |
|
| 2017 |
Bernard-Gauthier V, Collier TL, Liang SH, Vasdev N. Discovery of PET radiopharmaceuticals at the academia-industry interface. Drug Discovery Today. Technologies. 25: 19-26. PMID 29233263 DOI: 10.1016/J.Ddtec.2017.09.001 |
0.378 |
|
| 2017 |
Collier TL, Maresca KP, Normandin MD, Richardson P, McCarthy TJ, Liang SH, Waterhouse RN, Vasdev N. Brain Penetration of the ROS1/ALK Inhibitor Lorlatinib Confirmed by PET. Molecular Imaging. 16: 1536012117736669. PMID 29067878 DOI: 10.1177/1536012117736669 |
0.388 |
|
| 2017 |
Makaretz SJ, Quimby M, Collins J, Makris N, McGinnis S, Schultz A, Vasdev N, Johnson KA, Dickerson BC. Flortaucipir tau PET imaging in semantic variant primary progressive aphasia. Journal of Neurology, Neurosurgery, and Psychiatry. PMID 28986472 DOI: 10.1136/Jnnp-2017-316409 |
0.418 |
|
| 2017 |
Lin SF, Bois F, Holden D, Nabulsi N, Pracitto R, Gao H, Kapinos M, Teng JK, Shirali A, Ropchan J, Carson RE, Elmore CS, Vasdev N, Huang Y. The Search for a Subtype-Selective PET Imaging Agent for the GABAA Receptor Complex: Evaluation of the Radiotracer [(11)C]ADO in Nonhuman Primates. Molecular Imaging. 16: 1536012117731258. PMID 28929924 DOI: 10.1177/1536012117731258 |
0.361 |
|
| 2017 |
Kanthan M, Cumming P, Hooker JM, Vasdev N. Classics in Neuroimaging: Imaging the Dopaminergic Pathway with PET. Acs Chemical Neuroscience. PMID 28719177 DOI: 10.1021/Acschemneuro.7B00252 |
0.369 |
|
| 2017 |
Krishnan H, Ma L, Vasdev N, Liang S. ¹⁸F-Labeling of Sensitive Biomolecules for Positron Emission Tomography. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28704575 DOI: 10.1002/Chem.201701581 |
0.503 |
|
| 2017 |
Dahl K, Collier TL, Chang R, Zhang X, Sadovski O, Liang SH, Vasdev N. "In-Loop" [(11) C]CO2 -Fixation: Prototype and Proof-of-Concept. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 28600835 DOI: 10.1002/Jlcr.3528 |
0.317 |
|
| 2017 |
Collier TL, Normandin MD, Stephenson NA, Livni E, Liang SH, Wooten DW, Esfahani SA, Stabin MG, Mahmood U, Chen J, Wang W, Maresca K, Waterhouse RN, El Fakhri G, Richardson P, ... Vasdev N, et al. Synthesis and preliminary PET imaging of (11)C and (18)F isotopologues of the ROS1/ALK inhibitor lorlatinib. Nature Communications. 8: 15761. PMID 28594000 DOI: 10.1038/Ncomms15761 |
0.454 |
|
| 2017 |
Vasdev N, Alavi A. Novel PET Radiotracers with Potential Clinical Applications. Pet Clinics. 12: xi-xii. PMID 28576174 DOI: 10.1016/J.Cpet.2017.04.002 |
0.348 |
|
| 2017 |
Wang L, Cheng R, Fujinaga M, Yang J, Zhang Y, Hatori A, Kumata K, Yang J, Vasdev N, Du Y, Ran C, Zhang MR, Liang SH. A Facile Radiolabeling of [(18)F]FDPA via Spirocyclic Iodonium Ylides: Preliminary PET Imaging Studies in Preclinical Models of Neuroinflammation. Journal of Medicinal Chemistry. PMID 28530834 DOI: 10.1021/Acs.Jmedchem.7B00432 |
0.533 |
|
| 2017 |
Hu K, Patnaik D, Collier TL, Lee KN, Gao H, Swoyer MR, Rotstein BH, Krishnan HS, Liang SH, Wang J, Yan Z, Hooker JM, Vasdev N, Haggarty SJ, Ngai MY. Development of [(18)F]Maleimide-Based Glycogen Synthase Kinase-3β Ligands for Positron Emission Tomography Imaging. Acs Medicinal Chemistry Letters. 8: 287-292. PMID 28337318 DOI: 10.1021/Acsmedchemlett.6B00405 |
0.438 |
|
| 2017 |
Xia C, Makaretz SJ, Caso C, McGinnis S, Gomperts SN, Sepulcre J, Gomez-Isla T, Hyman BT, Schultz A, Vasdev N, Johnson KA, Dickerson BC. Association of In Vivo [18F]AV-1451 Tau PET Imaging Results With Cortical Atrophy and Symptoms in Typical and Atypical Alzheimer Disease. Jama Neurology. PMID 28241163 DOI: 10.1001/Jamaneurol.2016.5755 |
0.351 |
|
| 2017 |
Collier TL, Yokell DL, Livni E, Rice PA, Celen S, Serdons K, Neelamegam R, Bormans G, Harris D, Walji A, Hostetler ED, Bennacef I, Vasdev N. cGMP Production of the Radiopharmaceutical [(18) F]MK-6240 for PET imaging of Human Neurofibrillary Tangles. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 28185305 DOI: 10.1002/Jlcr.3496 |
0.541 |
|
| 2017 |
Khotavivattana T, Calderwood S, Verhoog S, Pfeifer L, Preshlock S, Vasdev N, Collier TL, Gouverneur V. Synthesis and Reactivity of (18)F-Labeled α,α-Difluoro-α-(aryloxy)acetic Acids. Organic Letters. PMID 28085289 DOI: 10.1021/Acs.Orglett.6B03730 |
0.464 |
|
| 2016 |
Yuan G, Wang F, Stephenson NA, Wang L, Rotstein BH, Vasdev N, Tang P, Liang SH. Metal-free (18)F-labeling of aryl-CF2H via nucleophilic radiofluorination and oxidative C-H activation. Chemical Communications (Cambridge, England). PMID 27917423 DOI: 10.1039/C6Cc07913J |
0.397 |
|
| 2016 |
Wooten D, Guehl NJ, Verwer EE, Shoup TM, Yokell DL, Zubcevik N, Vasdev N, Zafonte RD, Johnson KA, El Fakhri G, Normandin MD. Pharmacokinetic evaluation of the tau PET radiotracer [18F]T807 ([18F]AV-1451) in human subjects. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 27660144 DOI: 10.2967/Jnumed.115.170910 |
0.493 |
|
| 2016 |
Rotstein BH, Placzek MS, Krishnan HS, Pekošak A, Collier TL, Wang C, Liang SH, Burstein ES, Hooker JM, Vasdev N. Preclinical PET Neuroimaging of [11C]Bexarotene. Molecular Imaging. 15. PMID 27553293 DOI: 10.1177/1536012116663054 |
0.396 |
|
| 2016 |
Yuan G, Jones GB, Vasdev N, Liang SH. Radiosynthesis and preliminary PET evaluation of (18)F-labeled 2-(1-(3-fluorophenyl)-2-oxo-5-(pyrimidin-2-yl)-1,2-dihydropyridin-3-yl)benzonitrile for imaging AMPA receptors. Bioorganic & Medicinal Chemistry Letters. PMID 27546294 DOI: 10.1016/J.Bmcl.2016.07.078 |
0.562 |
|
| 2016 |
Rotstein BH, Wang L, Liu RY, Patteson J, Kwan EE, Vasdev N, Liang SH. Mechanistic Studies and Radiofluorination of Structurally Diverse Pharmaceuticals with Spirocyclic Iodonium(III) Ylides. Chemical Science. 7: 4407-4417. PMID 27540460 DOI: 10.1039/C6Sc00197A |
0.516 |
|
| 2016 |
Shi H, Braun A, Wang L, Liang SH, Vasdev N, Ritter T. Synthesis of (18) F-Difluoromethylarenes from Aryl (Pseudo) Halides. Angewandte Chemie (International Ed. in English). PMID 27491349 DOI: 10.1002/Anie.201604106 |
0.53 |
|
| 2016 |
Liang SH, Chen JM, Normandin MD, Chang JS, Chang GC, Taylor CK, Trapa P, Plummer MS, Para KS, Conn EL, Lopresti-Morrow L, Lanyon LF, Cook JM, Richter KE, Nolan CE, ... ... Vasdev N, et al. Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging. Angewandte Chemie (International Ed. in English). PMID 27355874 DOI: 10.1002/Anie.201603797 |
0.355 |
|
| 2016 |
Wang L, Mori W, Cheng R, Yui J, Hatori A, Ma L, Zhang Y, Rotstein BH, Fujinaga M, Shimoda Y, Yamasaki T, Xie L, Nagai Y, Minamimoto T, Higuchi M, ... Vasdev N, et al. Synthesis and Preclinical Evaluation of Sulfonamido-based [(11)C-Carbonyl]-Carbamates and Ureas for Imaging Monoacylglycerol Lipase. Theranostics. 6: 1145-59. PMID 27279908 DOI: 10.7150/Thno.15257 |
0.396 |
|
| 2016 |
Rotstein BH, Liang SH, Placzek MS, Hooker JM, Gee AD, Dollé F, Wilson AA, Vasdev N. (11)C[double bond, length as m-dash]O bonds made easily for positron emission tomography radiopharmaceuticals. Chemical Society Reviews. PMID 27276357 DOI: 10.1039/C6Cs00310A |
0.35 |
|
| 2016 |
Kassenbrock A, Vasdev N, Liang SH. Selected PET Radioligands for Ion Channel Linked Neuroreceptor Imaging: Focus on GABA, NMDA and nACh Receptors. Current Topics in Medicinal Chemistry. PMID 26975506 DOI: 10.2174/1568026616666160315142457 |
0.363 |
|
| 2015 |
Boros E, Bowen AM, Josephson L, Vasdev N, Holland JP. Chelate-free metal ion binding and heat-induced radiolabeling of iron oxide nanoparticles. Chemical Science. 6: 225-236. PMID 28553472 DOI: 10.1039/C4Sc02778G |
0.315 |
|
| 2015 |
Calderwood S, Collier TL, Gouverneur V, Liang SH, Vasdev N. Synthesis of (18)F-Arenes from Spirocyclic Iodonium(III) Ylides via Continuous-Flow Microfluidics. Journal of Fluorine Chemistry. 178: 249-253. PMID 27512233 DOI: 10.1016/J.Jfluchem.2015.08.006 |
0.51 |
|
| 2015 |
Liang SH, Vasdev N. Total Radiosynthesis: Thinking outside "the box". Australian Journal of Chemistry. 68: 1319-1328. PMID 27512156 DOI: 10.1071/Ch15406 |
0.473 |
|
| 2015 |
Wang L, Yui J, Wang Q, Zhang Y, Mori W, Shimoda Y, Fujinaga M, Kumata K, Yamasak TI, Hatori A, Rotstein BH, Collier TL, Ran C, Vasdev N, Zhang MR, et al. Synthesis and preliminary PET imaging studies of a FAAH radiotracer ([(11)C]MPPO) based on α-ketoheterocyclic scaffold. Acs Chemical Neuroscience. PMID 26505525 DOI: 10.1021/Acschemneuro.5B00248 |
0.386 |
|
| 2015 |
Marquié M, Normandin MD, Vanderburg CR, Costantino IM, Bien EA, Rycyna LG, Klunk WE, Mathis CA, Ikonomovic MD, Debnath ML, Vasdev N, Dickerson BC, Gomperts SN, Growdon JH, Johnson KA, et al. Validating novel tau positron emission tomography tracer [F-18]-AV-1451 (T807) on postmortem brain tissue. Annals of Neurology. PMID 26344059 DOI: 10.1002/Ana.24517 |
0.43 |
|
| 2015 |
Jacobson O, Weiss I, Wang L, Wang Z, Yang X, Dewhurst A, Ma Y, Zhu G, Niu G, Kiesewetter DO, Vasdev N, Liang S, Chen X. 18F-labeled Single-Stranded DNA Aptamer for PET Imaging of Protein Tyrosine Kinase-7 Expression. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 26315836 DOI: 10.2967/Jnumed.115.160960 |
0.368 |
|
| 2015 |
Wang L, Jacobson O, Avdic D, Rotstein BH, Weiss ID, Collier L, Chen X, Vasdev N, Liang SH. Ortho-Stabilized (18) F-Azido Click Agents and their Application in PET Imaging with Single-Stranded DNA Aptamers. Angewandte Chemie (International Ed. in English). PMID 26308650 DOI: 10.1002/Anie.201505927 |
0.51 |
|
| 2015 |
Rotstein BH, Liang SH, Belov VV, Livni E, Levine DB, Bonab AA, Papisov MI, Perlis RH, Vasdev N. Practical Radiosynthesis and Preclinical Neuroimaging of [11C]isradipine, a Calcium Channel Antagonist. Molecules (Basel, Switzerland). 20: 9550-9. PMID 26016546 DOI: 10.3390/Molecules20069550 |
0.35 |
|
| 2015 |
Liang SH, Holland JP, Stephenson NA, Kassenbrock A, Rotstein BH, Daignault CP, Lewis R, Collier L, Hooker JM, Vasdev N. PET neuroimaging studies of [(18)F]CABS13 in a double transgenic mouse model of Alzheimer's disease and nonhuman primates. Acs Chemical Neuroscience. 6: 535-41. PMID 25776827 DOI: 10.1021/Acschemneuro.5B00055 |
0.526 |
|
| 2015 |
Stephenson NA, Holland JP, Kassenbrock A, Yokell DL, Livni E, Liang SH, Vasdev N. Iodonium ylide-mediated radiofluorination of 18F-FPEB and validation for human use. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 56: 489-92. PMID 25655630 DOI: 10.2967/Jnumed.114.151332 |
0.523 |
|
| 2015 |
Heidari P, Deng F, Esfahani SA, Leece AK, Shoup TM, Vasdev N, Mahmood U. Pharmacodynamic imaging guides dosing of a selective estrogen receptor degrader. Clinical Cancer Research : An Official Journal of the American Association For Cancer Research. 21: 1340-7. PMID 25609068 DOI: 10.1158/1078-0432.Ccr-14-1178 |
0.354 |
|
| 2015 |
Hicks JW, Sadovski O, Parkes J, Houle S, Hay BA, Carter RL, Wilson AA, Vasdev N. Radiosynthesis and ex vivo evaluation of [(18)F]-(S)-3-(6-(3-fluoropropoxy)benzo[d]isoxazol-3-yl)-5-(methoxymethyl)oxazolidin-2-one for imaging MAO-B with PET. Bioorganic & Medicinal Chemistry Letters. 25: 288-91. PMID 25488845 DOI: 10.1016/J.Bmcl.2014.11.048 |
0.457 |
|
| 2015 |
Shoup TM, Bonab AA, Wilson AA, Vasdev N. Synthesis and preclinical evaluation of [¹⁸F]FCHC for neuroimaging of fatty acid amide hydrolase. Molecular Imaging and Biology : Mib : the Official Publication of the Academy of Molecular Imaging. 17: 257-63. PMID 25273322 DOI: 10.1007/S11307-014-0789-1 |
0.478 |
|
| 2015 |
Dickerson B, Makaretz S, Caso C, Stepanovic M, McGinnis SM, Xia C, Schultz AP, Vasdev N, Johnson KA. Imaging tau pathology in vivo in ftld with [18F] T807 PET Alzheimers & Dementia. 11: 545. DOI: 10.1016/J.Jalz.2015.06.690 |
0.482 |
|
| 2014 |
Liang SH, Yokell DL, Normandin MD, Rice PA, Jackson RN, Shoup TM, Brady TJ, Fakhri GE, Collier TL, Vasdev N. First Human Use of a Radiopharmaceutical Prepared by Continuous-Flow Microfluidic Radiofluorination: Proof of Concept with the Tau Imaging Agent [(18)F]T807. Molecular Imaging. 13: 7290201400025. PMID 28650281 DOI: 10.2310/7290.2014.00025 |
0.388 |
|
| 2014 |
Liang SH, Yokell DL, Jackson RN, Rice PA, Callahan R, Johnson KA, Alagille D, Tamagnan G, Collier TL, Vasdev N. Microfluidic continuous-flow radiosynthesis of [(18)F]FPEB suitable for human PET imaging. Medchemcomm. 5: 432-435. PMID 25431646 DOI: 10.1039/C3Md00335C |
0.509 |
|
| 2014 |
Liang SH, Yokell DL, Normandin MD, Rice PA, Jackson RN, Shoup TM, Brady TJ, El Fakhri G, Collier TL, Vasdev N. First human use of a radiopharmaceutical prepared by continuous-flow microfluidic radiofluorination: proof of concept with the tau imaging agent [18F]T807. Molecular Imaging. 13. PMID 25248283 DOI: 10.2310/7290.2014.00025 |
0.486 |
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| 2014 |
Rotstein BH, Stephenson NA, Vasdev N, Liang SH. Spirocyclic hypervalent iodine(III)-mediated radiofluorination of non-activated and hindered aromatics. Nature Communications. 5: 4365. PMID 25007318 DOI: 10.1038/Ncomms5365 |
0.497 |
|
| 2014 |
Rotstein BH, Wey HY, Shoup TM, Wilson AA, Liang SH, Hooker JM, Vasdev N. PET imaging of fatty acid amide hydrolase with [(18)F]DOPP in nonhuman primates. Molecular Pharmaceutics. 11: 3832-8. PMID 25004399 DOI: 10.1021/Mp500316H |
0.543 |
|
| 2014 |
Hicks JW, Parkes J, Tong J, Houle S, Vasdev N, Wilson AA. Radiosynthesis and ex vivo evaluation of [(11)C-carbonyl]carbamate- and urea-based monoacylglycerol lipase inhibitors. Nuclear Medicine and Biology. 41: 688-94. PMID 24969632 DOI: 10.1016/J.Nucmedbio.2014.05.001 |
0.349 |
|
| 2014 |
Rotstein BH, Hooker JM, Woo J, Collier TL, Brady TJ, Liang SH, Vasdev N. Synthesis of [(11)C]Bexarotene by Cu-Mediated [(11)C]Carbon Dioxide Fixation and Preliminary PET Imaging. Acs Medicinal Chemistry Letters. 5: 668-72. PMID 24944741 DOI: 10.1021/Ml500065Q |
0.365 |
|
| 2014 |
Rusjan PM, Wilson AA, Miler L, Fan I, Mizrahi R, Houle S, Vasdev N, Meyer JH. Kinetic modeling of the monoamine oxidase B radioligand [¹¹C]SL25.1188 in human brain with high-resolution positron emission tomography. Journal of Cerebral Blood Flow and Metabolism : Official Journal of the International Society of Cerebral Blood Flow and Metabolism. 34: 883-9. PMID 24517979 DOI: 10.1038/Jcbfm.2014.34 |
0.302 |
|
| 2014 |
Holland JP, Liang SH, Rotstein BH, Collier TL, Stephenson NA, Greguric I, Vasdev N. Alternative approaches for PET radiotracer development in Alzheimer's disease: imaging beyond plaque. Journal of Labelled Compounds & Radiopharmaceuticals. 57: 323-31. PMID 24327420 DOI: 10.1002/Jlcr.3158 |
0.376 |
|
| 2014 |
Shoup TM, McCauley JP, Lee DF, Chen R, Normandin MD, Bonab AA, El Fakhri G, Vasdev N. Synthesis of the dopamine D2/D3 receptor agonist (+)-PHNO via supercritical fluid chromatography: Preliminary PET imaging study with [3-11C]-(+)PHNO Tetrahedron Letters. 55: 682-685. DOI: 10.1016/J.Tetlet.2013.11.113 |
0.373 |
|
| 2014 |
Johnson KA, Schultz A, Becker A, Hyman B, Rentz D, Sepulcre J, Vasdev N, Sperling R, Brady T. Tau Pet Using F18-T807: Initial Experience In Normal Elderly And Ad Dementia Alzheimers & Dementia. 10: 242. DOI: 10.1016/J.Jalz.2014.04.365 |
0.414 |
|
| 2014 |
Liang SH, Vasdev N. C(sp3)-18F-Bindungsbildung durch übergangsmetallvermittelte [18F]Fluorierung Angewandte Chemie. 126: 11600-11602. DOI: 10.1002/Ange.201407065 |
0.505 |
|
| 2013 |
Shoup TM, Yokell DL, Rice PA, Jackson RN, Livni E, Johnson KA, Brady TJ, Vasdev N. A concise radiosynthesis of the tau radiopharmaceutical, [(18) F]T807. Journal of Labelled Compounds & Radiopharmaceuticals. 56: 736-40. PMID 24339014 DOI: 10.1002/Jlcr.3098 |
0.501 |
|
| 2013 |
Liang SH, Collier TL, Rotstein BH, Lewis R, Steck M, Vasdev N. Rapid microfluidic flow hydrogenation for reduction or deprotection of 18F-labeled compounds. Chemical Communications (Cambridge, England). 49: 8755-7. PMID 23948863 DOI: 10.1039/C3Cc45166F |
0.468 |
|
| 2013 |
Hicks JW, Parkes J, Sadovski O, Tong J, Houle S, Vasdev N, Wilson AA. Synthesis and preclinical evaluation of [11C-carbonyl]PF-04457845 for neuroimaging of fatty acid amide hydrolase. Nuclear Medicine and Biology. 40: 740-6. PMID 23731552 DOI: 10.1016/J.Nucmedbio.2013.04.008 |
0.347 |
|
| 2013 |
Sadovski O, Hicks JW, Parkes J, Raymond R, Nobrega J, Houle S, Cipriano M, Fowler CJ, Vasdev N, Wilson AA. Development and characterization of a promising fluorine-18 labelled radiopharmaceutical for in vivo imaging of fatty acid amide hydrolase. Bioorganic & Medicinal Chemistry. 21: 4351-7. PMID 23712084 DOI: 10.1016/J.Bmc.2013.04.077 |
0.522 |
|
| 2013 |
Rotstein BH, Liang SH, Holland JP, Collier TL, Hooker JM, Wilson AA, Vasdev N. 11CO2 fixation: a renaissance in PET radiochemistry. Chemical Communications (Cambridge, England). 49: 5621-9. PMID 23673726 DOI: 10.1039/C3Cc42236D |
0.324 |
|
| 2013 |
Vasdev N, Green DE, Vines DC, McLarty K, McCormick PN, Moran MD, Houle S, Wilson AA, Reilly RM. Positron-emission tomography imaging of the TSPO with [18F]FEPPA in a preclinical breast cancer model Cancer Biotherapy and Radiopharmaceuticals. 28: 254-259. PMID 23350894 DOI: 10.1089/Cbr.2012.1196 |
0.716 |
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| 2013 |
Wilson AA, Hicks JW, Sadovski O, Parkes J, Tong J, Houle S, Fowler CJ, Vasdev N. Radiosynthesis and evaluation of [¹¹C-carbonyl]-labeled carbamates as fatty acid amide hydrolase radiotracers for positron emission tomography. Journal of Medicinal Chemistry. 56: 201-9. PMID 23214511 DOI: 10.1021/Jm301492Y |
0.394 |
|
| 2012 |
Carroll L, Perumal M, Vasdev N, Robins E, Aboagye EO. Radiosynthesis and in vivo tumor uptake of 2-deoxy-2-[(18)F]fluoro-myo-inositol. Bioorganic & Medicinal Chemistry Letters. 22: 6148-50. PMID 22944120 DOI: 10.1016/J.Bmcl.2012.08.022 |
0.523 |
|
| 2012 |
Holland JP, Cumming P, Vasdev N. PET of signal transduction pathways in cancer. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 53: 1333-6. PMID 22879078 DOI: 10.2967/Jnumed.112.105387 |
0.32 |
|
| 2012 |
Moran MD, Wilson AA, Elmore CS, Parkes J, Ng A, Sadovski O, Graff A, Daskalakis ZJ, Houle S, Chapdelaine MJ, Vasdev N. Development of new carbon-11 labelled radiotracers for imaging GABA A- and GABA B-benzodiazepine receptors Bioorganic and Medicinal Chemistry. 20: 4482-4488. PMID 22717238 DOI: 10.1016/J.Bmc.2012.05.046 |
0.646 |
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| 2012 |
Hicks JW, Wilson AA, Rubie EA, Woodgett JR, Houle S, Vasdev N. Towards the preparation of radiolabeled 1-aryl-3-benzyl ureas: Radiosynthesis of [(11)C-carbonyl] AR-A014418 by [(11)C]CO(2) fixation. Bioorganic & Medicinal Chemistry Letters. 22: 2099-101. PMID 22321216 DOI: 10.1016/J.Bmcl.2011.12.139 |
0.306 |
|
| 2012 |
Vasdev N, Cao P, Oosten EMV, Wilson AA, Houle S, Hao G, Sun X, Slavine NV, Alhasan M, Antich PP, Bonte FJ, Kulkarni PV. Synthesis and PET imaging studies of [18F]2-fluoroquinolin-8-ol ([18F]CABS13) in transgenic mouse models of Alzheimer's disease Medchemcomm. 3: 1228-1230. DOI: 10.1039/C2Md20075A |
0.53 |
|
| 2012 |
Kulkarni P, Alhasan M, Slavine N, Chiguru S, Hao G, Vasdev N, Thomas P, Bonte F, Sun X. Assessment of disease progression in Alzheimer's transgenic mice by PET imaging with F-18 quinoline Alzheimers & Dementia. 8: 155. DOI: 10.1016/J.Jalz.2012.05.417 |
0.328 |
|
| 2011 |
McLarty K, Moran MD, Scollard DA, Chan C, Sabha N, Mukherjee J, Guha A, McLaurin J, Nitz M, Houle S, Wilson AA, Reilly RM, Vasdev N. Comparisons of [18F]-1-deoxy-1-fluoro-scyllo-inositol with [18F]-FDG for PET imaging of inflammation, breast and brain cancer xenografts in athymic mice. Nuclear Medicine and Biology. 38: 953-9. PMID 21982567 DOI: 10.1016/J.Nucmedbio.2011.02.017 |
0.731 |
|
| 2011 |
Vasdev N, Sadovski O, Moran MD, Parkes J, Meyer JH, Houle S, Wilson AA. Development of new radiopharmaceuticals for imaging monoamine oxidase B. Nuclear Medicine and Biology. 38: 933-43. PMID 21982565 DOI: 10.1016/J.Nucmedbio.2011.03.003 |
0.699 |
|
| 2011 |
Vasdev N, Dorff PN, O'Neil JP, Chin FT, Hanrahan S, VanBrocklin HF. Metabolic stability of 6,7-dialkoxy-4-(2-, 3- and 4-[18F]fluoroanilino)quinazolines, potential EGFR imaging probes. Bioorganic & Medicinal Chemistry. 19: 2959-65. PMID 21478021 DOI: 10.1016/J.Bmc.2011.03.032 |
0.487 |
|
| 2011 |
Wilson AA, Garcia A, Parkes J, Houle S, Tong J, Vasdev N. [11C]CURB: Evaluation of a novel radiotracer for imaging fatty acid amide hydrolase by positron emission tomography. Nuclear Medicine and Biology. 38: 247-53. PMID 21315280 DOI: 10.1016/J.Nucmedbio.2010.08.001 |
0.372 |
|
| 2011 |
Wilson AA, Garcia A, Houle S, Sadovski O, Vasdev N. Synthesis and application of isocyanates radiolabeled with carbon-11. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 259-64. PMID 21207622 DOI: 10.1002/Chem.201002345 |
0.395 |
|
| 2011 |
Van Oosten EM, Gerken M, Hazendonk P, Shank R, Houle S, Wilson AA, Vasdev N. Regioselective ring opening of 2-methylaziridine derivatives with 18F- and 19F-fluoride Tetrahedron Letters. 52: 4114-4116. DOI: 10.1016/J.Tetlet.2011.05.139 |
0.501 |
|
| 2011 |
Kulkarni P, Arora V, Chiguru S, Hao G, Gupta A, Slavine N, Qu B, Vasdev N, Sun X, Bennett M, Antich P, Bonte F. PET imaging of Alzheimer's transgenic mice at an early age with F-18 quinoline Alzheimers & Dementia. 7. DOI: 10.1016/J.Jalz.2011.05.021 |
0.449 |
|
| 2011 |
Vasdev N, Sadovski O, Garcia A, Dollé F, Meyer JH, Houle S, Wilson AA. Radiosynthesis of [11C]SL25.1188 via [11C]CO2 fixation for imaging monoamine oxidase B Journal of Labelled Compounds and Radiopharmaceuticals. 54: 678-680. DOI: 10.1002/Jlcr.1908 |
0.314 |
|
| 2010 |
Vasdev N, Moran MD, Tuononen HM, Chirakal R, Suontamo RJ, Bain AD, Schrobilgen GJ. NMR spectroscopic evidence for the intermediacy of XeF(3)(-) in XeF(2)/F(-) exchange, attempted syntheses and thermochemistry of XeF(3)(-) salts, and theoretical studies of the XeF(3)(-) anion. Inorganic Chemistry. 49: 8997-9004. PMID 20799721 DOI: 10.1021/Ic101275M |
0.785 |
|
| 2010 |
Wilson AA, Garcia A, Houle S, Vasdev N. Direct fixation of [(11)C]-CO(2) by amines: formation of [(11)C-carbonyl]-methylcarbamates. Organic & Biomolecular Chemistry. 8: 428-32. PMID 20066280 DOI: 10.1039/B916419G |
0.345 |
|
| 2010 |
Wilson AA, Garcia A, Houle S, Vasdev N. [11C]-URB694 for FAAH PET imaging: A novel radiotracer for a new target Neuroimage. 52: S24. DOI: 10.1016/J.Neuroimage.2010.04.208 |
0.387 |
|
| 2010 |
Vasdev N, Sadovski O, Parkes J, Moran MD, Meyer JH, Houle S, Wilson AA. Development of New PET radiopharmaceuticals for imaging monoamine oxidase-B Neuroimage. 52. DOI: 10.1016/J.Neuroimage.2010.04.201 |
0.363 |
|
| 2010 |
Kulkarni PV, Vasdev N, Arora V, Hao G, Long M, Slavine N, Qu B, Sun X, Bennett M, Antich PP, Bonte FJ. PET imaging of Alzheimer's disease (AD) transgenic mice with F-18 labeled 8-hydroxy quinoline Alzheimers & Dementia. 6. DOI: 10.1016/J.Jalz.2010.05.017 |
0.441 |
|
| 2010 |
Vasdev N, Chirakal R, Schrobilgen GJ, Nahmias C. ChemInform Abstract: Selectivity of Elemental Fluorine Towards L-Tyrosine and L-α-Methyltyrosine in Acidic Media and the Syntheses of Their [18F]3-Fluoro and [18F]3,5-Difluoro Derivatives. Cheminform. 33: no-no. DOI: 10.1002/CHIN.200220158 |
0.729 |
|
| 2009 |
Vasdev N, Chio J, van Oosten EM, Nitz M, McLaurin J, Vines DC, Houle S, Reilly RM, Wilson AA. Synthesis and preliminary biological evaluations of [18F]-1-deoxy-1-fluoro-scyllo-inositol. Chemical Communications (Cambridge, England). 5527-9. PMID 19753345 DOI: 10.1039/B913317H |
0.508 |
|
| 2009 |
van Oosten EM, Wilson AA, Stephenson KA, Mamo DC, Pollock BG, Mulsant BH, Yudin AK, Houle S, Vasdev N. An improved radiosynthesis of the muscarinic M2 radiopharmaceutical, [18F]FP-TZTP. Applied Radiation and Isotopes : Including Data, Instrumentation and Methods For Use in Agriculture, Industry and Medicine. 67: 611-6. PMID 19186063 DOI: 10.1016/J.Apradiso.2008.12.015 |
0.531 |
|
| 2009 |
Vasdev N, van Oosten EM, Stephenson KA, Zadikian N, Yudin AK, Lough AJ, Houle S, Wilson AA. [18F]Fluoroamines via ring-opening of N-Cbz-2-methylaziridine with [18F]-fluoride Tetrahedron Letters. 50: 544-547. DOI: 10.1016/J.Tetlet.2008.11.074 |
0.527 |
|
| 2008 |
Stephenson KA, van Oosten EM, Wilson AA, Meyer JH, Houle S, Vasdev N. Synthesis and preliminary evaluation of [(18)F]-fluoro-(2S)-Exaprolol for imaging cerebral beta-adrenergic receptors with PET. Neurochemistry International. 53: 173-9. PMID 18675864 DOI: 10.1016/J.Neuint.2008.06.013 |
0.472 |
|
| 2008 |
Stephenson KA, Wilson AA, Meyer JH, Houle S, Vasdev N. Facile radiosynthesis of fluorine-18 labeled beta-blockers. Synthesis, radiolabeling, and ex vivo biodistribution of [18F]-(2S and 2R)-1-(1-fluoropropan-2-ylamino)-3-(m-tolyloxy)propan-2-ol. Journal of Medicinal Chemistry. 51: 5093-100. PMID 18656910 DOI: 10.1021/Jm800227H |
0.452 |
|
| 2008 |
Wilson AA, Garcia A, Parkes J, McCormick P, Stephenson KA, Houle S, Vasdev N. Radiosynthesis and initial evaluation of [18F]-FEPPA for PET imaging of peripheral benzodiazepine receptors. Nuclear Medicine and Biology. 35: 305-14. PMID 18355686 DOI: 10.1016/J.Nucmedbio.2007.12.009 |
0.523 |
|
| 2008 |
Vasdev N, LaRonde FJ, Woodgett JR, Garcia A, Rubie EA, Meyer JH, Houle S, Wilson AA. Rationally designed PKA inhibitors for positron emission tomography: Synthesis and cerebral biodistribution of N-(2-(4-bromocinnamylamino)ethyl)-N-[11C]methyl-isoquinoline-5-sulfonamide. Bioorganic & Medicinal Chemistry. 16: 5277-84. PMID 18346896 DOI: 10.1016/J.Bmc.2008.03.013 |
0.341 |
|
| 2008 |
Vasdev N, Stephenson KA, Oosten EMv, Meyer JH, Houle S, Wilson AA. Recent advances towards imaging cerebral β-adrenergic receptors with PET Neuroimage. 41. DOI: 10.1016/J.Neuroimage.2008.04.165 |
0.336 |
|
| 2007 |
Vasdev N, Seeman P, Garcia A, Stableford WT, Nobrega JN, Houle S, Wilson AA. Syntheses and in vitro evaluation of fluorinated naphthoxazines as dopamine D2/D3 receptor agonists: radiosynthesis, ex vivo biodistribution and autoradiography of [(18)F]F-PHNO. Nuclear Medicine and Biology. 34: 195-203. PMID 17307127 DOI: 10.1016/J.Nucmedbio.2006.11.001 |
0.415 |
|
| 2006 |
Vasdev N, Natesan S, Galineau L, Garcia A, Stableford WT, McCormick P, Seeman P, Houle S, Wilson AA. Radiosynthesis, ex vivo and in vivo evaluation of [11C]preclamol as a partial dopamine D2 agonist radioligand for positron emission tomography. Synapse (New York, N.Y.). 60: 314-8. PMID 16786538 DOI: 10.1002/Syn.20304 |
0.337 |
|
| 2005 |
Vasdev N, Garcia A, Stableford WT, Young AB, Meyer JH, Houle S, Wilson AA. Synthesis and ex vivo evaluation of carbon-11 labelled N-(4-methoxybenzyl)-N'-(5-nitro-1,3-thiazol-2-yl)urea ([11C]AR-A014418): a radiolabelled glycogen synthase kinase-3beta specific inhibitor for PET studies. Bioorganic & Medicinal Chemistry Letters. 15: 5270-3. PMID 16202587 DOI: 10.1016/J.Bmcl.2005.08.037 |
0.336 |
|
| 2005 |
Vasdev N, Dorff PN, Gibbs AR, Nandanan E, Reid LM, O'Neil JP, VanBrocklin HF. Synthesis of 6-acrylamido-4-(2-[18F]fluoroanilino)quinazoline: A prospective irreversible EGFR binding probe Journal of Labelled Compounds and Radiopharmaceuticals. 48: 109-115. DOI: 10.1002/Jlcr.903 |
0.502 |
|
| 2003 |
Vasdev N, Chirakal R, Ashique R, Schrobilgen GJ, Gulenchyn K. Syntheses of [18F]5-fluoro-3-nitro-L-tyrosine Journal of Fluorine Chemistry. 121: 9-14. DOI: 10.1016/S0022-1139(02)00334-2 |
0.787 |
|
| 2002 |
Vasdev N, Pointner BE, Chirakal R, Schrobilgen GJ. On the preparation of fluorine-18 labelled XeF(2) and chemical exchange between fluoride ion and XeF(2). Journal of the American Chemical Society. 124: 12863-8. PMID 12392433 DOI: 10.1021/Ja020604Y |
0.771 |
|
| 2002 |
Vasdev N, Pointner BE, Chirakal R, Schrobilgen GJ. On the preparation of fluorine-18 labelled XeF2 and chemical exchange between fluoride ion and XeF2 Journal of the American Chemical Society. 124: 12863-12868. DOI: 10.1021/ja020604y |
0.675 |
|
| 2002 |
Chirakal R, Vasdev N, Asselin MC, Schrobilgen GJ, Nahmias C. The effect of aromatic fluorine substitution in L-DOPA on the in vivo behaviour of [18F]2-, [18F]5- and [18F]6-fluoro-L-DOPA in the human brain Journal of Fluorine Chemistry. 115: 33-39. DOI: 10.1016/S0022-1139(02)00025-8 |
0.782 |
|
| 2001 |
Vasdev N, Chirakal R, Schrobilgen GJ, Nahmias C. Selectivity of elemental fluorine towards L-tyrosine and L-α-methyltyrosine in acidic media and the syntheses of their [18F]3-fluoro and [18F]3,5-difluoro derivatives Journal of Fluorine Chemistry. 111: 17-25. DOI: 10.1016/S0022-1139(01)00406-7 |
0.767 |
|
| 2001 |
Chirakal R, Vasdev N, Schrobilgen GJ, Amano S, Nahmias C. A comparative study of the in vivo behaviour of [18F] 2-, 5- and 6-fluoro-L-dopa in the human brain Journal of Labelled Compounds and Radiopharmaceuticals. 44: S219-S221. DOI: 10.1002/Jlcr.2580440176 |
0.764 |
|
| 2001 |
Vasdev N, Chirakal R, Schrobilgen GJ, Nahmias C. Selectivity of [18F]F2 towards L-α-methyltyrosine and L-tyrosine: A radiochemical and NMR spectroscopic study Journal of Labelled Compounds and Radiopharmaceuticals. 44: S863-S865. DOI: 10.1002/Jlcr.25804401303 |
0.773 |
|
| 1999 |
Chirakal R, Vasdev N, Schrobilgen GJ, Nahmias C. Radiochemical and NMR spectroscopic investigation of the solvent effect on the electrophilic elemental fluorination of L-DOPA: Synthesis of [ 18F ]5-fluoro-L-DOPA Journal of Fluorine Chemistry. 99: 87-94. DOI: 10.1016/S0022-1139(99)00123-2 |
0.739 |
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