Year |
Citation |
Score |
2023 |
Ferrins L, Buskes MJ, Kapteyn MM, Engels HN, Enos SE, Lu C, Klug DM, Singh B, Quotadamo A, Bachovchin K, Tear WF, Spaulding AE, Forbes KC, Bag S, Rivers M, et al. Corrigendum: Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes. Frontiers in Microbiology. 14: 1304196. PMID 37954236 DOI: 10.3389/fmicb.2023.1304196 |
0.728 |
|
2023 |
Ferrins L, Buskes MJ, Kapteyn MM, Engels HN, Enos SE, Lu C, Klug DM, Singh B, Quotadamo A, Bachovchin K, Tear WF, Spaulding AE, Forbes KC, Bag S, Rivers M, et al. Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes. Frontiers in Microbiology. 14: 1149145. PMID 37234530 DOI: 10.3389/fmicb.2023.1149145 |
0.745 |
|
2023 |
Singh B, Sharma A, Gunaganti N, Rivers M, Gadekar PK, Greene B, Chichioco M, Sanz-Rodriguez CE, Fu C, LeBlanc C, Burchfield E, Sharif N, Hoffman B, Kumar G, Purmal A, et al. Chemical Optimization of CBL0137 for Human African Trypanosomiasis Lead Drug Discovery. Journal of Medicinal Chemistry. PMID 36695630 DOI: 10.1021/acs.jmedchem.2c01767 |
0.609 |
|
2022 |
Sanz-Rodriguez CE, Hoffman B, Guyett PJ, Purmal A, Singh B, Pollastri M, Mensa-Wilmot K. . Molecular Pharmacology. PMID 35605992 DOI: 10.1124/molpharm.121.000430 |
0.569 |
|
2020 |
Singh B, Diaz-Gonzalez R, Ceballos-Perez G, Rojas-Barros DI, Gunaganti N, Gillingwater K, Martinez-Martinez MS, Manzano P, Navarro M, Pollastri MP. Medicinal Chemistry Optimization of a Diaminopurine Chemotype: Toward a Lead for Inhibitors. Journal of Medicinal Chemistry. PMID 32786222 DOI: 10.1021/Acs.Jmedchem.0C01017 |
0.646 |
|
2020 |
Buskes MJ, Clements M, Bachovchin KA, Jalani HB, Leonard A, Bag S, Klug DM, Singh B, Campbell RF, Sciotti RJ, El-Sakkary N, Caffrey CR, Pollastri MP, Ferrins L. Structure-Bioactivity Relationships of Lapatinib Derived Analogs against . Acs Medicinal Chemistry Letters. 11: 258-265. PMID 32184954 DOI: 10.1021/Acsmedchemlett.9B00455 |
0.765 |
|
2020 |
Singh B, Bernatchez JA, McCall LI, Calvet CM, Ackermann J, Souza JM, Thomas D, Silva EM, Bachovchin KA, Klug DM, Jalani HB, Bag S, Buskes MJ, Leed SE, Roncal NE, et al. Scaffold and Parasite Hopping: Discovery of New Protozoal Proliferation Inhibitors. Acs Medicinal Chemistry Letters. 11: 249-257. PMID 32184953 DOI: 10.1021/Acsmedchemlett.9B00453 |
0.768 |
|
2018 |
Bachovchin KA, Sharma A, Bag S, Klug DM, Schneider KM, Singh B, Jalani HB, Buskes M, Mehta N, Tanghe S, Momper JD, Sciotti RJ, Rodriguez A, Mensa-Wilmot K, Pollastri MP, et al. Improvement of Aqueous Solubility of Lapatinib-derived Analogs: Identification of a Quinolinimine as a Lead for Human African Trypanosomiasis Drug Development. Journal of Medicinal Chemistry. PMID 30565932 DOI: 10.1021/Acs.Jmedchem.8B01365 |
0.768 |
|
2018 |
Woodring JL, Behera R, Sharma A, Wiedeman J, Patel G, Singh B, Guyett P, Amata E, Erath J, Roncal N, Penn E, Leed SE, Rodriguez A, Sciotti RJ, Mensa-Wilmot K, et al. Series of Alkynyl-Substituted Thienopyrimidines as Inhibitors of Protozoan Parasite Proliferation. Acs Medicinal Chemistry Letters. 9: 996-1001. PMID 30344906 DOI: 10.1021/Acsmedchemlett.8B00245 |
0.764 |
|
2016 |
Kumar A, Singh B, Mahajan G, Sharma PR, Bharate SB, Mintoo MJ, Mondhe DM. A novel colchicine-based microtubule inhibitor exhibits potent antitumor activity by inducing mitochondrial mediated apoptosis in MIA PaCa-2 pancreatic cancer cells. Tumour Biology : the Journal of the International Society For Oncodevelopmental Biology and Medicine. PMID 27449046 DOI: 10.1007/S13277-016-5160-5 |
0.643 |
|
2016 |
Gupta S, Kaul S, Singh B, Vishwakarma RA, Dhar MK. Production of Gentisyl Alcohol from Phoma herbarum Endophytic in Curcuma longa L. and Its Antagonistic Activity Towards Leaf Spot Pathogen Colletotrichum gloeosporioides. Applied Biochemistry and Biotechnology. PMID 27288000 DOI: 10.1007/S12010-016-2154-0 |
0.5 |
|
2016 |
Bharate SB, Singh B, Kachler S, Oliveira A, Kumar V, Bharate SS, Vishwakarma RA, Klotz KN, Gutiérrez-de-Terán H. Discovery of 7-(prolinol-N-yl)-2-phenylamino-thiazolo[5,4-d]pyrimidines as novel non-nucleoside partial agonists for the A2A adenosine receptor: Prediction from molecular modeling. Journal of Medicinal Chemistry. PMID 27227326 DOI: 10.1021/Acs.Jmedchem.6B00552 |
0.695 |
|
2016 |
Kumar A, Singh B, Sharma PR, Bharate SB, Saxena AK, Mondhe DM. A novel microtubule depolymerizing colchicine analogue triggers apoptosis and autophagy in HCT-116 colon cancer cells. Cell Biochemistry and Function. 34: 69-81. PMID 26919061 DOI: 10.1002/Cbf.3166 |
0.651 |
|
2015 |
Singh B, Sinha N, Sharma R, Parekh N. Non Surgical Correction of Mandibular Deviation and Neuromuscular Coordination after Two years of Mandibular Guidance Therapy: A Case Report. Journal of Clinical and Diagnostic Research : Jcdr. 9: ZD07-9. PMID 26673016 DOI: 10.7860/JCDR/2015/16309.6730 |
0.316 |
|
2015 |
Singh B, Jain SK, Bharate SB, Kushwaha M, Gupta AP, Vishwakarma RA. Simultaneous Quantification of Five Bioactive Flavonoids in High Altitude Plant Actinocarya tibetica by LC-ESI-MS/MS. Journal of Aoac International. 98: 907-12. PMID 26268971 DOI: 10.5740/Jaoacint.14-270 |
0.75 |
|
2015 |
Singh B, Kumar A, Joshi P, Guru SK, Kumar S, Wani ZA, Mahajan G, Hussain A, Qazi AK, Kumar A, Bharate SS, Gupta BD, Sharma PR, Hamid A, Saxena AK, et al. Colchicine derivatives with potent anticancer activity and reduced P-glycoprotein induction liability. Organic & Biomolecular Chemistry. 13: 5674-89. PMID 25895604 DOI: 10.1039/C5Ob00406C |
0.761 |
|
2014 |
Singh B, Guru SK, Sharma R, Bharate SS, Khan IA, Bhushan S, Bharate SB, Vishwakarma RA. Synthesis and anti-proliferative activities of new derivatives of embelin. Bioorganic & Medicinal Chemistry Letters. 24: 4865-70. PMID 25240254 DOI: 10.1016/J.Bmcl.2014.08.052 |
0.723 |
|
2014 |
Joshi P, Singh S, Wani A, Sharma S, Jain SK, Singh B, Gupta BD, Satti NK, Koul S, Khan IA, Kumar A, Bharate SB, Vishwakarma RA. Osthol and curcumin as inhibitors of human Pgp and multidrug efflux pumps of Staphylococcus aureus: Reversing the resistance against frontline antibacterial drugs Medchemcomm. 5: 1540-1547. DOI: 10.1039/C4Md00196F |
0.764 |
|
2013 |
Singh B, Guru SK, Kour S, Jain SK, Sharma R, Sharma PR, Singh SK, Bhushan S, Bharate SB, Vishwakarma RA. Synthesis, antiproliferative and apoptosis-inducing activity of thiazolo[5,4-d]pyrimidines. European Journal of Medicinal Chemistry. 70: 864-74. PMID 24262379 DOI: 10.1016/J.Ejmech.2013.10.039 |
0.764 |
|
2013 |
Jain SK, Pathania AS, Meena S, Sharma R, Sharma A, Singh B, Gupta BD, Bhushan S, Bharate SB, Vishwakarma RA. Semisynthesis of mallotus B from rottlerin: evaluation of cytotoxicity and apoptosis-inducing activity. Journal of Natural Products. 76: 1724-30. PMID 24041234 DOI: 10.1021/Np400433G |
0.763 |
|
2013 |
Singh B, Vishwakarma RA, Bharate SB. QSAR and pharmacophore modeling of natural and synthetic antimalarial prodiginines. Current Computer-Aided Drug Design. 9: 350-9. PMID 24010933 DOI: 10.2174/15734099113099990020 |
0.703 |
|
2013 |
Singh B, Sidiq T, Joshi P, Jain SK, Lawaniya Y, Kichlu S, Khajuria A, Vishwakarma RA, Bharate SB. Anti-inflammatory and immunomodulatory flavones from Actinocarya tibetica Benth. Natural Product Research. 27: 2227-30. PMID 23768253 DOI: 10.1080/14786419.2013.805334 |
0.753 |
|
2013 |
Bharate SB, Bharate JB, Khan SI, Tekwani BL, Jacob MR, Mudududdla R, Yadav RR, Singh B, Sharma PR, Maity S, Singh B, Khan IA, Vishwakarma RA. Discovery of 3,3'-diindolylmethanes as potent antileishmanial agents. European Journal of Medicinal Chemistry. 63: 435-43. PMID 23517732 DOI: 10.1016/J.Ejmech.2013.02.024 |
0.771 |
|
2013 |
Singh B, Parshad R, Khajuria R, Guru SK, Pathania AS, Sharma R, Chib R, Aravinda S, Gupta VK, Khan IA, Bhushan S, Bharate SB, Vishwakarma RA. Saccharonol B, a new cytotoxic methylated isocoumarin from Saccharomonospora azurea Tetrahedron Letters. 54: 6695-6699. DOI: 10.1016/J.Tetlet.2013.09.060 |
0.64 |
|
2012 |
Singh B, Nadkarni JR, Vishwakarma RA, Bharate SB, Nivsarkar M, Anandjiwala S. The hydroalcoholic extract of Cassia alata (Linn.) leaves and its major compound rhein exhibits antiallergic activity via mast cell stabilization and lipoxygenase inhibition. Journal of Ethnopharmacology. 141: 469-73. PMID 22449441 DOI: 10.1016/J.Jep.2012.03.012 |
0.63 |
|
2012 |
Bharate SB, Singh B, Vishwakarma RA. Modulation of k-Ras signaling by natural products. Current Medicinal Chemistry. 19: 2273-2291. PMID 22414109 DOI: 10.2174/092986712800229050 |
0.602 |
|
2012 |
Jain SK, Meena S, Singh B, Bharate JB, Joshi P, Singh VP, Vishwakarma RA, Bharate SB. KF/alumina catalyzed regioselective benzylation and benzoylation using solvent-free grind-stone chemistry Rsc Advances. 2: 8929. DOI: 10.1039/C2Ra21154H |
0.755 |
|
2012 |
Bharate SB, Manda S, Joshi P, Singh B, Vishwakarma RA. Total synthesis and anti-cholinesterase activity of marine-derived bis-indole alkaloid fascaplysin Medchemcomm. 3: 1098. DOI: 10.1039/C2Md20076G |
0.721 |
|
2012 |
Singh O, Usha K, Saboki E, Srivastav M, Dahuja A, Singh B. Enzymatic reactive oxygen species (ROS) scavenging system in mango varieties resistant and susceptible to malformation Scientia Horticulturae. 138: 81-89. DOI: 10.1016/J.Scienta.2011.12.031 |
0.302 |
|
2012 |
Bharate SB, Singh B, Bharate JB, Jain SK, Meena S, Vishwakarma RA. QSAR and pharmacophore modeling of N-acetyl-2-aminobenzothiazole class of phosphoinositide-3-kinase-α inhibitors Medicinal Chemistry Research. 22: 890-899. DOI: 10.1007/S00044-012-0081-3 |
0.734 |
|
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