| Grégoire Altan-Bonnet | Systems Immunology | | | | |
| Ettore Appella | | | | | |
| Omer Aras | Radiology and Nuclear Medicine | | | | |
| Joseph J. Barchi | Chemical Biology | | | | |
| Pedro J Batista | | | | | |
| Federico Bernal | Cancer Chemical Biology | | | | |
| John Albert Beutler | natural products, cancer | | 2004 | | Stuart F.J. LeGrice (collaborator) |
| Minou Bina | transcriptional control elements in human chromosomes | | 1975 | 1977 | Maxine F. Singer (post-doc) |
| Adrian Blackman | | Laboratory of Drug Discovery Research & Development | 1994 | 1994 | John Albert Beutler (research scientist) |
| Donald P Bottaro | cancer biology, cancer genetics, cell and molecular biology | Laboratory of Cellular and Molecular Biology Urologic Oncology Branch | 2003 | 1999 | Stuart A Aaronson (collaborator), W Marston Linehan (collaborator) |
| Quinton Brail | | | | | |
| George Bosworth Brown | amino acids, nucleic acids, pharmacology, carcinogens, tumors | | | | |
| Dalen Chan | | | 2019 | 2022 | Pedro J Batista (post-doc) |
| Namki Cho | | Molecular Targets Program | 2014 | 2016 | John Albert Beutler (post-doc) |
| Sarah Choyke | | Urologic Oncology Branch | 2005 | 2006 | Gagani Athauda (research assistant), Donald P Bottaro (research assistant), Benedetta Peruzzi (research assistant) |
| Maira Alves Constantino | Biophysics | | | | |
| Valeria Culotta | Cell Biology of Metals | | | 1990 | Dean H. Hamer (post-doc) |
| Marcos da Cunha | | Molecular Targets Laboratory | 2013 | 2014 | John Albert Beutler (grad student) |
| Yamini Dalal | gene regulation | | | | |
| Riccardo Dalla-Favera | Oncology, Pathology, Biochemistry | Laboratory of Tumor Cell Biology | 1978 | 1982 | Robert Charles Gallo (post-doc) |
| Sarath Parakumge Dayani | | | | | |
| Krishna Devkota | | Molecular Targets Laboratory | 2010 | 2013 | John Albert Beutler (post-doc) |
| Paul G Donlin-Asp | | | | | |
| Renata Dusi | | Molecular Targets Program | 2015 | 2015 | John Albert Beutler (grad student) |
| Amir Erez | | Immunology | 2015 | 2018 | Grégoire Altan-Bonnet (post-doc) |
| Fatma Memnune Eruҫar | | Molecular Targets Program | 2019 | | John Albert Beutler (grad student) |
| Laila Salmen Espindola | | Molecular Targets Program | 2014 | 2015 | John Albert Beutler (research scientist) |
| Christina M Fitzsimmons | chemical biology, epitranscriptomics, metabolism | Laboratory of Cell Biology | 2017 | | Pedro J Batista (post-doc) |
| Cecilia Florio | | | | | |
| Arun Ganesan | | | 2018 | | Yamini Dalal (post-doc) |
| Otto A. Gansow | Nuclear magnetic resonance | | | | |
| Harry V. Gelboin | cytochrome P450 metabolism of carcinogens and drugs | | | | |
| Jeffrey Gildersleeve | | | | | |
| Atul Goel | | | 1999 | 2001 | Ettore Appella (post-doc) |
| Michael M. Gottesman | resistance of cancer cells to anticancer drugs | | | | |
| Jesse Philip Greenstein | Production and Analysis of Optically Pure Amino Acid Stereoisomers | | | | |
| Benjamin Hoffman | | | 2006 | 2007 | Donald P Bottaro (research assistant) |
| Christine A. Hrycyna | multidrug resistance in human cancer | | 1993 | 2000 | Michael M. Gottesman (post-doc) |
| Amanda B. Hummon | transcriptome and the proteome in cancer cells | | 2005 | 2009 | Thomas Ried (post-doc) |
| Deborah R Kaye | | | 2009 | 2010 | Donald P Bottaro (post-doc) |
| Rinat Khannanov | | Molecular Targets Laboratory | 2013 | 2013 | John Albert Beutler (research scientist) |
| Young Ho Kim | | Molecular Targets Laboratory | 2004 | 2006 | John Albert Beutler (research scientist) |
| Ik-Soo Lee | | Molecular Targets Laboratory | 2007 | 2007 | John Albert Beutler (research scientist) |
| Molly M. Lee | | | | | |
| Stuart F.J. LeGrice | | | | | |
| Zhitao Li | Organic Chemistry, Molecular Biology | | | | Jeffrey Gildersleeve (post-doc) |
| Brandon M. Liu | singlet oxygen, metal-organic frameworks, synthetic organic chemistry, glycochemistry | Chemical Biology Laboratory | 2019 | | Joseph J. Barchi (research assistant) |
| Lawrence A. Loeb | mutations and human cancer | | 1962 | 1964 | Harry V. Gelboin (research assistant) |
| Judith Lunger | | | | | |
| Siddhardha Maligireddy | | Laboratory of Cell Biology | 2021 | | Pedro J Batista (research assistant) |
| Mariana Mandler | | | 2019 | | Pedro J Batista (research scientist) |
| Joseph C. Manimala | Supramolecular Chemistry | | | | Jeffrey Gildersleeve (post-doc) |
| Charles R. Maxwell | | | | | |
| Alton Meister | glutathione | | | 1947 | Jesse Philip Greenstein (research scientist) |
| H. Tai Nguyen | | Laboratory of Cell Biology | 2021 | | Pedro J Batista (research assistant) |
| Barry O'Keefe | | Laboratory of Drug Discovery Research & Development | 1994 | 1996 | John Albert Beutler (post-doc) |
| Oyindasola Omolara Oyelaran | | | | | Jeffrey Gildersleeve (post-doc) |
| Alon Oyler-Yaniv | | Immunology | 2014 | 2017 | Grégoire Altan-Bonnet (post-doc) |
| Esra Eroglu Ozkan | | Molecular Targets Laboratory | 2017 | 2018 | John Albert Beutler (research scientist) |
| Mary Pitman | | | 2015 | | Yamini Dalal (grad student) |
| Ranjala Ratnayake | | Molecular Targets Laboratory | 2007 | 2009 | John Albert Beutler (post-doc) |
| Joseph Reilly | | Urologic Oncology Branch | 2009 | 2011 | Fabiola Cecchi (research assistant) |
| Thomas Ried | genomic instability and associated gene expression changes during cancer development | | | | |
| Phillip Sanchez | | | | | Jun O. Liu (grad student) |
| Allix M. Sanders | | | 2015 | | Joel P. Schneider (post-doc) |
| Alexandra Schmiechen | | | 2017 | 2019 | Pedro J Batista (research assistant) |
| Joel P. Schneider | Biomaterial Science | | | | |
| Sarath P. Senadeera | | Molecular Targets Program | 2019 | | John Albert Beutler (post-doc) |
| Charles Sherr | | | | | George J. Todaro (post-doc) |
| Junfeng Shi | Peptide chemistry | | | 2015 | Joel P. Schneider (post-doc) |
| Haley M Simpson | | | 2009 | 2010 | Donald P Bottaro (research assistant) |
| Maxine F. Singer | RNA synthesis, the role of enzymes in DNA and RNA synthesis and metabolism, genetic recombination in defective viruses, and the structure of the DNA-protein complex called chromatin | | | | |
| MacKinzie Smith | | | | | |
| Eric R. Sterner | Heparin | | | | Jeffrey Gildersleeve (post-doc) |
| Sriram Subramaniam | Three-Dimensional Electron Microscopy at Molecular Resolution | | | | |
| Dennis J. Thiele | Molecular Biology, Biochemistry | | 1984 | 1987 | Dean H. Hamer (post-doc) |
| Mark Tischler | | Laboratory of Drug Discovery Research & Development | 1990 | 1991 | John Albert Beutler (post-doc) |
| George J. Todaro | | | | | |
| Taylor B. Updegrove | RNA; DNA; biophysics | | | | |
| Dongdong Wang | | Molecular Targets Program | 2016 | | John Albert Beutler (post-doc) |
| Sue Wickner | Molecular Chaperones | | | | |
| Li Xia | Glycobiology | | | | Jeffrey Gildersleeve (post-doc) |
| Zendra Elizabeth Zehner | Molecular Biology, Biochemistry | | 1979 | 1982 | Bruce Macdonald Paterson (post-doc) |