Brian H. Heasley, Ph.D.
Affiliations: | University of Virginia, Charlottesville, VA |
Area:
Bioorganic and Synthetic Organic ChemistryGoogle:
"Brian Heasley"Mean distance: 8.25 | S | N | B | C | P |
Parents
Sign in to add mentor| Timothy L. Macdonald | grad student | 2005 | UVA | |
| (Design, synthesis and evaluation of subtype-selective and non-hydrolyzable lysophosphatidic acid receptor agonists and antagonists.) | ||||
BETA: Related publications
See more...
Publications
|
You can help our author matching system! If you notice any publications incorrectly attributed to this author, please sign in and mark matches as correct or incorrect. |
| Yu HN, Richardson TE, Nataraja S, et al. (2014) Discovery of substituted benzamides as follicle stimulating hormone receptor allosteric modulators. Bioorganic & Medicinal Chemistry Letters. 24: 2168-72 |
| Heasley BH, Pacofsky GJ, Mamai A, et al. (2012) Synthesis and biological evaluation of antifungal derivatives of enfumafungin as orally bioavailable inhibitors of β-1,3-glucan synthase. Bioorganic & Medicinal Chemistry Letters. 22: 6811-6 |
| Heasley B. (2011) Synthesis of limonoid natural products European Journal of Organic Chemistry. 19-46 |
| Joshi EM, Heasley BH, MacDonald TL. (2009) 2-ABT-S-oxide detoxification by glutathione S-transferases A1-1, M1-1 and P1-1: Implications for toxicity associated with zileuton Xenobiotica. 39: 197-204 |
| Heasley BH, Jarosz R, Carter KM, et al. (2004) A novel series of 2-pyridyl-containing compounds as lysophosphatidic acid receptor antagonists: development of a nonhydrolyzable LPA3 receptor-selective antagonist. Bioorganic & Medicinal Chemistry Letters. 14: 4069-74 |
| Santos WL, Heasley BH, Jarosz R, et al. (2004) Synthesis and biological evaluation of phosphonic and thiophosphoric acid derivatives of lysophosphatidic acid. Bioorganic & Medicinal Chemistry Letters. 14: 3473-6 |
| Heasley BH, Jarosz R, Lynch KR, et al. (2004) Initial structure-activity relationships of lysophosphatidic acid receptor antagonists: discovery of a high-affinity LPA1/LPA3 receptor antagonist. Bioorganic & Medicinal Chemistry Letters. 14: 2735-40 |
| Joshi EM, Heasley BH, Chordia MD, et al. (2004) In Vitro Metabolism of 2-Acetylbenzothiophene: Relevance to Zileuton Hepatotoxicity Chemical Research in Toxicology. 17: 137-143 |
| Heise CE, Santos WL, Schreihofer AM, et al. (2001) Activity of 2-substituted lysophosphatidic acid (LPA) analogs at LPA receptors: discovery of a LPA1/LPA3 receptor antagonist. Molecular Pharmacology. 60: 1173-80 |