Ricardo Gallardo-Macias, Ph.D.
Affiliations: | 2014 | Yale University, New Haven, CT |
Area:
computational chemistry and molecular designGoogle:
"Ricardo Gallardo-Macias"Mean distance: 8.16 | S | N | B | C | P |
Parents
Sign in to add mentor| William L. Jorgensen | grad student | 2014 | Yale | |
| (Synthesis and Optimization of Novel Non-Nucleoside Reverse Transcriptase Inhibitors.) | ||||
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Publications
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| Rudraraju RS, Daher SS, Gallardo-Macias R, et al. (2022) KasA as a drug target: Structure-based inhibitor design. Frontiers in Cellular and Infection Microbiology. 12: 1008213 |
| Lee WG, Frey KM, Gallardo-Macias R, et al. (2015) Discovery and crystallography of bicyclic arylaminoazines as potent inhibitors of HIV-1 reverse transcriptase. Bioorganic & Medicinal Chemistry Letters. 25: 4824-7 |
| Lee WG, Frey KM, Gallardo-Macias R, et al. (2015) Discovery and crystallography of bicyclic arylaminoazines as potent inhibitors of HIV-1 reverse transcriptase Bioorganic and Medicinal Chemistry Letters |
| Lee WG, Frey KM, Gallardo-Macias R, et al. (2014) Picomolar Inhibitors of HIV-1 Reverse Transcriptase: Design and Crystallography of Naphthyl Phenyl Ethers. Acs Medicinal Chemistry Letters. 5: 1259-62 |
| Frey KM, Gray WT, Spasov KA, et al. (2014) Structure-based evaluation of C5 derivatives in the catechol diether series targeting HIV-1 reverse transcriptase. Chemical Biology & Drug Design. 83: 541-9 |
| Lee WG, Gallardo-Macias R, Frey KM, et al. (2013) Picomolar inhibitors of HIV reverse transcriptase featuring bicyclic replacement of a cyanovinylphenyl group. Journal of the American Chemical Society. 135: 16705-13 |
| Bollini M, Gallardo-Macias R, Spasov KA, et al. (2013) Optimization of benzyloxazoles as non-nucleoside inhibitors of HIV-1 reverse transcriptase to enhance Y181C potency. Bioorganic & Medicinal Chemistry Letters. 23: 1110-3 |
| Frey KM, Bollini M, Mislak AC, et al. (2012) Crystal structures of HIV-1 reverse transcriptase with picomolar inhibitors reveal key interactions for drug design. Journal of the American Chemical Society. 134: 19501-3 |
| Bollini M, Domaoal RA, Thakur VV, et al. (2011) Computationally-guided optimization of a docking hit to yield catechol diethers as potent anti-HIV agents. Journal of Medicinal Chemistry. 54: 8582-91 |