Rishi K. Jain, Ph.D.
Affiliations: | 2002 | Yale University, New Haven, CT |
Area:
chemical biologyGoogle:
"Rishi Jain"Mean distance: 8.23 | S | N | B | C | P |
Parents
Sign in to add mentor| Andrew D. Hamilton | grad student | 2002 | Yale | |
| (Protein surface recognition by synthetic receptors based on macrocyclic scaffolds: Designs and applications.) | ||||
| Jonathan A. Ellman | post-doc | 2004 | Novartis Institute for BioMedical Research | |
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Publications
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| Wang AC, Pham HT, Lipps JM, et al. (2018) Previously uncharacterized v-ATPase binding site discovered from structurally similar compounds with distinct mechanisms of action. Acs Chemical Biology |
| Thomas JR, Brittain SM, Lipps J, et al. (2017) A Photoaffinity Labeling-Based Chemoproteomics Strategy for Unbiased Target Deconvolution of Small Molecule Drug Candidates. Methods in Molecular Biology (Clifton, N.J.). 1647: 1-18 |
| Wong ML, Murphy J, Harrington E, et al. (2016) Examining the influence of specificity ligands and ATP-competitive ligands on the overall effectiveness of bivalent kinase inhibitors. Proteome Science. 15: 17 |
| Gower CM, Thomas JR, Harrington E, et al. (2016) Conversion of a Single Polypharmacological Agent into Selective Bivalent Inhibitors of Intracellular Kinase Activity. Acs Chemical Biology. 11: 121-31 |
| Carelli JD, Sethofer SG, Smith GA, et al. (2015) Ternatin and improved synthetic variants kill cancer cells by targeting the elongation factor-1A ternary complex. Elife. 4 |
| Bassilana F, Carlson A, DaSilva JA, et al. (2014) Target identification for a Hedgehog pathway inhibitor reveals the receptor GPR39. Nature Chemical Biology. 10: 343-9 |
| Jain RK, Tsou LK, Hamilton AD. (2009) Combined solid/solution phase synthesis of large surface area scaffolds derived from aminomethyl-benzoates. Tetrahedron Letters. 50: 2787-2789 |
| Miller-Moslin K, Peukert S, Jain RK, et al. (2009) 1-amino-4-benzylphthalazines as orally bioavailable smoothened antagonists with antitumor activity. Journal of Medicinal Chemistry. 52: 3954-68 |
| Peukert S, Jain RK, Geisser A, et al. (2009) Identification and structure-activity relationships of ortho-biphenyl carboxamides as potent Smoothened antagonists inhibiting the Hedgehog signaling pathway. Bioorganic & Medicinal Chemistry Letters. 19: 328-31 |
| Jecklin MC, Touboul D, Jain R, et al. (2009) Affinity classification of kinase inhibitors by mass spectrometric methods and validation using standard IC50 measurements Analytical Chemistry. 81: 408-419 |