Ganeshsingh A. Thakur

Chemistry & Chemical Biology Northeastern University, Boston, MA, United States 
Organic Chemistry
"Ganeshsingh Thakur"
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Garai S, Schaffer PC, Laprairie RB, et al. (2021) Design, synthesis, and pharmacological profiling of cannabinoid 1 receptor allosteric modulators: Preclinical efficacy of C2-group GAT211 congeners for reducing intraocular pressure. Bioorganic & Medicinal Chemistry. 50: 116421
Pismataro MC, Horenstein NA, Stokes C, et al. (2021) Stable desensitization of α nicotinic acetylcholine receptors by NS6740 requires interaction with S36 in the orthosteric agonist binding site. European Journal of Pharmacology. 905: 174179
Mizrachi T, Marsha O, Brusin K, et al. (2021) Suppression of neuroinflammation by an allosteric agonist and positive allosteric modulator of the α7 nicotinic acetylcholine receptor GAT107. Journal of Neuroinflammation. 18: 99
Garai S, Leo LM, Szczesniak AM, et al. (2021) Discovery of a Biased Allosteric Modulator for Cannabinoid 1 Receptor: Preclinical Anti-Glaucoma Efficacy. Journal of Medicinal Chemistry
Jiang S, Iliopoulos-Tsoutsouvas C, Tong F, et al. (2021) Novel Functionalized Cannabinoid Receptor Probes: Development of Exceptionally Potent Agonists. Journal of Medicinal Chemistry
McElroy DL, Roebuck AJ, Scott GA, et al. (2021) Antipsychotic potential of the type 1 cannabinoid receptor positive allosteric modulator GAT211: preclinical in vitro and in vivo studies. Psychopharmacology
Schaffer PC, Kulkarni PM, Janero DR, et al. (2020) Focused structure-activity relationship profiling around the 2-phenylindole scaffold of a cannabinoid type-1 receptor agonist-positive allosteric modulator: site-III aromatic-ring congeners with enhanced activity and solubility. Bioorganic & Medicinal Chemistry. 28: 115727
Papke RL, Garai S, Stokes C, et al. (2020) Differing activity profiles of the stereoisomers of 2,3,5,6TMP-TQS, a putative silent allosteric modulator of α7nAChR. Molecular Pharmacology
Thapa D, Cairns EA, Szczesniak AM, et al. (2020) Allosteric Cannabinoid Receptor 1 (CB1) Ligands Reduce Ocular Pain and Inflammation. Molecules (Basel, Switzerland). 25
Garai S, Kulkarni PM, Schaffer PC, et al. (2019) Application of Fluorine- And Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of CB1 Receptor Positive Allosteric Modulators. Journal of Medicinal Chemistry
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