Ad P. IJzerman
Affiliations: | Leiden University, Leiden, Netherlands |
Area:
PharmacochemistryWebsite:
https://hoogleraren.leidenuniv.nl/id/3592Google:
"Ad IJzerman"Mean distance: 14.62 | S | N | B | C | P |
Parents
Sign in to add mentor| Henk Timmerman | grad student | 1985 | VU Amsterdam | |
| (The β‐adrenoceptor complex; requirements for the interaction with its ligands) | ||||
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Publications
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| Dudley MW, Peet NP, Demeter DA, et al. (2024) Adenosine A Receptor and Ligand Molecular Modeling. Drug Development Research. 28: 237-243 |
| Jacobson KA, IJzerman AP, Linden J. (2024) 1,3-Dialkylxanthine Derivatives Having High Potency as Antagonists at Human A Adenosine Receptors. Drug Development Research. 47: 45-53 |
| Burggraaff L, van Veen A, Lam CC, et al. (2020) Annotation of Allosteric Compounds to Enhance Bioactivity Modeling for Class A GPCRs. Journal of Chemical Information and Modeling |
| Yang X, Dilweg MA, Osemwengie D, et al. (2020) Design and Pharmacological Profile of a Novel Covalent Partial Agonist for the Adenosine A Receptor. Biochemical Pharmacology. 114144 |
| Wang X, Jespers W, Bongers BJ, et al. (2020) Characterization of cancer-related somatic mutations in the adenosine A receptor. European Journal of Pharmacology. 173126 |
| Burggraaff L, Lenselink EB, Jespers W, et al. (2020) Successive Statistical and Structure-Based Modeling to Identify Chemically Novel Kinase Inhibitors. Journal of Chemical Information and Modeling |
| Ortiz Zacarías NV, van Veldhoven JPD, den Hollander LS, et al. (2019) Synthesis and pharmacological evaluation of triazolo-pyrimidinone derivatives as noncompetitive, intracellular antagonists for CC chemokine receptors 2 and 5. Journal of Medicinal Chemistry |
| Massink A, Amelia T, Karamychev A, et al. (2019) Allosteric modulation of G protein-coupled receptors by amiloride and its derivatives. Perspectives for drug discovery? Medicinal Research Reviews. 40: 683-708 |
| Bouzo-Lorenzo M, Stoddart LA, Xia L, et al. (2019) A live cell NanoBRET binding assay allows the study of ligand-binding kinetics to the adenosine A receptor. Purinergic Signalling |
| Yun Y, Chen J, Liu R, et al. (2019) Long residence time adenosine A receptor agonists produce sustained wash-resistant antilipolytic effect in rat adipocytes. Biochemical Pharmacology |