Tad Holak
Affiliations: | Biochemistry |
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Collaborators
Sign in to add collaborator| Rudrakshula MadhavaChary | collaborator | 2015-2018 | Biochemistry |
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Publications
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| Doemling A, Ricardo M, Ali A, et al. (2020) Multicomponent Peptide Stapling as a Diversity-Driven Tool for the Development of Inhibitors of Protein-Protein Interactions. Angewandte Chemie (International Ed. in English) |
| van der Vlag R, Yagiz Unver M, Felicetti T, et al. (2019) Optimized Inhibitors of MDM2 via an Attempted Protein-Templated Reductive Amination. Chemmedchem |
| Neochoritis CG, Atmaj J, Twarda-Clapa A, et al. (2019) Hitting on the move: Targeting intrinsically disordered protein states of the MDM2-p53 interaction. European Journal of Medicinal Chemistry. 182: 111588 |
| Neochoritis CG, Kazemi Miraki M, Abdelraheem EMM, et al. (2019) Design of indole- and MCR-based macrocycles as p53-MDM2 antagonists. Beilstein Journal of Organic Chemistry. 15: 513-520 |
| Estrada-Ortiz N, Neochoritis CG, Twarda-Clapa A, et al. (2017) Artificial Macrocycles as Potent p53-MDM2 Inhibitors. Acs Medicinal Chemistry Letters. 8: 1025-1030 |
| Surmiak E, Neochoritis CG, Musielak B, et al. (2016) Rational design and synthesis of 1,5-disubstituted tetrazoles as potent inhibitors of the MDM2-p53 interaction. European Journal of Medicinal Chemistry. 126: 384-407 |
| Surmiak E, Twarda-Clapa A, Zak KM, et al. (2016) A Unique Mdm2-Binding Mode of the 3-Pyrrolin-2-one- and 2-Furanone-Based Antagonists of the p53-Mdm2 Interaction. Acs Chemical Biology. 11: 3310-3318 |
| Golestanian S, Sharifi A, Popowicz GM, et al. (2015) Discovery of novel dual inhibitors against Mdm2 and Mdmx proteins by in silico approaches and binding assay. Life Sciences |
| Neochoritis CG, Wang K, Estrada-Ortiz N, et al. (2015) 2,3'-Bis(1'H-indole) heterocycles: New p53/MDM2/MDMX antagonists. Bioorganic & Medicinal Chemistry Letters |
| Boltjes A, Huang Y, van de Velde R, et al. (2014) Fragment-based library generation for the discovery of a peptidomimetic p53-Mdm4 inhibitor. Acs Combinatorial Science. 16: 393-6 |