| Year |
Citation |
Score |
| 2020 |
Gallagher WP, Beutner GL, Wadzinski TJ, Deshpande PP. Selective opening of nucleoside derived acetals to form highly functionalized vinyl ethers Tetrahedron Letters. 61: 151750. DOI: 10.1016/J.Tetlet.2020.151750 |
0.457 |
|
| 2019 |
Xiang J, Shang M, Kawamata Y, Lundberg H, Reisberg SH, Chen M, Mykhailiuk P, Beutner G, Collins MR, Davies A, Del Bel M, Gallego GM, Spangler JE, Starr J, Yang S, et al. Hindered dialkyl ether synthesis with electrogenerated carbocations. Nature. PMID 31501569 DOI: 10.1038/S41586-019-1539-Y |
0.454 |
|
| 2019 |
Fraunhoffer KJ, DelMonte AJ, Beutner GL, Bultman MS, Camacho K, Cohen B, Dixon DD, Fan Y, Fanfair D, Freitag AJ, Glace AW, Gonzalez-Bobes F, Gujjar M, Haley MW, Hickey MR, et al. Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor Organic Process Research & Development. 23: 2482-2498. DOI: 10.1021/Acs.Oprd.9B00359 |
0.33 |
|
| 2019 |
Beutner GL, Bultman MS, Cohen BM, Fan J, Marshall J, Sfouggatakis C. Follow the Silyl Cation: Insights into the Vorbrüggen Reaction Organic Process Research & Development. 23: 2050-2056. DOI: 10.1021/Acs.Oprd.9B00304 |
0.389 |
|
| 2019 |
Beutner GL, Coombs JR, Green RA, Inankur B, Lin D, Qiu J, Roberts F, Simmons EM, Wisniewski SR. Palladium-Catalyzed Amidation and Amination of (Hetero)aryl Chlorides under Homogeneous Conditions Enabled by a Soluble DBU/NaTFA Dual-Base System Organic Process Research & Development. 23: 1529-1537. DOI: 10.1021/Acs.Oprd.9B00196 |
0.43 |
|
| 2019 |
Beutner GL, Cohen BM, DelMonte AJ, Dixon DD, Fraunhoffer KJ, Glace AW, Lo E, Stevens JM, Vanyo D, Wilbert C. Revisiting the Cleavage of Evans Oxazolidinones with LiOH/H2O2 Organic Process Research & Development. 23: 1378-1385. DOI: 10.1021/Acs.Oprd.9B00124 |
0.36 |
|
| 2018 |
Stevens JM, Parra-Rivera AC, Dixon DD, Beutner GL, DelMonte AJ, Frantz DE, Janey JM, Paulson J, Talley MR. Direct Lewis Acid-Catalyzed Conversion of Enantioenriched N-Acyl Oxazolidinones to Chiral Esters, Amides, and Acids. The Journal of Organic Chemistry. PMID 30412670 DOI: 10.1021/Acs.Joc.8B02451 |
0.401 |
|
| 2018 |
Fox RJ, Cuniere NL, Bakrania L, Wei C, Strotman NA, Hay M, Fanfair D, Regens C, Beutner GL, Lawler M, Lobben P, Soumeillant MC, Cohen B, Zhu K, Skliar D, et al. C-H Arylation in the Formation of a Complex Pyrrolopyridine, the Commercial Synthesis of the Potent JAK2 Inhibitor, BMS-911543. The Journal of Organic Chemistry. PMID 30388009 DOI: 10.1021/Acs.Joc.8B02383 |
0.717 |
|
| 2018 |
Beutner GL, Young IS, Davies ML, Hickey MR, Park H, Stevens JM, Ye Q. TCFH-NMI: Direct Access to N-Acyl Imidazoliums for Challenging Amide Bond Formations. Organic Letters. PMID 29956545 DOI: 10.1021/Acs.Orglett.8B01591 |
0.333 |
|
| 2018 |
Beutner G, Carrasquillo R, Geng P, Hsiao Y, Huang EC, Janey J, Katipally K, Kolotuchin S, La Porte T, Lee A, Lobben P, Lora-Gonzalez F, Mack B, Mudryk B, Qiu Y, et al. Adventures in Atropisomerism: Total Synthesis of a Complex Active Pharmaceutical Ingredient with Two Chirality Axes. Organic Letters. PMID 29909639 DOI: 10.1021/Acs.Orglett.8B01218 |
0.365 |
|
| 2018 |
Beutner G, Wertjes W, Ayers S, Gao Q, Simmons E. A Divergent Nickel-Catalyzed Synthesis of Quinazolinediones and Benzoxazinone Imines Synthesis. 50: 4453-4461. DOI: 10.1055/S-0037-1610140 |
0.418 |
|
| 2017 |
Ayothiraman R, Rangaswamy S, Maity P, Simmons EM, Beutner GL, Janey J, Treitler DS, Eastgate MD, Vaidyanathan R. Zinc Acetate-Promoted Buchwald-Hartwig Couplings of Heteroaromatic Amines. The Journal of Organic Chemistry. PMID 28677970 DOI: 10.1021/Acs.Joc.7B01101 |
0.378 |
|
| 2017 |
Beutner GL, Hsiao Y, Razler T, Simmons EM, Wertjes W. Nickel-Catalyzed Synthesis of Quinazolinediones. Organic Letters. 19: 1052-1055. PMID 28253632 DOI: 10.1021/Acs.Orglett.7B00052 |
0.441 |
|
| 2017 |
Gallagher WP, Soumeillant M, Chen K, Fox RJ, Hsiao Y, Mack B, Iyer V, Fan J, Zhu J, Beutner G, Silverman SM, Fanfair DD, Glace AW, Freitag A, Sweeney J, et al. Preparation of the HIV Attachment Inhibitor BMS-663068. Part 7. Development of a Regioselective Ullmann–Goldberg–Buchwald Reaction Organic Process Research & Development. 21: 1156-1165. DOI: 10.1021/Acs.Oprd.7B00191 |
0.404 |
|
| 2017 |
Fox RJ, Cohen B, La Cruz TE, Simpson JH, Freitag A, Saurer E, Tripp JC, Chen C, Beutner GL, Rosso VW, Borgeson E, Glace AW, Eastgate MD, Schild RL, Sweeney JT, et al. Preparation of the HIV Attachment Inhibitor BMS-663068. Part 8. Installation of the Phosphonoxymethyl Prodrug Moiety Organic Process Research & Development. 21: 1166-1173. DOI: 10.1021/Acs.Oprd.7B00135 |
0.372 |
|
| 2017 |
Beutner GL, Albrecht J, Fan J, Fanfair D, Lawler MJ, Bultman M, Chen K, Ivy S, Schild RL, Tripp JC, Murugesan S, Dambalas K, McLeod DD, Sweeney JT, Eastgate MD, et al. Preparation of the HIV Attachment Inhibitor BMS-663068. Part 3. Mechanistic Studies Enable a Scale-Independent Friedel–Crafts Acylation Organic Process Research & Development. 21: 1122-1130. DOI: 10.1021/Acs.Oprd.7B00115 |
0.374 |
|
| 2017 |
Benkovics T, Ortiz A, Beutner GL, Sfouggatakis C. Enantioselective Preparation of 5‐Oxo‐5,6‐Dihydro‐2H‐Pyran‐2‐yl Phenylacetate via Organocatalytic Dynamic Kinetic Asymmetric Transformation (DyKAT) Organic Syntheses. 94: 292-302. DOI: 10.1002/0471264229.Os094.21 |
0.343 |
|
| 2015 |
Ortiz A, Benkovics T, Beutner GL, Shi Z, Bultman M, Nye J, Sfouggatakis C, Kronenthal DR. Scalable Synthesis of the Potent HIV Inhibitor BMS-986001 by Non-Enzymatic Dynamic Kinetic Asymmetric Transformation (DYKAT). Angewandte Chemie (International Ed. in English). 54: 7185-8. PMID 25925234 DOI: 10.1002/Anie.201502290 |
0.419 |
|
| 2015 |
Tran K, Beutner GL, Schmidt M, Janey J, Chen K, Rosso V, Eastgate MD. Development of a Diastereoselective Phosphorylation of a Complex Nucleoside via Dynamic Kinetic Resolution. The Journal of Organic Chemistry. 80: 4994-5003. PMID 25840459 DOI: 10.1021/Acs.Joc.5B00392 |
0.358 |
|
| 2015 |
Ji Y, Benkovics T, Beutner GL, Sfouggatakis C, Eastgate MD, Blackmond DG. Mechanistic insights into the vanadium-catalyzed Achmatowicz rearrangement of furfurol. The Journal of Organic Chemistry. 80: 1696-702. PMID 25562708 DOI: 10.1021/Jo502641D |
0.427 |
|
| 2014 |
Limanto J, Ashley ER, Yin J, Beutner GL, Grau BT, Kassim AM, Kim MM, Klapars A, Liu Z, Strotman HR, Truppo MD. A highly efficient asymmetric synthesis of vernakalant. Organic Letters. 16: 2716-9. PMID 24786635 DOI: 10.1021/Ol501002A |
0.461 |
|
| 2014 |
Beutner GL, Desai L, Fanfair D, Lobben P, Anderson E, Leung SW, Eastgate MD. A method for heteroaromatic nitration demonstrating remarkable thermal stability Organic Process Research and Development. 18: 1812-1820. DOI: 10.1021/Op5001572 |
0.369 |
|
| 2013 |
Beutner GL, Denmark SE. Lewis base catalysis of the Mukaiyama directed aldol reaction: 40 years of inspiration and advances. Angewandte Chemie (International Ed. in English). 52: 9086-96. PMID 23843275 DOI: 10.1002/Anie.201302084 |
0.568 |
|
| 2013 |
Beutner GL, Denmark SE. The interplay of invention, observation, and discovery in the development of lewis base activation of lewis acids for catalytic enantioselective synthesis Topics in Organometallic Chemistry. 44: 55-89. DOI: 10.1007/3418-2012-43 |
0.49 |
|
| 2013 |
Beutner GL, Denmark SE. ChemInform Abstract: Lewis Base Catalysis of the Mukaiyama Directed Aldol Reaction: 40 Years of Inspiration and Advances Cheminform. 44: no-no. DOI: 10.1002/chin.201347233 |
0.468 |
|
| 2013 |
Beutner GL, Denmark SE. Lewis‐Base‐Katalyse der gerichteten Mukaiyama‐Aldolreaktion: 40 Jahre Inspiration und Fortschritt Angewandte Chemie. 125: 9256-9266. DOI: 10.1002/Ange.201302084 |
0.457 |
|
| 2012 |
Bassan EM, Baxter CA, Beutner GL, Emerson KM, Fleitz FJ, Johnson S, Keen S, Kim MM, Kuethe JT, Leonard WR, Mullens PR, Muzzio DJ, Roberge C, Yasuda N. Multikilogram-scale synthesis of a chiral cyclopropanol and an investigation of the safe use of lithium acetylide-ethylene diamine complex Organic Process Research and Development. 16: 87-95. DOI: 10.1021/Op2002497 |
0.364 |
|
| 2010 |
Denmark SE, Williams BJ, Eklov BM, Pham SM, Beutner GL. Design, validation, and implementation of a rapid-injection NMR system. The Journal of Organic Chemistry. 75: 5558-72. PMID 20672809 DOI: 10.1021/Jo100837A |
0.608 |
|
| 2009 |
Beutner GL, Kuethe JT, Yasuda N. A facile synthesis of 2,3-disubstituted furo[2,3-b]pyridines Tetrahedron Letters. 50: 781-784. DOI: 10.1016/J.Tetlet.2008.11.125 |
0.378 |
|
| 2009 |
Kuethe JT, Zhong YL, Alam M, Alorati AD, Beutner GL, Cai D, Fleitz FJ, Gibb AD, Kassim A, Linn K, Mancheno D, Marcune B, Pye PJ, Scott JP, Tellers DM, et al. Development of practical syntheses of potent non-nucleoside reverse transcriptase inhibitors Tetrahedron. 65: 5013-5023. DOI: 10.1016/J.Tet.2009.03.084 |
0.416 |
|
| 2009 |
Kuethe JT, Beutner GL. Synthesis of 2‐Arylindole‐4‐Carboxylic Amides: [2‐(4‐Fluorophenyl)‐1H‐Indol‐4‐YL]‐1‐Pyrrolidinylmethanone Organic Syntheses. 86: 92-104. DOI: 10.1002/0471264229.Os086.10 |
0.398 |
|
| 2009 |
Kuethe JT, Beutner GL, Denmark SE, Muhuhi JM. Synthesis of 2-arylindole-4-carboxylic amides: [2(4-Fluorophenyl)-1H-indol- 4-yl]-1-pyrrolidinylmethanone Organic Syntheses. 86: 92-104. |
0.442 |
|
| 2008 |
Denmark SE, Beutner GL. Lewis base catalysis in organic synthesis. Angewandte Chemie (International Ed. in English). 47: 1560-638. PMID 18236505 DOI: 10.1002/Anie.200604943 |
0.529 |
|
| 2008 |
Denmark SE, Beutner GL. ChemInform Abstract: Lewis Base Catalysis in Organic Synthesis Cheminform. 39. DOI: 10.1002/chin.200821255 |
0.444 |
|
| 2008 |
Denmark S, Beutner G. Lewis-Base-Katalyse in der organischen Synthese Angewandte Chemie. 120: 1584-1663. DOI: 10.1002/Ange.200604943 |
0.491 |
|
| 2007 |
Kuethe JT, Gauthier DR, Beutner GL, Yasuda N. A concise synthesis of (S)-N-ethoxycarbonyl-alpha-methylvaline. The Journal of Organic Chemistry. 72: 7469-72. PMID 17713956 DOI: 10.1021/Jo7012862 |
0.358 |
|
| 2007 |
Beutner GL, Kuethe JT, Yasuda N. A practical method for preparation of 4-hydroxyquinolinone esters. The Journal of Organic Chemistry. 72: 7058-61. PMID 17676920 DOI: 10.1021/Jo071200X |
0.375 |
|
| 2007 |
Denmark SE, Barsanti PA, Beutner GL, Wilson TW. Enantioselective ring opening of epoxides with silicon tetrachloride in the presence of a chiral lewis base: Mechanism studies Advanced Synthesis and Catalysis. 349: 566-582. DOI: 10.1002/Adsc.200600551 |
0.736 |
|
| 2006 |
Morrill C, Beutner GL, Grubbs RH. Rhenium-catalyzed 1,3-isomerization of allylic alcohols: scope and chirality transfer. The Journal of Organic Chemistry. 71: 7813-25. PMID 16995691 DOI: 10.1021/Jo061436L |
0.351 |
|
| 2005 |
Denmark SE, Heemstra JR, Beutner GL. Catalytic, enantioselective, vinylogous aldol reactions. Angewandte Chemie (International Ed. in English). 44: 4682-98. PMID 15940727 DOI: 10.1002/Anie.200462338 |
0.73 |
|
| 2005 |
Denmark SE, Beutner GL, Wynn T, Eastgate MD. Lewis base activation of Lewis acids: catalytic, enantioselective addition of silyl ketene acetals to aldehydes. Journal of the American Chemical Society. 127: 3774-89. PMID 15771512 DOI: 10.1021/Ja047339W |
0.583 |
|
| 2005 |
Denmark SE, Heemstra JR, Beutner GL. Katalytische enantioselektive vinyloge Aldolreaktionen Angewandte Chemie. 117: 4760-4777. DOI: 10.1002/Ange.200462338 |
0.687 |
|
| 2003 |
Denmark SE, Beutner GL. Lewis base activation of Lewis acids. Vinylogous aldol reactions. Journal of the American Chemical Society. 125: 7800-1. PMID 12822988 DOI: 10.1021/Ja035448P |
0.605 |
|
| 2002 |
Denmark SE, Wynn T, Beutner GL. Lewis base activation of lewis acids. Addition of silyl ketene acetals to aldehydes. Journal of the American Chemical Society. 124: 13405-7. PMID 12418891 DOI: 10.1021/Ja0282947 |
0.602 |
|
| 2002 |
Ronsheim MD, Hilgenkamp RK, Zercher CK, Denmark SE, Beutner GL. Formation of γ-keto esters from -keto esters: Methyl 5.5-dimethyl-4-oxohexanoate Organic Syntheses. 79: 146-152. DOI: 10.15227/Orgsyn.079.0146 |
0.468 |
|
| 2002 |
Kitamura M, Oka H, Suga S, Noyori R, Kaelin DE, Martin SF, Beutner GL, Denmark SE. Catalytic enantioselective addition of dialkylzincs to aldehydes using (2s)-(-)-3-exo-(dimethylamino)isoborneol [(2S)DAIB]: (S)-1-phenyl-1-propanol Organic Syntheses. 79: 139-145. DOI: 10.15227/Orgsyn.079.0139 |
0.454 |
|
| Show low-probability matches. |