Year |
Citation |
Score |
2009 |
Saito Y, Takahashi S, Azer N, Eldefrawi AT, Eldefrawi ME, Takahata H. Catalytic asymmetric synthesis of both enantiomers of pyrrolizidines 223H', 239K', 265H', and 267H' found in madagascan frogs (Mantella) and their affinities for nicotinic acetylcholine receptor Heterocycles. 79: 1043-1060. DOI: 10.3987/COM-08-S(D)81 |
0.322 |
|
2003 |
Menegatti R, Cunha AC, Ferreira VF, Perreira EF, El-Nabawi A, Eldefrawi AT, Albuquerque EX, Neves G, Rates SM, Fraga CA, Barreiro EJ. Design, synthesis and pharmacological profile of novel dopamine D2 receptor ligands. Bioorganic & Medicinal Chemistry. 11: 4807-13. PMID 14556797 DOI: 10.1016/S0968-0896(03)00487-5 |
0.36 |
|
2000 |
El-Nabawi A, Quesenberry M, Saito K, Silbergeld E, Vasta G, Eldefrawi A. The N-methyl-D-aspartate neurotransmitter receptor is a mammalian brain target for the dinoflagellate Pfiesteria piscicida toxin. Toxicology and Applied Pharmacology. 169: 84-93. PMID 11076700 DOI: 10.1006/Taap.2000.9042 |
0.521 |
|
2000 |
Takahata H, Takahashi S, Azer N, Eldefrawi AT, Eldefrawi ME. Total synthesis of pyrrolizidines 223H', 239K', 265H', and 267H' found in Madagascan frogs (Mantella) and their affinities for nicotinic acetylcholine receptor. Bioorganic & Medicinal Chemistry Letters. 10: 1293-5. PMID 10866403 DOI: 10.1016/S0960-894X(00)00221-3 |
0.324 |
|
1998 |
Takahata H, Kubota M, Ihara K, Okamoto N, Momose T, Azer N, Eldefrawi AT, Eldefrawi ME. New synthesis of all the four stereoisomers of indolizidine 209D and their affinity for nicotinic acetylcholine receptor Tetrahedron Asymmetry. 9: 3289-3301. DOI: 10.1016/S0957-4166(98)00338-3 |
0.404 |
|
1997 |
Katz EJ, Cortes VI, Eldefrawi ME, Eldefrawi AT. Chlorpyrifos, parathion, and their oxons bind to and desensitize a nicotinic acetylcholine receptor: relevance to their toxicities. Toxicology and Applied Pharmacology. 146: 227-36. PMID 9344890 DOI: 10.1006/taap.1997.8201 |
0.482 |
|
1997 |
Eldefrawi ME, Eldefrawi AT. Comparative Molecular and Pharmacological Properties of Cholinergic Receptors in Insects and Mammals Acs Symposium Series. 658: 327-338. |
0.402 |
|
1994 |
Jett DA, Fernando JC, Eldefrawi ME, Eldefrawi AT. Differential regulation of muscarinic receptor subtypes in rat brain regions by repeated injections of parathion. Toxicology Letters. 73: 33-41. PMID 8042201 DOI: 10.1016/0378-4274(94)90186-4 |
0.33 |
|
1994 |
Nakanishi K, Choi SK, Hwang D, Lerro K, Orlando M, Kalivretenos AG, Eldefrawi A, Eldefrawi M, Usherwood PNR. Bioorganic studies of transmitter receptors with philanthotoxin analogs Pure and Applied Chemistry. 66: 671-678. DOI: 10.1351/Pac199466040671 |
0.582 |
|
1993 |
Eldefrawi ME, Anis NA, Eldefrawi AT. Glutamate receptor inhibitors as potential insecticides. Archives of Insect Biochemistry and Physiology. 22: 25-39. PMID 8431599 DOI: 10.1002/arch.940220105 |
0.51 |
|
1993 |
Jett DA, Hill EF, Fernando JC, Eldefrawi ME, Eldefrawi AT. Down-regulation of muscarinic receptors and the m3 subtype in white-footed mice by dietary exposure to parathion. Journal of Toxicology and Environmental Health. 39: 395-415. PMID 8350385 DOI: 10.1080/15287399309531760 |
0.344 |
|
1993 |
Jett DA, Eldefrawi AT, Eldefrawi ME. Receptor binding assay applied to monitoring the neurotoxicity of parathion to peromyscus after oral exposure Astm Special Technical Publication. 253-262. |
0.407 |
|
1992 |
Abdallah EA, Jett DA, Eldefrawi ME, Eldefrawi AT. Differential effects of paraoxon on the M3 muscarinic receptor and its effector system in rat submaxillary gland cells. Journal of Biochemical Toxicology. 7: 125-32. PMID 1328639 |
0.489 |
|
1991 |
Abdallah EA, Eldefrawi ME, Eldefrawi AT. Pharmacologic characterization of muscarinic receptors of insect brains. Archives of Insect Biochemistry and Physiology. 17: 107-18. PMID 1802028 DOI: 10.1002/arch.940170205 |
0.492 |
|
1991 |
Goodnow RA, Bukownik R, Nakanishi K, Usherwood PN, Eldefrawi AT, Anis NA, Eldefrawi ME. Synthesis and binding of [125I2]philanthotoxin-343, [125I2]philanthotoxin-343-lysine, and [125I2]philanthotoxin-343-arginine to rat brain membranes. Journal of Medicinal Chemistry. 34: 2389-94. PMID 1652018 DOI: 10.1021/Jm00112A012 |
0.557 |
|
1991 |
Jett DA, Abdallah EAM, El-Fakahany EE, Eldefrawi ME, Eldefrawi AT. High-affinity activation by paraoxon of a muscarinic receptor subtype in rat brain striatum Pesticide Biochemistry and Physiology. 39: 149-157. DOI: 10.1016/0048-3575(91)90135-9 |
0.508 |
|
1990 |
Silveira CL, Eldefrawi AT, Eldefrawi ME. Putative M2 muscarinic receptors of rat heart have high affinity for organophosphorus anticholinesterases. Toxicology and Applied Pharmacology. 103: 474-81. PMID 2339420 DOI: 10.1016/0041-008X(90)90320-T |
0.471 |
|
1990 |
Anis N, Sherby S, Goodnow R, Niwa M, Konno K, Kallimopoulos T, Bukownik R, Nakanishi K, Usherwood P, Eldefrawi A. Structure-activity relationships of philanthotoxin analogs and polyamines on N-methyl-D-aspartate and nicotinic acetylcholine receptors. The Journal of Pharmacology and Experimental Therapeutics. 254: 764-73. PMID 2168484 |
0.538 |
|
1990 |
Bruce M, Bukownik R, Eldefrawi AT, Eldefrawi ME, Goodnow R, Kallimopoulos T, Konno K, Nakanishi K, Niwa M, Usherwood PN. Structure-activity relationships of analogues of the wasp toxin philanthotoxin: non-competitive antagonists of quisqualate receptors. Toxicon : Official Journal of the International Society On Toxinology. 28: 1333-46. PMID 1965063 DOI: 10.1016/0041-0101(90)90098-R |
0.491 |
|
1990 |
Nakanishi K, Goodnow R, Konno K, Niwa M, Bukownik R, Thomas T, Kallimopoulos A, Usherwood P, Eldefrawi AT, Eldefrawi ME. Philanthotoxin-433 (PhTX-433), a non-competitive glutamate receptor inhibitor Pure and Applied Chemistry. 62: 1223-1230. DOI: 10.1351/Pac199062071223 |
0.506 |
|
1989 |
Ragsdale D, Gant DB, Anis NA, Eldefrawi AT, Eldefrawi ME, Konno K, Miledi R. Inhibition of rat brain glutamate receptors by philanthotoxin. The Journal of Pharmacology and Experimental Therapeutics. 251: 156-63. PMID 2571715 |
0.539 |
|
1989 |
Sattelle DB, Buckingham SD, Wafford KA, Sherby SM, Bakry NM, Eldefrawi AT, Eldefrawi ME, May TE. Actions of the insecticide 2(nitromethylene)tetrahydro-1,3-thiazine on insect and vertebrate nicotinic acetylcholine receptors. Proceedings of the Royal Society of London. Series B, Biological Sciences. 237: 501-14. PMID 2479949 DOI: 10.1098/Rspb.1989.0062 |
0.536 |
|
1989 |
Rozental R, Scoble GT, Albuquerque EX, Idriss M, Sherby S, Sattelle DB, Nakanishi K, Konno K, Eldefrawi AT, Eldefrawi ME. Allosteric inhibition of nicotinic acetylcholine receptors of vertebrates and insects by philanthotoxin. The Journal of Pharmacology and Experimental Therapeutics. 249: 123-30. PMID 2468760 |
0.513 |
|
1989 |
Wafford KA, Sattelle DB, Gant DB, Eldefrawi AT, Eldefrawi ME. Noncompetitive inhibition of GABA receptors in insect and vertebrate CNS by endrin and lindane Pesticide Biochemistry and Physiology. 33: 213-219. DOI: 10.1016/0048-3575(89)90119-3 |
0.362 |
|
1988 |
Bakry NM, el-Rashidy AH, Eldefrawi AT, Eldefrawi ME. Direct actions of organophosphate anticholinesterases on nicotinic and muscarinic acetylcholine receptors. Journal of Biochemical Toxicology. 3: 235-59. PMID 3236334 |
0.545 |
|
1988 |
Eldefrawi AT, Eldefrawi ME, Konno K, Mansour NA, Nakanishi K, Oltz E, Usherwood PN. Structure and synthesis of a potent glutamate receptor antagonist in wasp venom. Proceedings of the National Academy of Sciences of the United States of America. 85: 4910-3. PMID 2838850 DOI: 10.1073/Pnas.85.13.4910 |
0.482 |
|
1988 |
Matsumoto K, Eldefrawi ME, Eldefrawi AT. Action of polychlorocycloalkane insecticides on binding of [35S]t-butylbicyclophosphorothionate to Torpedo electric organ membranes and stereospecificity of the binding site. Toxicology and Applied Pharmacology. 95: 220-9. PMID 2458634 DOI: 10.1016/0041-008X(88)90158-5 |
0.419 |
|
1988 |
Ramadan AA, Bakry NM, Marei ASM, Eldefrawi AT, Eldefrawi ME. Actions of pyrethroids on the peripheral benzodiazepine receptor Pesticide Biochemistry and Physiology. 32: 106-113. DOI: 10.1016/0048-3575(88)90003-X |
0.428 |
|
1988 |
Ramadan AA, Bakry NM, Marei ASM, Eldefrawi AT, Eldefrawi ME. Action of pyrethroids on GABAA receptor function Pesticide Biochemistry and Physiology. 32: 97-105. DOI: 10.1016/0048-3575(88)90002-8 |
0.401 |
|
1987 |
Gant DB, Eldefrawi ME, Eldefrawi AT. Cyclodiene insecticides inhibit GABAA receptor-regulated chloride transport. Toxicology and Applied Pharmacology. 88: 313-21. PMID 3033845 DOI: 10.1016/0041-008X(87)90206-7 |
0.32 |
|
1987 |
Sherby SM, Eldefrawi ME, Wafford KA, Sattelle DB, Eldefrawi AT. Pharmacology of putative glutamate receptors from insect skeletal muscles, insect central nervous system and rat brain. Comparative Biochemistry and Physiology. C, Comparative Pharmacology and Toxicology. 87: 99-106. PMID 2885148 DOI: 10.1016/0742-8413(87)90189-7 |
0.38 |
|
1987 |
Gant DB, Eldefrawi ME, Eldefrawi AT. Action of organophosphates on GABAA receptor and voltage-dependent chloride channels. Fundamental and Applied Toxicology : Official Journal of the Society of Toxicology. 9: 698-704. PMID 2446940 DOI: 10.1093/toxsci/9.4.698 |
0.353 |
|
1987 |
Gant DB, Cole RJ, Valdes JJ, Eldefrawi ME, Eldefrawi AT. Action of tremorgenic mycotoxins on GABAA receptor. Life Sciences. 41: 2207-14. PMID 2444852 DOI: 10.1016/0024-3205(87)90517-0 |
0.506 |
|
1987 |
Eldefrawi AT, Eldefrawi ME. Receptors for gamma-aminobutyric acid and voltage-dependent chloride channels as targets for drugs and toxicants. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 1: 262-71. PMID 2443413 |
0.472 |
|
1986 |
Bakry NM, Sherby SM, Eldefrawi AT, Eldefrawi ME. Oxadiazolidinones: irreversible inhibition of cholinesterases and effects on acetylcholine receptors. Neurotoxicology. 7: 1-10. PMID 3822252 |
0.424 |
|
1986 |
Abalis IM, Eldefrawi ME, Eldefrawi AT. Effects of insecticides on GABA-induced chloride influx into rat brain microsacs. Journal of Toxicology and Environmental Health. 18: 13-23. PMID 3009836 DOI: 10.1080/15287398609530844 |
0.34 |
|
1986 |
Abalis IM, Eldefrawi AT, Eldefrawi ME. Actions of avermectin B1a on the gamma-aminobutyric acidA receptor and chloride channels in rat brain. Journal of Biochemical Toxicology. 1: 69-82. PMID 2856070 |
0.367 |
|
1986 |
Sherby SM, Eldefrawi AT, Deshpande SS, Albuquerque EX, Eldefrawi ME. Effects of pyrethroids on nicotinic acetylcholine receptor binding and function Pesticide Biochemistry and Physiology. 26: 107-115. DOI: 10.1016/0048-3575(86)90082-9 |
0.539 |
|
1986 |
Abalis IM, Eldefrawi AT. [3H]Muscimol binding to a putative GABA receptor in honey bee brain and its interaction with avermectin B1a Pesticide Biochemistry and Physiology. 25: 279-287. DOI: 10.1016/0048-3575(86)90001-5 |
0.381 |
|
1986 |
Sherby SM, Eldefrawi AT, David JA, Sattelle DB, Eldefrawi ME. Interactions of charatoxins and nereistoxin with the nicotinic acetylcholine receptors of insect cns andTorpedo electric organ Archives of Insect Biochemistry and Physiology. 3: 431-445. DOI: 10.1002/Arch.940030504 |
0.56 |
|
1985 |
Sherby SM, Eldefrawi AT, Albuquerque EX, Eldefrawi ME. Comparison of the actions of carbamate anticholinesterases on the nicotinic acetylcholine receptor. Molecular Pharmacology. 27: 343-8. PMID 3974572 |
0.553 |
|
1985 |
Filbin MT, Eldefrawi ME, Eldefrawi AT. Biochemical identification of a putative glutamate receptor in housefly thoracic membranes. Life Sciences. 36: 1531-9. PMID 2858805 DOI: 10.1016/0024-3205(85)90377-7 |
0.373 |
|
1985 |
Eldefrawi ME, Sherby SM, Abalis IM, Eldefrawi AT. Interactions of pyrethroid and cyclodiene insecticides with nicotinic acetylcholine and GABA receptors. Neurotoxicology. 6: 47-62. PMID 2410832 |
0.362 |
|
1985 |
Abalis IM, Eldefrawi ME, Eldefrawi AT. Binding of GABA receptor channel drugs to a putative voltage-dependent chloride channel in Torpedo electric organ. Biochemical Pharmacology. 34: 2579-82. PMID 2409983 DOI: 10.1016/0006-2952(85)90550-7 |
0.324 |
|
1985 |
Abalis IM, Eldefrawi ME, Eldefrawi AT. High-affinity stereospecific binding of cyclodiene insecticides and γ-hexachlorocyclohexane to γ-aminobutyric acid receptors of rat brain Pesticide Biochemistry and Physiology. 24: 95-102. DOI: 10.1016/0048-3575(85)90118-X |
0.361 |
|
1985 |
Sattelle DB, Hue B, Pelhate M, Sherby SM, Eldefrawi AT, Eldefrawi ME. Actions of phencyclidine and its thienylpyrrolidine analogue on synaptic transmission and axonal conduction in the central nervous system of the cockroach Periplaneta americana Journal of Insect Physiology. 31: 917-924. DOI: 10.1016/0022-1910(85)90025-3 |
0.39 |
|
1984 |
El-Fakahany EE, Eldefrawi AT, Murphy DL, Aguayo LG, Triggle DJ, Albuquerque EX, Eldefrawi ME. Interactions of phencyclidine with crayfish muscle membranes. Sensitivity to calcium channel antagonists and other drugs. Molecular Pharmacology. 25: 369-78. PMID 6328263 |
0.34 |
|
1984 |
El-Fakahany EE, Triggle DJ, Eldefrawi AT, Eldefrawi ME. Distinction between high-affinity [3H]phencyclidine binding sites and muscarinic receptors in guinea-pig ileum muscle. The Journal of Pharmacology and Experimental Therapeutics. 229: 447-54. PMID 6325665 |
0.438 |
|
1984 |
Idriss MH, Filbin MT, Eldefrawi AT. Effects of chlorisondamine and philanthotoxin on the glutamate receptor/channel complex of locus muscle Federation Proceedings. 43: no. 335. |
0.374 |
|
1983 |
Eldefrawi ME, Eldefrawi AT. Neurotransmitter receptors as targets for pesticides. Journal of Environmental Science and Health. Part. B, Pesticides, Food Contaminants, and Agricultural Wastes. 18: 65-88. PMID 6339601 DOI: 10.1080/03601238309372358 |
0.569 |
|
1983 |
Abbassy MA, Eldefrawi ME, Eldefrawi AT. Influence of the alcohol moiety of pyrethroids on their interactions with the nicotinic acetylcholine receptor. Journal of Toxicology and Environmental Health. 12: 575-90. PMID 6321746 DOI: 10.1080/15287398309530450 |
0.476 |
|
1983 |
Ei-Fakahany EF, Miller ER, Abbassy MA, Eldefrawi AT, Eldefrawi ME. Alcohol modulation of drug binding to the channel sites of the nicotinic acetylcholine receptor. The Journal of Pharmacology and Experimental Therapeutics. 224: 289-96. PMID 6296354 |
0.384 |
|
1983 |
Abalis IM, Eldefrawi ME, Eldefrawi AT. Biochemical identification of putative GABA/benzodiazepine receptors in house fly thorax muscles Pesticide Biochemistry and Physiology. 20: 39-48. DOI: 10.1016/0048-3575(83)90119-0 |
0.306 |
|
1983 |
Abbassy MA, Eldefrawi ME, Eldefrawi AT. Pyrethroid action on the nicotinic acetylcholine receptor/channel Pesticide Biochemistry and Physiology. 19: 299-308. DOI: 10.1016/0048-3575(83)90058-5 |
0.413 |
|
1982 |
Bakry NM, Eldefrawi AT, Eldefrawi ME, Riker WF. Interactions of quaternary ammonium drugs with acetylcholinesterase and acetylcholine receptor of Torpedo electric organ. Molecular Pharmacology. 22: 63-71. PMID 7121452 |
0.316 |
|
1982 |
El-Fakahany EF, Eldefrawi AT, Eldefrawi ME. Nicotinic acetylcholine receptor desensitization studied by [3H]perhydrohistrionicotoxin binding. The Journal of Pharmacology and Experimental Therapeutics. 221: 694-700. PMID 7086681 |
0.523 |
|
1982 |
Eldefrawi AT, Mansour NA, Eldefrawi ME. Insecticides affecting acetylcholine receptor interactions. Pharmacology & Therapeutics. 16: 45-65. PMID 6752971 DOI: 10.1016/0163-7258(82)90031-6 |
0.431 |
|
1982 |
Abbassy MA, Eldefrawi ME, Eldefrawi AT. Allethrin interactions with the nicotinic acetylcholine receptor channel. Life Sciences. 31: 1547-52. PMID 6292640 DOI: 10.1016/0024-3205(82)90045-5 |
0.5 |
|
1982 |
Eldefrawi AT, Miller ER, Eldefrawi ME. Binding of depolarizing drugs to the ionic channel sites of the nicotinic acetylcholine receptor. Biochemical Pharmacology. 31: 1819-22. PMID 6285933 DOI: 10.1016/0006-2952(82)90697-9 |
0.446 |
|
1982 |
Shaker N, Eldefrawi AT, Aguayo LG, Warnick JE, Albuquerque EX, Eldefrawi ME. Interactions of d-tubocurarine with the nicotinic acetylcholine receptor/channel molecule. The Journal of Pharmacology and Experimental Therapeutics. 220: 172-7. PMID 6273528 |
0.327 |
|
1982 |
Warnick JE, Maleque MA, Bakry N, Eldefrawi AT, Albuquerque EX. Structure-activity relationships of amantadine. I. Interaction of the N-alkyl analogues with the ionic channels of the nicotinic acetylcholine receptor and electrically excitable membrane. Molecular Pharmacology. 22: 82-93. PMID 6126806 |
0.403 |
|
1982 |
Eldefrawi AT, Miller ER, Murphy DL, Eldefrawi ME. [3H]Phencyclidine interactions with the nicotinic acetylcholine receptor channel and its inhibition by psychotropic, antipsychotic, opiate, antidepressant, antibiotic, antiviral, and antiarrhythmic drugs. Molecular Pharmacology. 22: 72-81. PMID 6126805 |
0.399 |
|
1982 |
El-Fakahany EF, Eldefrawi ME, Eldefrawi AT. Desensitization of torpedo nicotinic acetylcholine receptors Federation Proceedings. 41: No. 6146. |
0.434 |
|
1981 |
Desouki A, Eldefrawi AT, Eldefrawi ME. A new mechanism revealed for the action of antibodies on acetylcholine receptor function. Experimental Neurology. 73: 440-50. PMID 7262247 DOI: 10.1016/0014-4886(81)90278-8 |
0.33 |
|
1981 |
Aronstam RS, Eldefrawi AT, Pessah IN, Daly JW, Albuquerque EX, Eldefrawi ME. Regulation of [3H]perhydrohistrionicotoxin binding to Torpedo ocellata electroplax by effectors of the acetylcholine receptor. The Journal of Biological Chemistry. 256: 2843-50. PMID 7204378 |
0.51 |
|
1981 |
Albuquerque EX, Warnick JE, Mayer RF, Eldefrawi AT, Eldefrawi ME. Recent advances in the molecular mechanisms of human and animal models of myasthenia gravis. Annals of the New York Academy of Sciences. 377: 496-518. PMID 6280564 DOI: 10.1111/J.1749-6632.1981.Tb33756.X |
0.303 |
|
1981 |
Shaker N, Eldefrawi AT, Miller ER, Eldefrawi ME. Interaction of tricyclic antidepressants with the ionic channel of the acetylcholine receptor of Torpedo electric organ. Molecular Pharmacology. 20: 511-8. PMID 6276711 |
0.35 |
|
1981 |
Eldefrawi ME, Warnick JE, Schofield GG, Albuquerque EX, Eldefrawi AT. Interaction of imipramine with the ionic channel of the acetylcholine receptor of motor endplate and electric organ. Biochemical Pharmacology. 30: 1391-4. PMID 6268097 DOI: 10.1016/0006-2952(81)90331-2 |
0.303 |
|
1981 |
Shaker N, Eldefrawi A. Muscarinic receptor in house fly brain and its interaction with chlorobenzilate Pesticide Biochemistry and Physiology. 15: 14-20. DOI: 10.1016/0048-3575(81)90030-4 |
0.585 |
|
1981 |
Shaker N, Eldefrawi AT. [3H]ONB binding to housefly brain: Relation to muscarinic acetylcholine receptors Federation Proceedings. 40: 490. |
0.465 |
|
1981 |
Shaker N, Eldefrawi ME, Eldefrawi AT. Interaction of imipramine (IMIP) with the ionic channel of the nicotinic acetylcholine receptor Federation Proceedings. 40: 147. |
0.41 |
|
1980 |
Aronstam RS, Eldefrawi ME, Eldefrawi AT, Albuquerque EX, Jim KF, Triggle DJ. Sites of action of phencyclidine. III. Interactions with muscarinic receptors. Molecular Pharmacology. 18: 179-84. PMID 7421791 |
0.395 |
|
1980 |
Albuquerque EX, Tsai MC, Aronstam RS, Witkop B, Eldefrawi AT, Eldefrawi ME. Phencyclidine interactions with the ionic channel of the acetylcholine receptor and electrogenic membrane. Proceedings of the National Academy of Sciences of the United States of America. 77: 1224-8. PMID 6928673 DOI: 10.1073/Pnas.77.2.1224 |
0.463 |
|
1980 |
Eldefrawi ME, Eldefrawi AT, Aronstam RS, Maleque MA, Warnick JE, Albuquerque EX. [3H]Phencyclidine: a probe for the ionic channel of the nicotinic receptor. Proceedings of the National Academy of Sciences of the United States of America. 77: 7458-62. PMID 6261260 DOI: 10.1073/Pnas.77.12.7458 |
0.486 |
|
1980 |
Eldefrawi ME, Eldefrawi AT. Coupling between the nicotinic acetylcholine receptor site and the ionic channel site. Annals of the New York Academy of Sciences. 358: 239-52. PMID 6259991 |
0.384 |
|
1980 |
Albuquerque EX, Tsai MC, Aronstam RS, Eldefrawi AT, Eldefrawi ME. Sites of action of phencyclidine. II. Interaction with the ionic channel of the nicotinic receptor. Molecular Pharmacology. 18: 167-78. PMID 6252436 |
0.386 |
|
1980 |
Aronstam RS, Eldefrawi AT, Eldefrawi ME. Similarities in the binding sites of the muscarinic receptor and the ionic channel of the nicotinic receptor. Biochemical Pharmacology. 29: 1311-4. PMID 6249329 DOI: 10.1016/0006-2952(80)90292-0 |
0.534 |
|
1980 |
Eldefrawi AT, Bakry NM, Eldefrawi ME, Tsai MC, Albuquerque EX. Nereistoxin interaction with the acetylcholine receptor-ionic channel complex. Molecular Pharmacology. 17: 172-9. PMID 6248754 |
0.349 |
|
1980 |
Eldefrawi ME, Aronstam RS, Bakry NM, Eldefrawi AT, Albuquerque EX. Activation, inactivation, and desensitization of acetylcholine receptor channel complex detected by binding of perhydrohistrionicotoxin. Proceedings of the National Academy of Sciences of the United States of America. 77: 2309-13. PMID 6246539 DOI: 10.1073/Pnas.77.4.2309 |
0.453 |
|
1979 |
Adler M, Oliveira AC, Albuquerque EX, Mansour NA, Eldefrawi AT. Reaction of tetraethylammonium with the open and closed conformations of the acetylcholine receptor ionic channel complex. The Journal of General Physiology. 74: 129-52. PMID 486241 DOI: 10.1085/jgp.74.1.129 |
0.356 |
|
1979 |
Eldefrawi ME, Copio DS, Hudson CS, Rash J, Mansour NA, Eldefrawi AT, Albuguergue EX. Effects of antibodies to Torpedo acetylcholine receptor on the acetylcholine receptor--ionic channel complex of Torpedo electroplax and rabbit intercostal muscle. Experimental Neurology. 64: 428-44. PMID 428517 DOI: 10.1016/0014-4886(79)90281-4 |
0.512 |
|
1979 |
Eldefrawi ME, Eldefrawi AT. Biochemical studies on the ionic channel of Torpedo acetylcholine receptor. Advances in Cytopharmacology. 3: 213-23. PMID 382785 |
0.482 |
|
1979 |
Tiedt TN, Albuquerque EX, Bakry NM, Eldefrawi ME, Eldefrawi AT. Voltage- and time-dependent actions of piperocaine on the ion channel of the acetylcholine receptor. Molecular Pharmacology. 16: 909-21. PMID 316855 |
0.325 |
|
1979 |
Tsai MC, Oliveira AC, Albuquerque EX, Eldefrawi ME, Eldefrawi AT. Mode of action of quinacrine on the acetylcholine receptor ionic channel complex. Molecular Pharmacology. 16: 382-92. PMID 316101 |
0.327 |
|
1978 |
Sarvey JM, Albuquerque EX, Eldefrawi AT, Eldefrawi M. Effects of alpha-bungarotoxin and reversible cholinergic ligands on normal and denervated mammalian skeletal muscle. Membrane Biochemistry. 1: 131-57. PMID 756485 DOI: 10.3109/09687687809064163 |
0.318 |
|
1978 |
Eldefrawi ME, Eldefrawi AT, Mansour NA, Daly JW, Witkop B, Albuquerque EX. Acetylcholine receptor and ionic channel of Torpedo electroplax: binding of perhydrohistrionicotoxin to membrane and solubilized preparations. Biochemistry. 17: 5474-84. PMID 728410 DOI: 10.1021/Bi00618A023 |
0.428 |
|
1978 |
Rübsamen H, Eldefrawi AT, Eldefrawi ME, Hess GP. Characterization of calcium-binding sites of the purified acetylcholine receptor and identification of the calcium-binding subunit. Biochemistry. 17: 3818-25. PMID 698199 DOI: 10.1021/Bi00611A022 |
0.326 |
|
1978 |
Albuquerque EX, Eldefrawi AT, Eldefrawi ME, Mansour NA, Tsai MC. Amantadine: neuromuscular blockade by suppression of ionic conductance of the acetylcholine receptor. Science (New York, N.Y.). 199: 788-90. PMID 622570 DOI: 10.1126/Science.622570 |
0.461 |
|
1978 |
Tsai MC, Bakry NM, Eldefrawi AT, Albuquerque EX. Rimantadine on the ion conductance modulator of the cholinergic receptor Federation Proceedings. 37: No. 3008. |
0.307 |
|
1977 |
Eldefrawi ME, Mansour NA, Eldefrawi AT. Interactions of acetylcholine receptors with organic mercury compounds. Advances in Experimental Medicine and Biology. 84: 449-63. PMID 899953 |
0.521 |
|
1977 |
Eldefrawi AT, Mansour NA, Brattsten LB, Ahrens VD, Lisk DJ. Further toxicologic studies with commercial and candidate flame retardant chemicals. Part II. Bulletin of Environmental Contamination and Toxicology. 17: 720-6. PMID 880389 DOI: 10.1007/BF01685960 |
0.323 |
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1977 |
Eldefrawi AT, Eldefrawi ME, Albuquerque EX, Oliveira AC, Mansour N, Adler M, Daly JW, Brown GB, Burgermeister W, Witkop B. Perhydrohistrionicotoxin: a potential ligand for the ion conductance modulator of the acetylcholine receptor. Proceedings of the National Academy of Sciences of the United States of America. 74: 2172-6. PMID 301278 DOI: 10.1073/Pnas.74.5.2172 |
0.419 |
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1977 |
Mansour NA, Elderfrawi ME, Eldefrawi AT. Isolation of putative acetylcholine receptor proteins from housefly brain. Biochemistry. 16: 4126-32. PMID 71919 |
0.346 |
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1977 |
Mansour NA, Eldefrawi AT. Interaction of pesticides with the acetylcholine receptor Federation Proceedings. 36: No. 676. |
0.422 |
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1976 |
Rübsamen H, Hess GP, Eldefrawi AT, Eldefrawi ME. Interaction between calcium and ligand-binding sites of the purified acetylcholine receptor studied by use of a fluorescent lanthanide. Biochemical and Biophysical Research Communications. 68: 56-63. PMID 942851 DOI: 10.1016/0006-291X(76)90009-7 |
0.324 |
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1976 |
Eldefrawi AT, Eldefrawi ME. Identification of a calcium-binding subunit of the acetylcholine receptor. Biochemical and Biophysical Research Communications. 70: 1020-7. PMID 938522 DOI: 10.1016/0006-291X(76)90694-X |
0.376 |
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1975 |
Eldefrawi ME, Eldefrawi AT, Wilson DB. Tryptophan and cystein residues of the acetylcholine receptors of Torpedo species. Relationship to binding of cholinergic ligands. Biochemistry. 14: 4304-10. PMID 1182102 |
0.439 |
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1975 |
Edelstein SJ, Beyer WB, Eldefrawi AT, Eldefrawi ME. Molecular weight of the acetylcholine receptors of electric organs and the effect of Triton X 100 Journal of Biological Chemistry. 250: 6101-6106. PMID 1150674 |
0.385 |
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1975 |
Eldefrawi ME, Eldefrawi AT, Penfield LA, O'Brien RD, Van Campen D. Binding of calcium and zinc to the acetylcholine receptor purified from Torpedo Californica Life Sciences. 16: 925-935. PMID 1128162 DOI: 10.1016/0024-3205(75)90008-9 |
0.391 |
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1973 |
Eldefrawi ME, Eldefrawi AT. Purification and molecular properties of the acetylcholine receptor from Torpedo electroplax. Archives of Biochemistry and Biophysics. 159: 362-73. PMID 4806354 DOI: 10.1016/0003-9861(73)90462-1 |
0.416 |
|
1973 |
Eldefrawi ME, Eldefrawi AT. Cooperativities in the binding of acetylcholine to its receptor. Biochemical Pharmacology. 22: 3145-50. PMID 4761574 DOI: 10.1016/0006-2952(73)90209-8 |
0.523 |
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1972 |
Eldefrawi ME, Eldefrawi AT, Seifert S, O'Brien RD. Properties of lubrol-solubilized acetylcholine receptor from Torpedo electroplax. Archives of Biochemistry and Biophysics. 150: 210-8. PMID 5028075 DOI: 10.1016/0003-9861(72)90028-8 |
0.456 |
|
1972 |
Eldefrawi ME, Eldefrawi AT. Characterization and partial purification of the acetylcholine receptor from Torpedo electroplax. Proceedings of the National Academy of Sciences of the United States of America. 69: 1776-80. PMID 4505655 |
0.444 |
|
1972 |
O'Brien RD, Eldefrawi ME, Eldefrawi AT. Isolation of acetylcholine receptors. Annual Review of Pharmacology. 12: 19-34. PMID 4339017 DOI: 10.1146/annurev.pa.12.040172.000315 |
0.431 |
|
1971 |
Eldefrawi ME, Britten AG, Eldefrawi AT. Acetylcholine binding to Torpedo electroplax: relationship to acetylcholine receptors. Science (New York, N.Y.). 173: 338-40. PMID 5559905 |
0.494 |
|
1971 |
Eldefrawi ME, Eldefrawi AT, O'Brien RD. Binding of five cholinergic ligands to housefly brain and Torpedo electroplax. Relationship to acetylcholine receptors. Molecular Pharmacology. 7: 104-10. PMID 5552246 |
0.432 |
|
1971 |
Eldefrawi ME, Eldefrawi AT, O'Brien RD. Binding sites for cholinergic ligands in a particulate fraction of Electrophorus electroplax. Proceedings of the National Academy of Sciences of the United States of America. 68: 1047-50. PMID 4102561 |
0.411 |
|
1970 |
Eldefrawi AT, O'Brien RD. Binding of muscarone by extracts of housefly brain: relationship to receptors for acetylcholine. Journal of Neurochemistry. 17: 1287-93. PMID 5457631 |
0.398 |
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Low-probability matches (unlikely to be authored by this person) |
1979 |
Adler M, Oliveira AC, Eldefrawi ME, Eldefrawi AT, Albuquerque EX. Tetraethylammonium: voltage-dependent action on endplate conductance and inhibition of ligand binding to postsynaptic proteins. Proceedings of the National Academy of Sciences of the United States of America. 76: 531-5. PMID 284372 DOI: 10.1073/Pnas.76.1.531 |
0.283 |
|
1971 |
Eldefrawi ME, Eldefrawi AT, Gilmour LP, O'Brien RD. Multiple affinities for binding of cholinergic ligands to a particulate fraction of Torpedo electroplax. Molecular Pharmacology. 7: 420-8. PMID 5165342 |
0.274 |
|
1982 |
Eldefrawi ME, El-Fakahany EF, Murphy DL, Eldefrawi AT, Triggle DJ. High affinity binding of phencyclidine (PCP) to crayfish muscle. Displacement by calcium antagonists. Biochemical Pharmacology. 31: 2549-52. PMID 7126268 DOI: 10.1016/0006-2952(82)90069-7 |
0.272 |
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1987 |
Wafford KA, Sattelle DB, Abalis I, Eldefrawi AT, Eldefrawi ME. gamma-Aminobutyric acid-activated 36Cl- influx: a functional in vitro assay for CNS gamma-aminobutyric acid receptors of insects. Journal of Neurochemistry. 48: 177-80. PMID 3025362 DOI: 10.1111/j.1471-4159.1987.tb13144.x |
0.261 |
|
1979 |
Albuquerque EX, Eldefrawi AT, Oliveira AC, Copio DS, Eldefrawi ME. Myasthenia gravis animal model: quantitative analysis of the efficiency of pre- and postjunctional regions of intercostal muscles in rabbits immunized with Torpedo acetylcholine receptor. Experimental Neurology. 66: 109-22. PMID 225189 DOI: 10.1016/0014-4886(79)90067-0 |
0.259 |
|
1985 |
Filbin MT, Eldefrawi ME, Eldefrawi AT. Binding of [3H]phencyclidine to membranes from housefly thoracic muscles Archives of Insect Biochemistry and Physiology. 2: 181-190. DOI: 10.1002/arch.940020206 |
0.248 |
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1984 |
Abalis IM, Eldefrawi ME, Eldefrawi AT. Binding of [3H]strychnine to insect skeletal muscle Federation Proceedings. 43: no. 3755. |
0.24 |
|
1984 |
Filbin MT, Eldefrawi AT. Effects of organophosphate anticholinesterases, phencyclidine analogs and calcium channel antagonists on acetylcholine synthesis, release and choline uptake Federation Proceedings. 43: no. 337. |
0.21 |
|
1999 |
Cao CJ, Mioduszewski RJ, Menking DE, Valdes JJ, Katz EJ, Eldefrawi ME, Eldefrawi AT. Cytotoxicity of organophosphate anticholinesterases. In Vitro Cellular & Developmental Biology. Animal. 35: 493-500. PMID 10548430 DOI: 10.1007/s11626-999-0059-8 |
0.206 |
|
1977 |
Eldefrawi ME, Eldefrawi AT, Albuquerque EX. Binding of [3H]perhydrohistrionicotoxin to torpedo electric organ membranes: relation to ion conductance modulator Federation Proceedings. 36: No.3796. |
0.2 |
|
1988 |
Ramadan AA, Bakry NM, Marei ASM, Eldefrawi AT, Eldefrawi ME. Action of pyrethroids on K+-stimulated calcium uptake by, and [3H]nimodipine binding to, rat brain synaptosomes Pesticide Biochemistry and Physiology. 32: 114-122. DOI: 10.1016/0048-3575(88)90004-1 |
0.186 |
|
1990 |
Cao CJ, Eldefrawi AT, Eldefrawi ME. ATP-regulated neuronal catecholamine uptake: a new mechanism. Life Sciences. 47: 655-67. PMID 2402189 DOI: 10.1016/0024-3205(90)90578-F |
0.163 |
|
1991 |
Rogers KR, Cao CJ, Valdes JJ, Eldefrawi AT, Eldefrawi ME. Acetylcholinesterase fiber-optic biosensor for detection of anticholinesterases. Fundamental and Applied Toxicology : Official Journal of the Society of Toxicology. 16: 810-20. PMID 1909249 DOI: 10.1016/0272-0590(91)90166-2 |
0.159 |
|
1970 |
Eldefrawi ME, Eldefrawi AT, O'Brien RD. Mode of action of nicotine in the housefly Journal of Agricultural and Food Chemistry. 18: 1113-1116. |
0.155 |
|
1980 |
Tsai MC, Albuquerque EX, Aronstam RS, Eldefrawi AT, Eldefrawi ME, Triggle DJ. Sites of action of phencyclidine. I. Effects on the electrical excitability and chemosensitive properties of the neuromuscular junction of skeletal muscle. Molecular Pharmacology. 18: 159-66. PMID 6968397 |
0.146 |
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1994 |
Dehlawi MS, Eldefrawi AT, Eldefrawi ME, Anis NA, Valdes JJ. Choline derivatives and sodium fluoride protect acetylcholinesterase against irreversible inhibition and aging by DFP and paraoxon. Journal of Biochemical Toxicology. 9: 261-8. PMID 7853361 |
0.121 |
|
1998 |
Cao CJ, Eldefrawi ME, Eldefrawi AT, Burnett JW, Mioduszewski RJ, Menking DE, Valdes JJ. Toxicity of sea nettle toxin to human hepatocytes and the protective effects of phosphorylating and alkylating agents. Toxicon : Official Journal of the International Society On Toxinology. 36: 269-81. PMID 9620575 DOI: 10.1016/S0041-0101(97)00122-0 |
0.109 |
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1997 |
Cao CJ, Mioduszewski RJ, Menking DE, Valdes JJ, Cortes VI, Eldefrawi ME, Eldefrawi AT. Validation of the cytosensor for in vitro cytotoxicity studies. Toxicology in Vitro : An International Journal Published in Association With Bibra. 11: 285-93. PMID 20654314 DOI: 10.1016/S0887-2333(97)00009-X |
0.103 |
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1998 |
Mileson BE, Chambers JE, Chen WL, Dettbarn W, Ehrich M, Eldefrawi AT, Gaylor DW, Hamernik K, Hodgson E, Karczmar AG, Padilla S, Pope CN, Richardson RJ, Saunders DR, Sheets LP, et al. Common mechanism of toxicity: a case study of organophosphorus pesticides. Toxicological Sciences : An Official Journal of the Society of Toxicology. 41: 8-20. PMID 9520337 DOI: 10.1006/Toxs.1997.2431 |
0.095 |
|
1978 |
Tsai MC, Mansour NA, Eldefrawi AT, Eldefrawi ME, Albuquerque EX. Mechanism of action of amantadine on neuromuscular transmission. Molecular Pharmacology. 14: 787-803. PMID 213703 |
0.079 |
|
1979 |
Bakry N, Tsai MC, Albuquerque EX, Eldefrawi AT. Nereistoxin on neuromuscular transmission Federation Proceedings. 38: No. 253. |
0.069 |
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1995 |
Devine PJ, Anis NA, Wright J, Kim S, Eldefrawi AT, Eldefrawi ME. A fiber-optic cocaine biosensor. Analytical Biochemistry. 227: 216-24. PMID 7668383 DOI: 10.1006/abio.1995.1273 |
0.048 |
|
1997 |
Toppozada AR, Wright J, Eldefrawi AT, Eldefrawi ME, Johnson EL, Emche SD, Helling CS. Evaluation of a fiber optic immunosensor for quantitating cocaine in coca leaf extracts. Biosensors & Bioelectronics. 12: 113-24. PMID 9011023 DOI: 10.1016/S0956-5663(97)87057-1 |
0.036 |
|
1991 |
Masler EP, Kelly TJ, Menn JJ, Nachman RJ, Holman GM, Zitnan D, Takeda M, Sauman I, Sehnal F, Segal D, Altaratz M, Richard DS, Gilbert LI, Applebaum SW, Shaaya E, ... ... Eldefrawi AT, et al. Abstracts of papers presented at the United States/Israel bard workshop on new targets for insect management in crop protection Phytoparasitica. 19: 331-358. DOI: 10.1007/Bf02980967 |
0.029 |
|
1993 |
Fernando JC, Rogers KR, Anis NA, Valdes JJ, Thompson RG, Eldefrawi AT, Eldefrawi ME. Rapid detection of anticholinesterase insecticides by a reusable light addressable potentiometric biosensor Journal of Agricultural and Food Chemistry. 41: 511-516. |
0.025 |
|
1998 |
Mioduszewski R, Menking D, Valdes J, Cao C, Eldefrawi M, Eldefrawi A. Cytotoxicity of organophosphate anticholinesterases to human liver and nerve cells Toxicology Letters. 95: 140. DOI: 10.1016/S0378-4274(98)80554-7 |
0.024 |
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1995 |
Zhao CQ, Anis NA, Rogers KR, Kline RH, Wright J, Eldefrawi AT, Eldefrawi ME. Fiber optic immunosensor for polychlorinated biphenyls Journal of Agricultural and Food Chemistry. 43: 2308-2315. |
0.013 |
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1991 |
Masler EP, Kelly TJ, Menn JJ, Nachman RJ, Holman GM, Zitnan D, Takeda M, Sauman I, Sehnal F, Segal D, Altaratz M, Richard DS, Gilbert LI, Applebaum SW, Shaaya E, ... ... Eldefrawi AT, et al. Corrections Phytoparasitica. 19: 311. DOI: 10.1007/BF02980968 |
0.01 |
|
Hide low-probability matches. |