Year |
Citation |
Score |
2014 |
Blizzard TA, Chen H, Kim S, Wu J, Bodner R, Gude C, Imbriglio J, Young K, Park YW, Ogawa A, Raghoobar S, Hairston N, Painter RE, Wisniewski D, Scapin G, et al. Discovery of MK-7655, a β-lactamase inhibitor for combination with Primaxin®. Bioorganic & Medicinal Chemistry Letters. 24: 780-5. PMID 24433862 DOI: 10.1016/j.bmcl.2013.12.101 |
0.359 |
|
2011 |
Chen H, Blizzard TA, Kim S, Wu J, Young K, Park YW, Ogawa AM, Raghoobar S, Painter RE, Wisniewski D, Hairston N, Fitzgerald P, Sharma N, Scapin G, Lu J, et al. Side chain SAR of bicyclic β-lactamase inhibitors (BLIs). 2. N-Alkylated and open chain analogs of MK-8712. Bioorganic & Medicinal Chemistry Letters. 21: 4267-70. PMID 21676616 DOI: 10.1016/j.bmcl.2011.05.065 |
0.401 |
|
2010 |
Blizzard TA, et al. ea. ChemInform Abstract: Side Chain SAR of Bicyclic β-Lactamase Inhibitors (BLIs). Part 1. Discovery of a Class C BLI for Combination with Imipinem. Cheminform. 41: no-no. DOI: 10.1002/chin.201039214 |
0.387 |
|
2010 |
WADDELL ST, SANTORELLI GM, BLIZZARD TA, GRAHAM A, OCCI J. ChemInform Abstract: Synthesis and Antibacterial Activity of O-Methyl Derivatives of Azalide Antibiotics. Part 2. 6-OMe Derivatives via Clarithromycin. Cheminform. 29: no-no. DOI: 10.1002/chin.199841247 |
0.331 |
|
1999 |
Wilkening RR, Ratcliffe RW, Wildonger KJ, Cama LD, Dykstra KD, DiNinno FP, Blizzard TA, Hammond ML, Heck JV, Dorso KL, St Rose E, Kohler J, Hammond GG. Synthesis and activity of 2-(sulfonamido)methyl-carbapenems: discovery of a novel, anti-MRSA 1,8-naphthosultam pharmacophore. Bioorganic & Medicinal Chemistry Letters. 9: 673-8. PMID 10201827 DOI: 10.1016/S0960-894X(99)00070-0 |
0.34 |
|
1998 |
Meinke PT, Shoop WL, Michael BF, Blizzard TA, Dawson GR, Fisher MH, Mrozik H. Synthesis of gem-difluoro-avermectin derivatives: potent anthelmintic and anticonvulsant agents. Bioorganic & Medicinal Chemistry Letters. 8: 3643-6. PMID 9934486 DOI: 10.1016/S0960-894X(98)00674-X |
0.382 |
|
1998 |
Waddell ST, Santorelli GM, Blizzard TA, Graham A, Occi J. Synthesis and antibacterial activity of O-methyl derivatives of azalide antibiotics: II. 6-OME derivatives via clarithromycin. Bioorganic & Medicinal Chemistry Letters. 8: 1321-6. PMID 9871759 DOI: 10.1016/S0960-894X(98)00227-3 |
0.34 |
|
1998 |
Waddell ST, Santorelli GM, Blizzard TA, Graham A, Occi J. Synthesis and antibacterial activity of O-methyl derivatives of azalide antibiotics: I. 4", 11 and 12-OMe derivatives via direct methylation. Bioorganic & Medicinal Chemistry Letters. 8: 549-54. PMID 9871616 DOI: 10.1016/S0960-894X(98)00070-5 |
0.337 |
|
1994 |
Shankaran K, Wilkening RR, Blizzard TA, Ratcliffe RW, Heck JV, Graham AC, Herbert CM. Preparation and activities of 4″-epi and 4″-deoxy-4″-amino analogs derived from 9-deoxo-8a-aza-8a-homoerythromycin A Bioorganic and Medicinal Chemistry Letters. 4: 1111-1116. DOI: 10.1016/S0960-894X(01)80238-9 |
0.321 |
|
1992 |
Shankaran K, Blizzard TA. Synthesis and activities of 9-pyrrolo-9-deoxoerythromycin a analogs Bioorganic and Medicinal Chemistry Letters. 2: 1555-1558. DOI: 10.1016/S0960-894X(00)80427-8 |
0.366 |
|
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