Chris Sfouggatakis, Ph.D. - Publications

2004 University of Pennsylvania, Philadelphia, PA, United States 
Natural product synthesis

13/18 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2021 La Cruz TE, González-Bobes F, Eastgate MD, Sfouggatakis C, Zheng B, Kopp N, Xiao Y, Fan Y, Galindo KA, Pathirana C, Galella MA, Deerberg J. Scalable Asymmetric Synthesis of the All Triamino Cyclohexane Core of BMS-813160. The Journal of Organic Chemistry. PMID 34355895 DOI: 10.1021/acs.joc.1c01162  1
2015 Ortiz A, Benkovics T, Beutner GL, Shi Z, Bultman M, Nye J, Sfouggatakis C, Kronenthal DR. Scalable Synthesis of the Potent HIV Inhibitor BMS-986001 by Non-Enzymatic Dynamic Kinetic Asymmetric Transformation (DYKAT). Angewandte Chemie (International Ed. in English). 54: 7185-8. PMID 25925234 DOI: 10.1002/Anie.201502290  1
2015 Ji Y, Benkovics T, Beutner GL, Sfouggatakis C, Eastgate MD, Blackmond DG. Mechanistic insights into the vanadium-catalyzed Achmatowicz rearrangement of furfurol. The Journal of Organic Chemistry. 80: 1696-702. PMID 25562708 DOI: 10.1021/Jo502641D  1
2014 Cohen B, Mahoney M, Remy B, Qiu J, Sfouggatakis C, Shi Z, Wang C. Development of a robust API crystallization in a multi-component solvent mixture: Using high throughput automation as an enabling technology to develop comprehensive solubility maps Pharmaceutical Discovery, Development and Manufacturing Forum 2014 - Core Programming Area At the 2014 Aiche Annual Meeting. 310.  1
2013 Pathirana C, Sfouggatakis C, Palaniswamy V. N-N migration of a carbamoyl group in a pyrazole derivative revealed by NMR. Magnetic Resonance in Chemistry : Mrc. 51: 184-7. PMID 23338988 DOI: 10.1002/mrc.3921  1
2011 Broxer S, Fitzgerald MA, Sfouggatakis C, Defreese JL, Barlow E, Powers GL, Peddicord M, Su BN, Tai-Yuen Y, Pathirana C, Sherbine JP. The development of a robust process for a CRF1 receptor antagonist Organic Process Research and Development. 15: 343-352. DOI: 10.1021/op100270u  1
2009 Smith AB, Sfouggatakis C, Risatti CA, Sperry JB, Zhu W, Doughty VA, Tomioka T, Gotchev DB, Bennett CS, Sakamoto S, Atasoylu O, Shirakami S, Bauer D, Takeuchi M, Koyanagi J, et al. Spongipyran Synthetic Studies. Evolution of a Scalable Total Synthesis of (+)-Spongistatin 1. Tetrahedron. 65: 6489-6509. PMID 20640040 DOI: 10.1016/J.Tet.2009.04.003  1
2009 Smith AB, Doughty VA, Sfouggatakis C, Bennett CS, Koyanagi J, Takeuchi M. Spongistatin synthetic studies. An efficient, second-generation construction of an advanced ABCD intermediate (Organic Letters (2002) 4) Organic Letters. 11: 785.  1
2008 Smith AB, Tomioka T, Risatti CA, Sperry JB, Sfouggatakis C. Gram-scale synthesis of (+)-spongistatin 1: development of an improved, scalable synthesis of the F-ring subunit, fragment union, and final elaboration. Organic Letters. 10: 4359-62. PMID 18754594 DOI: 10.1021/ol801792k  1
2004 Smith AB, Sfouggatakis C, Gotchev DB, Shirakami S, Bauer D, Zhu W, Doughty VA. Spongistatin synthetic studies. evolution of a scalable synthesis for the EF fragment of (+)-Spongistatin 1 exploiting a Petasis-Ferrier union/rearrangement tactic. Organic Letters. 6: 3637-40. PMID 15387567 DOI: 10.1021/ol048418f  1
2003 Smith AB, Pitram SM, Boldi AM, Gaunt MJ, Sfouggatakis C, Moser WH. Multicomponent linchpin couplings. Reaction of dithiane anions with terminal epoxides, epichlorohydrin, and vinyl epoxides: efficient, rapid, and stereocontrolled assembly of advanced fragments for complex molecule synthesis. Journal of the American Chemical Society. 125: 14435-45. PMID 14624591 DOI: 10.1021/ja0376238  1
2003 Smith AB, Zhu W, Shirakami S, Sfouggatakis C, Doughty VA, Bennett CS, Sakamoto Y. Total synthesis of (+)-spongistatin 1. An effective second-generation construction of an advanced EF Wittig salt, fragment union, and final elaboration. Organic Letters. 5: 761-4. PMID 12605509 DOI: 10.1021/Ol034037A  1
2002 Smith AB, Doughty VA, Sfouggatakis C, Bennett CS, Koyanagi J, Takeuchi M. Spongistatin synthetic studies. An efficient, second-generation construction of an advanced ABCD intermediate. Organic Letters. 4: 783-6. PMID 11869127 DOI: 10.1021/Ol017273Z  1
Low-probability matches
2019 Beutner GL, Bultman MS, Cohen BM, Fan J, Marshall J, Sfouggatakis C. Follow the Silyl Cation: Insights into the Vorbrüggen Reaction Organic Process Research & Development. 23: 2050-2056. DOI: 10.1021/Acs.Oprd.9B00304  0.01
2019 Rosso V, Simon J, Hickey M, Risatti C, Sfouggatakis C, Breckenridge L, Lou S, Forest R, Chiou G, Marshall J, Tom J. Engaging senior management to improve the safety culture of a chemical development organization thru the SPYDR (Safety as Part of Your Daily Routine) lab visit program Journal of Chemical Health and Safety. 26: 38-43. DOI: 10.1016/J.JCHAS.2019.03.005  0.01
2018 Maity P, Reddy VVR, Mohan J, Korapati S, Narayana H, Cherupally N, Chandrasekaran S, Ramachandran R, Sfouggatakis C, Eastgate MD, Simmons EM, Vaidyanathan R. Development of a Scalable Synthesis of BMS-978587 Featuring a Stereospecific Suzuki Coupling of a Cyclopropane Carboxylic Acid Organic Process Research & Development. 22: 888-897. DOI: 10.1021/Acs.Oprd.8B00171  0.01
2017 Smith MJ, Lawler MJ, Kopp N, Mcleod DD, Davulcu AH, Lin D, Katipally K, Sfouggatakis C. Development of a Concise Multikilogram Synthesis of LPA-1 Antagonist BMS-986020 via a Tandem Borylation–Suzuki Procedure Organic Process Research & Development. 21: 1859-1863. DOI: 10.1021/acs.oprd.7b00301  0.01
2016 Deerberg J, Prasad SJ, Sfouggatakis C, Eastgate MD, Fan Y, Chidambaram R, Sharma P, Li L, Schild R, Müslehiddinoğlu J, Chung H, Leung S, Rosso V. Stereoselective Bulk Synthesis of CCR2 Antagonist BMS-741672: Assembly of an All-cis(S,R,R)-1,2,4-Triaminocyclohexane (TACH) Core via Sequential Heterogeneous Asymmetric Hydrogenations Organic Process Research & Development. 20: 1949-1966. DOI: 10.1021/Acs.Oprd.6B00282  0.01
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