Year |
Citation |
Score |
2010 |
Yates CM, Brown PJ, Stewart EL, Patten C, Austin RJ, Holt JA, Maglich JM, Angell DC, Sasse RZ, Taylor SJ, Uings IJ, Trump RP. Structure guided design of 5-arylindazole glucocorticoid receptor agonists and antagonists. Journal of Medicinal Chemistry. 53: 4531-44. PMID 20469868 DOI: 10.1021/Jm100447C |
0.376 |
|
2010 |
Rimland J, Dunne A, Hunjan SS, Sasse R, Uings I, Montanari D, Caivano M, Shah P, Standing D, Gray D, Brown D, Cairns W, Trump R, Smith PW, Bertheleme N, et al. The identification a novel, selective, non-steroidal, functional glucocorticoid receptor antagonist. Bioorganic & Medicinal Chemistry Letters. 20: 2340-3. PMID 20202837 DOI: 10.1016/J.Bmcl.2010.01.133 |
0.331 |
|
2007 |
Trump RP, Blanc JB, Stewart EL, Brown PJ, Caivano M, Gray DW, Hoekstra WJ, Willson TM, Han B, Turnbull P. Design and synthesis of an array of selective androgen receptor modulators. Journal of Combinatorial Chemistry. 9: 107-14. PMID 17206838 DOI: 10.1021/Cc060096E |
0.368 |
|
2005 |
Yang Y, Nesterenko DV, Trump RP, Yamaguchi K, Bartlett PA, Drueckhammer DG. Virtual hydrocarbon and combinatorial databases for use with CAVEAT. Journal of Chemical Information and Modeling. 45: 1820-3. PMID 16309289 DOI: 10.1021/Ci050277O |
0.403 |
|
2005 |
Bledsoe RK, Madauss KP, Holt JA, Apolito CJ, Lambert MH, Pearce KH, Stanley TB, Stewart EL, Trump RP, Willson TM, Williams SP. A ligand-mediated hydrogen bond network required for the activation of the mineralocorticoid receptor. The Journal of Biological Chemistry. 280: 31283-93. PMID 15967794 DOI: 10.1074/Jbc.M504098200 |
0.309 |
|
2003 |
Trump RP, Bartlett PA. Amino acid-derived heterocycles as combinatorial library targets: spirocyclic ketal lactones. Journal of Combinatorial Chemistry. 5: 285-91. PMID 12739946 DOI: 10.1021/Cc020081Q |
0.423 |
|
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