Year |
Citation |
Score |
2008 |
Dyck B, Tamiya J, Jovic F, Pick RR, Bradbury MJ, O'Brien J, Wen J, Johns M, Madan A, Fleck BA, Foster AC, Li B, Zhang M, Tran JA, Vickers T, et al. Characterization of thien-2-yl 1S,2R-milnacipran analogues as potent norepinephrine/serotonin transporter inhibitors for the treatment of neuropathic pain. Journal of Medicinal Chemistry. 51: 7265-72. PMID 18954038 DOI: 10.1021/Jm8009537 |
0.434 |
|
2008 |
Zhang M, Jovic F, Vickers T, Dyck B, Tamiya J, Grey J, Tran JA, Fleck BA, Pick R, Foster AC, Chen C. Studies on the structure-activity relationship of bicifadine analogs as monoamine transporter inhibitors Bioorganic and Medicinal Chemistry Letters. 18: 3682-3686. PMID 18539031 DOI: 10.1016/J.Bmcl.2008.05.077 |
0.398 |
|
2008 |
Vickers T, Dyck B, Tamiya J, Zhang M, Jovic F, Grey J, Fleck BA, Aparicio A, Johns M, Jin L, Tang H, Foster AC, Chen C. Studies on a series of milnacipran analogs containing a heteroaromatic group as potent norepinephrine and serotonin transporter inhibitors. Bioorganic & Medicinal Chemistry Letters. 18: 3230-5. PMID 18468895 DOI: 10.1016/J.Bmcl.2008.04.045 |
0.469 |
|
2008 |
Tamiya J, Dyck B, Zhang M, Phan K, Fleck BA, Aparicio A, Jovic F, Tran JA, Vickers T, Grey J, Foster AC, Chen C. Identification of 1S,2R-milnacipran analogs as potent norepinephrine and serotonin transporter inhibitors. Bioorganic & Medicinal Chemistry Letters. 18: 3328-32. PMID 18445525 DOI: 10.1016/J.Bmcl.2008.04.025 |
0.456 |
|
2008 |
Chen C, Dyck B, Fleck BA, Foster AC, Grey J, Jovic F, Mesleh M, Phan K, Tamiya J, Vickers T, Zhang M. Studies on the SAR and pharmacophore of milnacipran derivatives as monoamine transporter inhibitors. Bioorganic & Medicinal Chemistry Letters. 18: 1346-9. PMID 18207394 DOI: 10.1016/J.Bmcl.2008.01.011 |
0.371 |
|
2007 |
Rowbottom MW, Vickers TD, Tamiya J, Zhang M, Dyck B, Grey J, Schwarz D, Heise CE, Hedrick M, Wen J, Tang H, Wang H, Fisher A, Aparicio A, Saunders J, et al. Synthesis and structure-activity relationships of spirohydantoin-derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Bioorganic & Medicinal Chemistry Letters. 17: 2171-8. PMID 17350839 DOI: 10.1016/J.Bmcl.2007.01.104 |
0.541 |
|
2007 |
Zhang M, Tamiya J, Nguyen L, Rowbottom MW, Dyck B, Vickers TD, Grey J, Schwarz DA, Heise CE, Haelewyn J, Mistry MS, Goodfellow VS. Thienopyrimidinone bis-aminopyrrolidine ureas as potent melanin-concentrating hormone receptor-1 (MCH-R1) antagonists. Bioorganic & Medicinal Chemistry Letters. 17: 2535-9. PMID 17329101 DOI: 10.1016/J.Bmcl.2007.02.012 |
0.46 |
|
2006 |
Rowbottom MW, Vickers TD, Dyck B, Grey J, Tamiya J, Zhang M, Kiankarimi M, Wu D, Dwight W, Wade WS, Schwarz D, Heise CE, Madan A, Fisher A, Petroski R, et al. Synthesis and structure-activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 1. Bioorganic & Medicinal Chemistry Letters. 16: 4450-7. PMID 16814542 DOI: 10.1016/J.Bmcl.2006.06.045 |
0.557 |
|
2006 |
Dyck B, Markison S, Zhao L, Tamiya J, Grey J, Rowbottom MW, Zhang M, Vickers T, Sorensen K, Norton C, Wen J, Heise CE, Saunders J, Conlon P, Madan A, et al. A thienopyridazinone-based melanin-concentrating hormone receptor 1 antagonist with potent in vivo anorectic properties. Journal of Medicinal Chemistry. 49: 3753-6. PMID 16789729 DOI: 10.1021/Jm051263C |
0.344 |
|
2006 |
Dyck B, Zhao L, Tamiya J, Pontillo J, Hudson S, Ching B, Heise CE, Wen J, Norton C, Madan A, Schwarz D, Wade W, Goodfellow VS. Substituted chromones and quinolones as potent melanin-concentrating hormone receptor 1 antagonists. Bioorganic & Medicinal Chemistry Letters. 16: 4237-42. PMID 16762549 DOI: 10.1016/J.Bmcl.2006.05.075 |
0.433 |
|
2005 |
Rowbottom MW, Vickers TD, Dyck B, Tamiya J, Zhang M, Zhao L, Grey J, Provencal D, Schwarz D, Heise CE, Mistry M, Fisher A, Dong T, Hu T, Saunders J, et al. Synthesis and structure-activity relationships of biarylcarboxamide bis-aminopyrrolidine urea derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Bioorganic & Medicinal Chemistry Letters. 15: 3439-45. PMID 15950467 DOI: 10.1016/J.Bmcl.2005.05.015 |
0.528 |
|
2005 |
Grey J, Dyck B, Rowbottom MW, Tamiya J, Vickers TD, Zhang M, Zhao L, Heise CE, Schwarz D, Saunders J, Goodfellow VS. Bis(aminopyrrolidine)-derived ureas (APUs) as potent MCH1 receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 15: 999-1004. PMID 15686900 DOI: 10.1016/J.Bmcl.2004.12.036 |
0.439 |
|
2003 |
Tamiya J, Sorensen EJ. A spontaneous bicyclization facilitates a synthesis of (-)-hispidospermidin Tetrahedron. 59: 6921-6932. DOI: 10.1016/S0040-4020(03)00936-0 |
0.519 |
|
2000 |
Tamiya J, Sorensen EJ. A concise synthesis of (-)-hispidospermidin guided by a postulated biogenesis [10] Journal of the American Chemical Society. 122: 9556-9557. DOI: 10.1021/Ja0026758 |
0.454 |
|
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