Year |
Citation |
Score |
2022 |
Bresinsky M, Strasser JM, Vallaster B, Liu P, McCue WM, Fuller J, Hubmann A, Singh G, Nelson KM, Cuellar ME, Wilmot CM, Finzel BC, Ashe KH, Walters MA, Pockes S. Structure-Based Design and Biological Evaluation of Novel Caspase-2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314. Acs Pharmacology & Translational Science. 5: 20-40. PMID 35059567 DOI: 10.1021/acsptsci.1c00251 |
0.313 |
|
2020 |
Priebbenow DL, Leaver D, Nguyen N, Cleary B, Lagiakos HR, Sanchez J, Xue L, Huang F, Sun Y, Mujumdar P, Mudududdla R, Varghese S, Teguh SC, Charman SA, White KL, ... ... Cuellar ME, et al. Discovery of Acylsulfonohydrazide-Derived Lysine Acetyltransferase (KAT6A) Inhibitors as Potent Senescence-Inducing Anti-Cancer Agents. Journal of Medicinal Chemistry. PMID 32118427 DOI: 10.1021/Acs.Jmedchem.9B02071 |
0.324 |
|
2020 |
Xie Y, Tummala P, Oakley AJ, Deora GS, Nakano Y, Rooke M, Cuellar M, Strasser J, Dahlin JL, Walters MA, Casarotto MG, Board PG, Baell JB. Development of Benzenesulfonamide Derivatives as Potent Glutathione Transferase Omega-1 Inhibitors. Journal of Medicinal Chemistry. PMID 32105470 DOI: 10.1021/Acs.Jmedchem.9B01391 |
0.308 |
|
2020 |
Xie Y, Tummala P, Oakley AJ, Deora GS, Nakano Y, Rooke M, Cuellar ME, Strasser JM, Dahlin JL, Walters MA, Casarotto MG, Board PG, Baell JB. Development ofBenzenesulfonamide Derivatives as PotentGlutathione Transferase Omega‑1 Inhibitors Journal of Medicinal Chemistry. DOI: 10.1021/Acs.Jmedchem.9B01391.S001 |
0.308 |
|
2019 |
Leaver D, Cleary B, Nguyen NT, Priebbenow DL, Lagiakos HR, Sanchez J, Xue L, Huang F, Sun Y, Mujumdar P, Mudududdla R, Varghese S, Teguh S, Charman SA, White K, ... ... Cuellar M, et al. Discovery of benzoylsulfonohydrazides as potent inhibitors of the histone acetyltransferase KAT6A. Journal of Medicinal Chemistry. PMID 31256587 DOI: 10.2210/Pdb6Oio/Pdb |
0.338 |
|
2011 |
Wilger DJ, Park JH, Hughes RM, Cuellar ME, Waters ML. Induced-fit binding of a polyproline helix by a β-hairpin peptide. Angewandte Chemie (International Ed. in English). 50: 12201-4. PMID 22038775 DOI: 10.1002/Anie.201106177 |
0.448 |
|
2010 |
Ingerman LA, Cuellar ME, Waters ML. A small molecule receptor that selectively recognizes trimethyl lysine in a histone peptide with native protein-like affinity. Chemical Communications (Cambridge, England). 46: 1839-41. PMID 20198226 DOI: 10.1039/C000255K |
0.489 |
|
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