Kittichoat Tiyanont, Ph.D. - Related publications

2007 Princeton University, Princeton, NJ 
Chemical biology, enzymology, antibiotics, glycosyltransferases, inhibitors
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50 most relevant papers in past 60 days:
Year Citation  Score
2021 Amelia T, van Veldhoven JPD, Falsini M, Liu R, Heitman LH, van Westen GJP, Segala E, Verdon G, Cheng RKY, Cooke RM, van der Es D, IJzerman AP. Crystal Structure and Subsequent Ligand Design of a Nonriboside Partial Agonist Bound to the Adenosine A Receptor. Journal of Medicinal Chemistry. PMID 33764785 DOI: 10.1021/acs.jmedchem.0c01856   
2021 Moriwaki K, Chan FKM, Miyoshi E. Sweet modification and regulation of death receptor signaling pathway. Journal of Biochemistry. PMID 33752241 DOI: 10.1093/jb/mvab034   
2021 Slosky LM, Caron MG, Barak LS. Biased Allosteric Modulators: New Frontiers in GPCR Drug Discovery. Trends in Pharmacological Sciences. PMID 33581873 DOI: 10.1016/   
2021 Wang F, Chau B, West SM, Kimberlin CR, Cao F, Schwarz F, Aguilar B, Han M, Morishige W, Bee C, Dollinger G, Rajpal A, Strop P. Structures of mouse and human GITR-GITRL complexes reveal unique TNF superfamily interactions. Nature Communications. 12: 1378. PMID 33654081 DOI: 10.1038/s41467-021-21563-z   
2021 Deganutti G, Barkan K, Preti B, Leuenberger M, Wall M, Frenguelli BG, Lochner M, Ladds G, Reynolds CA. Deciphering the Agonist Binding Mechanism to the Adenosine A1 Receptor. Acs Pharmacology & Translational Science. 4: 314-326. PMID 33615181 DOI: 10.1021/acsptsci.0c00195   
2021 Sánchez MF, Els-Heindl S, Beck-Sickinger AG, Wieneke R, Tampé R. Photo-induced receptor confinement drives ligand-independent GPCR signaling. Science (New York, N.Y.). PMID 33632896 DOI: 10.1126/science.abb7657   
2021 Mason EO, Goldgur Y, Robev D, Freywald A, Nikolov DB, Himanen JP. Structure of the EphB6 receptor ectodomain. Plos One. 16: e0247335. PMID 33770085 DOI: 10.1371/journal.pone.0247335   
2021 Hanneken A, Mercado M, Maher P. Constitutive and Regulated Shedding of Soluble FGF Receptors Releases Biologically Active Inhibitors of FGF-2. International Journal of Molecular Sciences. 22. PMID 33800200 DOI: 10.3390/ijms22052712   
2021 Jaiswal S, Rajnikanth PS, Thakur S, Deepak P, Anand S. A Review on Novel Ligand Targeted Delivery for Cardiovascular Disorder. Current Drug Delivery. PMID 33645481 DOI: 10.2174/1567201818666210301095046   
2021 Zlotos DP, Abdelmalek CM, Botros LS, Banoub MM, Mandour YM, Breitinger U, El Nady A, Breitinger HG, Sotriffer C, Villmann C, Jensen AA, Holzgrabe U. C-2-Linked Dimeric Strychnine Analogues as Bivalent Ligands Targeting Glycine Receptors. Journal of Natural Products. PMID 33596384 DOI: 10.1021/acs.jnatprod.0c01030   
2021 Bouwman KM, Tomris I, Turner HL, van der Woude R, Shamorkina TM, Bosman GP, Rockx B, Herfst S, Snijder J, Haagmans BL, Ward AB, Boons GJ, de Vries RP. Multimerization- and glycosylation-dependent receptor binding of SARS-CoV-2 spike proteins. Plos Pathogens. 17: e1009282. PMID 33556147 DOI: 10.1371/journal.ppat.1009282   
2021 James NG, Malik S, Sanstrum BJ, Rhéaume C, Broide RS, Jameson DM, Brideau-Andersen A, Jacky BS. Characterization of clostridium botulinum neurotoxin serotype A (BoNT/A) and fibroblast growth factor receptor interactions using novel receptor dimerization assay. Scientific Reports. 11: 7832. PMID 33837264 DOI: 10.1038/s41598-021-87331-7   
2021 Onaran HO, Costa T. Conceptual and experimental issues in biased agonism. Cellular Signalling. 82: 109955. PMID 33607257 DOI: 10.1016/j.cellsig.2021.109955   
2021 Okamoto Y, Shikano S. Tyrosine sulfation and O-glycosylation of chemoattractant receptor GPR15 differentially regulate interaction with GPR15L. Journal of Cell Science. PMID 33758080 DOI: 10.1242/jcs.247833   
2021 Nakamura S, Saito R, Yamamoto S, Kobayashi I, Takeda R, Suzuki R, Kawai K, Takimoto-Kamimura M, Kurita N. Proposal of novel potent inhibitors against androgen receptor based on ab initio molecular orbital calculations. Journal of Molecular Graphics & Modelling. 105: 107873. PMID 33640786 DOI: 10.1016/j.jmgm.2021.107873   
2021 Schüß C, Vu O, Schubert M, Du Y, Mishra NM, Tough IR, Stichel J, Weaver CD, Emmitte KA, Cox HM, Meiler J, Beck-Sickinger AG. Highly Selective Y Receptor Antagonist Binds in an Allosteric Binding Pocket. Journal of Medicinal Chemistry. PMID 33595306 DOI: 10.1021/acs.jmedchem.0c02000   
2021 Raita Y, Zhu Z, Freishtat RJ, Fujiogi M, Liang L, Patregnani JT, Camargo CA, Hasegawa K. Soluble receptor for advanced glycation end products (sRAGE) and asthma: Mendelian randomisation study. Pediatric Allergy and Immunology : Official Publication of the European Society of Pediatric Allergy and Immunology. PMID 33599351 DOI: 10.1111/pai.13478   
2021 Deganutti G, Barkan K, Ladds G, Reynolds CA. Multisite Model of Allosterism for the Adenosine A1 Receptor. Journal of Chemical Information and Modeling. PMID 33779168 DOI: 10.1021/acs.jcim.0c01331   
2021 Mingle D, Ospanov M, Radwan MO, Ashpole N, Otsuka M, Ross SA, Walker L, Shilabin AG, Ibrahim MA. First In Class (,)-11-[2-(Arylmethylene)Hydrazono]-PBD Analogs As Selective CB2 Modulators Targeting Neurodegenerative Disorders. Medicinal Chemistry Research : An International Journal For Rapid Communications On Design and Mechanisms of Action of Biologically Active Agents. 30: 98-108. PMID 33776384 DOI: 10.1007/s00044-020-02640-2   
2021 Stroberg W, Schnell S. Concentration Sensing in Crowded Environments. Biophysical Journal. PMID 33675760 DOI: 10.1016/j.bpj.2021.02.035   
2021 Lin B, Wang Q, Liu K, Dong X, Zhu M, Li M. Alpha-Fetoprotein Binding Mucin and Scavenger Receptors: An Available Bio-Target for Treating Cancer. Frontiers in Oncology. 11: 625936. PMID 33718192 DOI: 10.3389/fonc.2021.625936   
2021 Yeliseev A, Iyer MR, Joseph TT, Coffey NJ, Cinar R, Zoubak L, Kunos G, Gawrisch K. Cholesterol as a modulator of cannabinoid receptor CB signaling. Scientific Reports. 11: 3706. PMID 33580091 DOI: 10.1038/s41598-021-83245-6   
2021 Siddiqa MA, Rao DS, Suvarna G, Chennamachetty VK, Verma MK, Rao MVR. In-Silico Drug Designing of Spike Receptor with Its ACE2 Receptor and Nsp10/Nsp16 MTase Complex Against SARS-CoV-2. International Journal of Peptide Research and Therapeutics. 1-8. PMID 33746660 DOI: 10.1007/s10989-021-10196-x   
2021 Sharma DS, Paddibhatla I, Raghuwanshi S, Malleswarapu M, Sangeeth A, Kovuru N, Dahariya S, Gautam DK, Pallepati A, Gutti RK. Endocannabinoid system: Role in blood cell development, neuroimmune interactions and associated disorders. Journal of Neuroimmunology. 353: 577501. PMID 33571815 DOI: 10.1016/j.jneuroim.2021.577501   
2021 McNeill SM, Baltos JA, White PJ, May LT. Biased agonism at adenosine receptors. Cellular Signalling. 109954. PMID 33610717 DOI: 10.1016/j.cellsig.2021.109954   
2021 Lazki-Hagenbach P, Ali H, Sagi-Eisenberg R. Authentic and Ectopically Expressed MRGPRX2 Elicit Similar Mechanisms to Stimulate Degranulation of Mast Cells. Cells. 10. PMID 33673037 DOI: 10.3390/cells10020376   
2021 Soriano Jerez EM, Gibbins JM, Hughes CE. Targeting platelet inhibition receptors for novel therapies: PECAM-1 and G6b-B. Platelets. 1-9. PMID 33646086 DOI: 10.1080/09537104.2021.1882668   
2021 Radaeva M, Ban F, Zhang F, LeBlanc E, Lallous N, Rennie PS, Gleave ME, Cherkasov A. Development of Novel Inhibitors Targeting the D-Box of the DNA Binding Domain of Androgen Receptor. International Journal of Molecular Sciences. 22. PMID 33801338 DOI: 10.3390/ijms22052493   
2021 Zhang T, Hu W, Chen W. Plasma Membrane Integrates Biophysical and Biochemical Regulation to Trigger Immune Receptor Functions. Frontiers in Immunology. 12: 613185. PMID 33679752 DOI: 10.3389/fimmu.2021.613185   
2021 Chan KK, Tan TJC, Narayanan KK, Procko E. An engineered decoy receptor for SARS-CoV-2 broadly binds protein S sequence variants. Science Advances. 7. PMID 33597251 DOI: 10.1126/sciadv.abf1738   
2021 Jiang S, Iliopoulos-Tsoutsouvas C, Tong F, Brust CA, Keenan CM, Raghav JG, Hua T, Wu S, Ho JH, Wu Y, Grim TW, Zvonok N, Thakur GA, Liu ZJ, Sharkey KA, et al. Novel Functionalized Cannabinoid Receptor Probes: Development of Exceptionally Potent Agonists. Journal of Medicinal Chemistry. PMID 33761251 DOI: 10.1021/acs.jmedchem.0c02053   
2021 Gao J, Xu X, Huang K, Liang Z. Fungal G-Protein-Coupled Receptors: A Promising Mediator of the Impact of Extracellular Signals on Biosynthesis of Ochratoxin A. Frontiers in Microbiology. 12: 631392. PMID 33643259 DOI: 10.3389/fmicb.2021.631392   
2021 Branch JR, Bush TL, Pande V, Connolly PJ, Zhang Z, Hickson I, Ondrus J, Jaensch S, Bischoff JR, Habineza G, Van Hecke G, Meerpoel L, Packman K, Parrett CJ, Chong YT, et al. Discovery of JNJ-63576253, a next-generation androgen receptor antagonist active against wild-type and clinically-relevant ligand binding domain mutations in mCRPC. Molecular Cancer Therapeutics. PMID 33649102 DOI: 10.1158/1535-7163.MCT-20-0510   
2021 Lin C, Li J, Wu C, Bao J. Identifying selective agonists targeting LXRβ from terpene compounds of alismatis rhizoma. Journal of Molecular Modeling. 27: 91. PMID 33616795 DOI: 10.1007/s00894-021-04699-z   
2021 Nguyen AH, Lefkowitz RJ. Signaling at the endosome: cryo-EM structure of a GPCR-G protein-beta-arrestin megacomplex. The Febs Journal. PMID 33605032 DOI: 10.1111/febs.15773   
2021 Pezzanite LM, Chow L, Johnson V, Griffenhagen GM, Goodrich L, Dow S. Toll-like receptor activation of equine mesenchymal stromal cells to enhance antibacterial activity and immunomodulatory cytokine secretion. Veterinary Surgery : Vs. PMID 33797775 DOI: 10.1111/vsu.13628   
2021 Divine R, Dang HV, Ueda G, Fallas JA, Vulovic I, Sheffler W, Saini S, Zhao YT, Raj IX, Morawski PA, Jennewein MF, Homad LJ, Wan YH, Tooley MR, Seeger F, et al. Designed proteins assemble antibodies into modular nanocages. Science (New York, N.Y.). 372. PMID 33795432 DOI: 10.1126/science.abd9994   
2021 Cook LB, Ophardt HD, Shen R, Pratt BH, Galbier LA. Transcriptome analysis of ciliary-dependent MCH signaling in differentiating 3T3-L1 pre-adipocytes. Scientific Reports. 11: 4880. PMID 33649390 DOI: 10.1038/s41598-021-84138-4   
2021 Koretz KS, McGraw CE, Stradley S, Elbaradei A, Malmstadt N, Robinson AS. Characterization of binding kinetics of AR to Gα protein by surface plasmon resonance. Biophysical Journal. PMID 33675761 DOI: 10.1016/j.bpj.2021.02.032   
2021 Pedersen MH, Pham J, Mancebo H, Inoue A, Asher WB, Javitch JA. A novel luminescence-based-β-arrestin recruitment assay for unmodified receptors. The Journal of Biological Chemistry. 100503. PMID 33684444 DOI: 10.1016/j.jbc.2021.100503   
2021 Elek M, Djokovic N, Frank A, Oljacic S, Zivkovic A, Nikolic K, Stark H. Synthesis, in silico, and in vitro studies of novel dopamine D and D receptor ligands. Archiv Der Pharmazie. e2000486. PMID 33615541 DOI: 10.1002/ardp.202000486   
2021 Liu K, Shen L, Wu M, Liu ZJ, Hua T. Structural insights into the activation of chemokine receptor CXCR2. The Febs Journal. PMID 33835690 DOI: 10.1111/febs.15865   
2021 Sabu V, Krishnan S, Peter J, Aswathy IS, Lal Preethi SS, Simon M, Radhakrishna GP, Helen A. Synergistic effect of Betulinic acid, Apigenin and Skimmianine (BASk) in high cholesterol diet rabbit: Involvement of CD36-TLR2 signaling pathway. Cytokine. 142: 155475. PMID 33667961 DOI: 10.1016/j.cyto.2021.155475   
2021 Stoddart LA, Kilpatrick LE, Corriden R, Kellam B, Briddon SJ, Hill SJ. Efficient G protein coupling is not required for agonist-mediated internalization and membrane reorganization of the adenosine A receptor. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 35: e21211. PMID 33710641 DOI: 10.1096/fj.202001729RR   
2021 Qu C, Mao C, Xiao P, Shen Q, Zhong YN, Yang F, Shen DD, Tao X, Zhang H, Yan X, Zhao RJ, He J, Guan Y, Zhang C, Hou G, et al. Ligand recognition, unconventional activation, and G protein coupling of the prostaglandin E receptor EP2 subtype. Science Advances. 7. PMID 33811074 DOI: 10.1126/sciadv.abf1268   
2021 Freyn AW, Han J, Guthmiller JJ, Bailey MJ, Neu K, Turner HL, Rosado VC, Chromikova V, Huang M, Strohmeier S, Liu STH, Simon V, Krammer F, Ward AB, Palese P, et al. Influenza hemagglutinin-specific IgA Fc-effector functionality is restricted to stalk epitopes. Proceedings of the National Academy of Sciences of the United States of America. 118. PMID 33593910 DOI: 10.1073/pnas.2018102118   
2021 Chevigné A, Janji B, Meyrath M, Reynders N, D'Uonnolo G, Uchański T, Xiao M, Berchem G, Ollert M, Kwon YJ, Noman MZ, Szpakowska M. CXCL10 Is an Agonist of the CC Family Chemokine Scavenger Receptor ACKR2/D6. Cancers. 13. PMID 33801414 DOI: 10.3390/cancers13051054   
2021 Day CJ, Lo AW, Hartley-Tassell LE, Argente MP, Poole J, King NP, Tiralongo J, Jennings MP, Schembri MA. Discovery of Bacterial Fimbria-Glycan Interactions Using Whole-Cell Recombinant Escherichia coli Expression. Mbio. 12. PMID 33622724 DOI: 10.1128/mBio.03664-20   
2021 Deluigi M, Klipp A, Klenk C, Merklinger L, Eberle SA, Morstein L, Heine P, Mittl PRE, Ernst P, Kamenecka TM, He Y, Vacca S, Egloff P, Honegger A, Plückthun A. Complexes of the neurotensin receptor 1 with small-molecule ligands reveal structural determinants of full, partial, and inverse agonism. Science Advances. 7. PMID 33571132 DOI: 10.1126/sciadv.abe5504   
2021 Schierle S, Chaikuad A, Lillich FF, Ni X, Woltersdorf S, Schallmayer E, Renelt B, Ronchetti R, Knapp S, Proschak E, Merk D. Oxaprozin Analogues as Selective RXR Agonists with Superior Properties and Pharmacokinetics. Journal of Medicinal Chemistry. PMID 33793232 DOI: 10.1021/acs.jmedchem.1c00235