| Year |
Citation |
Score |
| 2019 |
More SS, Beach JM, McClelland C, Mokhtarzadeh A, Vince R. In Vivo Assessment of Retinal Biomarkers by Hyperspectral Imaging: Early Detection of Alzheimer's Disease. Acs Chemical Neuroscience. PMID 31603648 DOI: 10.1021/acschemneuro.9b00331 |
1 |
|
| 2019 |
Xie W, Xie J, Vince R, More SS. Guanabenz Attenuates Acetaminophen-Induced Liver Toxicity and Synergizes Analgesia in Mice. Chemical Research in Toxicology. PMID 31524377 DOI: 10.1021/acs.chemrestox.9b00162 |
1 |
|
| 2019 |
Singh R, Xie W, Williams J, Vince R, More SS. Discovery of anticancer clinical candidate, tosedostat, as an analgesic agent. Acs Chemical Neuroscience. PMID 31415151 DOI: 10.1021/acschemneuro.9b00230 |
1 |
|
| 2017 |
Singh R, Williams J, Vince R. Puromycin based inhibitors of aminopeptidases for the potential treatment of hematologic malignancies. European Journal of Medicinal Chemistry. 139: 325-336. PMID 28803047 DOI: 10.1016/j.ejmech.2017.07.048 |
1 |
|
| 2017 |
More SS, Nugent J, Vartak AP, Nye SM, Vince R. Hepatoprotective Effect of ψ-GSH in a Murine Model of Acetaminophen-Induced Liver Toxicity. Chemical Research in Toxicology. PMID 28165728 DOI: 10.1021/acs.chemrestox.6b00291 |
1 |
|
| 2016 |
More SS, Beach JM, Vince R. Early Detection of Amyloidopathy in Alzheimer's Mice by Hyperspectral Endoscopy. Investigative Ophthalmology & Visual Science. 57: 3231-8. PMID 27333181 DOI: 10.1167/iovs.15-17406 |
1 |
|
| 2016 |
Patterson SE, Moeller B, Nagasawa HT, Vince R, Crankshaw DL, Briggs J, Stutelberg MW, Vinnakota CV, Logue BA. Development of sulfanegen for mass cyanide casualties. Annals of the New York Academy of Sciences. PMID 27308865 DOI: 10.1111/nyas.13114 |
1 |
|
| 2016 |
Wezena CA, Urscher M, Vince R, More SS, Deponte M. Hemolytic and antimalarial effects of tight-binding glyoxalase 1 inhibitors on the host-parasite unit of erythrocytes infected with Plasmodium falciparum. Redox Biology. 8: 348-353. PMID 26972115 DOI: 10.1016/j.redox.2016.02.006 |
1 |
|
| 2015 |
Nugent JS, Vince R, Raza A. Topical Acyclothymidine Dinucleosides (aTds) Promote Non-UV-Mediated Endogenous Defense Mechanisms in Guinea Pig Skin. The Journal of Investigative Dermatology. 135: 1687-9. PMID 25699520 DOI: 10.1038/jid.2015.57 |
1 |
|
| 2015 |
More SS, Vince R. Hyperspectral imaging signatures detect amyloidopathy in Alzheimer's mouse retina well before onset of cognitive decline. Acs Chemical Neuroscience. 6: 306-15. PMID 25354367 DOI: 10.1021/cn500242z |
1 |
|
| 2014 |
Felczak K, Vince R, Pankiewicz KW. NAD-based inhibitors with anticancer potential. Bioorganic & Medicinal Chemistry Letters. 24: 332-6. PMID 24269162 DOI: 10.1016/j.bmcl.2013.11.005 |
1 |
|
| 2014 |
Raza A, Ericson ME, Nugent JS, Dreis CD, Vince R. A bio-mimetic approach to DNA photoprotection. The Journal of Investigative Dermatology. 134: 559-62. PMID 23938461 DOI: 10.1038/jid.2013.344 |
1 |
|
| 2013 |
More SS, Vartak AP, Vince R. Restoration of glyoxalase enzyme activity precludes cognitive dysfunction in a mouse model of Alzheimer's disease. Acs Chemical Neuroscience. 4: 330-8. PMID 23421684 DOI: 10.1021/cn3001679 |
1 |
|
| 2013 |
Patterson SE, Monteil AR, Cohen JF, Crankshaw DL, Vince R, Nagasawa HT. Cyanide antidotes for mass casualties: water-soluble salts of the dithiane (sulfanegen) from 3-mercaptopyruvate for intramuscular administration. Journal of Medicinal Chemistry. 56: 1346-9. PMID 23301495 DOI: 10.1021/jm301633x |
1 |
|
| 2013 |
Raza A, Dreis CD, Vince R. Photoprotection of DNA (in vitro) by acyclothymidine dinucleosides. Bioorganic & Medicinal Chemistry Letters. 23: 620-3. PMID 23290453 DOI: 10.1016/j.bmcl.2012.12.023 |
1 |
|
| 2012 |
More SS, Vince R. Potential of a γ-glutamyl-transpeptidase-stable glutathione analogue against amyloid-β toxicity. Acs Chemical Neuroscience. 3: 204-10. PMID 22860189 DOI: 10.1021/cn200113z |
1 |
|
| 2012 |
Chen YL, Zacharias J, Vince R, Geraghty RJ, Wang Z. C-6 aryl substituted 4-quinolone-3-carboxylic acids as inhibitors of hepatitis C virus. Bioorganic & Medicinal Chemistry. 20: 4790-800. PMID 22748708 DOI: 10.1016/j.bmc.2012.05.066 |
1 |
|
| 2012 |
More SS, Vartak AP, Vince R. The butter flavorant, diacetyl, exacerbates β-amyloid cytotoxicity. Chemical Research in Toxicology. 25: 2083-91. PMID 22731744 DOI: 10.1021/tx3001016 |
1 |
|
| 2012 |
Singh R, Vince R. 2-Azabicyclo[2.2.1]hept-5-en-3-one: chemical profile of a versatile synthetic building block and its impact on the development of therapeutics. Chemical Reviews. 112: 4642-86. PMID 22681478 DOI: 10.1021/cr2004822 |
1 |
|
| 2012 |
Urscher M, More SS, Alisch R, Vince R, Deponte M. Tight-binding inhibitors efficiently inactivate both reaction centers of monomeric Plasmodium falciparum glyoxalase 1. The Febs Journal. 279: 2568-78. PMID 22607473 DOI: 10.1111/j.1742-4658.2012.08640.x |
1 |
|
| 2012 |
Belani KG, Singh H, Beebe DS, George P, Patterson SE, Nagasawa HT, Vince R. Cyanide toxicity in juvenile pigs and its reversal by a new prodrug, sulfanegen sodium. Anesthesia and Analgesia. 114: 956-61. PMID 22392971 DOI: 10.1213/ANE.0b013e31824c4eb5 |
1 |
|
| 2012 |
More SS, Raza A, Vince R. The butter flavorant, diacetyl, forms a covalent adduct with 2-deoxyguanosine, uncoils DNA, and leads to cell death. Journal of Agricultural and Food Chemistry. 60: 3311-7. PMID 22385266 DOI: 10.1021/jf300180e |
1 |
|
| 2012 |
Chen YL, Tang J, Kesler MJ, Sham YY, Vince R, Geraghty RJ, Wang Z. The design, synthesis and biological evaluations of C-6 or C-7 substituted 2-hydroxyisoquinoline-1,3-diones as inhibitors of hepatitis C virus. Bioorganic & Medicinal Chemistry. 20: 467-79. PMID 22100256 DOI: 10.1016/j.bmc.2011.10.058 |
1 |
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| 2011 |
Tang J, Maddali K, Dreis CD, Sham YY, Vince R, Pommier Y, Wang Z. N-3 Hydroxylation of Pyrimidine-2,4-diones Yields Dual Inhibitors of HIV Reverse Transcriptase and Integrase. Acs Medicinal Chemistry Letters. 2: 63-67. PMID 21499541 DOI: 10.1021/ml1002162 |
1 |
|
| 2011 |
Raza A, Vince R. Dehydroascorbic acid adducts of guanosine residues: possible biological implications. Chembiochem : a European Journal of Chemical Biology. 12: 1015-7. PMID 21425230 DOI: 10.1002/cbic.201000748 |
1 |
|
| 2011 |
Tang J, Maddali K, Dreis CD, Sham YY, Vince R, Pommier Y, Wang Z. 6-Benzoyl-3-hydroxypyrimidine-2,4-diones as dual inhibitors of HIV reverse transcriptase and integrase. Bioorganic & Medicinal Chemistry Letters. 21: 2400-2. PMID 21392991 DOI: 10.1016/j.bmcl.2011.02.069 |
1 |
|
| 2011 |
Tang J, Maddali K, Metifiot M, Sham YY, Vince R, Pommier Y, Wang Z. 3-Hydroxypyrimidine-2,4-diones as an inhibitor scaffold of HIV integrase. Journal of Medicinal Chemistry. 54: 2282-92. PMID 21381765 DOI: 10.1021/jm1014378 |
1 |
|
| 2011 |
Felczak K, Chen L, Wilson D, Williams J, Vince R, Petrelli R, Jayaram HN, Kusumanchi P, Kumar M, Pankiewicz KW. Cofactor-type inhibitors of inosine monophosphate dehydrogenase via modular approach: targeting the pyrophosphate binding sub-domain. Bioorganic & Medicinal Chemistry. 19: 1594-605. PMID 21324702 DOI: 10.1016/j.bmc.2011.01.042 |
1 |
|
| 2010 |
Wang Z, Tang J, Salomon CE, Dreis CD, Vince R. Pharmacophore and structure-activity relationships of integrase inhibition within a dual inhibitor scaffold of HIV reverse transcriptase and integrase. Bioorganic & Medicinal Chemistry. 18: 4202-11. PMID 20576573 DOI: 10.1016/j.bmc.2010.05.004 |
1 |
|
| 2010 |
Lu D, Sham YY, Vince R. Design, asymmetric synthesis, and evaluation of pseudosymmetric sulfoximine inhibitors against HIV-1 protease. Bioorganic & Medicinal Chemistry. 18: 2037-48. PMID 20138769 DOI: 10.1016/j.bmc.2010.01.020 |
1 |
|
| 2009 |
More SS, Vince R. Inhibition of glyoxalase I: the first low-nanomolar tight-binding inhibitors. Journal of Medicinal Chemistry. 52: 4650-6. PMID 19610604 DOI: 10.1021/jm900382u |
1 |
|
| 2008 |
Raza A, Sham YY, Vince R. Design and synthesis of sulfoximine based inhibitors for HIV-1 protease. Bioorganic & Medicinal Chemistry Letters. 18: 5406-10. PMID 18829317 DOI: 10.1016/j.bmcl.2008.09.044 |
1 |
|
| 2008 |
More SS, Vince R. Design, synthesis and biological evaluation of glutathione peptidomimetics as components of anti-Parkinson prodrugs. Journal of Medicinal Chemistry. 51: 4581-8. PMID 18651729 DOI: 10.1021/jm800239v |
1 |
|
| 2008 |
Wang Z, Vince R. Design and synthesis of dual inhibitors of HIV reverse transcriptase and integrase: introducing a diketoacid functionality into delavirdine. Bioorganic & Medicinal Chemistry. 16: 3587-95. PMID 18314335 DOI: 10.1016/j.bmc.2008.02.007 |
1 |
|
| 2008 |
Wang Z, Vince R. Synthesis of pyrimidine and quinolone conjugates as a scaffold for dual inhibitors of HIV reverse transcriptase and integrase. Bioorganic & Medicinal Chemistry Letters. 18: 1293-6. PMID 18226894 DOI: 10.1016/j.bmcl.2008.01.025 |
1 |
|
| 2008 |
Lu D, Vince R. Corrigendum to "Discovery of potent HIV-1 protease inhibitors incorporating sulfoximine functionality" [Bioorg. Med. Chem. Lett. 17 (2007) 5614-5619] (DOI:10.1016/j.bmcl.2007.07.095) Bioorganic and Medicinal Chemistry Letters. 18: 2228. DOI: 10.1016/j.bmcl.2008.02.004 |
1 |
|
| 2008 |
Vince R. A brief history of the development of ziagen Chemtracts. 21: 127-134. |
1 |
|
| 2007 |
Nagasawa HT, Goon DJ, Crankshaw DL, Vince R, Patterson SE. Novel, orally effective cyanide antidotes. Journal of Medicinal Chemistry. 50: 6462-4. PMID 18038966 DOI: 10.1021/jm7011497 |
1 |
|
| 2007 |
Lu D, Vince R. Discovery of potent HIV-1 protease inhibitors incorporating sulfoximine functionality. Bioorganic & Medicinal Chemistry Letters. 17: 5614-9. PMID 17822899 DOI: 10.1016/j.bmcl.2007.07.095 |
1 |
|
| 2007 |
Wang Z, Bennett EM, Wilson DJ, Salomon C, Vince R. Rationally designed dual inhibitors of HIV reverse transcriptase and integrase. Journal of Medicinal Chemistry. 50: 3416-9. PMID 17608468 DOI: 10.1021/jm070512p |
1 |
|
| 2007 |
More SS, Vince R. Design, synthesis, and binding studies of bidentate Zn-chelating peptidic inhibitors of glyoxalase-I. Bioorganic & Medicinal Chemistry Letters. 17: 3793-7. PMID 17513107 DOI: 10.1016/j.bmcl.2006.12.056 |
1 |
|
| 2007 |
Pham PT, Vince R. Carbovir-related compounds and phosphonate analogues Phosphorus, Sulfur and Silicon and the Related Elements. 182: 779-791. DOI: 10.1080/10426500601047578 |
1 |
|
| 2006 |
Vince R, Hua M. Synthesis of carbovir and abacavir from a carbocyclic precursor. Current Protocols in Nucleic Acid Chemistry / Edited by Serge L. Beaucage ... [Et Al.]. Unit 14.4. PMID 18428951 DOI: 10.1002/0471142700.nc1404s25 |
1 |
|
| 2006 |
More SS, Vince R. A metabolically stable tight-binding transition-state inhibitor of glyoxalase-I. Bioorganic & Medicinal Chemistry Letters. 16: 6039-42. PMID 16997560 DOI: 10.1016/j.bmcl.2006.08.121 |
1 |
|
| 2006 |
Tang Y, Muthyala R, Vince R. Synthesis and biological evaluation of carboacyclic nucleosides with (Z) and (E)-9-[4,4-bis(hydroxymethyl)]-2-butenyl side chain. Bioorganic & Medicinal Chemistry. 14: 5866-75. PMID 16759867 DOI: 10.1016/j.bmc.2006.05.029 |
1 |
|
| 2006 |
Li X, Vince R. Synthesis and biological evaluation of purine derivatives incorporating metal chelating ligands as HIV integrase inhibitors. Bioorganic & Medicinal Chemistry. 14: 5742-55. PMID 16753300 DOI: 10.1016/j.bmc.2006.04.011 |
1 |
|
| 2006 |
Li X, Vince R. Conformationally restrained carbazolone-containing alpha,gamma-diketo acids as inhibitors of HIV integrase. Bioorganic & Medicinal Chemistry. 14: 2942-55. PMID 16386908 DOI: 10.1016/j.bmc.2005.12.013 |
1 |
|
| 2004 |
Muthyala R, Vince R. Vinyl and aryl metals Comprehensive Organic Functional Group Transformations Ii. 2: 1025-1057. |
1 |
|
| 2002 |
Quirk Dorr DR, Vince R. Synthesis and biological evaluation of endocyclic 2',3'-didehydro-2',3'-dideoxymethanocarba adenosine. Nucleosides, Nucleotides & Nucleic Acids. 21: 665-80. PMID 12502282 DOI: 10.1002/chin.200318194 |
1 |
|
| 2002 |
Bhushan RG, Vince R. Synthesis of conformationally restricted 2',3'-exo-methylene carbocyclic nucleosides built on a bicyclo[3.1.0]hexane template. Bioorganic & Medicinal Chemistry. 10: 2325-33. PMID 11983530 DOI: 10.1016/S0968-0896(02)00063-9 |
1 |
|
| 2000 |
Parker WB, Shaddix SC, Rose LM, Pham PT, Hua M, Vince R. Metabolism of O6-propyl and N6-propyl-carbovir in CEM cells. Nucleosides, Nucleotides & Nucleic Acids. 19: 795-804. PMID 10960036 DOI: 10.1080/15257770008035025 |
1 |
|
| 1999 |
Antle VD, Donat N, Hua M, Liao PL, Vince R, Carperelli CA. Substrate specificity of human glycinamide ribonucleotide transformylase. Archives of Biochemistry and Biophysics. 370: 231-5. PMID 10577357 DOI: 10.1006/abbi.1999.1428 |
1 |
|
| 1999 |
Vince R, Brownell J, Akella LB. Synthesis and activity of γ-(L-γ-azaglutamyl)-S-(p-bromobenzyl)-L- cysteinylglycine: A metabolically stable inhibitor of glyoxalase I Bioorganic and Medicinal Chemistry Letters. 9: 853-856. PMID 10206549 DOI: 10.1016/S0960-894X(99)00097-9 |
1 |
|
| 1998 |
Katagiri N, Kokufuda H, Makino M, Vince R, Kaneko C. Deamination of cyclaradine by adenosine deaminase under high pressure Nucleosides and Nucleotides. 17: 81-89. PMID 9708342 |
1 |
|
| 1997 |
Katagiri N, Kokufuda H, Makino M, Matsuhashi Y, Kaneko C, Vince R. A highly efficient synthesis of cyclaradine and its behaviour towards adenosine deaminase Nucleic Acids Symposium Series. 3-4. PMID 9585970 |
1 |
|
| 1997 |
Parker WB, Shaddix SC, Vince R, Bennett LL. Lack of mitochondrial toxicity in CEM cells treated with carbovir Antiviral Research. 34: 131-136. PMID 9191020 DOI: 10.1016/S0166-3542(97)01033-4 |
1 |
|
| 1996 |
Konkel MJ, Vince R. Palladium-Catalyzed Allylic Coupling of 1,2,3-Triazolo[4,5-d]pyrimidines (8-Azapurines). The Journal of Organic Chemistry. 61: 6199-6204. PMID 11667455 DOI: 10.1021/jo960815j |
1 |
|
| 1996 |
Antle VD, Liu D, McKellar BR, Caperelli CA, Hua M, Vince R. Substrate specificity of glycinamide ribonucleotide synthetase from chicken liver. The Journal of Biological Chemistry. 271: 8192-5. PMID 8626510 DOI: 10.1074/jbc.271.14.8192 |
1 |
|
| 1996 |
Antle VD, Liu D, McKellars BR, Caperelli CA, Hua M, Vince R. Substrate specificity of glycinamide ribonucleotide transformylase from chicken liver. The Journal of Biological Chemistry. 271: 6045-9. PMID 8626389 DOI: 10.1074/jbc.271.11.6045 |
1 |
|
| 1996 |
Konkel MJ, Vince R. Cyclohexenyl nucleosides: Synthesis and biological activity of trans-3-(purin-9-yl)-4-cyclohexenylcarbinols Tetrahedron. 52: 8969-8978. DOI: 10.1016/0040-4020(96)00445-0 |
1 |
|
| 1996 |
Akella LB, Vince R. Enantioselective synthesis of 2-[5-(9H-purin-9-yl)-2-cyclopenten-1-yl]-ethanol analogues as potential antiviral agents Tetrahedron. 52: 8407-8412. DOI: 10.1016/0040-4020(96)00412-7 |
1 |
|
| 1996 |
Akella LB, Vince R. Palladium-catalyzed synthesis of cw-2-[4-(9H-purin-9-yl)-2-cyclopenten-1-yl]ethanol analogues Tetrahedron. 52: 2789-2794. DOI: 10.1016/0040-4020(96)00015-4 |
1 |
|
| 1996 |
Konkel MJ, Vince R. Cyclohexenyl nucleosides: Synthesis of cis-4-(9H-purin-9-yl)-2-cyclohexenylcarbinols Tetrahedron. 52: 799-808. DOI: 10.1016/0040-4020(95)00926-4 |
1 |
|
| 1996 |
Vince R, Hua M, Caperelli CA. Phosphonate analogs of carbocyclic phosphoribosylamine and carbocyclic glycinamide ribonucleotide Nucleosides and Nucleotides. 15: 1711-1718. |
1 |
|
| 1995 |
Wen YD, Remmel RP, Pham PT, Vince R, Zimmerman CL. Comparative brain exposure to (-)-carbovir after (-)-carbovir or (-)-6-aminocarbovir intravenous infusion in rats. Pharmaceutical Research. 12: 911-5. PMID 7667200 DOI: 10.1023/A:1016229624703 |
1 |
|
| 1995 |
Vince R, Brownell J, Beers SA. 6-Deoxycarbovir: A Xanthine Oxidase Activated Prodrug Of Carbovir Nucleosides and Nucleotides. 14: 39-44. DOI: 10.1080/15257779508014651 |
1 |
|
| 1995 |
Konkel MJ, Vince R. Synthesis and Biological Activity of Cyclohexenyl Nucleosides, cis-5-(9H-Purin-9-YL)-3-Cyclohexenyl Carbinols and their 8-Azapurinyl Analogs Nucleosides and Nucleotides. 14: 2061-2077. DOI: 10.1080/15257779508010724 |
1 |
|
| 1995 |
Vince R, Pham PT. The Synthesis and Biological Evaluation of Sulfamoyl Nucleosides Related to Carbovir and Azt Nucleosides and Nucleotides. 14: 2051-2060. DOI: 10.1080/15257779508010723 |
1 |
|
| 1995 |
Vince R, Kilama J, Pham PT, Beers SA, Bowdon BJ, Keith KA, Parker WB. 6-substituted derivatives of carbovir: Anti-HIV activity Nucleosides and Nucleotides. 14: 1703-1708. DOI: 10.1080/15257779508009751 |
1 |
|
| 1993 |
Parker WB, Shaddix SC, Bowdon BJ, Rose LM, Vince R, Shannon WM, Bennett LL. Metabolism of carbovir, a potent inhibitor of human immunodeficiency virus type 1, and its effects on cellular metabolism Antimicrobial Agents and Chemotherapy. 37: 1004-1009. PMID 7685993 |
1 |
|
| 1992 |
Peterson EM, Brownell J, Vince R. Synthesis and biological evaluation of 5'-sulfamoylated purinyl carbocyclic nucleosides. Journal of Medicinal Chemistry. 35: 3991-4000. PMID 1433208 |
1 |
|
| 1992 |
Zimmerman CL, Remmel RP, Ibrahim SS, Beers SA, Vince R. Pharmacokinetic evaluation of (-)-6-aminocarbovir as a prodrug for (-)-carbovir in rats. Drug Metabolism and Disposition: the Biological Fate of Chemicals. 20: 47-51. PMID 1346995 |
1 |
|
| 1991 |
Vince R. Synthesis and anti-HIV activity of carbovir and related carbocyclic nucleosides Nucleic Acids Symposium Series. 193-194. PMID 1842080 |
1 |
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| 1991 |
Parker WB, White EL, Shaddix SC, Ross LJ, Buckheit RW, Germany JM, Secrist JA, Vince R, Shannon WM. Mechanism of inhibition of human immunodeficiency virus type 1 reverse transcriptase and human DNA polymerases α, β, and γ by the 5′-triphosphates of carbovir, 3′-azido-3′-deoxythymidine, 2′,3′-dideoxyguanosine, and 3′-deoxythymidine: A novel RNA template for the evaluation of antiretroviral drugs Journal of Biological Chemistry. 266: 1754-1762. PMID 1703154 |
1 |
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| 1991 |
Peterson ML, Vince R. Synthesis and biological evaluation of 4-purinylpyrrolidine nucleosides Journal of Medicinal Chemistry. 34: 2787-2797. PMID 1654429 DOI: 10.1021/jm00113a017 |
1 |
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| 1990 |
Vince R, Brownell J. Resolution of racemic carbovir and selective inhibition of human immunodeficiency virus by the (-) enantiomer Biochemical and Biophysical Research Communications. 168: 912-916. PMID 2346492 DOI: 10.1016/0006-291X(90)91115-9 |
1 |
|
| 1990 |
Vince R, Hua M. Synthesis and anti-HIV activity of carbocyclic 2',3'-didehydro-2',3'-dideoxy 2,6-disubstituted purine nucleosides. Journal of Medicinal Chemistry. 33: 17-21. PMID 2296018 |
1 |
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| 1990 |
Bondoc LL, Shannon WM, Secrist JA, Vince R, Fridland A. Metabolism of the carbocyclic nucleoside analogue carbovir, an inhibitor of human immunodeficiency virus, in human lymphoid cells Biochemistry. 29: 9839-9843. PMID 2271622 |
1 |
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| 1990 |
Peterson ML, Vince R. Synthesis and biological evaluation of carbocyclic analogues of lyxofuranosides of 2-amino-6-substituted-purines and 2-amino-6-substituted-8-azapurines Journal of Medicinal Chemistry. 33: 1214-1219. PMID 2157013 DOI: 10.1021/jm00166a020 |
1 |
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| 1989 |
Remmel RP, Yeom YH, Hua M, Vince R, Zimmerman CL. Liquid chromatographic assay of carbovir, a carbocyclic nucleoside active against human immunodeficiency virus. Journal of Chromatography. 489: 323-31. PMID 2753956 DOI: 10.1016/S0378-4347(00)82910-2 |
1 |
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| 1989 |
Yeom YH, Remmel RP, Huang SH, Hua M, Vince R, Zimmerman CL. Pharmacokinetics and bioavailability of carbovir, a carbocyclic nucleoside active against human immunodeficiency virus, in rats. Antimicrobial Agents and Chemotherapy. 33: 171-5. PMID 2719460 |
1 |
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| 1989 |
White EL, Parker WB, Macy LJ, Shaddix SC, McCaleb G, Secrist JA, Vince R, Shannon WM. Comparison of the effect of Carbovir, AZT, and dideoxynucleoside triphosphates on the activity of human immunodeficiency virus reverse transcriptase and selected human polymerases Biochemical and Biophysical Research Communications. 161: 393-398. PMID 2472136 DOI: 10.1016/0006-291X(89)92611-9 |
1 |
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| 1989 |
Vince R, Lavelle GC, Hua M, Qualls J, Brownell J, Shannon WM. Carbovir: A carbocyclic nucleoside with potent and selective activity against human immunodeficiency virus (HIV) in vitro Nucleosides and Nucleotides. 8: 1127-1128. DOI: 10.1080/07328318908054307 |
1 |
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| 1988 |
Vince R, Hua M, Brownell J, Daluge S, Lee FC, Shannon WM, Lavelle GC, Qualls J, Weislow OS, Kiser R. Potent and selective activity of a new carbocyclic nucleoside analog (carbovir: NSC 614846) against human immunodeficiency virus in vitro. Biochemical and Biophysical Research Communications. 156: 1046-53. PMID 2847711 DOI: 10.1016/S0006-291X(88)80950-1 |
1 |
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| 1987 |
Hua M, Korkowski PM, Vince R. Synthesis and biological evaluation of acyclic neplanocin analogues. Journal of Medicinal Chemistry. 30: 198-200. PMID 3027333 |
1 |
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| 1987 |
Vince R, Turakhia RH, Shannon WM, Arnett G. Synthesis and antiviral activity of carbocyclic analogues of xylofuranosides of 2-amino-6-substituted-purines and 2-amino-6-substituted-8-azapurines Journal of Medicinal Chemistry. 30: 2026-2030. PMID 2822928 |
1 |
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| 1986 |
Vince R, Daluge S, Brownell J. Carbocyclic puromycin: Synthesis and inhibition of protein biosynthesis Journal of Medicinal Chemistry. 29: 2400-2403. PMID 3783599 |
1 |
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| 1986 |
Dunham EW, Vince R. Hypotensive and renal vasodilator effects of carbocyclic adenosine (aristeromycin) in anesthetized spontaneously hypertensive rats Journal of Pharmacology and Experimental Therapeutics. 238: 954-959. PMID 3018227 |
1 |
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| 1984 |
Vince R, Brownell J, Daluge S. Carbocyclic analogues of xylofuranosylpurine nucleosides. Synthesis and antitumor activity Journal of Medicinal Chemistry. 27: 1358-1360. PMID 6481772 |
1 |
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| 1984 |
McFarlan SC, Vince R. Inhibition of peptidyltransferase and possible mode of action of a dipeptidyl chloramphenicol analog Biochemical and Biophysical Research Communications. 122: 748-754. PMID 6380501 DOI: 10.1016/S0006-291X(84)80097-2 |
1 |
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| 1983 |
Vince R, Daluge S, Lee H, Shannon WM, Arnett G, Schafer TW, Nagabhushan TL, Reichert P, Tsai H. Carbocyclic arabinofuranosyladenine (cyclaradine): efficacy against genital herpes in guinea pigs. Science (New York, N.Y.). 221: 1405-6. PMID 6684328 |
1 |
|
| 1983 |
Shannon WM, Westbrook L, Arnett G, Daluge S, Lee H, Vince R. Comparison of the efficacy of vidarabine, its carbocyclic analog (cyclaradine), and cyclaradine-5'-methoxyacetate in the treatment of herpes simplex virus type 1 encephalitis in mice Antimicrobial Agents and Chemotherapy. 24: 538-543. PMID 6651280 |
1 |
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| 1981 |
Vince R, Lee H, Narang AS, Shirota FN. 5′-Chloropuromycin. Inhibition of protein synthesis and antitrypanosomal activity Journal of Medicinal Chemistry. 24: 1511-1514. PMID 7310828 |
1 |
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| 1981 |
Lee H, Fong KL, Vince R. Puromycin analogues. Effect of aryl-substituted puromycin analogues on the ribosomal peptidyltransferase reaction Journal of Medicinal Chemistry. 24: 304-308. PMID 7265117 |
1 |
|
| 1981 |
Cermak RC, Vince R. (±) 4β-amino-2α,3α-dihydroxy-1β-cyclopentanemethanol hydrochloride. Carbocyclic ribofuranosylamine for the synthesis of carbocyclic nucleosides Tetrahedron Letters. 22: 2331-2332. DOI: 10.1016/S0040-4039(01)82898-7 |
1 |
|
| 1980 |
Lee H, Vince R. Carbocyclic analogs of arabinosylpurine nucleosides Journal of Pharmaceutical Sciences. 69: 1019-1021. PMID 6251197 |
1 |
|
| 1980 |
Vince R, Daluge S. Facile synthesis of carbocyclic lyxo- and ribonucleosides Journal of Organic Chemistry. 45: 531-533. |
1 |
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| 1979 |
Broom AD, Amarnath V, Vince R, Brownell J. Poly(2-fluoroadenylic acid) The role of basicity in the stabilization of complementary helices Bba Section Nucleic Acids and Protein Synthesis. 563: 508-517. PMID 37911 DOI: 10.1016/0005-2787(79)90069-8 |
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| 1978 |
Fong KLL, Vince R. Peptidyl transferase substrate specificity with nonaromatic aminoacyl analogues of puromycin Journal of Medicinal Chemistry. 21: 792-795. PMID 691004 |
1 |
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| 1978 |
Vince R. Photoaffinity labeling of the ribosomal peptidyl transferase site with synthetic puromycin analogues Biochemistry. 17: 5489-5493. PMID 365231 |
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| 1978 |
Brandt Rauf P, Vince R, LeMahieu R, Pestlea S. Fluorescent assay for estimating the biding of erythromycin derivatives to ribosomes Antimicrobial Agents and Chemotherapy. 14: 88-94. PMID 356727 |
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| 1978 |
Vince R, Fong KLL. Peptidyl transferase substrate activity and inhibition of protein biosynthesis by a hydrophilic-aminoacyl analogue of puromycin Biochemical and Biophysical Research Communications. 81: 559-564. PMID 352348 DOI: 10.1016/0006-291X(78)91571-1 |
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| 1978 |
Lee CK, Vince R. Effect of sparsomycin analogues on the puromycin-peptidyl transferase reaction on ribosomes Journal of Medicinal Chemistry. 21: 176-179. PMID 340693 |
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| 1978 |
Daluge S, Vince R. Synthesis of carbocyclic aminonucleosides Journal of Organic Chemistry. 43: 2311-2320. |
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| 1977 |
Vince R, Brownell J, Kiu Lee C. Inhibition of protein biosynthesis: The first active sparsomycin analog Biochemical and Biophysical Research Communications. 75: 563-567. PMID 856177 DOI: 10.1016/0006-291X(77)91509-1 |
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| 1977 |
Lyon PA, Vince R. Synthesis and kinetic evaluation of S- and N-substituted cysteinylglycines as inhibitors of glyoxalase I Journal of Medicinal Chemistry. 20: 77-80. PMID 833829 |
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| 1977 |
Vince R, Daluge S. Synthesis of cyclohexyl carbocyclic puromycin and its inhibition of protein synthesis Journal of Medicinal Chemistry. 20: 930-934. PMID 327067 |
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| 1977 |
Langlois R, Cantor CR, Vince R, Pestka S. Interaction between the Erythromycin and chloramphenicol binding sites on the Escherichia coli ribosome Biochemistry. 16: 2349-2356. PMID 324517 DOI: 10.1021/bi00630a007 |
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| 1977 |
Narang AS, Vince R. 1,2,4-Triazole amino nucleosides. 1-β-D-3′-amino-3′-deoxyribofuranosyl-1,2,4-triazole-3- carboxamide and related nucleosides Journal of Medicinal Chemistry. 20: 1684-1687. PMID 201758 |
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| 1977 |
Vince R, Daluge S. Carbocyclic arabinosyladenine, an adenosine deaminase resistant antiviral agent Journal of Medicinal Chemistry. 20: 612-613. PMID 191615 |
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| 1976 |
Pestka S, Vince R, LeMahieu R, Weiss F, Fern L, Unowsky J. Induction of erythromycin resistance in Staphyloccus aureus by erythromycin derivatives. Antimicrobial Agents and Chemotherapy. 9: 128-30. PMID 1259386 |
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| 1976 |
Pestka S, Weiss D, Vince R, Wienen B, Stöffler G, Smith I. Thiostrepton-resistant mutants of Bacillus subtilis: Localization of resistance to the 50S subunit Mgg Molecular & General Genetics. 144: 235-241. PMID 818503 DOI: 10.1007/BF00341721 |
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| 1976 |
Vince R, Weiss D, Gordon J, Howard G, Smith I, Pestka S. Binding of thiostrepton to ribosomes from thiostrepton sensitive and -resistant Bacillus subtilis strains Antimicrobial Agents and Chemotherapy. 9: 665-667. PMID 817664 |
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| 1976 |
Langlois R, Lee CC, Cantor CR, Vince R, Pestka S. The distance between two functionally significant regions of the 50 S Escherichia coli ribosome: the erythromycin binding site and proteins L7 L12 Journal of Molecular Biology. 106: 297-313. PMID 789892 DOI: 10.1016/0022-2836(76)90087-5 |
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| 1976 |
Pestka S, Weiss D, Vince R. Partition of ribosomes in two-polymer aqueous phase systems Analytical Biochemistry. 71: 137-142. PMID 776031 DOI: 10.1016/0003-2697(76)90020-8 |
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| 1976 |
Vince R, Weiss D, Pestka S. Binding of N substituted erythromycylamines to ribosomes Antimicrobial Agents and Chemotherapy. 9: 131-136. PMID 769668 |
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| 1976 |
Vince R, Almquist RG, Ritter CL, Shirota FN, Nagasawa HT. An active puromycin analog derived from a non nephrotoxic aminonucleoside Life Sciences. 18: 345-350. PMID 768682 DOI: 10.1016/S0140-6736(76)93103-2 |
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| 1976 |
Daluge S, Vince R. A synthetic route to carbocyclic aminonucleosides Tetrahedron Letters. 17: 3005-3008. DOI: 10.1016/0040-4039(76)80055-X |
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| 1976 |
Vince R, Almquist RG, Ritter CL, Shirota FN, Nagasawa HT. An active puromycin analog derived from a non-nephrotoxic aminonucleoside Life Sciences. 18: 345-349. DOI: 10.1016/0024-3205(76)90063-1 |
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| 1976 |
Pestka S, Weiss D, Vince R, Wienen B, Stöffler G, Smith I. Errata Mgg Molecular & General Genetics. 147: 233. DOI: 10.1007/BF00267576 |
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| 1971 |
Schaeffer HJ, Gurwara S, Vince R, Bittner S. Novel substrate of adenosine deaminase. Journal of Medicinal Chemistry. 14: 367-9. PMID 5553754 |
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| 1968 |
Schaeffer HJ, Vince R. Enzyme inhibitors. XIX. The synthesis of some 1-hydroxy-2-hydroxymethyl-4-(6-substituted-9-purinyl)cyclohexanes as nucleoside analogs. Journal of Medicinal Chemistry. 11: 15-20. PMID 5637163 |
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| 1967 |
Schaeffer HJ, Vince R. Enzyme inhibitors. 18. Studies on the stereoselectivity of inhibition of adenosine deaminase by DL-, D-, and L-9-(2-hydroxypropyl)adenine. Journal of Medicinal Chemistry. 10: 689-91. PMID 6037062 |
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| 1965 |
SCHAEFFER HJ, VINCE R. ENZYME INHIBITORS. VI. STUDIES ON THE BULK TOLERANCE OF ADENOSINE DEAMINASE FOR 6-SUBSTITUTED AMINO-9-(3-HYDROXYPROPYL)PURINES. Journal of Medicinal Chemistry. 8: 33-5. PMID 14287263 |
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| 1965 |
Schaeffer HJ, Gvogel D, Vince R. Enzyme inhibitors. 8. Studies on the mode of binding of some 6-substituted 9-(hydroxyalkyl)purines to adenosine deaminase. Journal of Medicinal Chemistry. 8: 502-6. PMID 5883714 |
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