| Year |
Citation |
Score |
| 2023 |
Dobariya P, Xie W, Rao SP, Xie J, Seelig DM, Vince R, Lee MK, More SS. Deletion of Glyoxalase 1 exacerbates acetaminophen-induced hepatotoxicity in mice. Biorxiv : the Preprint Server For Biology. PMID 38187538 DOI: 10.1101/2023.12.21.572856 |
0.537 |
|
| 2023 |
Xie W, Jiang R, Xie J, Vince R, More SS. Geometric Isomer of Guanabenz Confers Hepatoprotection to a Murine Model of Acetaminophen Toxicity. Chemical Research in Toxicology. PMID 37348131 DOI: 10.1021/acs.chemrestox.3c00047 |
0.536 |
|
| 2022 |
Xie W, Cao B, Zhu H, Raza A, Juckel N, Xie J, Jiang R, Vince R, Lee MK, More SS. Orally Bioavailable Prodrugs of ψ-GSH: A Potential Treatment for Alzheimer's Disease. Journal of Medicinal Chemistry. 65: 14441-14455. PMID 36353871 DOI: 10.1021/acs.jmedchem.2c00779 |
0.571 |
|
| 2022 |
Rao SP, Xie W, Christopher Kwon YI, Juckel N, Xie J, Dronamraju VR, Vince R, Lee MK, More SS. Sulfanegen stimulates 3-mercaptopyruvate sulfurtransferase activity and ameliorates Alzheimer's disease pathology and oxidative stress in vivo. Redox Biology. 57: 102484. PMID 36183541 DOI: 10.1016/j.redox.2022.102484 |
0.555 |
|
| 2022 |
Raza A, Xie W, Kim KH, Dronamraju VR, Williams J, Vince R, More SS. Dipeptide of ψ-GSH Inhibits Oxidative Stress and Neuroinflammation in an Alzheimer's Disease Mouse Model. Antioxidants (Basel, Switzerland). 11. PMID 35739972 DOI: 10.3390/antiox11061075 |
0.574 |
|
| 2021 |
Beach JM, Rizvi M, Lichtenfels CB, Vince R, More SS. Topical Review: Studies of Ocular Function and Disease Using Hyperspectral Imaging. Optometry and Vision Science : Official Publication of the American Academy of Optometry. PMID 34897230 DOI: 10.1097/OPX.0000000000001853 |
0.498 |
|
| 2021 |
Christopher Kwon YI, Xie W, Zhu H, Xie J, Shinn K, Juckel N, Vince R, More SS, Lee MK. γ-Glutamyl-Transpeptidase-Resistant Glutathione Analog Attenuates Progression of Alzheimer's Disease-like Pathology and Neurodegeneration in a Mouse Model. Antioxidants (Basel, Switzerland). 10. PMID 34829667 DOI: 10.3390/antiox10111796 |
0.537 |
|
| 2021 |
Xie W, Kim KH, Vince R, More SS. The Amyloid Aggregation Accelerator Diacetyl Prevents Cognitive Decline in Alzheimer's Mouse Models. Chemical Research in Toxicology. PMID 33857375 DOI: 10.1021/acs.chemrestox.1c00089 |
0.529 |
|
| 2019 |
More SS, Beach JM, McClelland C, Mokhtarzadeh A, Vince R. In Vivo Assessment of Retinal Biomarkers by Hyperspectral Imaging: Early Detection of Alzheimer's Disease. Acs Chemical Neuroscience. PMID 31603648 DOI: 10.1021/Acschemneuro.9B00331 |
0.56 |
|
| 2019 |
Xie W, Xie J, Vince R, More SS. Guanabenz Attenuates Acetaminophen-Induced Liver Toxicity and Synergizes Analgesia in Mice. Chemical Research in Toxicology. PMID 31524377 DOI: 10.1021/Acs.Chemrestox.9B00162 |
0.577 |
|
| 2019 |
Singh R, Xie W, Williams J, Vince R, More SS. Discovery of anticancer clinical candidate, tosedostat, as an analgesic agent. Acs Chemical Neuroscience. PMID 31415151 DOI: 10.1021/Acschemneuro.9B00230 |
0.646 |
|
| 2017 |
Singh R, Williams J, Vince R. Puromycin based inhibitors of aminopeptidases for the potential treatment of hematologic malignancies. European Journal of Medicinal Chemistry. 139: 325-336. PMID 28803047 DOI: 10.1016/J.Ejmech.2017.07.048 |
0.571 |
|
| 2017 |
More SS, Nugent J, Vartak AP, Nye SM, Vince R. Hepatoprotective Effect of ψ-GSH in a Murine Model of Acetaminophen-Induced Liver Toxicity. Chemical Research in Toxicology. PMID 28165728 DOI: 10.1021/Acs.Chemrestox.6B00291 |
0.6 |
|
| 2016 |
More SS, Beach JM, Vince R. Early Detection of Amyloidopathy in Alzheimer's Mice by Hyperspectral Endoscopy. Investigative Ophthalmology & Visual Science. 57: 3231-8. PMID 27333181 DOI: 10.1167/Iovs.15-17406 |
0.56 |
|
| 2016 |
Wezena CA, Urscher M, Vince R, More SS, Deponte M. Hemolytic and antimalarial effects of tight-binding glyoxalase 1 inhibitors on the host-parasite unit of erythrocytes infected with Plasmodium falciparum. Redox Biology. 8: 348-353. PMID 26972115 DOI: 10.1016/J.Redox.2016.02.006 |
0.611 |
|
| 2015 |
More SS, Vince R. Hyperspectral imaging signatures detect amyloidopathy in Alzheimer's mouse retina well before onset of cognitive decline. Acs Chemical Neuroscience. 6: 306-15. PMID 25354367 DOI: 10.1021/Cn500242Z |
0.569 |
|
| 2014 |
Felczak K, Vince R, Pankiewicz KW. NAD-based inhibitors with anticancer potential. Bioorganic & Medicinal Chemistry Letters. 24: 332-6. PMID 24269162 DOI: 10.1016/J.Bmcl.2013.11.005 |
0.394 |
|
| 2013 |
More SS, Vartak AP, Vince R. Restoration of glyoxalase enzyme activity precludes cognitive dysfunction in a mouse model of Alzheimer's disease. Acs Chemical Neuroscience. 4: 330-8. PMID 23421684 DOI: 10.1021/Cn3001679 |
0.598 |
|
| 2012 |
More SS, Vince R. Potential of a γ-glutamyl-transpeptidase-stable glutathione analogue against amyloid-β toxicity. Acs Chemical Neuroscience. 3: 204-10. PMID 22860189 DOI: 10.1021/Cn200113Z |
0.609 |
|
| 2012 |
Chen YL, Zacharias J, Vince R, Geraghty RJ, Wang Z. C-6 aryl substituted 4-quinolone-3-carboxylic acids as inhibitors of hepatitis C virus. Bioorganic & Medicinal Chemistry. 20: 4790-800. PMID 22748708 DOI: 10.1016/J.Bmc.2012.05.066 |
0.701 |
|
| 2012 |
More SS, Vartak AP, Vince R. The butter flavorant, diacetyl, exacerbates β-amyloid cytotoxicity. Chemical Research in Toxicology. 25: 2083-91. PMID 22731744 DOI: 10.1021/Tx3001016 |
0.586 |
|
| 2012 |
Singh R, Vince R. 2-Azabicyclo[2.2.1]hept-5-en-3-one: chemical profile of a versatile synthetic building block and its impact on the development of therapeutics. Chemical Reviews. 112: 4642-86. PMID 22681478 DOI: 10.1021/Cr2004822 |
0.461 |
|
| 2012 |
Urscher M, More SS, Alisch R, Vince R, Deponte M. Tight-binding inhibitors efficiently inactivate both reaction centers of monomeric Plasmodium falciparum glyoxalase 1. The Febs Journal. 279: 2568-78. PMID 22607473 DOI: 10.1111/J.1742-4658.2012.08640.X |
0.63 |
|
| 2012 |
More SS, Raza A, Vince R. The butter flavorant, diacetyl, forms a covalent adduct with 2-deoxyguanosine, uncoils DNA, and leads to cell death. Journal of Agricultural and Food Chemistry. 60: 3311-7. PMID 22385266 DOI: 10.1021/Jf300180E |
0.578 |
|
| 2012 |
Chen YL, Tang J, Kesler MJ, Sham YY, Vince R, Geraghty RJ, Wang Z. The design, synthesis and biological evaluations of C-6 or C-7 substituted 2-hydroxyisoquinoline-1,3-diones as inhibitors of hepatitis C virus. Bioorganic & Medicinal Chemistry. 20: 467-79. PMID 22100256 DOI: 10.1016/J.Bmc.2011.10.058 |
0.698 |
|
| 2012 |
Vartak AP, More SS, Vince R. Could the artificial butter flavoring, diacetyl, cause Alzheimer’s disease? Neurodegenerative Disease Management. 2: 557-559. DOI: 10.2217/Nmt.12.59 |
0.592 |
|
| 2011 |
Tang J, Maddali K, Dreis CD, Sham YY, Vince R, Pommier Y, Wang Z. N-3 Hydroxylation of Pyrimidine-2,4-diones Yields Dual Inhibitors of HIV Reverse Transcriptase and Integrase. Acs Medicinal Chemistry Letters. 2: 63-67. PMID 21499541 DOI: 10.1021/Ml1002162 |
0.657 |
|
| 2011 |
Tang J, Maddali K, Dreis CD, Sham YY, Vince R, Pommier Y, Wang Z. 6-Benzoyl-3-hydroxypyrimidine-2,4-diones as dual inhibitors of HIV reverse transcriptase and integrase. Bioorganic & Medicinal Chemistry Letters. 21: 2400-2. PMID 21392991 DOI: 10.1016/J.Bmcl.2011.02.069 |
0.655 |
|
| 2011 |
Tang J, Maddali K, Metifiot M, Sham YY, Vince R, Pommier Y, Wang Z. 3-Hydroxypyrimidine-2,4-diones as an inhibitor scaffold of HIV integrase. Journal of Medicinal Chemistry. 54: 2282-92. PMID 21381765 DOI: 10.1021/Jm1014378 |
0.65 |
|
| 2011 |
Felczak K, Chen L, Wilson D, Williams J, Vince R, Petrelli R, Jayaram HN, Kusumanchi P, Kumar M, Pankiewicz KW. Cofactor-type inhibitors of inosine monophosphate dehydrogenase via modular approach: targeting the pyrophosphate binding sub-domain. Bioorganic & Medicinal Chemistry. 19: 1594-605. PMID 21324702 DOI: 10.1016/J.Bmc.2011.01.042 |
0.337 |
|
| 2010 |
Wang Z, Tang J, Salomon CE, Dreis CD, Vince R. Pharmacophore and structure-activity relationships of integrase inhibition within a dual inhibitor scaffold of HIV reverse transcriptase and integrase. Bioorganic & Medicinal Chemistry. 18: 4202-11. PMID 20576573 DOI: 10.1016/J.Bmc.2010.05.004 |
0.791 |
|
| 2010 |
Lu D, Sham YY, Vince R. Design, asymmetric synthesis, and evaluation of pseudosymmetric sulfoximine inhibitors against HIV-1 protease. Bioorganic & Medicinal Chemistry. 18: 2037-48. PMID 20138769 DOI: 10.1016/J.Bmc.2010.01.020 |
0.63 |
|
| 2009 |
More SS, Vince R. Inhibition of glyoxalase I: the first low-nanomolar tight-binding inhibitors. Journal of Medicinal Chemistry. 52: 4650-6. PMID 19610604 DOI: 10.1021/Jm900382U |
0.646 |
|
| 2008 |
Raza A, Sham YY, Vince R. Design and synthesis of sulfoximine based inhibitors for HIV-1 protease. Bioorganic & Medicinal Chemistry Letters. 18: 5406-10. PMID 18829317 DOI: 10.1016/J.Bmcl.2008.09.044 |
0.44 |
|
| 2008 |
More SS, Vince R. Design, synthesis and biological evaluation of glutathione peptidomimetics as components of anti-Parkinson prodrugs. Journal of Medicinal Chemistry. 51: 4581-8. PMID 18651729 DOI: 10.1021/Jm800239V |
0.582 |
|
| 2008 |
Wang Z, Vince R. Design and synthesis of dual inhibitors of HIV reverse transcriptase and integrase: introducing a diketoacid functionality into delavirdine. Bioorganic & Medicinal Chemistry. 16: 3587-95. PMID 18314335 DOI: 10.1016/J.Bmc.2008.02.007 |
0.641 |
|
| 2008 |
Wang Z, Vince R. Synthesis of pyrimidine and quinolone conjugates as a scaffold for dual inhibitors of HIV reverse transcriptase and integrase. Bioorganic & Medicinal Chemistry Letters. 18: 1293-6. PMID 18226894 DOI: 10.1016/J.Bmcl.2008.01.025 |
0.662 |
|
| 2008 |
Lu D, Vince R. Corrigendum to "Discovery of potent HIV-1 protease inhibitors incorporating sulfoximine functionality" [Bioorg. Med. Chem. Lett. 17 (2007) 5614-5619] (DOI:10.1016/j.bmcl.2007.07.095) Bioorganic and Medicinal Chemistry Letters. 18: 2228. DOI: 10.1016/J.Bmcl.2008.02.004 |
0.6 |
|
| 2008 |
WANG Z, VINCE R. From RT Inhibitor to RT/IN Dual Inhibitor: An Rational Design Antiviral Research. 78: A51-A51. DOI: 10.1016/J.Antiviral.2008.01.103 |
0.612 |
|
| 2007 |
Nagasawa HT, Goon DJ, Crankshaw DL, Vince R, Patterson SE. Novel, orally effective cyanide antidotes. Journal of Medicinal Chemistry. 50: 6462-4. PMID 18038966 DOI: 10.1021/Jm7011497 |
0.337 |
|
| 2007 |
Lu D, Vince R. Discovery of potent HIV-1 protease inhibitors incorporating sulfoximine functionality. Bioorganic & Medicinal Chemistry Letters. 17: 5614-9. PMID 17822899 DOI: 10.1016/J.Bmcl.2007.07.095 |
0.601 |
|
| 2007 |
Wang Z, Bennett EM, Wilson DJ, Salomon C, Vince R. Rationally designed dual inhibitors of HIV reverse transcriptase and integrase. Journal of Medicinal Chemistry. 50: 3416-9. PMID 17608468 DOI: 10.1021/Jm070512P |
0.781 |
|
| 2007 |
More SS, Vince R. Design, synthesis, and binding studies of bidentate Zn-chelating peptidic inhibitors of glyoxalase-I. Bioorganic & Medicinal Chemistry Letters. 17: 3793-7. PMID 17513107 DOI: 10.1016/J.Bmcl.2006.12.056 |
0.638 |
|
| 2007 |
Pham PT, Vince R. Carbovir-related compounds and phosphonate analogues Phosphorus, Sulfur and Silicon and the Related Elements. 182: 779-791. DOI: 10.1080/10426500601047578 |
0.301 |
|
| 2006 |
Vince R, Hua M. Synthesis of carbovir and abacavir from a carbocyclic precursor. Current Protocols in Nucleic Acid Chemistry / Edited by Serge L. Beaucage ... [Et Al.]. Unit 14.4. PMID 18428951 DOI: 10.1002/0471142700.Nc1404S25 |
0.606 |
|
| 2006 |
More SS, Vince R. A metabolically stable tight-binding transition-state inhibitor of glyoxalase-I. Bioorganic & Medicinal Chemistry Letters. 16: 6039-42. PMID 16997560 DOI: 10.1016/J.Bmcl.2006.08.121 |
0.649 |
|
| 2006 |
Tang Y, Muthyala R, Vince R. Synthesis and biological evaluation of carboacyclic nucleosides with (Z) and (E)-9-[4,4-bis(hydroxymethyl)]-2-butenyl side chain. Bioorganic & Medicinal Chemistry. 14: 5866-75. PMID 16759867 DOI: 10.1016/J.Bmc.2006.05.029 |
0.532 |
|
| 2006 |
Li X, Vince R. Synthesis and biological evaluation of purine derivatives incorporating metal chelating ligands as HIV integrase inhibitors. Bioorganic & Medicinal Chemistry. 14: 5742-55. PMID 16753300 DOI: 10.1016/J.Bmc.2006.04.011 |
0.605 |
|
| 2006 |
Li X, Vince R. Conformationally restrained carbazolone-containing alpha,gamma-diketo acids as inhibitors of HIV integrase. Bioorganic & Medicinal Chemistry. 14: 2942-55. PMID 16386908 DOI: 10.1016/J.Bmc.2005.12.013 |
0.585 |
|
| 2002 |
Quirk Dorr DR, Vince R. Synthesis and biological evaluation of endocyclic 2',3'-didehydro-2',3'-dideoxymethanocarba adenosine. Nucleosides, Nucleotides & Nucleic Acids. 21: 665-80. PMID 12502282 DOI: 10.1081/Ncn-120015724 |
0.772 |
|
| 2002 |
Bhushan RG, Vince R. Synthesis of conformationally restricted 2',3'-exo-methylene carbocyclic nucleosides built on a bicyclo[3.1.0]hexane template. Bioorganic & Medicinal Chemistry. 10: 2325-33. PMID 11983530 DOI: 10.1016/S0968-0896(02)00063-9 |
0.784 |
|
| 2000 |
Parker WB, Shaddix SC, Rose LM, Pham PT, Hua M, Vince R. Metabolism of O6-propyl and N6-propyl-carbovir in CEM cells. Nucleosides, Nucleotides & Nucleic Acids. 19: 795-804. PMID 10960036 DOI: 10.1080/15257770008035025 |
0.591 |
|
| 1999 |
Antle VD, Donat N, Hua M, Liao PL, Vince R, Carperelli CA. Substrate specificity of human glycinamide ribonucleotide transformylase. Archives of Biochemistry and Biophysics. 370: 231-5. PMID 10577357 DOI: 10.1006/Abbi.1999.1428 |
0.577 |
|
| 1999 |
Vince R, Brownell J, Akella LB. Synthesis and activity of γ-(L-γ-azaglutamyl)-S-(p-bromobenzyl)-L- cysteinylglycine: A metabolically stable inhibitor of glyoxalase I Bioorganic and Medicinal Chemistry Letters. 9: 853-856. PMID 10206549 DOI: 10.1016/S0960-894X(99)00097-9 |
0.375 |
|
| 1997 |
Parker WB, Shaddix SC, Vince R, Bennett LL. Lack of mitochondrial toxicity in CEM cells treated with carbovir Antiviral Research. 34: 131-136. PMID 9191020 DOI: 10.1016/S0166-3542(97)01033-4 |
0.341 |
|
| 1996 |
Antle VD, Liu D, McKellar BR, Caperelli CA, Hua M, Vince R. Substrate specificity of glycinamide ribonucleotide synthetase from chicken liver. The Journal of Biological Chemistry. 271: 8192-5. PMID 8626510 DOI: 10.1074/Jbc.271.14.8192 |
0.573 |
|
| 1996 |
Antle VD, Liu D, McKellars BR, Caperelli CA, Hua M, Vince R. Substrate specificity of glycinamide ribonucleotide transformylase from chicken liver. The Journal of Biological Chemistry. 271: 6045-9. PMID 8626389 DOI: 10.1074/Jbc.271.11.6045 |
0.592 |
|
| 1996 |
Vince R, Hua M, Caperelli CA. Phosphonate analogs of carbocyclic phosphoribosylamine and carbocyclic glycinamide ribonucleotide Nucleosides and Nucleotides. 15: 1711-1718. DOI: 10.1080/07328319608002726 |
0.631 |
|
| 1996 |
Konkel MJ, Vince R. Cyclohexenyl nucleosides: Synthesis of cis-4-(9H-purin-9-yl)-2-cyclohexenylcarbinols Tetrahedron. 52: 799-808. DOI: 10.1016/0040-4020(95)00926-4 |
0.313 |
|
| 1995 |
Vince R, Brownell J, Beers SA. 6-Deoxycarbovir: A Xanthine Oxidase Activated Prodrug Of Carbovir Nucleosides and Nucleotides. 14: 39-44. DOI: 10.1080/15257779508014651 |
0.333 |
|
| 1995 |
Konkel MJ, Vince R. Synthesis and Biological Activity of Cyclohexenyl Nucleosides, cis-5-(9H-Purin-9-YL)-3-Cyclohexenyl Carbinols and their 8-Azapurinyl Analogs Nucleosides and Nucleotides. 14: 2061-2077. DOI: 10.1080/15257779508010724 |
0.311 |
|
| 1995 |
Vince R, Pham PT. The Synthesis and Biological Evaluation of Sulfamoyl Nucleosides Related to Carbovir and Azt Nucleosides and Nucleotides. 14: 2051-2060. DOI: 10.1080/15257779508010723 |
0.384 |
|
| 1995 |
Vince R, Kilama J, Pham PT, Beers SA, Bowdon BJ, Keith KA, Parker WB. 6-substituted derivatives of carbovir: Anti-HIV activity Nucleosides and Nucleotides. 14: 1703-1708. DOI: 10.1080/15257779508009751 |
0.399 |
|
| 1993 |
Parker WB, Shaddix SC, Bowdon BJ, Rose LM, Vince R, Shannon WM, Bennett LL. Metabolism of carbovir, a potent inhibitor of human immunodeficiency virus type 1, and its effects on cellular metabolism Antimicrobial Agents and Chemotherapy. 37: 1004-1009. PMID 7685993 DOI: 10.1128/Aac.37.5.1004 |
0.366 |
|
| 1992 |
Peterson EM, Brownell J, Vince R. Synthesis and biological evaluation of 5'-sulfamoylated purinyl carbocyclic nucleosides. Journal of Medicinal Chemistry. 35: 3991-4000. PMID 1433208 DOI: 10.1021/Jm00100A003 |
0.372 |
|
| 1991 |
Peterson ML, Vince R. Synthesis and biological evaluation of 4-purinylpyrrolidine nucleosides Journal of Medicinal Chemistry. 34: 2787-2797. PMID 1654429 DOI: 10.1021/Jm00113A017 |
0.381 |
|
| 1990 |
Vince R, Brownell J. Resolution of racemic carbovir and selective inhibition of human immunodeficiency virus by the (-) enantiomer Biochemical and Biophysical Research Communications. 168: 912-916. PMID 2346492 DOI: 10.1016/0006-291X(90)91115-9 |
0.332 |
|
| 1990 |
Vince R, Hua M. Synthesis and anti-HIV activity of carbocyclic 2',3'-didehydro-2',3'-dideoxy 2,6-disubstituted purine nucleosides. Journal of Medicinal Chemistry. 33: 17-21. PMID 2296018 DOI: 10.1021/Jm00163A004 |
0.555 |
|
| 1990 |
Bondoc LL, Shannon WM, Secrist JA, Vince R, Fridland A. Metabolism of the carbocyclic nucleoside analogue carbovir, an inhibitor of human immunodeficiency virus, in human lymphoid cells Biochemistry. 29: 9839-9843. PMID 2271622 DOI: 10.1021/Bi00494A013 |
0.353 |
|
| 1989 |
Remmel RP, Yeom YH, Hua M, Vince R, Zimmerman CL. Liquid chromatographic assay of carbovir, a carbocyclic nucleoside active against human immunodeficiency virus. Journal of Chromatography. 489: 323-31. PMID 2753956 DOI: 10.1016/S0378-4347(00)82910-2 |
0.54 |
|
| 1989 |
Yeom YH, Remmel RP, Huang SH, Hua M, Vince R, Zimmerman CL. Pharmacokinetics and bioavailability of carbovir, a carbocyclic nucleoside active against human immunodeficiency virus, in rats. Antimicrobial Agents and Chemotherapy. 33: 171-5. PMID 2719460 DOI: 10.1128/Aac.33.2.171 |
0.533 |
|
| 1989 |
White EL, Parker WB, Macy LJ, Shaddix SC, McCaleb G, Secrist JA, Vince R, Shannon WM. Comparison of the effect of Carbovir, AZT, and dideoxynucleoside triphosphates on the activity of human immunodeficiency virus reverse transcriptase and selected human polymerases Biochemical and Biophysical Research Communications. 161: 393-398. PMID 2472136 DOI: 10.1016/0006-291X(89)92611-9 |
0.381 |
|
| 1989 |
Vince R, Lavelle GC, Hua M, Qualls J, Brownell J, Shannon WM. Carbovir: A carbocyclic nucleoside with potent and selective activity against human immunodeficiency virus (HIV) in vitro Nucleosides and Nucleotides. 8: 1127-1128. DOI: 10.1080/07328318908054307 |
0.606 |
|
| 1988 |
Vince R, Hua M, Brownell J, Daluge S, Lee FC, Shannon WM, Lavelle GC, Qualls J, Weislow OS, Kiser R. Potent and selective activity of a new carbocyclic nucleoside analog (carbovir: NSC 614846) against human immunodeficiency virus in vitro. Biochemical and Biophysical Research Communications. 156: 1046-53. PMID 2847711 DOI: 10.1016/S0006-291X(88)80950-1 |
0.608 |
|
| 1987 |
Hua M, Korkowski PM, Vince R. Synthesis and biological evaluation of acyclic neplanocin analogues. Journal of Medicinal Chemistry. 30: 198-200. PMID 3027333 DOI: 10.1021/Jm00384A033 |
0.558 |
|
| 1987 |
Vince R, Turakhia RH, Shannon WM, Arnett G. Synthesis and antiviral activity of carbocyclic analogues of xylofuranosides of 2-amino-6-substituted-purines and 2-amino-6-substituted-8-azapurines Journal of Medicinal Chemistry. 30: 2026-2030. PMID 2822928 DOI: 10.1021/Jm00394A017 |
0.301 |
|
| 1986 |
Vince R, Daluge S, Brownell J. Carbocyclic puromycin: Synthesis and inhibition of protein biosynthesis Journal of Medicinal Chemistry. 29: 2400-2403. PMID 3783599 DOI: 10.1021/Jm00161A044 |
0.339 |
|
| 1984 |
McFarlan SC, Vince R. Inhibition of peptidyltransferase and possible mode of action of a dipeptidyl chloramphenicol analog Biochemical and Biophysical Research Communications. 122: 748-754. PMID 6380501 DOI: 10.1016/S0006-291X(84)80097-2 |
0.363 |
|
| 1981 |
Vince R, Lee H, Narang AS, Shirota FN. 5′-Chloropuromycin. Inhibition of protein synthesis and antitrypanosomal activity Journal of Medicinal Chemistry. 24: 1511-1514. PMID 7310828 DOI: 10.1002/Chin.198222340 |
0.361 |
|
| 1980 |
Lee H, Vince R. Carbocyclic analogs of arabinosylpurine nucleosides Journal of Pharmaceutical Sciences. 69: 1019-1021. PMID 6251197 DOI: 10.1002/Chin.198110368 |
0.354 |
|
| 1978 |
Fong KLL, Vince R. Peptidyl transferase substrate specificity with nonaromatic aminoacyl analogues of puromycin Journal of Medicinal Chemistry. 21: 792-795. PMID 691004 DOI: 10.1002/Chin.197851358 |
0.334 |
|
| 1978 |
Vince R, Fong KLL. Peptidyl transferase substrate activity and inhibition of protein biosynthesis by a hydrophilic-aminoacyl analogue of puromycin Biochemical and Biophysical Research Communications. 81: 559-564. PMID 352348 DOI: 10.1016/0006-291X(78)91571-1 |
0.369 |
|
| 1978 |
Lee CK, Vince R. Effect of sparsomycin analogues on the puromycin-peptidyl transferase reaction on ribosomes Journal of Medicinal Chemistry. 21: 176-179. PMID 340693 DOI: 10.1002/Chin.197825305 |
0.315 |
|
| 1977 |
Vince R, Brownell J, Kiu Lee C. Inhibition of protein biosynthesis: The first active sparsomycin analog Biochemical and Biophysical Research Communications. 75: 563-567. PMID 856177 DOI: 10.1016/0006-291X(77)91509-1 |
0.362 |
|
| 1977 |
Lyon PA, Vince R. Synthesis and kinetic evaluation of S- and N-substituted cysteinylglycines as inhibitors of glyoxalase I Journal of Medicinal Chemistry. 20: 77-80. PMID 833829 DOI: 10.1002/Chin.197721180 |
0.365 |
|
| 1977 |
Narang AS, Vince R. 1,2,4-Triazole amino nucleosides. 1-β-D-3′-amino-3′-deoxyribofuranosyl-1,2,4-triazole-3- carboxamide and related nucleosides Journal of Medicinal Chemistry. 20: 1684-1687. PMID 201758 DOI: 10.1021/Jm00222A032 |
0.329 |
|
| 1976 |
Vince R, Weiss D, Pestka S. Binding of N substituted erythromycylamines to ribosomes Antimicrobial Agents and Chemotherapy. 9: 131-136. PMID 769668 DOI: 10.1128/Aac.9.1.131 |
0.307 |
|
| 1976 |
Vince R, Almquist RG, Ritter CL, Shirota FN, Nagasawa HT. An active puromycin analog derived from a non nephrotoxic aminonucleoside Life Sciences. 18: 345-350. PMID 768682 DOI: 10.1016/0024-3205(76)90063-1 |
0.316 |
|
| 1975 |
Duquette PH, Ritter CL, Vince R. Puromycin analogs. Ribosomal binding and peptidyl transferase substrate activity of a carbocyclic analog of 8-azapuromycin. Biochemistry. 13: 4855-9. PMID 4609468 DOI: 10.1021/Bi00720A026 |
0.307 |
|
| 1974 |
Pestka S, Vince R, Daluge S, Harris R. Effect of puromycin analogues and other agents on peptidyl-puromycin synthesis on polyribosomes. Antimicrobial Agents and Chemotherapy. 4: 37-43. PMID 4598844 DOI: 10.1128/Aac.4.1.37 |
0.314 |
|
| 1974 |
ALMQUIST RG, VINCE R. ChemInform Abstract: PUROMYCIN ANALOGS, SYNTHESIS AND BIOLOGICAL ACTIVITY OF 5′-DEOXYPUROMYCIN AND ITS AMINONUCLEOSIDE, 6-DIMETHYLAMINO-9-(3′-AMINO-3′,5′-DIDEOXY-BETA-D-RIBOFURANOSYL)-PURINE Chemischer Informationsdienst. 5: no-no. DOI: 10.1002/Chin.197417484 |
0.302 |
|
| 1972 |
Vince R, Daluge S, Wadd WB. Studies on the inhibition of glyoxalase I by S-substituted glutathiones. Journal of Medicinal Chemistry. 14: 402-4. PMID 5117686 DOI: 10.1021/Jm00287A006 |
0.338 |
|
| 1972 |
Vince R, Daluge S, Palm M. Inhibition of in vitro protein synthesis by a carbocyclic puromycin analog. Biochemical and Biophysical Research Communications. 46: 866-70. PMID 4550700 DOI: 10.1016/S0006-291X(72)80221-3 |
0.33 |
|
| 1971 |
Schaeffer HJ, Gurwara S, Vince R, Bittner S. Novel substrate of adenosine deaminase. Journal of Medicinal Chemistry. 14: 367-9. PMID 5553754 DOI: 10.1021/Jm00286A024 |
0.597 |
|
| 1971 |
Vince R, Daluge S. Glyoxalase inhibitors. A possible approach to anticancer agents. Journal of Medicinal Chemistry. 14: 35-7. PMID 5099673 DOI: 10.1021/Jm00283A009 |
0.323 |
|
| 1971 |
SCHAEFFER HJ, GURWARA S, VINCE R, BITTNER A. ChemInform Abstract: EIN NEUES SUBSTRAT FUER ADENOSIN-DESAMINASE Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197130327 |
0.555 |
|
| 1969 |
Vince R, Wadd WB. Glyoxalase inhibitors as potential anticancer agents. Biochemical and Biophysical Research Communications. 35: 593-8. PMID 5794079 DOI: 10.1016/0006-291X(69)90445-8 |
0.385 |
|
| 1968 |
Schaeffer HJ, Vince R. Enzyme inhibitors. XIX. The synthesis of some 1-hydroxy-2-hydroxymethyl-4-(6-substituted-9-purinyl)cyclohexanes as nucleoside analogs. Journal of Medicinal Chemistry. 11: 15-20. PMID 5637163 DOI: 10.1021/Jm00307A003 |
0.66 |
|
| 1967 |
Schaeffer HJ, Vince R. Enzyme inhibitors. 18. Studies on the stereoselectivity of inhibition of adenosine deaminase by DL-, D-, and L-9-(2-hydroxypropyl)adenine. Journal of Medicinal Chemistry. 10: 689-91. PMID 6037062 DOI: 10.1021/Jm00316A037 |
0.625 |
|
| 1965 |
SCHAEFFER HJ, VINCE R. ENZYME INHIBITORS. VI. STUDIES ON THE BULK TOLERANCE OF ADENOSINE DEAMINASE FOR 6-SUBSTITUTED AMINO-9-(3-HYDROXYPROPYL)PURINES. Journal of Medicinal Chemistry. 8: 33-5. PMID 14287263 DOI: 10.1021/Jm00325A008 |
0.644 |
|
| 1965 |
Schaeffer HJ, Gvogel D, Vince R. Enzyme inhibitors. 8. Studies on the mode of binding of some 6-substituted 9-(hydroxyalkyl)purines to adenosine deaminase. Journal of Medicinal Chemistry. 8: 502-6. PMID 5883714 DOI: 10.1021/Jm00328A020 |
0.621 |
|
| 1965 |
Schaeffer HJ, Vince R. Enzyme Inhibitors. X. A Reinvestigation of the Alkylation of 6-Chloropurine by 3-Bromo-1-propanol1 Journal of Medicinal Chemistry. 8: 710-712. DOI: 10.1021/Jm00329A040 |
0.624 |
|
| 1963 |
Schaeffer HJ, Vince R. Intramolecular Reactions of Some Cyclic β-Diketones1 The Journal of Organic Chemistry. 28: 1653-1656. DOI: 10.1021/Jo01041A055 |
0.55 |
|
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