Hak-Sung Kim - Publications

1999-2003 Wonkwang University, Iksan, South Korea 

79 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Choi Y, Jeong S, Choi JM, Ndong C, Griswold KE, Bailey-Kellogg C, Kim HS. Computer-guided binding mode identification and affinity improvement of an LRR protein binder without structure determination. Plos Computational Biology. 16: e1008150. PMID 32866140 DOI: 10.1371/journal.pcbi.1008150  0.44
2020 Jeong S, Sohn YK, Choi Y, Park J, Kim HS. A regulatory SH2 domain-targeting protein binder effectively inhibits the activity of Bruton's tyrosine kinase and its drug-resistant variants. Biochemical and Biophysical Research Communications. PMID 32192770 DOI: 10.1016/j.bbrc.2020.03.006  0.44
2020 Sohn YK, Son S, Choi Y, Hwang DE, Seo HD, Lee JJ, Kim HS. Effective inhibition of C3a-mediated pro-inflammatory response by a human C3a-specific protein binder. Biotechnology and Bioengineering. PMID 32068245 DOI: 10.1002/bit.27309  0.44
2019 Yu TG, Kim HS, Choi Y. B-SIDER: Computational Algorithm for the Design of Complementary β-sheet Sequences. Journal of Chemical Information and Modeling. PMID 31512871 DOI: 10.1021/acs.jcim.9b00548  0.44
2018 Ryu Y, Kang JA, Kim D, Kim SR, Kim S, Park SJ, Kwon SH, Kim KN, Lee DE, Lee JJ, Kim HS. Programed Assembly of Nucleoprotein Nanoparticles Using DNA and Zinc Fingers for Targeted Protein Delivery. Small (Weinheim An Der Bergstrasse, Germany). e1802618. PMID 30398698 DOI: 10.1002/smll.201802618  0.32
2018 Heu W, Choi JM, Kyeong HH, Choi Y, Kim HY, Kim HS. Repeat module-based rational design of a photo-switchable protein for light-driven control of biological processes. Angewandte Chemie (International Ed. in English). PMID 29952059 DOI: 10.1002/anie.201803993  0.44
2017 Kyeong HH, Choi Y, Kim HS. GradDock: Rapid Simulation and Tailored Ranking Functions for Peptide-MHC Class I Docking. Bioinformatics (Oxford, England). PMID 28968726 DOI: 10.1093/bioinformatics/btx589  0.44
2016 An JH, Jin F, Kim HS, Ryu HC, Kim JS, Kim HM, Kiyonga AN, Min DS, Youn W, Kim KH, Jung K. Application of ionic liquid to polymorphic transformation of anti-viral/HIV drug adefovir dipivoxil. Archives of Pharmacal Research. PMID 26908332 DOI: 10.1007/s12272-016-0721-0  0.36
2016 Ryou JH, Sohn YK, Hwang DE, Park WY, Kim N, Heo WD, Kim MY, Kim HS. Engineering of bacterial exotoxins for highly efficient and receptor-specific intracellular delivery of diverse cargos. Biotechnology and Bioengineering. PMID 26773973 DOI: 10.1002/bit.25935  0.52
2015 Kim YP, Kim HS. Nanoparticles for Use in Enzyme Assays. Chembiochem : a European Journal of Chemical Biology. PMID 26662229 DOI: 10.1002/cbic.201500512  0.96
2015 Lee JJ, Choi HJ, Yun M, Kang Y, Jung JE, Ryu Y, Kim TY, Cha YJ, Cho HS, Min JJ, Chung CW, Kim HS. Enzymatic Prenylation and Oxime Ligation for the Synthesis of Stable and Homogeneous Protein-Drug Conjugates for Targeted Therapy. Angewandte Chemie (International Ed. in English). PMID 26315561 DOI: 10.1002/anie.201505964  0.52
2015 Bae JH, Jo SM, Kim HS. Comprehensive detection of diverse exon 19 deletion mutations of EGFR in lung Cancer by a single probe set. Biosensors & Bioelectronics. 74: 849-55. PMID 26233641 DOI: 10.1016/j.bios.2015.07.043  0.52
2015 Min H, Jo SM, Kim HS. Efficient capture and simple quantification of circulating tumor cells using quantum dots and magnetic beads. Small (Weinheim An Der Bergstrasse, Germany). 11: 2536-42. PMID 25630488 DOI: 10.1002/smll.201403126  0.52
2015 Jo SM, Lee JJ, Heu W, Kim HS. Nanotentacle-structured magnetic particles for efficient capture of circulating tumor cells. Small (Weinheim An Der Bergstrasse, Germany). 11: 1975-82. PMID 25504978 DOI: 10.1002/smll.201402619  0.52
2015 Ryu Y, Jin Z, Lee JJ, Noh SH, Shin TH, Jo SM, Choi J, Park H, Cheon J, Kim HS. Size-controlled construction of magnetic nanoparticle clusters using DNA-binding zinc finger protein. Angewandte Chemie (International Ed. in English). 54: 923-6. PMID 25425202 DOI: 10.1002/anie.201408593  0.52
2014 Yeo SJ, Huong DT, Hong NN, Li CY, Choi K, Yu K, Choi DY, Chong CK, Choi HS, Mallik SK, Kim HS, Sung HW, Park H. Rapid and quantitative detection of zoonotic influenza A virus infection utilizing coumarin-derived dendrimer-based fluorescent immunochromatographic strip test (FICT). Theranostics. 4: 1239-49. PMID 25285172 DOI: 10.7150/thno.10255  0.56
2014 Ryou JH, Park K, Lee JJ, Kim D, Kim HS. Soluble expression of human glycoprotein Ibα in Escherichia coli through replacement of the N-terminal capping domain. Protein Expression and Purification. 101: 21-7. PMID 24925643 DOI: 10.1016/j.pep.2014.06.001  0.52
2014 Jeong YS, Choi JM, Kyeong HH, Choi JY, Kim EJ, Kim HS. Rational design of organophosphorus hydrolase with high catalytic efficiency for detoxifying a V-type nerve agent. Biochemical and Biophysical Research Communications. 449: 263-7. PMID 24824182 DOI: 10.1016/j.bbrc.2014.04.155  0.52
2014 Seo MH, Park J, Kim E, Hohng S, Kim HS. Protein conformational dynamics dictate the binding affinity for a ligand. Nature Communications. 5: 3724. PMID 24758940 DOI: 10.1038/ncomms4724  0.52
2014 Lee JJ, Kim HJ, Yang CS, Kyeong HH, Choi JM, Hwang DE, Yuk JM, Park K, Kim YJ, Lee SG, Kim D, Jo EK, Cheong HK, Kim HS. A high-affinity protein binder that blocks the IL-6/STAT3 signaling pathway effectively suppresses non-small cell lung cancer. Molecular Therapy : the Journal of the American Society of Gene Therapy. 22: 1254-65. PMID 24682171 DOI: 10.1038/mt.2014.59  0.52
2014 Eum JY, Hwang SY, Ju Y, Shim JM, Piao Y, Lee J, Kim HS, Kim J. A highly sensitive immunoassay using antibody-conjugated spherical mesoporous silica with immobilized enzymes. Chemical Communications (Cambridge, England). 50: 3546-8. PMID 24402353 DOI: 10.1039/c3cc48044e  0.36
2014 Choi SL, Rha E, Lee SJ, Kim H, Kwon K, Jeong YS, Rhee YH, Song JJ, Kim HS, Lee SG. Toward a generalized and high-throughput enzyme screening system based on artificial genetic circuits. Acs Synthetic Biology. 3: 163-71. PMID 24295047 DOI: 10.1021/sb400112u  0.52
2013 Choi JM, Seo MH, Kyeong HH, Kim E, Kim HS. Molecular basis for the role of glucokinase regulatory protein as the allosteric switch for glucokinase. Proceedings of the National Academy of Sciences of the United States of America. 110: 10171-6. PMID 23733961 DOI: 10.1073/pnas.1300457110  0.52
2013 Jo SM, Kim Y, Jeong YS, Hee Oh Y, Park K, Kim HS. Rapid detection of exon 2-deleted AIMP2 mutation as a potential biomarker for lung cancer by molecular beacons. Biosensors & Bioelectronics. 46: 142-9. PMID 23537880 DOI: 10.1016/j.bios.2013.02.037  0.52
2013 Kim E, Lee S, Jeon A, Choi JM, Lee HS, Hohng S, Kim HS. A single-molecule dissection of ligand binding to a protein with intrinsic dynamics. Nature Chemical Biology. 9: 313-8. PMID 23502425 DOI: 10.1038/nchembio.1213  0.52
2013 Kim J, Seo MH, Lee S, Cho K, Yang A, Woo K, Kim HS, Park HS. Simple and efficient strategy for site-specific dual labeling of proteins for single-molecule fluorescence resonance energy transfer analysis. Analytical Chemistry. 85: 1468-74. PMID 23276151 DOI: 10.1021/ac303089v  0.52
2012 Jeong YS, Choi SL, Kyeong HH, Kim JH, Kim EJ, Pan JG, Rha E, Song JJ, Lee SG, Kim HS. High-throughput screening system based on phenolics-responsive transcription activator for directed evolution of organophosphate-degrading enzymes. Protein Engineering, Design & Selection : Peds. 25: 725-31. PMID 23077277 DOI: 10.1093/protein/gzs071  0.52
2012 Oh BJ, Seo MH, Kim HS. Insignificant role of the N-terminal cobalt-binding site of albumin in the assessment of acute coronary syndrome: discrepancy between the albumin cobalt-binding assay and N-terminal-targeted immunoassay. Biomarkers : Biochemical Indicators of Exposure, Response, and Susceptibility to Chemicals. 17: 394-401. PMID 22630368 DOI: 10.3109/1354750X.2012.672460  0.52
2012 Mallik SK, Li da Y, Cui M, Song HO, Park H, Kim HS. Synthesis and evaluation of peptidyl α,β-unsaturated carbonyl derivatives as anti-malarial calpain inhibitors. Archives of Pharmacal Research. 35: 469-79. PMID 22477194 DOI: 10.1007/s12272-012-0310-9  0.56
2011 Seo MH, Lee TS, Kim E, Cho YL, Park HS, Yoon TY, Kim HS. Efficient single-molecule fluorescence resonance energy transfer analysis by site-specific dual-labeling of protein using an unnatural amino acid. Analytical Chemistry. 83: 8849-54. PMID 22035235 DOI: 10.1021/ac202096t  0.52
2011 Park S, Han J, Kim W, Lee GM, Kim HS. Rapid selection of single cells with high antibody production rates by microwell array. Journal of Biotechnology. 156: 197-202. PMID 21925218 DOI: 10.1016/j.jbiotec.2011.08.031  0.52
2011 Seo MH, Han J, Jin Z, Lee DW, Park HS, Kim HS. Controlled and oriented immobilization of protein by site-specific incorporation of unnatural amino acid. Analytical Chemistry. 83: 2841-5. PMID 21428414 DOI: 10.1021/ac103334b  0.52
2011 Piao Y, Jin Z, Lee D, Lee HJ, Na HB, Hyeon T, Oh MK, Kim J, Kim HS. Sensitive and high-fidelity electrochemical immunoassay using carbon nanotubes coated with enzymes and magnetic nanoparticles Biosensors and Bioelectronics. 26: 3192-3199. PMID 21242086 DOI: 10.1016/j.bios.2010.12.025  0.52
2010 Oh YH, Kim Y, Kim YP, Seo SW, Mitsudomi T, Ahn MJ, Park K, Kim HS. Rapid detection of the epidermal growth factor receptor mutation in non-small-cell lung cancer for analysis of acquired resistance using molecular beacons. The Journal of Molecular Diagnostics : Jmd. 12: 644-52. PMID 20805561 DOI: 10.2353/jmoldx.2010.090208  0.96
2010 Park S, Kim W, Kim Y, Son YD, Lee SC, Kim E, Kim SH, Kim JH, Kim HS. Array-based analysis of secreted glycoproteins for rapid selection of a single cell producing a glycoprotein with desired glycosylation. Analytical Chemistry. 82: 5830-7. PMID 20550136 DOI: 10.1021/ac100992n  0.52
2010 Jin XY, Lee SH, Park PH, Hur J, Kim SA, Kim HS, Sohn DH. 2'-Methoxy-4'6'-bis(methoxymethoxy)chalcone inhibits nitric oxide production in lipopolysaccharide-stimulated RAW 264.7 macrophages. Basic & Clinical Pharmacology & Toxicology. 106: 454-60. PMID 20088848 DOI: 10.1111/j.1742-7843.2009.00524.x  0.36
2009 Han MK, Oh YH, Kang J, Kim YP, Seo S, Kim J, Park K, Kim HS. Protein profiling in human sera for identification of potential lung cancer biomarkers using antibody microarray. Proteomics. 9: 5544-52. PMID 20017155 DOI: 10.1002/pmic.200800777  0.96
2009 Yang SH, Lee KB, Kong B, Kim JH, Kim HS, Choi IS. Biomimetic encapsulation of individual cells with silica. Angewandte Chemie (International Ed. in English). 48: 9160-3. PMID 19856355 DOI: 10.1002/anie.200903010  0.52
2009 Piao Y, Lee D, Lee J, Hyeon T, Kim J, Kim HS. Multiplexed immunoassay using the stabilized enzymes in mesoporous silica. Biosensors & Bioelectronics. 25: 906-12. PMID 19782556 DOI: 10.1016/j.bios.2009.09.005  0.52
2009 Yun KS, Lee D, Kim HS, Yoon E. Microfluidic chips designed for measuring biomolecules through a microbead-based quantum dot fluorescence assay. Methods in Molecular Biology (Clifton, N.J.). 544: 53-67. PMID 19488693 DOI: 10.1007/978-1-59745-483-4_5  0.52
2009 Jin Z, Hahn YK, Oh E, Kim YP, Park JK, Moon SH, Jang JT, Cheon J, Kim HS. Magnetic nanoclusters for ultrasensitive magnetophoretic assays. Small (Weinheim An Der Bergstrasse, Germany). 5: 2243-6. PMID 19472195 DOI: 10.1002/smll.200900311  0.96
2009 Piao Y, Lee D, Kim J, Kim J, Hyeon T, Kim HS. High performance immunoassay using immobilized enzyme in nanoporous carbon. The Analyst. 134: 926-32. PMID 19381386 DOI: 10.1039/b813451k  0.52
2009 Kim YP, Jin Z, Kim E, Park S, Oh YH, Kim HS. Analysis of in vitro SUMOylation using bioluminescence resonance energy transfer (BRET). Biochemical and Biophysical Research Communications. 382: 530-4. PMID 19289109 DOI: 10.1016/j.bbrc.2009.03.055  0.96
2009 Park PH, Kim HS, Hur J, Jin XY, Jin YL, Sohn DH. YL-I-108, a synthetic chalcone derivative, inhibits lipopolysaccharide-stimulated nitric oxide production in RAW 264.7 murine macrophages: involvement of heme oxygenase-1 induction and blockade of activator protein-1. Archives of Pharmacal Research. 32: 79-89. PMID 19183880 DOI: 10.1007/s12272-009-1121-5  0.36
2009 Kim SA, Jin YL, Kim HS. Structure-activity relationship studies of novel oxygen-incorporated SAHA analogues. Archives of Pharmacal Research. 32: 15-21. PMID 19183872 DOI: 10.1007/s12272-009-1113-5  0.36
2009 Park PH, Kim HS, Jin XY, Jin F, Hur J, Ko G, Sohn DH. KB-34, a newly synthesized chalcone derivative, inhibits lipopolysaccharide-stimulated nitric oxide production in RAW 264.7 macrophages via heme oxygenase-1 induction and blockade of activator protein-1. European Journal of Pharmacology. 606: 215-24. PMID 19174156 DOI: 10.1016/j.ejphar.2008.12.034  0.36
2009 Kim YP, Park S, Oh E, Oh YH, Kim HS. On-chip detection of protein glycosylation based on energy transfer between nanoparticles. Biosensors & Bioelectronics. 24: 1189-94. PMID 18722763 DOI: 10.1016/j.bios.2008.07.012  0.52
2008 Jin YL, Jin XY, Jin F, Sohn DH, Kim HS. Structure activity relationship studies of anti-inflammatory TMMC derivatives: 4-dimethylamino group on the B ring responsible for lowering the potency. Archives of Pharmacal Research. 31: 1145-52. PMID 18806957 DOI: 10.1007/s12272-001-1281-7  0.36
2008 Shin EM, Zhou HY, Guo LY, Kim JA, Lee SH, Merfort I, Kang SS, Kim HS, Kim S, Kim YS. Anti-inflammatory effects of glycyrol isolated from Glycyrrhiza uralensis in LPS-stimulated RAW264.7 macrophages. International Immunopharmacology. 8: 1524-32. PMID 18621150 DOI: 10.1016/j.intimp.2008.06.008  0.56
2008 Kim YP, Lee BS, Kim E, Choi IS, Moon DW, Lee TG, Kim HS. Activity-based assay of matrix metalloproteinase on nonbiofouling surfaces using time-of-flight secondary ion mass spectrometry. Analytical Chemistry. 80: 5094-102. PMID 18505270 DOI: 10.1021/ac800299d  0.52
2008 Pae HO, Jeong SO, Kim HS, Kim SH, Song YS, Kim SK, Chai KY, Chung HT. Dimethoxycurcumin, a synthetic curcumin analogue with higher metabolic stability, inhibits NO production, inducible NO synthase expression and NF-kappaB activation in RAW264.7 macrophages activated with LPS. Molecular Nutrition & Food Research. 52: 1082-91. PMID 18481332 DOI: 10.1002/mnfr.200700333  0.56
2008 Kim YP, Oh YH, Oh E, Ko S, Han MK, Kim HS. Energy transfer-based multiplexed assay of proteases by using gold nanoparticle and quantum dot conjugates on a surface. Analytical Chemistry. 80: 4634-41. PMID 18457412 DOI: 10.1021/ac702416e  0.52
2008 Kim YP, Oh YH, Kim HS. Protein kinase assay on peptide-conjugated gold nanoparticles. Biosensors & Bioelectronics. 23: 980-6. PMID 18024102 DOI: 10.1016/j.bios.2007.10.001  0.52
2007 Jin F, Jin XY, Jin YL, Sohn DW, Kim SA, Sohn DH, Kim YC, Kim HS. Structural requirements of 2',4',6'-tris(methoxymethoxy) chalcone derivatives for anti-inflammatory activity: the importance of a 2'-hydroxy moiety. Archives of Pharmacal Research. 30: 1359-67. PMID 18087801  0.44
2007 Kim YP, Cho K, Lee D, Piao Y, Ahn YH, Yoo JS, Hyun T, Kim HS. Efficient enrichment and desalting of protein digests using magnetic mesocellular carbon foams in matrix-assisted laser desorption/ionization mass spectrometry. Rapid Communications in Mass Spectrometry : Rcm. 21: 3435-42. PMID 17902195 DOI: 10.1002/rcm.3231  0.96
2007 Kim YP, Oh E, Oh YH, Moon DW, Lee TG, Kim HS. Protein kinase assay on peptide-conjugated gold nanoparticles by using secondary-ion mass spectrometric imaging. Angewandte Chemie (International Ed. in English). 46: 6816-9. PMID 17665386 DOI: 10.1002/anie.200701418  0.52
2007 Pae HO, Jeong GS, Jeong SO, Kim HS, Kim SA, Kim YC, Yoo SJ, Kim HD, Chung HT. Roles of heme oxygenase-1 in curcumin-induced growth inhibition in rat smooth muscle cells. Experimental & Molecular Medicine. 39: 267-77. PMID 17603281 DOI: 10.1038/emm.2007.30  0.44
2007 Han MK, Seo MH, Lee D, Kim SH, Park HS, Kim HS. Optimization of critical factors affecting the performance of an allergen chip for the analysis of an allergen-specific human IgE in serum. Analytical Sciences : the International Journal of the Japan Society For Analytical Chemistry. 23: 545-9. PMID 17495399 DOI: JST.JSTAGE/analsci/23.545  0.52
2007 Kim S, Sohn DW, Kim YC, Kim SA, Lee SK, Kim HS. Fine tuning of a reported synthetic route for biologically active flavonoid, baicalein. Archives of Pharmacal Research. 30: 18-21. PMID 17328237  0.44
2007 Kim YP, Hong MY, Kim J, Oh E, Shon HK, Moon DW, Kim HS, Lee TG. Quantitative analysis of surface-immobilized protein by TOF-SIMS: effects of protein orientation and trehalose additive. Analytical Chemistry. 79: 1377-85. PMID 17297937 DOI: 10.1021/ac0616005  0.52
2007 Hahn YK, Jin Z, Kang JH, Oh E, Han MK, Kim HS, Jang JT, Lee JH, Cheon J, Kim SH, Park HS, Park JK. Magnetophoretic immunoassay of allergen-specific IgE in an enhanced magnetic field gradient. Analytical Chemistry. 79: 2214-20. PMID 17288405 DOI: 10.1021/ac061522l  0.36
2007 Pae HO, Jeong SO, Jeong GS, Kim KM, Kim HS, Kim SA, Kim YC, Kang SD, Kim BN, Chung HT. Curcumin induces pro-apoptotic endoplasmic reticulum stress in human leukemia HL-60 cells. Biochemical and Biophysical Research Communications. 353: 1040-5. PMID 17198682 DOI: 10.1016/j.bbrc.2006.12.133  0.56
2006 Oh E, Lee D, Kim YP, Cha SY, Oh DB, Kang HA, Kim J, Kim HS. Nanoparticle-based energy transfer for rapid and simple detection of protein glycosylation. Angewandte Chemie (International Ed. in English). 45: 7959-63. PMID 17080470 DOI: 10.1002/anie.200601948  0.96
2006 Han MK, Hong MY, Lee D, Lee DE, Noh GY, Lee JH, Kim SH, Kim HS. Expression profiling of proteins in L-threonine biosynthetic pathway of Escherichia coli by using antibody microarray. Proteomics. 6: 5929-40. PMID 17051646 DOI: 10.1002/pmic.200600324  0.52
2004 Dunn PM, Kim HS, Jacobson KA, Burnstock G. Northern Ring Conformation of Methanocarba-Adenosine 5'-Triphosphate Required for Activation of P2X Receptors. Drug Development Research. 61: 227-232. PMID 22833693 DOI: 10.1002/ddr.10381  0.92
2004 Ohno M, Costanzi S, Kim HS, Kempeneers V, Vastmans K, Herdewijn P, Maddileti S, Gao ZG, Harden TK, Jacobson KA. Nucleotide analogues containing 2-oxa-bicyclo[2.2.1]heptane and l-alpha-threofuranosyl ring systems: interactions with P2Y receptors. Bioorganic & Medicinal Chemistry. 12: 5619-30. PMID 15465340 DOI: 10.1016/j.bmc.2004.07.067  0.92
2003 Kim HS, Ohno M, Xu B, Kim HO, Choi Y, Ji XD, Maddileti S, Marquez VE, Harden TK, Jacobson KA. 2-Substitution of adenine nucleotide analogues containing a bicyclo[3.1.0]hexane ring system locked in a northern conformation: enhanced potency as P2Y1 receptor antagonists. Journal of Medicinal Chemistry. 46: 4974-87. PMID 14584948 DOI: 10.1021/jm030127+  0.92
2003 Choi Y, George C, Comin MJ, Barchi JJ, Kim HS, Jacobson KA, Balzarini J, Mitsuya H, Boyer PL, Hughes SH, Marquez VE. A conformationally locked analogue of the anti-HIV agent stavudine. An important correlation between pseudorotation and maximum amplitude. Journal of Medicinal Chemistry. 46: 3292-9. PMID 12852759 DOI: 10.1021/jm030116g  0.56
2003 Kim HS, Jacobson KA. Synthesis of a novel conformationally locked carbocyclic nucleoside ring system. Organic Letters. 5: 1665-8. PMID 12735747 DOI: 10.1021/ol034326z  0.92
2002 Xu B, Stephens A, Kirschenheuter G, Greslin AF, Cheng X, Sennelo J, Cattaneo M, Zighetti ML, Chen A, Kim SA, Kim HS, Bischofberger N, Cook G, Jacobson KA. Acyclic analogues of adenosine bisphosphates as P2Y receptor antagonists: phosphate substitution leads to multiple pathways of inhibition of platelet aggregation. Journal of Medicinal Chemistry. 45: 5694-709. PMID 12477353  0.92
2002 Waldo GL, Corbitt J, Boyer JL, Ravi G, Kim HS, Ji XD, Lacy J, Jacobson KA, Harden TK. Quantitation of the P2Y(1) receptor with a high affinity radiolabeled antagonist. Molecular Pharmacology. 62: 1249-57. PMID 12391289 DOI: 10.1124/mol.62.5.1249  0.56
2002 Kim SA, Marshall MA, Melman N, Kim HS, Müller CE, Linden J, Jacobson KA. Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions. Journal of Medicinal Chemistry. 45: 2131-8. PMID 12014951 DOI: 10.1021/jm0104318  0.56
2002 Ravi RG, Kim HS, Servos J, Zimmermann H, Lee K, Maddileti S, Boyer JL, Harden TK, Jacobson KA. Adenine nucleotide analogues locked in a Northern methanocarba conformation: enhanced stability and potency as P2Y(1) receptor agonists. Journal of Medicinal Chemistry. 45: 2090-100. PMID 11985476 DOI: 10.1021/jm010538v  0.56
2002 Kim HS, Ravi RG, Marquez VE, Maddileti S, Wihlborg AK, Erlinge D, Malmsjö M, Boyer JL, Harden TK, Jacobson KA. Methanocarba modification of uracil and adenine nucleotides: high potency of Northern ring conformation at P2Y1, P2Y2, P2Y4, and P2Y11 but not P2Y6 receptors. Journal of Medicinal Chemistry. 45: 208-18. PMID 11754592 DOI: 10.1021/jm010369e  0.92
2001 Jacobson KA, Ravi RG, Nandanan E, Kim HS, Moro S, Kim YC, Lee K, Barak D, Marquez VE, Ji XD. Ribose modified nucleosides and nucleotides as ligands for purine receptors. Nucleosides, Nucleotides & Nucleic Acids. 20: 333-41. PMID 11563046 DOI: 10.1081/NCN-100002305  0.92
2001 Kim HS, Barak D, Harden TK, Boyer JL, Jacobson KA. Acyclic and cyclopropyl analogues of adenosine bisphosphate antagonists of the P2Y1 receptor: structure-activity relationships and receptor docking. Journal of Medicinal Chemistry. 44: 3092-108. PMID 11543678 DOI: 10.1021/jm010082h  0.92
2001 Ravi G, Lee K, Ji X, Kim HS, Soltysiak KA, Marquez VE, Jacobson KA. Synthesis and purine receptor affinity of 6-oxopurine nucleosides and nucleotides containing (N)-methanocarba-pseudoribose rings. Bioorganic & Medicinal Chemistry Letters. 11: 2295-300. PMID 11527718  0.92
2001 Jacobson KA, Moro S, Hoffmann C, Kim YC, Kim HS, Ravi RG, Harden TK, Boyer JL. Structurally related nucleotides as selective agonists and antagonists at P2Y1 receptors. Farmaco (Società Chimica Italiana : 1989). 56: 71-5. PMID 11347970 DOI: 10.1016/S0014-827X(01)01023-0  0.56
1999 Li AH, Ji XD, Kim HS, Melman N, Jacobson KA. Pyran Template Approach to the Design of Novel A3 Adenosine Receptor Antagonists. Drug Development Research. 48: 171-177. PMID 27182099 DOI: 10.1002/(SICI)1098-2299(199912)48:4<171::AID-DDR4>3.0.CO;2-5  0.92
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