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Stephen C. Bergmeier - Publications

Affiliations: 
Department of Chemistry and Biochemistry Ohio University, Athens, OH, United States 
Area:
Organic Chemistry, Pharmaceutical Chemistry
Website:
https://www.ohio.edu/cas/chemistry/contact/profiles.cfm?profile=bergmeis
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71 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2021 Ghazanfari D, Noori MS, Bergmeier SC, Hines JV, McCall KD, Goetz DJ. A novel GSK-3 inhibitor binds to GSK-3β via a reversible, time and Cys-199-dependent mechanism. Bioorganic & Medicinal Chemistry. 40: 116179. PMID 33991821 DOI: 10.1016/j.bmc.2021.116179  0.62
2021 Shriwas P, Roberts D, Li Y, Wang L, Qian Y, Bergmeier S, Hines J, Adhicary S, Nielsen C, Chen X. A small-molecule pan-class I glucose transporter inhibitor reduces cancer cell proliferation in vitro and tumor growth in vivo by targeting glucose-based metabolism. Cancer & Metabolism. 9: 14. PMID 33771231 DOI: 10.1186/s40170-021-00248-7  0.615
2020 Armstrong I, Aldhumani AH, Schopis JL, Fang F, Parsons E, Zeng C, Hossain MI, Bergmeier SC, Hines JV. RNA drug discovery: Conformational restriction enhances specific modulation of the T-box riboswitch function. Bioorganic & Medicinal Chemistry. 28: 115696. PMID 33069065 DOI: 10.1016/J.Bmc.2020.115696  0.717
2020 Roberts DA, Wang L, Zhang W, Liu Y, Shriwas P, Qian Y, Chen X, Bergmeier SC. Isosteres of ester derived glucose uptake inhibitors. Bioorganic & Medicinal Chemistry Letters. 30: 127406. PMID 32736210 DOI: 10.1016/J.Bmcl.2020.127406  0.533
2019 Noori MS, Bhatt PM, Courreges MC, Ghazanfari D, Cuckler C, Orac CM, McMills MC, Schwartz FL, Deosarkar SP, Bergmeier SC, McCall KD, Goetz DJ. Identification of a Novel Selective and Potent Inhibitor of Glycogen Synthase Kinase-3. American Journal of Physiology. Cell Physiology. PMID 31553649 DOI: 10.1152/Ajpcell.00061.2019  0.759
2019 Zheng Z, Bergmeier SC. Routes to N-glycinamide oxazolidinone derivatives: The reaction of 4-trityloxymethyl-3-oxa-1-azabicyclo[3.1.0]hexan-2-one with active halides Arkivoc. 2019: 40-52. DOI: 10.24820/Ark.5550190.P010.812  0.31
2017 Armstrong I, Bergmeier S. Development of a Method for the Synthesis of 4-Aryl-Functionalized 2-Azabicyclo[3.2.1]octanes Synthesis. 49: 2733-2742. DOI: 10.1055/S-0036-1558973  0.342
2015 Zeng C, Zhou S, Bergmeier SC, Hines JV. Factors that influence T box riboswitch efficacy and tRNA affinity. Bioorganic & Medicinal Chemistry. 23: 5702-8. PMID 26220520 DOI: 10.1016/J.Bmc.2015.07.018  0.69
2015 Alapati A, Deosarkar SP, Lanier OL, Qi C, Carlson GE, Burdick MM, Schwartz FL, McCall KD, Bergmeier SC, Goetz DJ. Simple modifications to methimazole that enhance its inhibitory effect on tumor necrosis factor-α-induced vascular cell adhesion molecule-1 expression by human endothelial cells. European Journal of Pharmacology. 751: 59-66. PMID 25641748 DOI: 10.1016/J.Ejphar.2015.01.032  0.31
2013 Bergmeier SC, Lapinsky DJ. Chapter 2 - Three-Membered Ring Systems Progress in Heterocyclic Chemistry. 25. DOI: 10.1016/B978-0-08-099406-2.00002-9  0.336
2012 Henderson BJ, González-Cestari TF, Yi B, Pavlovicz RE, Boyd RT, Li C, Bergmeier SC, McKay DB. Defining the putative inhibitory site for a selective negative allosteric modulator of human α4β2 neuronal nicotinic receptors. Acs Chemical Neuroscience. 3: 682-92. PMID 23019495 DOI: 10.1021/Cn300035F  0.325
2012 Liu Y, Cao Y, Zhang W, Bergmeier S, Qian Y, Akbar H, Colvin R, Ding J, Tong L, Wu S, Hines J, Chen X. A small-molecule inhibitor of glucose transporter 1 downregulates glycolysis, induces cell-cycle arrest, and inhibits cancer cell growth in vitro and in vivo Molecular Cancer Therapeutics. 11: 1672-1682. PMID 22689530 DOI: 10.1158/1535-7163.Mct-12-0131  0.717
2012 Fang F, Vogel M, Hines JV, Bergmeier SC. Fused ring aziridines as a facile entry into triazole fused tricyclic and bicyclic heterocycles. Organic & Biomolecular Chemistry. 10: 3080-91. PMID 22402729 DOI: 10.1039/C2Ob07042A  0.696
2012 Henderson BJ, Orac CM, Maciagiewicz I, Bergmeier SC, McKay DB. 3D-QSAR and 3D-QSSR models of negative allosteric modulators facilitate the design of a novel selective antagonist of human α4β2 neuronal nicotinic acetylcholine receptors. Bioorganic & Medicinal Chemistry Letters. 22: 1797-813. PMID 22285942 DOI: 10.1016/J.Bmcl.2011.11.051  0.773
2012 Zhou S, Means JA, Acquaah-Harrison G, Bergmeier SC, Hines JV. Characterization of a 1,4-disubstituted 1,2,3-triazole binding to T box antiterminator RNA. Bioorganic & Medicinal Chemistry. 20: 1298-302. PMID 22230198 DOI: 10.1016/J.Bmc.2011.12.017  0.776
2012 Zhou S, Acquaah-Harrison G, Jack KD, Bergmeier SC, Hines JV. Ligand-induced changes in T box antiterminator RNA stability. Chemical Biology & Drug Design. 79: 202-8. PMID 22117759 DOI: 10.1111/J.1747-0285.2011.01274.X  0.764
2012 Luesse SB, Wells G, Miller J, Bolstad E, Bergmeier SC, McMills MC, Priestley ND, Wright DL. Synthesis of a functionalized oxabicyclo[2.2.1]-heptene-based chemical library. Combinatorial Chemistry & High Throughput Screening. 15: 81-9. PMID 21774767 DOI: 10.2174/138620712798280835  0.394
2012 Liu Y, Cao Y, Zhang W, Bergmeier S, Qian Y, Akbar H, Colvin R, Ding J, Tong L, Wu S, Hines J, Chen X. Abstract 3231: A small molecule inhibitor of glucose transporter 1 (Glut1) down-regulates glycolysis, induces cell cycle arrest, and inhibits cancer cell growthin vitroandin vivo Cancer Research. 72: 3231-3231. DOI: 10.1158/1538-7445.Am2012-3231  0.719
2012 Bergmeier S, Maciagiewicz I, Fang F, Roberts D, Zhou S, Hines J. A Synthesis of 1,4-Disubstituted Imidazolidin-2-ones from Fused-Ring Aziridines Synthesis. 2012: 551-560. DOI: 10.1055/S-0031-1289684  0.691
2012 Wells GM, Dudding T, Belding L, Frick JA, Nayek A, Huang J, Katz SJ, Bergmeier SC. Studies on the ring opening reactions of 3-oxa-1-azabicyclo[3.1.0]hexan-2- ones. Synthesis of aminomethyl oxazolidinones and aziridinyl ureas Tetrahedron. 68: 3980-3987. DOI: 10.1016/J.Tet.2012.03.071  0.553
2012 Wells GM, Dudding T, Belding L, Frick JA, Nayek A, Huang J, Katz SJ, Bergmeier SC. ChemInform Abstract: Studies on the Ring Opening Reactions of 3-Oxa-1-azabicyclo[3.1.0]hexan-2-ones. Synthesis of Aminomethyl Oxazolidinones and Aziridinyl Ureas. Cheminform. 43: no-no. DOI: 10.1002/CHIN.201244035  0.523
2012 Maciagiewicz IM, Fang F, Roberts DA, Zhou S, Hines JV, Bergmeier SC. ChemInform Abstract: A Synthesis of 1,4-Disubstituted Imidazolidin-2-ones from Fused-Ring Aziridines. Cheminform. 43: no-no. DOI: 10.1002/CHIN.201224120  0.667
2011 Zhou S, Acquaah-Harrison G, Bergmeier SC, Hines JV. Anisotropy studies of tRNA-T box antiterminator RNA complex in the presence of 1,4-disubstituted 1,2,3-triazoles. Bioorganic & Medicinal Chemistry Letters. 21: 7059-63. PMID 22001091 DOI: 10.1016/J.Bmcl.2011.09.095  0.779
2011 Hurst WJ, Krake SH, Bergmeier SC, Payne MJ, Miller KB, Stuart DA. Impact of fermentation, drying, roasting and Dutch processing on flavan-3-ol stereochemistry in cacao beans and cocoa ingredients. Chemistry Central Journal. 5: 53. PMID 21917164 DOI: 10.1186/1752-153X-5-53  0.749
2011 Orac CM, Zhou S, Means JA, Boehm D, Bergmeier SC, Hines JV. Synthesis and stereospecificity of 4,5-disubstituted oxazolidinone ligands binding to T-box riboswitch RNA. Journal of Medicinal Chemistry. 54: 6786-95. PMID 21812425 DOI: 10.1021/Jm2006904  0.789
2011 Maciagiewicz I, Zhou S, Bergmeier SC, Hines JV. Structure-activity studies of RNA-binding oxazolidinone derivatives. Bioorganic & Medicinal Chemistry Letters. 21: 4524-7. PMID 21733684 DOI: 10.1016/J.Bmcl.2011.05.130  0.707
2011 Sumskaya YG, Swain PW, Bergmeier SC, McMills MC, Priestley ND, Wrighta DL. Natural feedstocks for diversity-oriented synthesis: Macrolide-like scaffolds from nonactate Arkivoc. 2011: 144-166. DOI: 10.3998/Ark.5550190.0012.513  0.344
2011 Liu Y, Zhang W, Cao Y, Bergmeier S, Akbar H, Colvin R, Qian Y, Ding J, Chen X. Abstract 4068: A novel antiglycolytic small compound inhibits cancer growth in vitro and in vivo by inhibiting glut1 Cancer Research. 71: 4068-4068. DOI: 10.1158/1538-7445.Am2011-4068  0.531
2010 Liu Y, Zhang W, Cao Y, Liu Y, Bergmeier S, Chen X. Small compound inhibitors of basal glucose transport inhibit cell proliferation and induce apoptosis in cancer cells via glucose-deprivation-like mechanisms. Cancer Letters. 298: 176-85. PMID 20678861 DOI: 10.1016/J.Canlet.2010.07.002  0.516
2010 Acquaah-Harrison G, Zhou S, Hines JV, Bergmeier SC. Library of 1,4-disubstituted 1,2,3-triazole analogs of oxazolidinone RNA-binding agents. Journal of Combinatorial Chemistry. 12: 491-6. PMID 20557032 DOI: 10.1021/Cc100029Y  0.79
2010 Henderson BJ, Pavlovicz RE, Allen JD, González-Cestari TF, Orac CM, Bonnell AB, Zhu MX, Boyd RT, Li C, Bergmeier SC, McKay DB. Negative allosteric modulators that target human alpha4beta2 neuronal nicotinic receptors. The Journal of Pharmacology and Experimental Therapeutics. 334: 761-74. PMID 20551292 DOI: 10.1124/Jpet.110.168211  0.788
2010 Zhang W, Liu Y, Chen X, Bergmeier SC. Novel inhibitors of basal glucose transport as potential anticancer agents. Bioorganic & Medicinal Chemistry Letters. 20: 2191-4. PMID 20194024 DOI: 10.1016/J.Bmcl.2010.02.027  0.516
2010 Bergmeier SC, Krake SH. Inter- and intramolecular reactions of epoxides and aziridines with π-nucleophiles Tetrahedron. 66: 7337-7360. DOI: 10.1016/J.Tet.2010.06.064  0.772
2010 HEIDT PC, BERGMEIER SC, PEARSON WH. ChemInform Abstract: Synthesis of Indolizidines by the 1,3-Dipolar Cycloaddition of Azides with Methyl Methylenecyclopropanes Followed by Cyclopropylimine Rearrangement. Cheminform. 22: no-no. DOI: 10.1002/chin.199141167  0.514
2009 González-Cestari TF, Henderson BJ, Pavlovicz RE, McKay SB, El-Hajj RA, Pulipaka AB, Orac CM, Reed DD, Boyd RT, Zhu MX, Li C, Bergmeier SC, McKay DB. Effect of novel negative allosteric modulators of neuronal nicotinic receptors on cells expressing native and recombinant nicotinic receptors: implications for drug discovery. The Journal of Pharmacology and Experimental Therapeutics. 328: 504-15. PMID 18984653 DOI: 10.1124/Jpet.108.144576  0.757
2009 Bergmeier SC, Lapinsky DJ. Chapter 3: Three-membered ring systems Progress in Heterocyclic Chemistry. 19: 47-73. DOI: 10.1016/S0959-6380(08)80005-0  0.363
2009 Orac CM, Bergmeier SC. A formal [3+2] cycloaddition for the synthesis of bicyclo[3.2.1]octanes Tetrahedron Letters. 50: 1261-1263. DOI: 10.1016/J.Tetlet.2008.12.098  0.771
2009 Lapinsky DJ, Pulipaka AB, Bergmeier SC. Substitution effects in intramolecular aziridine-allylsilane cyclizations Tetrahedron. 65: 741-747. DOI: 10.1016/J.Tet.2008.11.043  0.778
2009 Orac CM, Bergmeier SC. ChemInform Abstract: A Formal [3 + 2] Cycloaddition for the Synthesis of Bicyclo[3.2.1]octanes. Cheminform. 40. DOI: 10.1002/chin.200926069  0.783
2008 Emelda N, Bergmeier SC. Ring expansion of substituted norbornadienes for the synthesis of mono- and disubstituted 2-azabicyclo[3.2.1]octadienes. Tetrahedron Letters. 49: 5363-5365. PMID 19746153 DOI: 10.1016/J.Tetlet.2008.06.123  0.374
2008 Huang J, Bergmeier SC. Diastereoselective Synthesis of a Highly Substituted cis-Decahydroquinoline via a Knoevenagel Condensation. Tetrahedron. 64: 6434-6439. PMID 19572008 DOI: 10.1016/J.Tet.2008.04.073  0.543
2008 Luesse SB, Wells G, Nayek A, Smith AE, Kusche BR, Bergmeier SC, McMills MC, Priestley ND, Wright DL. Natural products in parallel synthesis: triazole libraries of nonactic acid. Bioorganic & Medicinal Chemistry Letters. 18: 3946-9. PMID 18585037 DOI: 10.1016/J.Bmcl.2008.06.020  0.337
2008 Anupam R, Nayek A, Green NJ, Grundy FJ, Henkin TM, Means JA, Bergmeier SC, Hines JV. 4,5-Disubstituted oxazolidinones: High affinity molecular effectors of RNA function. Bioorganic & Medicinal Chemistry Letters. 18: 3541-4. PMID 18502126 DOI: 10.1016/J.Bmcl.2008.05.015  0.694
2008 Huang J, Orac CM, McKay S, McKay DB, Bergmeier SC. The synthesis of 5-substituted ring E analogs of methyllycaconitine via the Suzuki-Miyaura cross-coupling reaction. Bioorganic & Medicinal Chemistry. 16: 3816-24. PMID 18272373 DOI: 10.1016/J.Bmc.2008.01.050  0.787
2008 Pulipaka AB, Bergmeier SC. A synthesis of 6-azabicyclo[3.2.1]octanes. The role of N-substitution. The Journal of Organic Chemistry. 73: 1462-7. PMID 18211092 DOI: 10.1021/Jo702444C  0.79
2008 Pulipaka AB, Bergmeier SC. Synthesis of hexahydro-1H-benzo[c]chromen-1-amines via the intramolecular ring-opening reactions of aziridines by π-nucleophiles Synthesis. 1420-1430. DOI: 10.1055/S-2008-1072561  0.784
2008 Pulipaka AB, Bergmeier SC. ChemInform Abstract: Synthesis of Hexahydro-1H-benzo[c]chromen-1-amines via the Intramolecular Ring-Opening Reactions of Aziridines by π-Nucleophiles. Cheminform. 39. DOI: 10.1002/chin.200837138  0.786
2007 McKay DB, Chang C, González-Cestari TF, McKay SB, El-Hajj RA, Bryant DL, Zhu MX, Swaan PW, Arason KM, Pulipaka AB, Orac CM, Bergmeier SC. Analogs of methyllycaconitine as novel noncompetitive inhibitors of nicotinic receptors: pharmacological characterization, computational modeling, and pharmacophore development. Molecular Pharmacology. 71: 1288-97. PMID 17308033 DOI: 10.1124/Mol.106.033233  0.763
2007 Reed DD, Bergmeier SC. A facile synthesis of a polyhydroxylated 2-azabicyclo[3.2.1]octane. The Journal of Organic Chemistry. 72: 1024-6. PMID 17253828 DOI: 10.1021/Jo0619231  0.317
2006 Means J, Katz S, Nayek A, Anupam R, Hines JV, Bergmeier SC. Structure-activity studies of oxazolidinone analogs as RNA-binding agents. Bioorganic & Medicinal Chemistry Letters. 16: 3600-4. PMID 16603349 DOI: 10.1016/J.Bmcl.2006.03.068  0.715
2006 Malki A, Pulipaka AB, Evans SC, Bergmeier SC. Structure-activity studies of quinuclidinone analogs as anti-proliferative agents in lung cancer cell lines. Bioorganic & Medicinal Chemistry Letters. 16: 1156-9. PMID 16361100 DOI: 10.1016/J.Bmcl.2005.11.085  0.754
2004 Bergmeier SC, Ismail KA, Arason KM, McKay S, Bryant DL, McKay DB. Structure activity studies of ring E analogues of methyllycaconitine. Part 2: Synthesis of antagonists to the alpha3beta4* nicotinic acetylcholine receptors through modifications to the ester. Bioorganic & Medicinal Chemistry Letters. 14: 3739-42. PMID 15203153 DOI: 10.1016/J.Bmcl.2004.05.001  0.394
2004 Bergmeier SC, Katz SJ, Huang J, McPherson H, Donoghue PJ, Reed DD. Intramolecular cyclization reactions of aziridines with π-nucleophiles Tetrahedron Letters. 45: 5011-5014. DOI: 10.1016/J.Tetlet.2004.05.009  0.555
2004 Bergmeier SC, Katz SJ, Huang J, McPherson H, Donoghue PJ, Reed DD. Intramolecular Cyclization Reactions of Aziridines with π-Nucleophiles. Cheminform. 35. DOI: 10.1002/chin.200440102  0.477
2003 Lapinsky DJ, Bergmeier SC. Aziridine—Allylsilane-Mediated Synthesis of Exocyclic γ-Amino Olefins and Azabicyclo[x.y.1]-Systems. Cheminform. 34. DOI: 10.1016/S0040-4020(02)00725-1  0.317
2002 Bryant DL, Free RB, Thomasy SM, Lapinsky DJ, Ismail KA, Arason KM, Bergmeier SC, McKay DB. Effects of methyllycaconitine and related analogues on bovine adrenal alpha3beta4* nicotinic acetylcholine receptors. Annals of the New York Academy of Sciences. 971: 139-41. PMID 12438104 DOI: 10.1111/J.1749-6632.2002.Tb04448.X  0.351
2002 Donaldson SF, Bergmeier SC, Hines JV, Gerdeman MS. Synthesis and hybridization studies of a 5-aminopentanoic acid nucleobase (APN) dimer. Nucleosides, Nucleotides & Nucleic Acids. 21: 111-23. PMID 11991139 DOI: 10.1081/Ncn-120003176  0.64
2002 Bergmeier SC, Katz SJ. A method for the parallel synthesis of multiply substituted oxazolidinones. Journal of Combinatorial Chemistry. 4: 162-6. PMID 11886291 DOI: 10.1021/Cc010050F  0.399
2002 Bryant DL, Free RB, Thomasy SM, Lapinsky DJ, Ismail KA, McKay SB, Bergmeier SC, McKay DB. Structure-activity studies with ring E analogues of methyllycaconitine on bovine adrenal alpha3beta4* nicotinic receptors. Neuroscience Research. 42: 57-63. PMID 11814609 DOI: 10.1016/S0168-0102(01)00304-2  0.382
2001 Lapinsky DJ, Bergmeier SC. A Suzuki cross-coupling route to substituted aziridines Tetrahedron Letters. 42: 8583-8586. DOI: 10.1016/S0040-4039(01)01903-7  0.341
2000 Bergmeier SC, Ismail KA. Synthesis of Monosubstituted Succinic Acids from tert-Butylsuccinate Synthesis. 2000: 1369-1371. DOI: 10.1055/S-2000-7110  0.301
1993 Bergmeier SC, Lee WK, Rapoport H. Chirospecific synthesis of (1S,3R)-1-amino-3-(hydroxymethyl)cyclopentane, a precursor for carbocyclic nucleoside synthesis. Intramolecular aziridine cyclizations The Journal of Organic Chemistry. 58: 5019-5022. DOI: 10.1021/Jo00070A050  0.326
1993 Bergmeier SC, Cobas AA, Rapoport H. Chirospecific synthesis of (1S,3R)-1-amino-3-(hydroxymethyl)cyclopentane, precursor for carbocyclic nucleoside synthesis. Dieckmann cyclization with an .alpha.-amino acid The Journal of Organic Chemistry. 58: 2369-2376. DOI: 10.1021/Jo00061A006  0.305
1992 Pearson WH, Bergmeier SC, Williams JP. Synthesis of (-)-slaframine and related indolizidines Journal of Organic Chemistry. 57: 3977-3987. DOI: 10.1021/Jo00040A045  0.588
1991 Pearson WH, Bergmeier SC. A synthesis of (-)-slaframine and (-)-1,8a-diepislaframine Journal of Organic Chemistry. 56: 1976-1978. DOI: 10.1021/Jo00006A002  0.563
1990 Jean JC, Wise LD, Caprathe BW, Tecle H, Bergmeier S, Humblet CC, Heffner TG, Meltzer LT, Pugsley TA. 4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: A novel class of compounds with central dopamine agonist properties Journal of Medicinal Chemistry. 33: 311-317. PMID 1967314 DOI: 10.1021/Jm00163A051  0.336
1990 Pearson WH, Bergmeier SC, Chytra JA. The Synthesis of Triazole Analogues of Antitumor Dehydropyrrolizidine Alkaloids Synthesis. 1990: 156-159. DOI: 10.1055/S-1990-26820  0.599
1990 Pearson WH, Bergmeier SC, Degan S, Lin KC, Poon YF, Schkeryantz JM, Williams JP. Synthesis of pyrrolizidines and indolizidines by the intramolecular cycloaddition of azides with electron-rich 1,3-dienes. A synthetic equivalent of a nitrene-diene cycloaddition Journal of Organic Chemistry. 55: 5719-5738. DOI: 10.1021/Jo00309A016  0.575
1990 Heidt. PC, Bergmeier SC, Pearson WH. Synthesis of indolidines by the 1,3-dipolar cycloaddition of azides with methylenecyclopropanes followed by cyclopropyumine rearrangement Tetrahedron Letters. 31: 5441-5444. DOI: 10.1016/S0040-4039(00)97867-5  0.558
1990 PEARSON WH, BERGMEIER S, CHYTRA JA. ChemInform Abstract: The Synthesis of Triazole Analogues of Antitumor Dehydropyrrolizidine Alkaloids. Cheminform. 21. DOI: 10.1002/chin.199028167  0.562
1989 Tecle H, Bergmeier SC, Wise LD, Hershenson FM, Coughenour LL, Heffner TG. Alkyl substituted3-PPPderivatives. Synthesis and biological investigation Journal of Heterocyclic Chemistry. 26: 1125-1128. DOI: 10.1002/Jhet.5570260441  0.362
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