Year |
Citation |
Score |
2012 |
Tarrant MK, Rho HS, Xie Z, Jiang YL, Gross C, Culhane JC, Yan G, Qian J, Ichikawa Y, Matsuoka T, Zachara N, Etzkorn FA, Hart GW, Jeong JS, Blackshaw S, et al. Regulation of CK2 by phosphorylation and O-GlcNAcylation revealed by semisynthesis. Nature Chemical Biology. 8: 262-9. PMID 22267120 DOI: 10.1038/Nchembio.771 |
0.477 |
|
2010 |
Culhane JC, Wang D, Yen PM, Cole PA. Comparative analysis of small molecules and histone substrate analogues as LSD1 lysine demethylase inhibitors. Journal of the American Chemical Society. 132: 3164-76. PMID 20148560 DOI: 10.1021/Ja909996P |
0.543 |
|
2007 |
Szewczuk LM, Saldanha SA, Ganguly S, Bowers EM, Javoroncov M, Karanam B, Culhane JC, Holbert MA, Klein DC, Abagyan R, Cole PA. De novo discovery of serotonin N-acetyltransferase inhibitors. Journal of Medicinal Chemistry. 50: 5330-8. PMID 17924613 DOI: 10.1021/Jm0706463 |
0.569 |
|
2007 |
Culhane JC, Cole PA. LSD1 and the chemistry of histone demethylation. Current Opinion in Chemical Biology. 11: 561-8. PMID 17851108 DOI: 10.1016/J.Cbpa.2007.07.014 |
0.531 |
|
2007 |
Yang M, Culhane JC, Szewczuk LM, Jalili P, Ball HL, Machius M, Cole PA, Yu H. Structural basis for the inhibition of the LSD1 histone demethylase by the antidepressant trans-2-phenylcyclopropylamine. Biochemistry. 46: 8058-65. PMID 17569509 DOI: 10.1021/Bi700664Y |
0.576 |
|
2007 |
Yang M, Culhane JC, Szewczuk LM, Gocke CB, Brautigam CA, Tomchick DR, Machius M, Cole PA, Yu H. Structural basis of histone demethylation by LSD1 revealed by suicide inactivation. Nature Structural & Molecular Biology. 14: 535-9. PMID 17529991 DOI: 10.1038/Nsmb1255 |
0.548 |
|
2007 |
Szewczuk LM, Culhane JC, Yang M, Majumdar A, Yu H, Cole PA. Mechanistic analysis of a suicide inactivator of histone demethylase LSD1. Biochemistry. 46: 6892-902. PMID 17511474 DOI: 10.1021/Bi700414B |
0.582 |
|
2006 |
Culhane JC, Szewczuk LM, Liu X, Da G, Marmorstein R, Cole PA. A mechanism-based inactivator for histone demethylase LSD1. Journal of the American Chemical Society. 128: 4536-7. PMID 16594666 DOI: 10.1021/Ja0602748 |
0.581 |
|
Low-probability matches (unlikely to be authored by this person) |
2008 |
Ebner DC, Culhane JC, Winkelman TN, Haustein MD, Ditty JL, Ippoliti JT. Synthesis of novel oxazolidinone antimicrobial agents. Bioorganic & Medicinal Chemistry. 16: 2651-6. PMID 18077175 DOI: 10.1016/j.bmc.2007.11.040 |
0.14 |
|
2011 |
Culhane JC, Fokin VV. Synthesis and reactivity of sulfamoyl azides and 1-sulfamoyl-1,2,3-triazoles. Organic Letters. 13: 4578-80. PMID 21812453 DOI: 10.1021/Ol201705K |
0.095 |
|
2014 |
Culhane JC, Dawson PE. Peptide pharmaceuticals: Modifications to the peptide backbone that enhance stability and targeting Chimica Oggi/Chemistry Today. 32: 17-20. |
0.094 |
|
2016 |
Kaushik A, Heuer AM, Bell DT, Culhane JC, Ebner DC, Parrish N, Ippoliti JT, Lamichhane G. An evolved oxazolidinone with selective potency against Mycobacterium tuberculosis and gram positive bacteria. Bioorganic & Medicinal Chemistry Letters. PMID 27329794 DOI: 10.1016/J.Bmcl.2016.06.019 |
0.072 |
|
2015 |
Kong L, Kadam RU, Giang E, Ruwona TB, Nieusma T, Culhane JC, Stanfield RL, Dawson PE, Wilson IA, Law M. Structure of hepatitis C virus envelope glycoprotein E1 antigenic site 314-324 in complex with antibody IGH526. Journal of Molecular Biology. PMID 26135247 DOI: 10.1016/J.Jmb.2015.06.012 |
0.067 |
|
2021 |
Sato Y, Liu J, Kukor AJ, Culhane JC, Tucker JL, Kucera DJ, Cochran BM, Hein JE. Real-Time Monitoring of Solid-Liquid Slurries: Optimized Synthesis of Tetrabenazine. The Journal of Organic Chemistry. PMID 34213349 DOI: 10.1021/acs.joc.1c01098 |
0.048 |
|
2022 |
Kukor AJ, Depner N, Cai I, Tucker JL, Culhane JC, Hein JE. Enantioselective synthesis of (-)-tetrabenazine continuous crystallization-induced diastereomer transformation. Chemical Science. 13: 10765-10772. PMID 36320713 DOI: 10.1039/d2sc01825j |
0.043 |
|
Hide low-probability matches. |