Year |
Citation |
Score |
2017 |
Banerjee S, Norman DD, Lee SC, Parrill AL, Pham TC, Baker DL, Tigyi GG, Miller DD. Highly Potent Non-Carboxylic Acid Autotaxin Inhibitors Reduce Melanoma Metastasis and Chemotherapeutic Resistance of Breast Cancer Stem Cells. Journal of Medicinal Chemistry. PMID 28112925 DOI: 10.1021/Acs.Jmedchem.6B01270 |
0.641 |
|
2014 |
Fells JI, Lee SC, Norman DD, Tsukahara R, Kirby JR, Nelson S, Seibel W, Papoian R, Patil R, Miller DD, Parrill AL, Pham TC, Baker DL, Bittman R, Tigyi G. Targeting the hydrophobic pocket of autotaxin with virtual screening of inhibitors identifies a common aromatic sulfonamide structural motif. The Febs Journal. 281: 1017-28. PMID 24314137 DOI: 10.1111/Febs.12674 |
0.8 |
|
2013 |
Young JK, Clayton BT, Kikonyogo A, Pham TC, Parrill AL. Structural Characterization of an LPA1 Second Extracellular Loop Mimetic with a Self-Assembling Coiled-Coil Folding Constraint. International Journal of Molecular Sciences. 14: 2788-807. PMID 23434648 DOI: 10.3390/Ijms14022788 |
0.734 |
|
2011 |
Parrill AL, Wanjala IW, Pham TC, Baker DL. Computational identification and experimental characterization of substrate binding determinants of nucleotide pyrophosphatase/phosphodiesterase 7. Bmc Biochemistry. 12: 65. PMID 22177013 DOI: 10.1186/1471-2091-12-65 |
0.7 |
|
2011 |
Gupte R, Patil R, Liu J, Wang Y, Lee SC, Fujiwara Y, Fells J, Bolen AL, Emmons-Thompson K, Yates CR, Siddam A, Panupinthu N, Pham TC, Baker DL, Parrill AL, et al. Benzyl and naphthalene methylphosphonic acid inhibitors of autotaxin with anti-invasive and anti-metastatic activity. Chemmedchem. 6: 922-35. PMID 21465666 DOI: 10.1002/Cmdc.201000425 |
0.79 |
|
2010 |
Gupte R, Siddam A, Lu Y, Li W, Fujiwara Y, Panupinthu N, Pham TC, Baker DL, Parrill AL, Gotoh M, Murakami-Murofushi K, Kobayashi S, Mills GB, Tigyi G, Miller DD. Synthesis and pharmacological evaluation of the stereoisomers of 3-carba cyclic-phosphatidic acid. Bioorganic & Medicinal Chemistry Letters. 20: 7525-8. PMID 21051230 DOI: 10.1016/J.Bmcl.2010.09.115 |
0.649 |
|
2010 |
Valentine WJ, Kiss GN, Liu J, E S, Gotoh M, Murakami-Murofushi K, Pham TC, Baker DL, Parrill AL, Lu X, Sun C, Bittman R, Pyne NJ, Tigyi G. (S)-FTY720-vinylphosphonate, an analogue of the immunosuppressive agent FTY720, is a pan-antagonist of sphingosine 1-phosphate GPCR signaling and inhibits autotaxin activity. Cellular Signalling. 22: 1543-53. PMID 20566326 DOI: 10.1016/J.Cellsig.2010.05.023 |
0.633 |
|
2010 |
North EJ, Howard AL, Wanjala IW, Pham TC, Baker DL, Parrill AL. Pharmacophore development and application toward the identification of novel, small-molecule autotaxin inhibitors. Journal of Medicinal Chemistry. 53: 3095-105. PMID 20349977 DOI: 10.1021/Jm901718Z |
0.723 |
|
2010 |
Hoeglund AB, Howard AL, Wanjala IW, Pham TC, Parrill AL, Baker DL. Characterization of non-lipid autotaxin inhibitors. Bioorganic & Medicinal Chemistry. 18: 769-76. PMID 20005724 DOI: 10.1016/J.Bmc.2009.11.056 |
0.659 |
|
2008 |
Pham TC, Fells JI, Osborne DA, North EJ, Naor MM, Parrill AL. Molecular recognition in the sphingosine 1-phosphate receptor family. Journal of Molecular Graphics & Modelling. 26: 1189-201. PMID 18165127 DOI: 10.1016/J.Jmgm.2007.11.001 |
0.722 |
|
2008 |
Parrill AL, Echols U, Nguyen T, Pham TC, Hoeglund A, Baker DL. Virtual screening approaches for the identification of non-lipid autotaxin inhibitors. Bioorganic & Medicinal Chemistry. 16: 1784-95. PMID 18036821 DOI: 10.1016/J.Bmc.2007.11.018 |
0.771 |
|
2007 |
Pham TC, Kriwacki RW, Parrill AL. Peptide design and structural characterization of a GPCR loop mimetic. Biopolymers. 86: 298-310. PMID 17443712 DOI: 10.1002/Bip.20745 |
0.582 |
|
1985 |
Pham TC, Leluk J, Polanowski A, Wilusz T. Purification and characterization of the trypsin inhibitor from Cucurbita pepo var. patissonina fruits. Biological Chemistry Hoppe-Seyler. 366: 939-44. PMID 3933527 DOI: 10.1515/bchm3.1985.366.2.939 |
0.321 |
|
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