Year |
Citation |
Score |
2019 |
Vaidya AS, Helander JDM, Peterson FC, Elzinga D, Dejonghe W, Kaundal A, Park SY, Xing Z, Mega R, Takeuchi J, Khanderahoo B, Bishay S, Volkman BF, Todoroki Y, Okamoto M, et al. Dynamic control of plant water use using designed ABA receptor agonists. Science (New York, N.Y.). 366. PMID 31649167 DOI: 10.1126/Science.Aaw8848 |
0.313 |
|
2019 |
Elzinga D, Sternburg E, Sabbadin D, Bartsch M, Park SY, Vaidya A, Mosquna A, Kaundal A, Wendeborn S, Lachia M, Karginov FV, Cutler SR. Defining and Exploiting Hypersensitivity Hotspots to Facilitate Abscisic Acid Agonist Optimization. Acs Chemical Biology. PMID 30668093 DOI: 10.1021/Acschembio.8B00955 |
0.359 |
|
2017 |
Petukhov PA, Abdelkarim H, Neelarapu R, Madriaga A, Kastrati I, Wang YT, Vaidya AS, Taha TY, Thatcher GRJ, Frasor J. Design, Synthesis, Molecular Modeling, and Biological Evaluation of Novel Amine-based Histone Deacetylase Inhibitors. Chemmedchem. PMID 29080240 DOI: 10.1002/Cmdc.201700449 |
0.601 |
|
2017 |
Vaidya AS, Peterson FC, Yarmolinsky D, Merilo E, Verstraeten I, Park SY, Elzinga D, Kaundal A, Helander J, Lozano-Juste J, Otani M, Wu K, Jensen DR, Kollist H, Volkman BF, et al. A rationally designed agonist defines subfamily IIIA ABA receptors as critical targets for manipulating transpiration. Acs Chemical Biology. PMID 28949512 DOI: 10.1021/Acschembio.7B00650 |
0.334 |
|
2014 |
Patel HK, Siklos MI, Abdelkarim H, Mendonca EL, Vaidya A, Petukhov PA, Thatcher GR. A chimeric SERM-histone deacetylase inhibitor approach to breast cancer therapy. Chemmedchem. 9: 602-13. PMID 23956109 DOI: 10.1002/Cmdc.201300270 |
0.589 |
|
2014 |
Patel HK, Siklos MI, Abdelkarim H, Mendonca EL, Vaidya A, Petukhov PA, Thatcher GRJ. Cover Picture: A Chimeric SERM-Histone Deacetylase Inhibitor Approach to Breast Cancer Therapy (ChemMedChem 3/2014) Chemmedchem. 9: 413-413. DOI: 10.1002/Cmdc.201490005 |
0.581 |
|
2012 |
Vaidya AS, Neelarapu R, Madriaga A, Bai H, Mendonca E, Abdelkarim H, van Breemen RB, Blond SY, Petukhov PA. Novel histone deacetylase 8 ligands without a zinc chelating group: exploring an 'upside-down' binding pose. Bioorganic & Medicinal Chemistry Letters. 22: 6621-7. PMID 23010266 DOI: 10.1016/J.Bmcl.2012.08.104 |
0.566 |
|
2012 |
Vaidya AS, Karumudi B, Mendonca E, Madriaga A, Abdelkarim H, van Breemen RB, Petukhov PA. Design, synthesis, modeling, biological evaluation and photoaffinity labeling studies of novel series of photoreactive benzamide probes for histone deacetylase 2. Bioorganic & Medicinal Chemistry Letters. 22: 5025-30. PMID 22771007 DOI: 10.1016/J.Bmcl.2012.06.017 |
0.576 |
|
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