Keykavous Parang - Related publications

2000-2013 Biomedical and Pharmaceutical Sciences University of Rhode Island, Providence, RI, United States 
 2013- Medicinal Chemistry and Pharmacology Chapman University, Orange, CA, United States 
Pharmaceutical Chemistry, Pharmacology
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50 most relevant papers in past 60 days:
Year Citation  Score
2021 Khan SN, Shaheen F, Aleem U, Sheikh SF, Tamfu AN, Ashraf S, Ul-Haq Z, Ullah S, Wahab AT, Choudhary MI, Jahan H. Peptide Conjugates of 18β-Glycyrrhetinic Acid as Potent Inhibitors of α-Glucosidase and AGEs-Induced Oxidation. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. 106045. PMID 34666184 DOI: 10.1016/j.ejps.2021.106045   
2021 Mirgany TO, Abdalla AN, Arifuzzaman M, Motiur Rahman AFM, Al-Salem HS. Quinazolin-4(3)-one based potential multiple tyrosine kinase inhibitors with excellent cytotoxicity. Journal of Enzyme Inhibition and Medicinal Chemistry. 36: 2055-2067. PMID 34551654 DOI: 10.1080/14756366.2021.1972992   
2021 Legru A, Verdirosa F, Hernandez JF, Tassone G, Sannio F, Benvenuti M, Conde PA, Bossis G, Thomas CA, Crowder MW, Dillenberger M, Becker K, Pozzi C, Mangani S, Docquier JD, et al. 1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity. European Journal of Medicinal Chemistry. 226: 113873. PMID 34626878 DOI: 10.1016/j.ejmech.2021.113873   
2021 Zhang JH, Xie HX, Li Y, Wang KM, Song Z, Zhu KK, Fang L, Zhang J, Jiang CS. Design, synthesis and biological evaluation of novel (E)-2-benzylidene-N-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)hydrazine-1-carboxamide derivatives as α-glucosidase inhibitors. Bioorganic & Medicinal Chemistry Letters. 128413. PMID 34634473 DOI: 10.1016/j.bmcl.2021.128413   
2021 Quratulain -, Abbas Khan M, Ahmad I, Hamad A, Ashraf M, Hussain S. Synthesis, characterization, SAR, antioxidant, anti-acetylcholinesterase and anti-butyrylcholinesterase activities of cephradine Schiff bases. Pakistan Journal of Pharmaceutical Sciences. 34: 1989-1994. PMID 34836871   
2021 Zhang L, Feng XZ, Xiao ZQ, Fan GR, Chen SX, Liao SL, Luo H, Wang ZD. Design, Synthesis, Antibacterial, Antifungal and Anticancer Evaluations of Novel -Pinene Quaternary Ammonium Salts. International Journal of Molecular Sciences. 22. PMID 34681957 DOI: 10.3390/ijms222011299   
2021 Kshirsagar RR, Gadekar PK, Khedkar VM, Vijayakumar V. Design, Synthesis, and the Effects of ()-9-Oxooctadec-10-en-12-ynoic Acid Analogues to Promote Glucose Uptake. Acs Omega. 6: 24118-24127. PMID 34568690 DOI: 10.1021/acsomega.1c03600   
2021 Zhang TJ, Tu S, Zhang X, Wang QY, Hu SS, Zhang Y, Zhang ZH, Wang ZR, Meng FH. Amide-based xanthine oxidase inhibitors bearing an N-(1-alkyl-3-cyano-1H-indol-5-yl) moiety: Design, synthesis and structure-activity relationship investigation. Bioorganic Chemistry. 117: 105417. PMID 34673452 DOI: 10.1016/j.bioorg.2021.105417   
2021 Dobie C, Montgomery AP, Szabo R, Yu H, Skropeta D. Synthesis and biological evaluation of selective phosphonate-bearing 1,2,3-triazole-linked sialyltransferase inhibitors. Rsc Medicinal Chemistry. 12: 1680-1689. PMID 34778769 DOI: 10.1039/d1md00079a   
2021 Toplak A, Teixeira de Oliveira EF, Schmidt M, Rozeboom HJ, Wijma HJ, Meekels LKM, de Visser R, Janssen DB, Nuijens T. From thiol-subtilisin to omniligase: Design and structure of a broadly applicable peptide ligase. Computational and Structural Biotechnology Journal. 19: 1277-1287. PMID 33717424 DOI: 10.1016/j.csbj.2021.02.002   
2021 Afzal O, Altamimi ASA, Shahroz MM, Sharma HK, Riadi Y, Hassan MQ. Analgesic and Anticancer Activity of Benzoxazole Clubbed 2-Pyrrolidinones as Novel Inhibitors of Monoacylglycerol Lipase. Molecules (Basel, Switzerland). 26. PMID 33924091 DOI: 10.3390/molecules26082389   
2021 Mancuso F, De Luca L, Bucolo F, Vrabel M, Angeli A, Capasso C, Supuran CT, Gitto R. 4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae. Chemmedchem. PMID 34592052 DOI: 10.1002/cmdc.202100510   
2021 Ghosh AK, Shahabi D, Yadav M, Kovela S, Anson BJ, Lendy EK, Bonham C, Sirohi D, Brito-Sierra CA, Hattori SI, Kuhn R, Mitsuya H, Mesecar AD. Chloropyridinyl Esters of Nonsteroidal Anti-Inflammatory Agents and Related Derivatives as Potent SARS-CoV-2 3CL Protease Inhibitors. Molecules (Basel, Switzerland). 26. PMID 34641337 DOI: 10.3390/molecules26195782   
2021 Wang Y, Zhai J, Yang D, Han N, Liu Z, Liu Z, Li S, Yin J. Antioxidant, Anti-Inflammatory, and Antidiabetic Activities of Bioactive Compounds from the Fruits of Based on Network Pharmacology Prediction. Oxidative Medicine and Cellular Longevity. 2021: 7807046. PMID 34707780 DOI: 10.1155/2021/7807046   
2021 Gao Z, Huang XY, Geng CA, Li TZ, Chen JJ. Artemicapillasins A-N, cytotoxic coumaric acid analogues against hepatic stellate cell LX2 from Artemisia capillaris (Yin-Chen). Bioorganic Chemistry. 117: 105441. PMID 34695731 DOI: 10.1016/j.bioorg.2021.105441   
2021 Sim J, Lanka S, Jo JW, Chaudhary CL, Vishwanath M, Jung CH, Lee YH, Kim EY, Kim YS, Hyun SS, Lee HS, Lee K, Seo SY, Viji M, Jung JK. Inhibitory Effect of Chlorogenic Acid Analogues Comprising Pyridine and Pyrimidine on α-MSH-Stimulated Melanogenesis and Stability of Acyl Analogues in Methanol. Pharmaceuticals (Basel, Switzerland). 14. PMID 34832958 DOI: 10.3390/ph14111176   
2021 Campos-Almazán MI, Flores-Ramos M, Hernández-Campos A, Castillo R, Sierra-Campos E, Torgeson K, Peti W, Valdez-Solana M, Oria-Hernández J, Méndez ST, Castillo-Villanueva A, Jiménez-de Jesús H, Avitia-Domínguez C, Téllez-Valencia A. Design, synthesis, kinetic, molecular dynamics, and hypoglycemic effect characterization of new and potential selective benzimidazole derivatives as Protein Tyrosine Phosphatase 1B inhibitors. Bioorganic & Medicinal Chemistry. 48: 116418. PMID 34563877 DOI: 10.1016/j.bmc.2021.116418   
2021 Thissera B, Sayed AM, Hassan MHA, Abdelwahab SF, Amaeze N, Semler VT, Alenezi FN, Yaseen M, Alhadrami HA, Belbahri L, Rateb ME. Bioguided Isolation of Cyclopenin Analogues as Potential SARS-CoV-2 M Inhibitors from TDPEF34. Biomolecules. 11. PMID 34572579 DOI: 10.3390/biom11091366   
2021 Pokhrel S, Bouback TA, Samad A, Nur SM, Alam R, Abdullah-Al-Mamun M, Nain Z, Imon RR, Talukder MEK, Tareq MMI, Hossen MS, Karpiński TM, Ahammad F, Qadri I, Rahman MS. Spike protein recognizer receptor ACE2 targeted identification of potential natural antiviral drug candidates against SARS-CoV-2. International Journal of Biological Macromolecules. PMID 34592225 DOI: 10.1016/j.ijbiomac.2021.09.146   
2021 Mishra A, Khan WH, Rathore AS. Synergistic Effects of Natural Compounds Toward Inhibition of SARS-CoV-2 3CL Protease. Journal of Chemical Information and Modeling. PMID 34694807 DOI: 10.1021/acs.jcim.1c00994   
2021 Wang X, Duan W, Lin G, Li B, Chen M, Lei F. Synthesis, 3D-QSAR and Molecular Docking Study of Nopol-Based 1,2,4-Triazole-Thioether Compounds as Potential Antifungal Agents. Frontiers in Chemistry. 9: 757584. PMID 34765587 DOI: 10.3389/fchem.2021.757584   
2021 Duong TH, Nguyen HT, Nguyen CH, Tran NM, Danova A, Tran TM, Vu-Huynh KL, Musa V, Jutakanoke R, Nguyen NH, Sichaem J. Identification of Highly Potent α-Glucosidase Inhibitors from Artocarpus integer and Molecular Docking Studies. Chemistry & Biodiversity. e2100499. PMID 34761862 DOI: 10.1002/cbdv.202100499   
2021 Wang Y, Wang J, Wang S, Cao Z, Gu D, Wang Y, Tian J, Yang Y. An efficient method based on an inhibitor-enzyme complex to screen an active compound against lipase from . Food & Function. PMID 34617090 DOI: 10.1039/d1fo01542g   
2021 Rocha K, Magallon J, Reeves C, Phan K, Vu P, Oakley-Havens CL, Kwan S, Ramirez MS, LaVoi T, Donow H, Chapagain P, Santos R, Pinilla C, Giulianotti MA, Tolmasky ME. Inhibition of Aminoglycoside 6'--acetyltransferase Type Ib (AAC(6')-Ib): Structure-Activity Relationship of Substituted Pyrrolidine Pentamine Derivatives as Inhibitors. Biomedicines. 9. PMID 34572404 DOI: 10.3390/biomedicines9091218   
2021 Yu Q, Xie L, Li Y, Bai L, Zhao YL, Wei D, Shi T. Exploring the Molecular Basis of Substrate and Product Selectivities of Nocardicin Bifunctional Thioesterase. Interdisciplinary Sciences, Computational Life Sciences. PMID 34699036 DOI: 10.1007/s12539-021-00482-z   
2021 Azimi F, Azizian H, Najafi M, Khodarahmi G, Saghaei L, Hassanzadeh M, Ghasemi JB, Faramarzi MA, Larijani B, Hassanzadeh F, Mahdavi M. Design, synthesis, biological evaluation, and molecular modeling studies of pyrazole-benzofuran hybrids as new α-glucosidase inhibitor. Scientific Reports. 11: 20776. PMID 34675367 DOI: 10.1038/s41598-021-99899-1   
2021 van Haren MJ, Gao Y, Buijs N, Campagna R, Sartini D, Emanuelli M, Mateuszuk L, Kij A, Chlopicki S, Escudé Martinez de Castilla P, Schiffelers R, Martin NI. Esterase-Sensitive Prodrugs of a Potent Bisubstrate Inhibitor of Nicotinamide -Methyltransferase (NNMT) Display Cellular Activity. Biomolecules. 11. PMID 34572571 DOI: 10.3390/biom11091357   
2021 Weiss M, Loi EM, Sterle M, Balsollier C, Tomašič T, Pieters RJ, Gobec M, Anderluh M. New Quinolinone O-GlcNAc Transferase Inhibitors Based on Fragment Growth. Frontiers in Chemistry. 9: 666122. PMID 33937202 DOI: 10.3389/fchem.2021.666122   
2021 Chen Y, Zhang D, Zhang X, Wang Z, Liu CF, Tam JP. Site-Specific Protein Modifications by an Engineered Asparaginyl Endopeptidase from . Frontiers in Chemistry. 9: 768854. PMID 34746098 DOI: 10.3389/fchem.2021.768854   
2021 Yin JY, Han YN, Liu MQ, Piao ZH, Zhang X, Xue YT, Zhang YH. Structure-guided discovery of antioxidant peptides bounded to the Keap1 receptor as hunter for potential dietary antioxidants. Food Chemistry. 373: 130999. PMID 34710694 DOI: 10.1016/j.foodchem.2021.130999   
2021 Chen YJ, Ma KY, Du SS, Zhang ZJ, Wu TL, Sun Y, Liu YQ, Yin XD, Zhou R, Yan YF, Wang RX, He YH, Chu QR, Tang C. Antifungal Exploration of Quinoline Derivatives against Phytopathogenic Fungi Inspired by Quinine Alkaloids. Journal of Agricultural and Food Chemistry. PMID 34623798 DOI: 10.1021/acs.jafc.1c05677   
2021 Pei X, Wang J, Zheng H, Xiao Q, Wang A, Su W. Catalytically active inclusion bodies (CatIBs) induced by terminally attached self-assembling coiled-coil domains: To enhance the stability of (R)-hydroxynitrile lyase. Enzyme and Microbial Technology. 153: 109915. PMID 34670185 DOI: 10.1016/j.enzmictec.2021.109915   
2021 Li Y, Zhang JH, Xie HX, Ge YX, Wang KM, Song ZL, Zhu KK, Zhang J, Jiang CS. Discovery of new 2-phenyl-1H-benzo[d]imidazole core-based potent α-glucosidase inhibitors: Synthesis, kinetic study, molecular docking, and in vivo anti-hyperglycemic evaluation. Bioorganic Chemistry. 117: 105423. PMID 34717239 DOI: 10.1016/j.bioorg.2021.105423   
2021 Wang S, Chen J, Shi J, Wang Z, Hu D, Song B. Novel Cinnamic Acid Derivatives Containing the 1,3,4-Oxadiazole Moiety: Design, Synthesis, Antibacterial Activities, and Mechanisms. Journal of Agricultural and Food Chemistry. PMID 34597041 DOI: 10.1021/acs.jafc.1c03087   
2021 Česnek M, Šafránek M, Dračínský M, Tloušťová E, Mertlíková-Kaiserová H, Hayes MP, Watts VJ, Janeba Z. Halogen Dance-Based Synthesis of Phosphonomethoxyethyl (PME) Substituted 2-Aminothiazoles as Potent Inhibitors of Bacterial Adenylate Cyclases. Chemmedchem. PMID 34636150 DOI: 10.1002/cmdc.202100568   
2021 Ma QG, Tang Y, Sang ZP, Dong JH, Wei RR. Structurally diverse biflavonoids from the fruits of Citrus medica L. var. sarcodactylis Swingle and their hypolipidemic and immunosuppressive activities. Bioorganic Chemistry. 117: 105450. PMID 34710667 DOI: 10.1016/j.bioorg.2021.105450   
2021 Pogorevc D, Müller R. Biotechnological production optimization of argyrins - a potent immunomodulatory natural product class. Microbial Biotechnology. PMID 34724343 DOI: 10.1111/1751-7915.13959   
2021 Low YS, Garcia MD, Lonhienne T, Fraser JA, Schenk G, Guddat LW. Triazolopyrimidine herbicides are potent inhibitors of Aspergillus fumigatus acetohydroxyacid synthase and potential antifungal drug leads. Scientific Reports. 11: 21055. PMID 34702838 DOI: 10.1038/s41598-021-00349-9   
2021 Dar'in D, Kantin G, Chupakhin E, Sharoyko V, Krasavin M. Natural-Like Spirocyclic Δ -Butenolides Obtained from Diazo Homophthalimides. Chemistry (Weinheim An Der Bergstrasse, Germany). 27: 8221-8227. PMID 33848018 DOI: 10.1002/chem.202100880   
2021 Zhang B, Duan Y, Yang Y, Mao Q, Lin F, Gao J, Dai X, Zhang P, Li Q, Li J, Dai R, Wang S. Design, synthesis, and biological evaluation of N-(3-cyano-1H-indol-5/6-yl)-6-oxo-1,6-dihydropyrimidine-4-carboxamides and 5-(6-oxo-1,6-dihydropyrimidin-2-yl)-1H-indole-3-carbonitriles as novel xanthine oxidase inhibitors. European Journal of Medicinal Chemistry. 227: 113928. PMID 34688012 DOI: 10.1016/j.ejmech.2021.113928   
2021 An X, Yu L, Wang S, Ao Y, Zhan X, Liu Q, Zhao Y, Li M, Shu X, Li F, He L, Zhao J. Kinetic Characterization and Inhibitor Screening of Pyruvate Kinase I From . Frontiers in Microbiology. 12: 710678. PMID 34603237 DOI: 10.3389/fmicb.2021.710678   
2021 Khobragade TP, Sarak S, Pagar AD, Jeon H, Giri P, Yun H. Synthesis of Sitagliptin Intermediate by a Multi-Enzymatic Cascade System Using Lipase and Transaminase With Benzylamine as an Amino Donor. Frontiers in Bioengineering and Biotechnology. 9: 757062. PMID 34692666 DOI: 10.3389/fbioe.2021.757062   
2021 An Y, Liu W, Xie H, Fan H, Han J, Sun B. Construction and activity evaluation of novel benzodioxane derivatives as dual-target antifungal inhibitors. European Journal of Medicinal Chemistry. 227: 113950. PMID 34731761 DOI: 10.1016/j.ejmech.2021.113950   
2021 Sharma V, Pugazhenthi G, Vasanth D. Production and characterization of a novel thermostable laccase from Bacillus licheniformis VNQ and its application in synthesis of bioactive 1,4-naphthoquinones. Journal of Bioscience and Bioengineering. PMID 34629297 DOI: 10.1016/j.jbiosc.2021.09.008   
2021 Wang Z, Zang R, Niu Z, Wang W, Wang X, Tang Y. Synthesis and antiviral effect of phosphamide modified vidarabine for treating HSV 1 infections. Bioorganic & Medicinal Chemistry Letters. 128405. PMID 34624489 DOI: 10.1016/j.bmcl.2021.128405   
2021 Guinan M, Huang N, Hawes CS, Lima MA, Smith M, Miller GJ. Chemical synthesis of 4'-thio and 4'-sulfinyl pyrimidine nucleoside analogues. Organic & Biomolecular Chemistry. PMID 34806745 DOI: 10.1039/d1ob02097h   
2021 Liew HT, To J, Zhang X, Hemu X, Chan NY, Serra A, Sze SK, Liu CF, Tam JP. The legumain McPAL1 from Momordica cochinchinensis is a highly stable Asx-specific splicing enzyme. The Journal of Biological Chemistry. 101325. PMID 34710371 DOI: 10.1016/j.jbc.2021.101325   
2021 N Vijayan A, Refaei MA, Silva RN, Tsang P, Zhang P. Detection of Sortase A and Identification of Its Inhibitors by Paramagnetic Nanoparticle-Assisted Nuclear Relaxation. Analytical Chemistry. PMID 34757710 DOI: 10.1021/acs.analchem.1c03271   
2021 Shanina E, Kuhaudomlarp S, Lal K, Seeberger PH, Imberty A, Rademacher C. Druggable allosteric sites in β-propeller lectins. Angewandte Chemie (International Ed. in English). PMID 34713573 DOI: 10.1002/anie.202109339   
2021 Dissanayake AA, Mills GL, Bonito G, Rennick B, Nair MG. Chemical Composition and Anti-Inflammatory and Antioxidant Activities of Extracts from Cultivated Morel Mushrooms, Species of Genus Morchella (Ascomycota). International Journal of Medicinal Mushrooms. 23: 73-83. PMID 34591400 DOI: 10.1615/IntJMedMushrooms.2021039297