Kuo-Shyan Lin, Ph.D. - Publications

Affiliations: 
2001 Johns Hopkins University, Baltimore, MD 
Area:
Pharmaceutical Chemistry

89 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2024 Wang L, Kuo HT, Zhang Z, Zhang C, Chen CC, Chapple D, Wilson R, Colpo N, Lin KS. Unnatural amino acid substitutions to improve in vivo stability and tumor uptake of Ga-labeled GRPR-targeted TacBOMB2 derivatives for cancer imaging with positron emission tomography. Ejnmmi Radiopharmacy and Chemistry. 9: 8. PMID 38305955 DOI: 10.1186/s41181-024-00241-7  0.304
2023 Lu K, Zhang C, Zhang Z, Kuo HT, Colpo N, Bénard F, Lin KS. Synthesis and Evaluation of Tc-Labeled PSMA-Targeted Tracers Based on the Lys-Urea-Aad Pharmacophore for Detecting Prostate Cancer with Single Photon Emission Computed Tomography. Molecules (Basel, Switzerland). 28. PMID 37446782 DOI: 10.3390/molecules28135120  0.316
2022 Kwon D, Zhang Z, Zeisler J, Kuo HT, Lin KS, Benard F. Reducing the Kidney Uptake of High Contrast CXCR4 PET Imaging Agents via Linker Modifications. Pharmaceutics. 14. PMID 35890397 DOI: 10.3390/pharmaceutics14071502  0.312
2021 Bratanovic IJ, Zhang C, Zhang Z, Kuo HT, Colpo N, Zeisler J, Merkens H, Uribe C, Lin KS, Bénard F. A Novel Radiotracer for Molecular Imaging and Therapy of Gastrin-Releasing Peptide Receptor Positive Prostate Cancer. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 34301778 DOI: 10.2967/jnumed.120.257758  0.322
2020 Wong AAWL, Lozada J, Lepage ML, Zhang C, Merkens H, Zeisler J, Lin KS, Bénard F, Perrin DM. Synthesis and F-radiolabeling of thymidine AMBF conjugates. Rsc Medicinal Chemistry. 11: 569-576. PMID 33479658 DOI: 10.1039/d0md00054j  0.34
2020 Kwon D, Lozada J, Zhang Z, Zeisler J, Poon R, Zhang C, Roxin Á, Lin KS, Perrin D, Benard F. High-Contrast CXCR4-Targeted F-PET Imaging Using a Potent and Selective Antagonist. Molecular Pharmaceutics. PMID 33253591 DOI: 10.1021/acs.molpharmaceut.0c00785  0.348
2020 Kuo HT, Lin KS, Zhang Z, Uribe CF, Merkens H, Zhang C, Benard F. Novel Lu-labeled Albumin-binder-conjugated PSMA-targeting Agents with Extremely High Tumor Uptake and Enhanced Tumor-to-kidney Absorbed Dose Ratio. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 32859704 DOI: 10.2967/Jnumed.120.250738  0.401
2020 Bendre S, Zhang Z, Kuo HT, Rousseau J, Zhang C, Merkens H, Roxin Á, Bénard F, Lin KS. Evaluation of Met-Val-Lys as a Renal Brush Border Enzyme-Cleavable Linker to Reduce Kidney Uptake of Ga-Labeled DOTA-Conjugated Peptides and Peptidomimetics. Molecules (Basel, Switzerland). 25. PMID 32854201 DOI: 10.3390/Molecules25173854  0.308
2020 Lau J, Rousseau J, Kwon D, Bénard F, Lin KS. A Systematic Review of Molecular Imaging Agents Targeting Bradykinin B1 and B2 Receptors. Pharmaceuticals (Basel, Switzerland). 13. PMID 32824565 DOI: 10.3390/Ph13080199  0.322
2020 Li L, Kuo HT, Wang X, Merkens H, Colpo N, Radchenko V, Schaffer P, Lin KS, Bénard F, Orvig C. Buoctapa-alkyl-NHS for metalloradiopeptide preparation. Dalton Transactions (Cambridge, England : 2003). PMID 32459231 DOI: 10.1039/D0Dt00845A  0.321
2020 Lau J, Rousseau E, Kwon D, Lin KS, Bénard F, Chen X. Insight into the Development of PET Radiopharmaceuticals for Oncology. Cancers. 12. PMID 32455729 DOI: 10.3390/Cancers12051312  0.35
2020 Zhang C, Zhang Z, Zeisler J, Colpo N, Lin KS, Bénard F. Selective Cyclized α-Melanocyte-Stimulating Hormone Derivative with Multiple -Methylations for Melanoma Imaging with Positron Emission Tomography. Acs Omega. 5: 10767-10773. PMID 32455196 DOI: 10.1021/acsomega.0c00310  0.319
2020 Sahylí Ortega Pijeira M, Sérgio Gonçalves Nunes P, Nascimento Dos Santos S, Zhang Z, Pérez Nario A, Araujo Perini E, Miguel Turato W, Rodríguez Riera Z, Chammas R, H Elsinga P, Lin KS, Carvalho I, Soares Bernardes E. Synthesis and Evaluation of [F]FEtLos and [F]AMBFLos as Novel F-Labelled Losartan Derivatives for Molecular Imaging of Angiotensin II Type 1 Receptors. Molecules (Basel, Switzerland). 25. PMID 32325695 DOI: 10.3390/Molecules25081872  0.404
2020 Li L, Rousseau J, Jaraquemada-Peláez MG, Wang X, Robertson A, Radchenko V, Schaffer P, Lin KS, Bénard F, Orvig C. 225Ac-H4py4pa for Targeted-Alpha-Therapy. Bioconjugate Chemistry. PMID 32216377 DOI: 10.1021/Acs.Bioconjchem.0C00171  0.308
2020 Lau J, Pan J, Rousseau E, Uribe CF, Seelam SR, Sutherland BW, Perrin DM, Lin KS, Bénard F. Pharmacokinetics, radiation dosimetry, acute toxicity and automated synthesis of [F]AmBF-TATE. Ejnmmi Research. 10: 25. PMID 32189151 DOI: 10.1186/S13550-020-0611-9  0.354
2020 Li L, Jaraquemada-Peláez MG, Aluicio-Sarduy E, Wang X, Jiang D, Sakheie M, Kuo HT, Barnhart TE, Cai W, Radchenko V, Schaffer P, Lin KS, Engle JW, Bénard F, Orvig C. [Sc(pypa)]: Thermodynamic Stability, Radiolabeling, and Biodistribution of a Prostate-Specific-Membrane-Antigen-Targeting Conjugate. Inorganic Chemistry. PMID 31976659 DOI: 10.1021/Acs.Inorgchem.9B03347  0.35
2019 Rousseau E, Lau J, Zhang Z, Zhang C, Kwon D, Uribe CF, Kuo HT, Zeisler J, Bratanovic I, Lin KS, Bénard F. Comparison of biological properties of [ Lu]Lu-ProBOMB1 and [ Lu]Lu-NeoBOMB1 for GRPR-targeting. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 31715025 DOI: 10.1002/Jlcr.3815  0.359
2019 Lepage ML, Kuo HT, Roxin A, Huh S, Zhang Z, Kandasamy RL, Merkens H, Kumlin J, Limoges A, Zeisler SK, Benard F, Lin KS, Perrin D. Toward 18F-Labeled Theranostics: A Single Agent that can be Labeled with 18F, 64Cu, or 177Lu. Chembiochem : a European Journal of Chemical Biology. PMID 31621172 DOI: 10.1002/Cbic.201900632  0.431
2019 Lau J, Kwon D, Rousseau E, Zhang Z, Zeisler J, Uribe CF, Kuo HT, Zhang C, Lin KS, Benard F. [68Ga]Ga/[177Lu]Lu-BL01, a Novel Theranostic Pair for Targeting C-X-C Chemokine Receptor 4. Molecular Pharmaceutics. PMID 31545614 DOI: 10.1021/Acs.Molpharmaceut.9B00808  0.316
2019 Zhang C, Zhang Z, Merkens H, Zeisler J, Colpo N, Hundal-Jabal N, Perrin DM, Lin KS, Bénard F. F-Labeled Cyclized α-Melanocyte-Stimulating Hormone Derivatives for Imaging Human Melanoma Xenograft with Positron Emission Tomography. Scientific Reports. 9: 13575. PMID 31537869 DOI: 10.1038/S41598-019-50014-5  0.466
2019 Li L, Jaraquemada-Peláez MG, Kuo HT, Merkens H, Choudhary N, Gitschalter K, Jermilova U, Colpo N, Uribe-Munoz C, Radchenko V, Schaffer P, Lin KS, Benard F, Orvig C. Functionally Versatile and Highly Stable Chelator for 111In and 177Lu: Proof-of-principle Prostate Specific Membrane Antigen Targeting. Bioconjugate Chemistry. PMID 31009566 DOI: 10.1021/Acs.Bioconjchem.9B00225  0.352
2019 Roxin A, Zhang C, Huh S, Lepage ML, Zhang Z, Lin KS, Bénard F, Perrin DM. A Metal-Free DOTA-Conjugated 18F-Labeled Radiotracer: [18F]DOTA-AMBF3-LLP2A for Imaging VLA-4 Over-Expression in Murine Melanoma with Improved Tumor Uptake and Greatly Enhanced Renal Clearance. Bioconjugate Chemistry. PMID 30896929 DOI: 10.1021/Acs.Bioconjchem.9B00146  0.469
2019 Kuo HT, Lepage M, Lin KS, Pan J, Zhang Z, Liu Z, Pryyma A, Zhang C, Merkens H, Roxin A, Perrin D, Benard F. One-step F-labeling and preclinical evaluation of prostate specific membrane antigen trifluoroborate probes for cancer imaging. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 30737299 DOI: 10.2967/Jnumed.118.216598  0.459
2019 Lau J, Jacobson O, Niu G, Lin KS, Bénard F, Chen X. Bench to Bedside: Albumin Binders for Improved Cancer Radioligand Therapies. Bioconjugate Chemistry. PMID 30616340 DOI: 10.1021/Acs.Bioconjchem.8B00919  0.34
2018 Čolović M, Rousseau E, Zhang Z, Lau J, Zhang C, Kuo HT, Yang H, Schaffer P, François Bénard, Lin KS. Synthesis and evaluation of an F-labeled boramino acid analog of aminosuberic acid for PET imaging of the antiporter system x. Bioorganic & Medicinal Chemistry Letters. PMID 30316632 DOI: 10.1016/J.Bmcl.2018.06.014  0.417
2018 Kuo HT, Merkens H, Zhang Z, Uribe CF, Lau J, Zhang C, Colpo N, Lin KS, Benard F. Enhancing treatment efficacy of 177Lu-PSMA-617 with the conjugation of an albumin-binding motif: preclinical dosimetry and endoradiotherapy studies. Molecular Pharmaceutics. PMID 30251544 DOI: 10.1021/Acs.Molpharmaceut.8B00720  0.396
2018 Rousseau E, Lau J, Kuo HT, Zhang Z, Merkens H, Hundal-Jabal N, Colpo N, Lin KS, Bénard F. Monosodium glutamate reduces Ga-PSMA-11 uptake in salivary glands and kidneys in preclinical prostate cancer model. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 30097503 DOI: 10.2967/Jnumed.118.215350  0.319
2018 Wang X, Jaraquemada-Peláez MG, Cao Y, Pan J, Lin KS, Patrick BO, Orvig C. Hhox: Dual-Channel Oxine-Derived Acyclic Chelating Ligand for Ga Radiopharmaceuticals. Inorganic Chemistry. PMID 29989801 DOI: 10.1021/Acs.Inorgchem.8B01208  0.319
2018 Kuo HT, Pan J, Zhang Z, Lau J, Merkens H, Zhang C, Colpo N, Lin KS, Benard F. Effects of linker modification on tumor-to-kidney contrast of 68Ga-labeled PSMA-targeted imaging probes. Molecular Pharmaceutics. PMID 29920108 DOI: 10.1021/Acs.Molpharmaceut.8B00499  0.354
2018 Nakai M, Pan J, Lin KS, Thompson JR, Nocentini A, Supuran CT, Nakabayashi Y, Storr T. Evaluation of Tc-sulfonamide and sulfocoumarin derivatives for imaging carbonic anhydrase IX expression. Journal of Inorganic Biochemistry. 185: 63-70. PMID 29778927 DOI: 10.1016/J.Jinorgbio.2018.04.009  0.34
2018 Zhang C, Zhang Z, Lin KS, Lau J, Zeisler J, Colpo N, Perrin DM, Benard F. Melanoma imaging using F-labeled α-melanocyte-stimulating hormone derivatives with positron emission tomography. Molecular Pharmaceutics. PMID 29714486 DOI: 10.1021/Acs.Molpharmaceut.7B01113  0.471
2018 Roxin Á, Zhang C, Huh S, Lepage ML, Zhang Z, Lin KS, Bénard F, Perrin DM. Preliminary evaluation ofF-labeled LLP2A-trifluoroborate conjugates as VLA-4 (αβintegrin) specific radiotracers for PET imaging of melanoma. Nuclear Medicine and Biology. 61: 11-20. PMID 29597141 DOI: 10.1016/J.Nucmedbio.2018.02.005  0.428
2018 Rousseau J, Zhang Z, Wang X, Zhang C, Lau J, Rousseau E, Čolović M, Hundal-Jabal N, Bénard F, Lin KS. Synthesis and evaluation of bifunctional tetrahydroxamate chelators for labeling antibodies with 89Zr for imaging with positron emission tomography. Bioorganic & Medicinal Chemistry Letters. PMID 29426769 DOI: 10.1016/J.Bmcl.2018.01.067  0.385
2017 Woods M, Leung L, Frantzen K, Garrick JG, Zhang Z, Zhang C, English W, Wilson D, Bénard F, Lin KS. Improving the stability ofC-labeled L-methionine with ascorbate. Ejnmmi Radiopharmacy and Chemistry. 2: 13. PMID 29503854 DOI: 10.1186/S41181-017-0032-X  0.337
2017 Dude I, Zhang Z, Rousseau J, Hundal-Jabal N, Colpo N, Merkens H, Lin KS, Bénard F. Evaluation of agonist and antagonist radioligands for somatostatin receptor imaging of breast cancer using positron emission tomography. Ejnmmi Radiopharmacy and Chemistry. 2: 4. PMID 29503845 DOI: 10.1186/S41181-017-0023-Y  0.373
2017 Dias GM, Ramogida CF, Rousseau J, Zacchia NA, Hoehr C, Schaffer P, Lin KS, Bénard F. 89Zr for antibody labeling and in vivo studies - A comparison between liquid and solid target production. Nuclear Medicine and Biology. 58: 1-7. PMID 29291493 DOI: 10.1016/J.Nucmedbio.2017.11.005  0.303
2017 Nunes PSG, Zhang Z, Kuo HT, Zhang C, Rousseau J, Rousseau E, Lau J, Kwon D, Carvalho I, Bénard F, Lin KS. Synthesis and evaluation of an 18 F-labeled trifluoroborate derivative of 2-nitroimidazole for imaging tumor hypoxia with positron emission tomography. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 29247455 DOI: 10.1002/Jlcr.3594  0.448
2017 Zhang C, Lin KS, Bénard F. Molecular Imaging and Radionuclide Therapy of Melanoma Targeting the Melanocortin 1 Receptor. Molecular Imaging. 16: 1536012117737919. PMID 29182034 DOI: 10.1177/1536012117737919  0.44
2017 Lau J, Lin KS, Bénard F. Past, Present, and Future: Development of Theranostic Agents Targeting Carbonic Anhydrase IX. Theranostics. 7: 4322-4339. PMID 29158829 DOI: 10.7150/Thno.21848  0.301
2017 Zhang Z, Lau J, Zhang C, Colpo N, Nocentini A, Supuran CT, Bénard F, Lin KS. Design, synthesis and evaluation of (18)F-labeled cationic carbonic anhydrase IX inhibitors for PET imaging. Journal of Enzyme Inhibition and Medicinal Chemistry. 32: 722-730. PMID 28385087 DOI: 10.1080/14756366.2017.1308928  0.437
2017 Zhang C, Zhang Z, Lin KS, Pan J, Dude I, Hundal-Jabal N, Colpo N, Bénard F. Preclinical Melanoma Imaging with (68)Ga-Labeled α-Melanocyte-Stimulating Hormone Derivatives Using PET. Theranostics. 7: 805-813. PMID 28382155 DOI: 10.7150/Thno.17117  0.427
2017 Zhang Z, Lau J, Kuo HT, Zhang C, Colpo N, Bénard F, Lin KS. Synthesis and evaluation of (18)F-labeled CJ-042794 for imaging prostanoid EP4 receptor expression in cancer with positron emission tomography. Bioorganic & Medicinal Chemistry Letters. PMID 28377057 DOI: 10.1016/J.Bmcl.2017.03.078  0.462
2017 Rousseau J, Zhang Z, Dias GM, Zhang C, Colpo N, Bénard F, Lin KS. Design, synthesis and evaluation of novel bifunctional tetrahydroxamate chelators for PET imaging of (89)Zr-labeled antibodies. Bioorganic & Medicinal Chemistry Letters. PMID 28131709 DOI: 10.1016/J.Bmcl.2017.01.052  0.366
2017 Kuo HT, Pan J, Lau J, Zhang C, Zeisler J, Colpo N, Benard F, Lin KS. Radiolabeled R954 derivatives for imaging bradykinin B1 receptor expression with positron emission tomography. Molecular Pharmaceutics. PMID 28094956 DOI: 10.1021/Acs.Molpharmaceut.6B01055  0.473
2016 Amouroux G, Zhang Z, Pan J, Jenni S, Zhang C, Hundal-Jabal N, Colpo N, Zeisler J, Lin KS, Bénard F. Synthesis and evaluation of a (68)Ga-labeled bradykinin B1 receptor agonist for imaging with positron emission tomography. Bioorganic & Medicinal Chemistry. PMID 27908753 DOI: 10.1016/J.Bmc.2016.11.038  0.423
2016 Zhang C, Pan J, Lin KS, Dude I, Lau J, Zeisler J, Merkens H, Jenni S, Guérin B, Benard F. Targeting the neuropeptide Y1 receptor for cancer imaging by positron emission tomography using novel truncated peptides. Molecular Pharmaceutics. PMID 27669056 DOI: 10.1021/Acs.Molpharmaceut.6B00464  0.469
2016 Zhang Z, Zhang C, Lau J, Colpo N, Bénard F, Lin KS. One-step synthesis of 4-[(18) F]fluorobenzyltriphenylphosphonium cation for imaging with positron emission tomography. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 27578168 DOI: 10.1002/Jlcr.3436  0.383
2016 Imamura Y, Tien AH, Pan J, Leung JK, Banuelos CA, Jian K, Wang J, Mawji NR, Fernandez JG, Lin KS, Andersen RJ, Sadar MD. An imaging agent to detect androgen receptor and its active splice variants in prostate cancer. Jci Insight. 1. PMID 27525313 DOI: 10.1172/Jci.Insight.87850  0.321
2016 Zhang Z, Kuo HT, Lau J, Jenni S, Zhang C, Zeisler J, Bénard F, Lin KS. Design, synthesis and evaluation of (18)F-labeled bradykinin B1 receptor-targeting small molecules for PET imaging. Bioorganic & Medicinal Chemistry Letters. PMID 27390067 DOI: 10.1016/J.Bmcl.2016.06.066  0.445
2016 Zhang Z, Amouroux G, Pan J, Jenni S, Zeisler J, Zhang C, Liu Z, Perrin DM, Benard F, Lin KS. Radiolabeled B9958 derivatives for imaging bradykinin B1 receptor expression with positron emission tomography: effect of the radiolabel-chelator complex on biodistribution and tumor uptake. Molecular Pharmaceutics. PMID 27348517 DOI: 10.1021/Acs.Molpharmaceut.6B00428  0.452
2016 Zhang Z, Jenni S, Zhang C, Merkens H, Lau J, Liu Z, Perrin DM, Bénard F, Lin KS. Synthesis and evaluation of (18)F-trifluoroborate derivatives of triphenylphosphonium for myocardial perfusion imaging. Bioorganic & Medicinal Chemistry Letters. PMID 26922139 DOI: 10.1016/J.Bmcl.2016.02.062  0.377
2015 Zhang Z, Lau J, Kuo HT, Zhang C, Hundal-Jabal N, Colpo N, Bénard F, Lin KS. Synthesis and evaluation of (18)F-labeled 4-nitrobenzyl derivatives for imaging tumor hypoxia with positron emission tomography: Comparison of 2-[(18)F]fluoroethyl carbonate and 2-[(18)F]fluoroethyl carbamate. Bioorganic & Medicinal Chemistry Letters. PMID 26646218 DOI: 10.1016/J.Bmcl.2015.11.066  0.418
2015 Liu Z, Lin KS, Bénard F, Pourghiasian M, Kiesewetter DO, Perrin DM, Chen X. One-step (18)F labeling of biomolecules using organotrifluoroborates. Nature Protocols. 10: 1423-32. PMID 26313478 DOI: 10.1038/Nprot.2015.090  0.399
2015 Amouroux G, Pan J, Jenni S, Zhang C, Zhang Z, Hundal-Jabal N, Colpo N, Liu Z, Bénard F, Lin KS. Imaging Bradykinin B1 Receptor with (68)Ga-Labeled [des-Arg(10)]Kallidin Derivatives: Effect of the Linker on Biodistribution and Tumor Uptake. Molecular Pharmaceutics. PMID 26101793 DOI: 10.1021/Acs.Molpharmaceut.5B00070  0.411
2015 Ramogida CF, Pan J, Ferreira CL, Patrick BO, Rebullar K, Yapp DT, Lin KS, Adam MJ, Orvig C. Nitroimidazole-Containing H2dedpa and H2CHXdedpa Derivatives as Potential PET Imaging Agents of Hypoxia with (68)Ga. Inorganic Chemistry. 54: 4953-65. PMID 25928800 DOI: 10.1021/Acs.Inorgchem.5B00554  0.384
2015 Normandin MD, Zheng MQ, Lin KS, Mason NS, Lin SF, Ropchan J, Labaree D, Henry S, Williams WA, Carson RE, Neumeister A, Huang Y. Imaging the cannabinoid CB1 receptor in humans with [(11)C]OMAR: assessment of kinetic analysis methods, test-retest reproducibility, and gender differences. Journal of Cerebral Blood Flow and Metabolism : Official Journal of the International Society of Cerebral Blood Flow and Metabolism. PMID 25833345 DOI: 10.1038/Jcbfm.2015.46  0.355
2015 Pourghiasian M, Liu Z, Pan J, Zhang Z, Colpo N, Lin KS, Perrin DM, Bénard F. (18)F-AmBF3-MJ9: a novel radiofluorinated bombesin derivative for prostate cancer imaging. Bioorganic & Medicinal Chemistry. 23: 1500-6. PMID 25757604 DOI: 10.1016/J.Bmc.2015.02.009  0.467
2015 Lin KS, Amouroux G, Pan J, Zhang Z, Jenni S, Lau J, Liu Z, Hundal-Jabal N, Colpo N, Bénard F. Comparative studies of three 68Ga-labeled [Des-Arg10]kallidin derivatives for imaging bradykinin B1 receptor expression with PET. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 56: 622-7. PMID 25745086 DOI: 10.2967/Jnumed.114.152132  0.4
2015 Liu Z, Amouroux G, Zhang Z, Pan J, Hundal-Jabal N, Colpo N, Lau J, Perrin DM, Bénard F, Lin KS. (18)F-trifluoroborate derivatives of [des-arg(10)]kallidin for imaging bradykinin b1 receptor expression with positron emission tomography. Molecular Pharmaceutics. 12: 974-82. PMID 25629412 DOI: 10.1021/Acs.Molpharmaceut.5B00003  0.441
2015 Lin KS, Pan J, Amouroux G, Turashvili G, Mesak F, Hundal-Jabal N, Pourghiasian M, Lau J, Jenni S, Aparicio S, Bénard F. In vivo radioimaging of bradykinin receptor b1, a widely overexpressed molecule in human cancer. Cancer Research. 75: 387-93. PMID 25488751 DOI: 10.1158/0008-5472.Can-14-1603  0.398
2015 Imamura Y, Tien AH, Kunzhong J, Pan J, Lin K, Andersen RJ, Sadar M. Development of an imaging approach to detect splice variants of androgen receptor in prostate cancer. Journal of Clinical Oncology. 33: 5058-5058. DOI: 10.1200/Jco.2015.33.15_Suppl.5058  0.322
2014 Liu Z, Radtke MA, Wong MQ, Lin KS, Yapp DT, Perrin DM. Dual mode fluorescent (18)F-PET tracers: efficient modular synthesis of rhodamine-[cRGD]2-[(18)F]-organotrifluoroborate, rapid, and high yielding one-step (18)F-labeling at high specific activity, and correlated in vivo PET imaging and ex vivo fluorescence. Bioconjugate Chemistry. 25: 1951-62. PMID 25265337 DOI: 10.1021/Bc5003357  0.396
2014 Liu Z, Pourghiasian M, Radtke MA, Lau J, Pan J, Dias GM, Yapp D, Lin KS, Bénard F, Perrin DM. An organotrifluoroborate for broadly applicable one-step 18F-labeling. Angewandte Chemie (International Ed. in English). 53: 11876-80. PMID 25196467 DOI: 10.1002/Anie.201406258  0.429
2014 Liu Z, Pourghiasian M, Bénard F, Pan J, Lin KS, Perrin DM. Preclinical evaluation of a high-affinity 18F-trifluoroborate octreotate derivative for somatostatin receptor imaging. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 55: 1499-505. PMID 24970911 DOI: 10.2967/Jnumed.114.137836  0.471
2014 Lau J, Pan J, Zhang Z, Hundal-Jabal N, Liu Z, Bénard F, Lin KS. Synthesis and evaluation of (18)F-labeled tertiary benzenesulfonamides for imaging carbonic anhydrase IX expression in tumours with positron emission tomography. Bioorganic & Medicinal Chemistry Letters. 24: 3064-8. PMID 24878197 DOI: 10.1016/J.Bmcl.2014.05.021  0.379
2014 Pan J, Lau J, Mesak F, Hundal N, Pourghiasian M, Liu Z, Bénard F, Dedhar S, Supuran CT, Lin KS. Synthesis and evaluation of 18F-labeled carbonic anhydrase IX inhibitors for imaging with positron emission tomography. Journal of Enzyme Inhibition and Medicinal Chemistry. 29: 249-55. PMID 23463940 DOI: 10.3109/14756366.2013.773994  0.372
2014 Imamura Y, Tien A, Pan J, Kunzhong J, Lin K, Andersen R, Sadar M. MP24-02 DEVELOPMENT OF AN IMAGING APPROACH TO DETECT SPLICE VARIANTS OF ANDROGEN RECEPTOR IN PROSTATE CANCER Journal of Urology. 191. DOI: 10.1016/J.Juro.2014.02.283  0.409
2013 Li Y, Liu Z, Lozada J, Wong MQ, Lin KS, Yapp D, Perrin DM. Single step 18F-labeling of dimeric cycloRGD for functional PET imaging of tumors in mice. Nuclear Medicine and Biology. 40: 959-66. PMID 24090672 DOI: 10.1016/J.Nucmedbio.2013.08.001  0.454
2013 Liu Z, Li Y, Lozada J, Wong MQ, Greene J, Lin KS, Yapp D, Perrin DM. Kit-like 18F-labeling of RGD-19F-arytrifluroborate in high yield and at extraordinarily high specific activity with preliminary in vivo tumor imaging. Nuclear Medicine and Biology. 40: 841-9. PMID 23810487 DOI: 10.1016/J.Nucmedbio.2013.05.002  0.455
2013 Pan J, Pourghiasian M, Hundal N, Lau J, Bénard F, Dedhar S, Lin KS. f-[18F]fluoroethanol and 3-[18F]fluoropropanol: facile preparation, biodistribution in mice, and their application as nucleophiles in the synthesis of [18F]fluoroalkyl aryl ester and ether PET tracers. Nuclear Medicine and Biology. 40: 850-7. PMID 23774003 DOI: 10.1016/J.Nucmedbio.2013.04.009  0.346
2013 Inkster J, Lin KS, Ait-Mohand S, Gosselin S, Bénard F, Guérin B, Pourghiasian M, Ruth T, Schaffer P, Storr T. 2-Fluoropyridine prosthetic compounds for the 18F labeling of bombesin analogues. Bioorganic & Medicinal Chemistry Letters. 23: 3920-6. PMID 23683595 DOI: 10.1016/J.Bmcl.2013.04.060  0.405
2013 Li Y, Liu Z, Harwig CW, Pourghiasian M, Lau J, Lin KS, Schaffer P, Benard F, Perrin DM. (18)F-click labeling of a bombesin antagonist with an alkyne-(18)F-ArBF(3) (-): in vivo PET imaging of tumors expressing the GRP-receptor. American Journal of Nuclear Medicine and Molecular Imaging. 3: 57-70. PMID 23342301  0.354
2012 Liu Z, Li Y, Lozada J, Pan J, Lin KS, Schaffer P, Perrin DM. Rapid, one-step, high yielding 18F-labeling of an aryltrifluoroborate bioconjugate by isotope exchange at very high specific activity Journal of Labelled Compounds and Radiopharmaceuticals. 55: 491-496. DOI: 10.1002/Jlcr.2990  0.368
2010 Normandin MD, Weinzimmer DP, Ropchan J, Labaree D, Lin K, Mason NS, Carson RE, D'Souza DC, Neumeister A, Huang Y. Modeling analysis of the CB1 PET tracer [11C]OMAR in rhesus monkeys and humans Neuroimage. 52: S13. DOI: 10.1016/J.Neuroimage.2010.04.198  0.302
2007 Kim SW, Ding YS, Alexoff D, Patel V, Logan J, Lin KS, Shea C, Muench L, Xu Y, Carter P, King P, Constanzo JR, Ciaccio JA, Fowler JS. Synthesis and positron emission tomography studies of C-11-labeled isotopomers and metabolites of GTS-21, a partial alpha7 nicotinic cholinergic agonist drug. Nuclear Medicine and Biology. 34: 541-51. PMID 17591554 DOI: 10.1016/J.Nucmedbio.2007.04.005  0.322
2007 Kil KE, Ding YS, Lin KS, Alexoff D, Kim SW, Shea C, Xu Y, Muench L, Fowler JS. Synthesis and positron emission tomography studies of carbon-11-labeled imatinib (Gleevec). Nuclear Medicine and Biology. 34: 153-63. PMID 17307123 DOI: 10.1016/J.Nucmedbio.2006.11.004  0.358
2006 Ding YS, Lin KS, Logan J. PET imaging of norepinephrine transporters. Current Pharmaceutical Design. 12: 3831-45. PMID 17073682 DOI: 10.2174/138161206778559687  0.36
2006 Ding YS, Kil KE, Lin KS, Ma W, Yokota Y, Carroll IF. A novel nicotinic acetylcholine receptor antagonist radioligand for PET studies. Bioorganic & Medicinal Chemistry Letters. 16: 1049-53. PMID 16289815 DOI: 10.1016/J.Bmcl.2005.10.075  0.39
2005 Ding YS, Lin KS, Logan J, Benveniste H, Carter P. Comparative evaluation of positron emission tomography radiotracers for imaging the norepinephrine transporter: (S,S) and (R,R) enantiomers of reboxetine analogs ([11C]methylreboxetine, 3-Cl-[11C]methylreboxetine and [18F]fluororeboxetine), (R)-[11C]nisoxetine, [11C]oxaprotiline and [11C]lortalamine. Journal of Neurochemistry. 94: 337-51. PMID 15998285 DOI: 10.1111/J.1471-4159.2005.03202.X  0.362
2005 Logan J, Ding YS, Lin KS, Pareto D, Fowler J, Biegon A. Modeling and analysis of PET studies with norepinephrine transporter ligands: the search for a reference region. Nuclear Medicine and Biology. 32: 531-42. PMID 15982584 DOI: 10.1016/J.Nucmedbio.2005.04.005  0.329
2005 Lin KS, Ding YS. Synthesis and C-11 labeling of three potent norepinephrine transporter selective ligands ((R)-nisoxetine, lortalamine, and oxaprotiline) for comparative PET studies in baboons. Bioorganic & Medicinal Chemistry. 13: 4658-66. PMID 15914010 DOI: 10.1016/J.Bmc.2005.04.062  0.344
2005 Lin KS, Ding YS, Kim SW, Kil KE. Synthesis, enantiomeric resolution, F-18 labeling and biodistribution of reboxetine analogs: promising radioligands for imaging the norepinephrine transporter with positron emission tomography. Nuclear Medicine and Biology. 32: 415-22. PMID 15878511 DOI: 10.1016/J.Nucmedbio.2005.02.005  0.348
2005 Lin KS, Luu A, Baidoo KE, Hashemzadeh-Gargari H, Chen MK, Brenneman K, Pili R, Pomper M, Carducci MA, Wagner HN. A new high affinity technetium-99m-bombesin analogue with low abdominal accumulation. Bioconjugate Chemistry. 16: 43-50. PMID 15656574 DOI: 10.1021/Bc049820H  0.638
2004 Lin KS, Luu A, Baidoo KE, Hashemzadeh-Gargari H, Chen MK, Pili R, Pomper M, Carducci M, Wagner HN. A new high affinity technetium analogue of bombesin containing DTPA as a pharmacokinetic modifier. Bioconjugate Chemistry. 15: 1416-23. PMID 15546210 DOI: 10.1021/Bc0498267  0.624
2004 Baidoo KE, Knight LC, Lin KS, Gabriel JL, Romano JE. Design and synthesis of a short-chain bitistatin analogue for imaging thrombi and emboli. Bioconjugate Chemistry. 15: 1068-75. PMID 15366961 DOI: 10.1021/Bc049954V  0.599
2004 Lin KS, Ding YS. Synthesis, enantiomeric resolution, and selective C-11 methylation of a highly selective radioligand for imaging the norepinephrine transporter with positron emission tomography. Chirality. 16: 475-81. PMID 15236345 DOI: 10.1002/Chir.20055  0.312
2003 Bettegowda C, Dang LH, Abrams R, Huso DL, Dillehay L, Cheong I, Agrawal N, Borzillary S, McCaffery JM, Watson EL, Lin KS, Bunz F, Baidoo K, Pomper MG, Kinzler KW, et al. Overcoming the hypoxic barrier to radiation therapy with anaerobic bacteria. Proceedings of the National Academy of Sciences of the United States of America. 100: 15083-8. PMID 14657371 DOI: 10.1073/Pnas.2036598100  0.558
2003 Ding YS, Lin KS, Garza V, Carter P, Alexoff D, Logan J, Shea C, Xu Y, King P. Evaluation of a new norepinephrine transporter PET ligand in baboons, both in brain and peripheral organs. Synapse (New York, N.Y.). 50: 345-52. PMID 14556239 DOI: 10.1002/Syn.10281  0.304
1998 Baidoo KE, Lin KS, Zhan Y, Finley P, Scheffel U, Wagner HN. Design, synthesis, and initial evaluation of high-affinity technetium bombesin analogues. Bioconjugate Chemistry. 9: 218-25. PMID 9548537 DOI: 10.1021/Bc9701959  0.628
Show low-probability matches.