Gijsbert A. van der Marel - Publications

Affiliations: 
chemistry Leiden University, Leiden, Netherlands 
Area:
Synthetic organic chemistry
Website:
https://www.universiteitleiden.nl/en/staffmembers/gijs-van-der-marel#tab-1

336 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2019 Artola M, Wouters S, Schröder SP, de Boer C, Chen Y, Petracca R, van den Nieuwendijk AMCH, Aerts JMFG, van der Marel GA, Codée JDC, Overkleeft HS. Direct Stereoselective Aziridination of Cyclohexenols with 3-Amino-2-(trifluoromethyl)quinazolin-4(3)-one in the Synthesis of Cyclitol Aziridine Glycosidase Inhibitors. European Journal of Organic Chemistry. 2019: 1397-1404. PMID 31787842 DOI: 10.1002/ejoc.201801703  0.6
2019 van der Vorm S, Hansen T, van Hengst JMA, Overkleeft HS, van der Marel GA, Codée JDC. Acceptor reactivity in glycosylation reactions. Chemical Society Reviews. PMID 31287452 DOI: 10.1039/c8cs00369f  0.6
2019 Schröder SP, de Boer C, McGregor NGS, Rowland RJ, Moroz O, Blagova E, Reijngoud J, Arentshorst M, Osborn D, Morant MD, Abbate E, Stringer MA, Krogh KBRM, Raich L, Rovira C, ... ... van der Marel GA, et al. Dynamic and Functional Profiling of Xylan-Degrading Enzymes in Secretomes Using Activity-Based Probes. Acs Central Science. 5: 1067-1078. PMID 31263766 DOI: 10.1021/acscentsci.9b00221  0.6
2019 Hansen T, Lebedel L, Remmerswaal WA, van der Vorm S, Wander DPA, Somers M, Overkleeft HS, Filippov DV, Désiré J, Mingot A, Bleriot Y, van der Marel GA, Thibaudeau S, Codée JDC. Defining the S1 Side of Glycosylation Reactions: Stereoselectivity of Glycopyranosyl Cations. Acs Central Science. 5: 781-788. PMID 31139714 DOI: 10.1021/acscentsci.9b00042  0.6
2019 Liu Q, van der Marel GA, Filippov DV. Chemical ADP-ribosylation: mono-ADPr-peptides and oligo-ADP-ribose. Organic & Biomolecular Chemistry. PMID 31112180 DOI: 10.1039/c9ob00501c  0.32
2019 Wang L, Overkleeft HS, van der Marel GA, Codée JDC. Reagent Controlled Stereoselective Assembly of α-(1,3)-Glucans. European Journal of Organic Chemistry. 2019: 1994-2003. PMID 31007571 DOI: 10.1002/ejoc.201800894  0.6
2019 Gential GPP, Hogervorst TP, Tondini E, van de Graaff MJ, Overkleeft HS, Codée JDC, van der Marel GA, Ossendorp F, Filippov DV. Peptides conjugated to 2-alkoxy-8-oxo-adenine as potential synthetic vaccines triggering TLR7. Bioorganic & Medicinal Chemistry Letters. PMID 30952595 DOI: 10.1016/j.bmcl.2019.03.048  0.6
2019 van der Vorm S, Hansen T, van Rijssel ER, Dekkers R, Madern JM, Overkleeft HS, Filippov DV, van der Marel GA, Codée JDC. Furanosyl oxocarbenium ion Conformational Energy Landscape maps as a tool to study the glycosylation stereoselectivity of 2-azidofuranoses, 2-fluorofuranoses and methyl furanosyl uronates. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 30882938 DOI: 10.1002/chem.201900651  0.6
2019 Zom GG, Willems MMJHP, Meeuwenoord N, Reintjens NRM, Tondini E, Khan S, Overkleeft HS, van der Marel GA, Codée JDC, Ossendorp F, Filippov DV. Dual Synthetic Peptide Conjugate Vaccine Simultaneously Triggers TLR2 and NOD2 and Activates Human Dendritic Cells. Bioconjugate Chemistry. PMID 30865430 DOI: 10.1021/acs.bioconjchem.9b00087  0.6
2019 Artola M, Kuo CL, Lelieveld LT, Rowland RJ, van der Marel GA, Codée JDC, Boot RG, Davies GJ, Aerts JMFG, Overkleeft HS. Functionalized cyclophellitols are selective glucocerebrosidase inhibitors and induce a bona fide neuropathic Gaucher model in zebrafish. Journal of the American Chemical Society. PMID 30811188 DOI: 10.1021/jacs.9b00056  0.6
2019 Xin BT, Huber E, de Bruin G, Heinemeyer W, Maurits E, Espinal C, Du Y, Janssens M, Weyburne ES, Kisselev A, Florea BI, Driessen C, van der Marel GA, Groll M, Overkleeft HS. Structure-based design of inhibitors selective for human proteasome β2c or β2i subunits. Journal of Medicinal Chemistry. PMID 30657666 DOI: 10.1021/acs.jmedchem.8b01884  0.6
2019 Madern JM, Hansen T, van Rijssel ER, Kistemaker HAV, van der Vorm S, Overkleeft HS, van der Marel GA, Filippov DV, Codée JDC. Synthesis, reactivity and stereoselectivity of 4-thiofuranosides. The Journal of Organic Chemistry. PMID 30605336 DOI: 10.1021/acs.joc.8b02536  0.6
2018 Zom GG, Willems MMJHP, Khan S, van der Sluis TC, Kleinovink JW, Camps MGM, van der Marel GA, Filippov DV, Melief CJM, Ossendorp F. Novel TLR2-binding adjuvant induces enhanced T cell responses and tumor eradication. Journal For Immunotherapy of Cancer. 6: 146. PMID 30541631 DOI: 10.1186/s40425-018-0455-2  0.32
2018 Artola M, Kuo CL, McMahon SA, Oehler V, Hansen T, van der Lienden M, He X, van den Elst H, Florea BI, Kermode AR, Gloster TM, van der Marel GA, Codée JDC, Overkleeft HS, Aerts JMFG. New irreversible α-L-iduronidase inhibitors and activity-based probes. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 30307091 DOI: 10.1002/chem.201804662  0.8
2018 Voorneveld J, Rack JGM, Ahel I, Overkleeft HS, van der Marel GA, Filippov DV. Synthetic α- and β-Ser-ADP-ribosylated Peptides Reveal α-Ser-ADPr as the Native Epimer. Organic Letters. PMID 29947522 DOI: 10.1021/acs.orglett.8b01742  0.6
2018 Schröder SP, Kallemeijn WW, Debets MF, Sobala LF, Hakki Z, Williams SJ, Beenakker TJM, Aerts JMFG, van der Marel GA, Codée JDC, Davies GJ, Overkleeft HS. Spiro-epoxyglycosides as activity-based probes for glycoside hydrolase family 99 endomannosidase/endomannanase. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29797675 DOI: 10.1002/chem.201801902  0.6
2018 van der Vorm S, van Hengst JMA, Bakker M, Overkleeft HS, van der Marel GA, Codée J. Mapping Glycosyl Acceptor Reactivity - Glycosylation Stereoselectivity Relationships. Angewandte Chemie (International Ed. in English). PMID 29603532 DOI: 10.1002/anie.201802899  0.6
2018 Schröder SP, Wu L, Artola M, Hansen T, Offen WA, Ferraz MJ, Li KY, Aerts JMFG, van der Marel GA, Codée JDC, Davies GJ, Overkleeft HS. Gluco-1H-imidazole: a new class of azole-type β-glucosidase inhibitor. Journal of the American Chemical Society. PMID 29601200 DOI: 10.1021/jacs.8b02399  0.6
2018 Wang L, Overkleeft HS, van der Marel GA, Codée JDC. Reagent controlled stereoselective synthesis of α-glucans. Journal of the American Chemical Society. PMID 29553729 DOI: 10.1021/jacs.8b00669  0.6
2018 van der Es D, Berni F, Hogendorf WFJ, Meeuwenoord N, Laverde D, van Diepen A, Overkleeft HS, Filippov DV, Hokke CH, Huebner J, van der Marel GA, Codée J. Streamlined synthesis and evaluation of teichoic acid fragments. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29389054 DOI: 10.1002/chem.201800153  0.6
2017 Liu Q, Kistemaker HAV, Bhogaraju S, Dikic I, Overkleeft HS, van der Marel GA, Ovaa H, van der Heden van Noort G, Filippov DV. A General Approach Towards Triazole-linked Adenosine Diphosphate Ribosylated Peptides and Proteins. Angewandte Chemie (International Ed. in English). PMID 29215186 DOI: 10.1002/anie.201710527  0.6
2017 Geert Volbeda A, van Mechelen J, Meeuwenoord N, Overkleeft HS, van der Marel GA, Codée JDC. The Cyanopivaloyl Ester in the Automated Solid Phase Synthesis of Oligorhamnans. The Journal of Organic Chemistry. PMID 29148768 DOI: 10.1021/acs.joc.7b02511  0.6
2017 Schröder SP, van de Sande JW, Kallemeijn WW, Kuo CL, Artola M, van Rooden EJ, Jiang J, Beenakker TJM, Florea BI, Offen WA, Davies GJ, Minnaard AJ, Aerts JMFG, Codée JDC, van der Marel GA, et al. Towards broad spectrum activity-based glycosidase probes: synthesis and evaluation of deoxygenated cyclophellitol aziridines. Chemical Communications (Cambridge, England). PMID 29116266 DOI: 10.1039/c7cc07730k  0.6
2017 Lahav D, Liu B, van den Berg RJBHN, van den Nieuwendijk AMCH, Wennekes T, Ghisaidoobe AT, Breen I, Ferraz MJ, Kuo CL, Wu L, Geurink PP, Ovaa H, van der Marel GA, van der Stelt M, Boot RG, et al. A Fluorescence Polarization Activity-Based Protein Profiling Assay in the Discovery of Potent, Selective Inhibitors for Human Non-lysosomal Glucosylceramidase. Journal of the American Chemical Society. PMID 28937220 DOI: 10.1021/jacs.7b07352  0.6
2017 Zhang Q, Overkleeft HS, van der Marel GA, Codée JD. Synthetic zwitterionic polysaccharides. Current Opinion in Chemical Biology. 40: 95-101. PMID 28888143 DOI: 10.1016/j.cbpa.2017.07.010  0.6
2017 Liu Q, Kistemaker HAV, Overkleeft HS, van der Marel GA, Filippov DV. Synthesis of ribosyl-ribosyl-adenosine-5',5'',5'''(triphosphate)-the naturally occurring branched fragment of poly(ADP ribose). Chemical Communications (Cambridge, England). PMID 28868552 DOI: 10.1039/c7cc05755e  0.6
2017 Zhang Q, Howell PL, Overkleeft HS, Filippov DV, van der Marel GA, Codée JDC. Chemical synthesis of guanosine diphosphate mannuronic acid (GDP-ManA) and its C-4-O-methyl and C-4-deoxy congeners. Carbohydrate Research. 450: 12-18. PMID 28822279 DOI: 10.1016/j.carres.2017.08.005  0.6
2017 Artola M, Wu L, Ferraz MJ, Kuo CL, Raich L, Breen IZ, Offen WA, Codée JDC, van der Marel GA, Rovira C, Aerts JMFG, Davies GJ, Overkleeft HS. 1,6-Cyclophellitol Cyclosulfates: A New Class of Irreversible Glycosidase Inhibitor. Acs Central Science. 3: 784-793. PMID 28776021 DOI: 10.1021/acscentsci.7b00214  0.6
2017 Narhe BD, Breman AC, Padwal J, Vandenput DAL, Scheidt JM, Benningshof JCJ, van der Marel GA, Overkleeft HS, van der Stelt M, Filippov DV. Piperidine and octahydropyrano[3,4-c] pyridine scaffolds for drug-like molecular libraries of the European Lead Factory. Bioorganic & Medicinal Chemistry. PMID 28720326 DOI: 10.1016/j.bmc.2017.07.016  0.6
2017 Jiang J, Kuo CL, Wu L, Franke C, Kallemeijn WW, Florea BI, van Meel E, van der Marel GA, Codée JDC, Boot RG, Davies GJ, Overkleeft HS, Aerts JMFG. Correction to "Detection of Active Mammalian GH31 α-Glucosidases in Health and Disease Using In-Class, Broad-Spectrum Activity-Based Probes". Acs Central Science. 3: 673. PMID 28691081 DOI: 10.1021/acscentsci.7b00185  0.6
2017 Wu L, Jiang J, Jin Y, Kallemeijn WW, Kuo CL, Artola M, Dai W, van Elk C, van Eijk M, van der Marel GA, Codée JDC, Florea BI, Aerts JMFG, Overkleeft HS, Davies GJ. Activity-based probes for functional interrogation of retaining β-glucuronidases. Nature Chemical Biology. PMID 28581485 DOI: 10.1038/nchembio.2395  0.6
2017 van der Vorm S, Hansen T, Overkleeft HS, van der Marel GA, Codée JDC. The influence of acceptor nucleophilicity on the glycosylation reaction mechanism. Chemical Science. 8: 1867-1875. PMID 28553477 DOI: 10.1039/c6sc04638j  0.6
2017 Hagen B, van Dijk JHM, Zhang Q, Overkleeft HS, van der Marel GA, Codée JDC. Synthesis of the Staphylococcus aureus Strain M Capsular Polysaccharide Repeating Unit. Organic Letters. PMID 28485610 DOI: 10.1021/acs.orglett.7b00747  0.6
2017 Beenakker TJM, Wander D, Offen WA, Artola M, Raich L, Ferraz MJ, Li KY, Houben JHPM, van Rijssel ER, Hansen T, van der Marel GA, Codée JDC, Aerts JMFG, Rovira C, Davies GJ, et al. Carba-Cyclophellitols are Neutral Retaining Glucosidase Inhibitors. Journal of the American Chemical Society. PMID 28463498 DOI: 10.1021/jacs.7b01773  0.6
2017 van der Vorm S, Overkleeft HS, van der Marel GA, Codée JD. Stereoselectivity of conformationally restricted glucosazide donors. The Journal of Organic Chemistry. PMID 28401764 DOI: 10.1021/acs.joc.7b00470  0.6
2017 van Rijssel E, Janssen A, Males A, Davies G, van der Marel G, Overkleeft HS, Codée J. Conformational behaviour of mannuronic acid based azasugars. Chembiochem : a European Journal of Chemical Biology. PMID 28256791 DOI: 10.1002/cbic.201700080  0.6
2017 Engelsma SB, Meeuwenoord NJ, Overkleeft HS, van der Marel GA, Filippov DV. Combined Phosphoramidite-Phosphodiester Reagents for the Synthesis of Methylene Bisphosphonates. Angewandte Chemie (International Ed. in English). PMID 28170152 DOI: 10.1002/anie.201611878  0.64
2017 Hagen B, Ali S, Overkleeft HS, van der Marel GA, Codée JD. Mapping the reactivity and selectivity of 2-azidofucosyl donors for the assembly of N-acetyl fucosamine containing bacterial oligosaccharides. The Journal of Organic Chemistry. PMID 28051314 DOI: 10.1021/acs.joc.6b02593  0.6
2016 Kistemaker HAV, Meeuwenoord NJ, Overkleeft HS, van der Marel GA, Filippov DV. Solid-Phase Synthesis of Oligo-ADP-Ribose. Current Protocols in Nucleic Acid Chemistry. 64: 4.68.1-4.68.27. PMID 31820580 DOI: 10.1002/0471142700.nc0468s64  0.64
2016 van der Es D, Hogendorf WF, Overkleeft HS, van der Marel GA, Codée JD. Teichoic acids: synthesis and applications. Chemical Society Reviews. PMID 27990523 DOI: 10.1039/c6cs00270f  0.6
2016 Zom GG, Welters MJ, Loof NM, Goedemans R, Lougheed S, Valentijn RR, Zandvliet ML, Meeuwenoord NJ, Melief CJ, de Gruijl TD, Van der Marel GA, Filippov DV, Ossendorp F, Van der Burg SH. TLR2 ligand-synthetic long peptide conjugates effectively stimulate tumor-draining lymph node T cells of cervical cancer patients. Oncotarget. PMID 27564262 DOI: 10.18632/oncotarget.11512  0.64
2016 Kistemaker HA, Nardozza AP, Overkleeft HS, van der Marel GA, Ladurner AG, Filippov DV. Synthesis and Macrodomain Binding of Mono-ADP-Ribosylated Peptides. Angewandte Chemie (International Ed. in English). 55: 10634-8. PMID 27464500 DOI: 10.1002/anie.201604058  0.6
2016 Xin BT, de Bruin G, Huber EM, Besse A, Florea BI, Filippov DV, van der Marel GA, Kisselev AF, van der Stelt M, Driessen C, Groll M, Overkleeft HS. Structure-Based Design of β5c Selective Inhibitors of Human Constitutive Proteasomes. Journal of Medicinal Chemistry. PMID 27438186 DOI: 10.1021/acs.jmedchem.6b00705  1
2016 Gential GP, Ho NI, Chiodo F, Meeuwenoord N, Ossendorp F, Overkleeft HS, van der Marel GA, Filippov DV. Synthesis and evaluation of fluorescent Pam3Cys peptide conjugates. Bioorganic & Medicinal Chemistry Letters. PMID 27289322 DOI: 10.1016/j.bmcl.2016.05.094  0.6
2016 Jiang J, Kuo CL, Wu L, Franke C, Kallemeijn WW, Florea BI, van Meel E, van der Marel GA, Codée JD, Boot RG, Davies GJ, Overkleeft HS, Aerts JM. Detection of Active Mammalian GH31 α-Glucosidases in Health and Disease Using In-Class, Broad-Spectrum Activity-Based Probes. Acs Central Science. 2: 351-8. PMID 27280170 DOI: 10.1021/acscentsci.6b00057  0.6
2016 Mirzaian M, Wisse P, Ferraz MJ, Marques AR, Gabriel TL, van Roomen CP, Ottenhoff R, van Eijk M, Codée JD, van der Marel GA, Overkleeft HS, Aerts JM. Accurate quantification of sphingosine-1-phosphate in normal and Fabry disease plasma, cells and tissues by LC-MS/MS with (13)C-encoded natural S1P as internal standard. Clinica Chimica Acta; International Journal of Clinical Chemistry. 459: 36-44. PMID 27221202 DOI: 10.1016/j.cca.2016.05.017  0.6
2016 Stolze SC, Liu N, Wijdeven RH, Tuin AW, van den Nieuwendijk AM, Florea BI, van der Stelt M, van der Marel GA, Neefjes JJ, Overkleeft HS. Photo-crosslinking of clinically relevant kinases using H89-derived photo-affinity probes. Molecular Biosystems. PMID 27138522 DOI: 10.1039/c6mb00257a  0.6
2016 Xin BT, Schimmack G, Du Y, Florea BI, van der Marel GA, Driessen C, Krappmann D, Overkleeft HS. Development of new Malt1 inhibitors and probes. Bioorganic & Medicinal Chemistry. PMID 27085674 DOI: 10.1016/j.bmc.2016.03.035  1
2016 van der Es D, Groenia NA, Laverde D, Overkleeft HS, Huebner J, van der Marel GA, Codée JD. Synthesis of E. faecium wall teichoic acid fragments. Bioorganic & Medicinal Chemistry. PMID 26993744 DOI: 10.1016/j.bmc.2016.03.019  0.6
2016 de Bruin G, Mock ED, Hoogendoorn S, van den Nieuwendijk AM, Mazurek J, van der Marel GA, Florea BI, Overkleeft HS. Enantioselective synthesis of adamantylalanine and carboranylalanine and their incorporation into the proteasome inhibitor bortezomib. Chemical Communications (Cambridge, England). PMID 26894389 DOI: 10.1039/c6cc01156j  0.6
2016 Xin BT, de Bruin G, Plomp JW, Florea BI, van der Marel GA, Overkleeft HS. Incorporation of the Constrained Peptidomimetic, 5-Methylpyridin-2-one into Peptide Vinyl Sulfones and Peptide Epoxy Ketones is Detrimental for Proteasome Inhibition European Journal of Organic Chemistry. DOI: 10.1002/ejoc.201501401  1
2015 Jiang J, Kallemeijn WW, Wright DW, van den Nieuwendijk AMCH, Rohde VC, Folch EC, van den Elst H, Florea BI, Scheij S, Donker-Koopman WE, Verhoek M, Li N, Schürmann M, Mink D, Boot RG, ... ... van der Marel GA, et al. In vitro and in vivo comparative and competitive activity-based protein profiling of GH29 α-l-fucosidases. Chemical Science. 6: 2782-false. PMID 29142681 DOI: 10.1039/c4sc03739a  0.8
2015 de Bruin G, Xin BT, Kraus M, van der Stelt M, van der Marel GA, Kisselev AF, Driessen C, Florea BI, Overkleeft HS. A Set of Activity-Based Probes to Visualize Human (Immuno)proteasome Activities. Angewandte Chemie (International Ed. in English). PMID 26511210 DOI: 10.1002/anie.201509092  1
2015 van den Berg RJ, van Rijssel ER, Ferraz MJ, Houben J, Strijland A, Donker-Koopman WE, Wennekes T, Bonger KM, Ghisaidoobe AB, Hoogendoorn S, van der Marel GA, Codée JD, Overkleeft HS, Aerts JM. Synthesis and Evaluation of Hybrid Structures Composed of Two Glucosylceramide Synthase Inhibitors. Chemmedchem. PMID 26492941 DOI: 10.1002/cmdc.201500407  0.56
2015 Kistemaker HA, Overkleeft HS, van der Marel GA, Filippov DV. Branching of poly(ADP-ribose): Synthesis of the Core Motif. Organic Letters. 17: 4328-31. PMID 26307949 DOI: 10.1021/acs.orglett.5b02143  1
2015 Volbeda AG, Kistemaker HA, Overkleeft HS, van der Marel GA, Filippov DV, Codée JD. Chemoselective Cleavage of p-Methoxybenzyl and 2-Naphthylmethyl Ethers Using a Catalytic Amount of HCl in Hexafluoro-2-propanol. The Journal of Organic Chemistry. 80: 8796-806. PMID 26230920 DOI: 10.1021/acs.joc.5b01030  1
2015 Jiang J, Beenakker TJ, Kallemeijn WW, van der Marel GA, van den Elst H, Codée JD, Aerts JM, Overkleeft HS. Comparing Cyclophellitol N-Alkyl and N-Acyl Cyclophellitol Aziridines as Activity-Based Glycosidase Probes. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 10861-9. PMID 26073749 DOI: 10.1002/chem.201501313  1
2015 Wisse P, de Geus MA, Cross G, van den Nieuwendijk AM, van Rooden EJ, van den Berg RJ, Aerts JM, van der Marel GA, Codée JD, Overkleeft HS. Synthesis of 6-Hydroxysphingosine and α-Hydroxy Ceramide Using a Cross-Metathesis Strategy. The Journal of Organic Chemistry. 80: 7258-65. PMID 26061009 DOI: 10.1021/acs.joc.5b00823  1
2015 Willems MM, Zom GG, Meeuwenoord N, Khan S, Ossendorp F, Overkleeft HS, van der Marel GA, Filippov DV, Codée JD. Lipophilic Muramyl Dipeptide-Antigen Conjugates as Immunostimulating Agents. Chemmedchem. PMID 26059481 DOI: 10.1002/cmdc.201500196  1
2015 Zhang Q, van Rijssel ER, Walvoort MT, Overkleeft HS, van der Marel GA, Codée JD. Acceptor reactivity in the total synthesis of alginate fragments containing α-L-guluronic acid and β-D-mannuronic acid. Angewandte Chemie (International Ed. in English). 54: 7670-3. PMID 25960101 DOI: 10.1002/anie.201502581  1
2015 Liu N, Hoogendoorn S, van de Kar B, Kaptein A, Barf T, Driessen C, Filippov DV, van der Marel GA, van der Stelt M, Overkleeft HS. Direct and two-step bioorthogonal probes for Bruton's tyrosine kinase based on ibrutinib: a comparative study. Organic & Biomolecular Chemistry. 13: 5147-57. PMID 25849561 DOI: 10.1039/c5ob00474h  1
2015 van Rijssel ER, van Delft P, van Marle DV, Bijvoets SM, Lodder G, Overkleeft HS, van der Marel GA, Filippov DV, Codée JD. Stereoselectivity in the Lewis acid mediated reduction of ketofuranoses. The Journal of Organic Chemistry. 80: 4553-65. PMID 25826382 DOI: 10.1021/acs.joc.5b00419  1
2015 Ouchaou K, Maire F, Salo O, Ali H, Hankemeier T, van der Marel GA, Filippov DV, Bovenberg RA, Vreeken RJ, Driessen AJ, Overkleeft HS. A mutasynthesis approach with a Penicillium chrysogenum ΔroqA strain yields new roquefortine D analogues. Chembiochem : a European Journal of Chemical Biology. 16: 915-23. PMID 25766600 DOI: 10.1002/cbic.201402686  1
2015 Ouairy CM, Ferraz MJ, Boot RG, Baggelaar MP, van der Stelt M, Appelman M, van der Marel GA, Florea BI, Aerts JM, Overkleeft HS. Development of an acid ceramidase activity-based probe. Chemical Communications (Cambridge, England). 51: 6161-3. PMID 25748248 DOI: 10.1039/c5cc00356c  1
2015 Kistemaker HA, Lameijer LN, Meeuwenoord NJ, Overkleeft HS, van der Marel GA, Filippov DV. Synthesis of well-defined adenosine diphosphate ribose oligomers. Angewandte Chemie (International Ed. in English). 54: 4915-8. PMID 25704172 DOI: 10.1002/anie.201412283  1
2015 Padwal JD, Filippov DV, Narhe BD, Aertssen S, Beuving RJ, Benningshof JC, van der Marel GA, Overkleeft HS, van der Stelt M. Cyclopentitol as a scaffold for a natural product-like compound library for drug discovery. Bioorganic & Medicinal Chemistry. 23: 2650-5. PMID 25691210 DOI: 10.1016/j.bmc.2015.01.040  1
2015 Jiang J, Kallemeijn WW, Wright DW, Van Den Nieuwendijk AMCH, Rohde VC, Folch EC, Van Den Elst H, Florea BI, Scheij S, Donker-Koopman WE, Verhoek M, Li N, Schürmann M, Mink D, Boot RG, ... ... Van Der Marel GA, et al. In vitro and in vivo comparative and competitive activity-based protein profiling of GH29 α-L-fucosidases Chemical Science. 6: 2782-2789. DOI: 10.1039/c4sc03739a  1
2015 Kistemaker HAV, Meeuwenoord NJ, Overkleeft HS, Van Der Marel GA, Filippov DV. On the Synthesis of Oligonucleotides Interconnected through Pyrophosphate Linkages European Journal of Organic Chemistry. 2015: 6084-6091. DOI: 10.1002/ejoc.201500911  1
2015 Hoogendoorn S, Mock ED, Strijland A, Donker-Koopman WE, van den Elst H, van den Berg RJBHN, Aerts JMFG, van der Marel GA, Overkleeft HS. ortho-Carborane-Modified N-Substituted Deoxynojirimycins European Journal of Organic Chemistry. DOI: 10.1002/ejoc.201500364  1
2015 Wisse P, Gold H, Mirzaian M, Ferraz MJ, Lutteke G, Van Den Berg RJBHN, Van Den Elst H, Lugtenburg J, Van Der Marel GA, Aerts JMFG, Codée JDC, Overkleeft HS. Synthesis of a panel of carbon-13-labelled (glyco)sphingolipids European Journal of Organic Chemistry. 2015: 2661-2677. DOI: 10.1002/ejoc.201500025  1
2015 Wong CS, Hoogendoorn S, Van Der Marel GA, Overkleeft HS, Codée JDC. Targeted delivery of fluorescent high-mannose-type oligosaccharide cathepsin inhibitor conjugates Chempluschem. 80: 928-937. DOI: 10.1002/cplu.201500004  1
2014 Zom GG, Filippov DV, van der Marel GA, Overkleeft HS, Melief CJ, Ossendorp F. Two in one: improving synthetic long peptide vaccines by combining antigen and adjuvant in one molecule. Oncoimmunology. 3: e947892. PMID 25610736 DOI: 10.4161/21624011.2014.947892  0.6
2014 Kallemeijn WW, Witte MD, Voorn-Brouwer TM, Walvoort MT, Li KY, Codée JD, van der Marel GA, Boot RG, Overkleeft HS, Aerts JM. A sensitive gel-based method combining distinct cyclophellitol-based probes for the identification of acid/base residues in human retaining β-glucosidases. The Journal of Biological Chemistry. 289: 35351-62. PMID 25344605 DOI: 10.1074/jbc.M114.593376  1
2014 Laverde D, Wobser D, Romero-Saavedra F, Hogendorf W, Van Der Marel G, Berthold M, Kropec A, Codee J, Huebner J. Synthetic teichoic acid conjugate vaccine against nosocomial Gram-positive bacteria Plos One. 9. PMID 25333799 DOI: 10.1371/journal.pone.0110953  1
2014 Ghisaidoobe AT, van den Berg RJ, Butt SS, Strijland A, Donker-Koopman WE, Scheij S, van den Nieuwendijk AM, Koomen GJ, van Loevezijn A, Leemhuis M, Wennekes T, van der Stelt M, van der Marel GA, van Boeckel CA, Aerts JM, et al. Identification and development of biphenyl substituted iminosugars as improved dual glucosylceramide synthase/neutral glucosylceramidase inhibitors. Journal of Medicinal Chemistry. 57: 9096-104. PMID 25250725 DOI: 10.1021/jm501181z  1
2014 Hoogendoorn S, van Puijvelde GH, Kuiper J, van der Marel GA, Overkleeft HS. A multivalent ligand for the mannose-6-phosphate receptor for endolysosomal targeting of an activity-based probe. Angewandte Chemie (International Ed. in English). 53: 10975-8. PMID 25163608 DOI: 10.1002/anie.201406842  1
2014 Li KY, Jiang J, Witte MD, Kallemeijn WW, Donker-Koopman WE, Boot RG, Aerts JM, Codée JD, van der Marel GA, Overkleeft HS. Exploring functional cyclophellitol analogues as human retaining beta-glucosidase inhibitors. Organic & Biomolecular Chemistry. 12: 7786-91. PMID 25156485 DOI: 10.1039/c4ob01611d  1
2014 Willems LI, Beenakker TJ, Murray B, Scheij S, Kallemeijn WW, Boot RG, Verhoek M, Donker-Koopman WE, Ferraz MJ, van Rijssel ER, Florea BI, Codée JD, van der Marel GA, Aerts JM, Overkleeft HS. Potent and selective activity-based probes for GH27 human retaining α-galactosidases. Journal of the American Chemical Society. 136: 11622-5. PMID 25105979 DOI: 10.1021/ja507040n  1
2014 Duivenvoorden BA, Ghauharali K, Scheij S, Boot RG, Aerts JM, van der Marel GA, Overkleeft HS, Codée JD. Design and synthesis of 4'-O-alkyl-chitobiosyl-4-methylumbelliferone as human chitinase fluorogenic substrates. Carbohydrate Research. 399: 26-37. PMID 25104395 DOI: 10.1016/j.carres.2014.07.007  1
2014 Willems LI, Jiang J, Li KY, Witte MD, Kallemeijn WW, Beenakker TJ, Schröder SP, Aerts JM, van der Marel GA, Codée JD, Overkleeft HS. From covalent glycosidase inhibitors to activity-based glycosidase probes. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 10864-72. PMID 25100671 DOI: 10.1002/chem.201404014  1
2014 van Rijssel ER, van Delft P, Lodder G, Overkleeft HS, van der Marel GA, Filippov DV, Codée JD. Furanosyl oxocarbenium ion stability and stereoselectivity. Angewandte Chemie (International Ed. in English). 53: 10381-5. PMID 25081839 DOI: 10.1002/anie.201405477  1
2014 Willems MM, Zom GG, Khan S, Meeuwenoord N, Melief CJ, van der Stelt M, Overkleeft HS, Codée JD, van der Marel GA, Ossendorp F, Filippov DV. N-tetradecylcarbamyl lipopeptides as novel agonists for Toll-like receptor 2. Journal of Medicinal Chemistry. 57: 6873-8. PMID 25019313 DOI: 10.1021/jm500722p  1
2014 de Bruin G, Huber EM, Xin BT, van Rooden EJ, Al-Ayed K, Kim KB, Kisselev AF, Driessen C, van der Stelt M, van der Marel GA, Groll M, Overkleeft HS. Structure-based design of β1i or β5i specific inhibitors of human immunoproteasomes. Journal of Medicinal Chemistry. 57: 6197-209. PMID 25006746 DOI: 10.1021/jm500716s  1
2014 Willems MM, Zom GG, Meeuwenoord N, Ossendorp FA, Overkleeft HS, van der Marel GA, Codée JD, Filippov DV. Design, automated synthesis and immunological evaluation of NOD2-ligand-antigen conjugates. Beilstein Journal of Organic Chemistry. 10: 1445-53. PMID 24991299 DOI: 10.3762/bjoc.10.148  1
2014 Xin BT, de Bruin G, Verdoes M, Filippov DV, van der Marel GA, Overkleeft HS. Exploring dual electrophiles in peptide-based proteasome inhibitors: carbonyls and epoxides. Organic & Biomolecular Chemistry. 12: 5710-8. PMID 24968066 DOI: 10.1039/c4ob00893f  1
2014 Castelli R, Schindler S, Walter SM, Kniep F, Overkleeft HS, Van der Marel GA, Huber SM, Codée JD. Activation of glycosyl halides by halogen bonding. Chemistry, An Asian Journal. 9: 2095-8. PMID 24962953 DOI: 10.1002/asia.201402259  1
2014 Zom GG, Khan S, Britten CM, Sommandas V, Camps MG, Loof NM, Budden CF, Meeuwenoord NJ, Filippov DV, van der Marel GA, Overkleeft HS, Melief CJ, Ossendorp F. Efficient induction of antitumor immunity by synthetic toll-like receptor ligand-peptide conjugates. Cancer Immunology Research. 2: 756-64. PMID 24950688 DOI: 10.1158/2326-6066.CIR-13-0223  1
2014 Engelsma SB, Willems LI, van Paaschen CE, van Kasteren SI, van der Marel GA, Overkleeft HS, Filippov DV. Acylazetine as a dienophile in bioorthogonal inverse electron-demand Diels-Alder ligation. Organic Letters. 16: 2744-7. PMID 24796604 DOI: 10.1021/ol501049c  1
2014 Van Delft P, De Witte W, Meeuwenoord NJ, Van Der Heden Van Noort GJ, Versluis F, Olsthoorn RCL, Overkleeft HS, Van Der Marel GA, Filippov DV. Design of a ribosyltriazole-annulated cyclooctyne for oligonucleotide labeling by strain-promoted alkyne-azide cycloaddition European Journal of Organic Chemistry. 2014: 7566-7571. DOI: 10.1002/ejoc.201403086  1
2014 Willems LI, Beenakker TJM, Murray B, Gagestein B, van den Elst H, van Rijssel ER, Codée JDC, Kallemeijn WW, Aerts JMFG, van der Marel GA, Overkleeft HS. Synthesis of α- and β-galactopyranose-configured isomers of cyclophellitol and cyclophellitol aziridine European Journal of Organic Chemistry. DOI: 10.1002/ejoc.201402589  1
2014 Li KY, Jiang J, Witte MD, Kallemeijn WW, van den Elst H, Wong CS, Chander SD, Hoogendoorn S, Beenakker TJM, Codée JDC, Aerts JMFG, van der Marel GA, Overkleeft HS. Synthesis of cyclophellitol, cyclophellitol aziridine, and their tagged derivatives European Journal of Organic Chemistry. DOI: 10.1002/ejoc.201402588  1
2014 Li KY, Kallemeijn W, Jiang J, Walvoort M, Willems L, Beenakker T, Van Den Elst H, Van Der Marel G, Codée J, Aerts H, Florea B, Boot R, Witte M, Overkleeft H. Rational Design of Activity-Based Retaining β-Exoglucosidase Probes Concepts and Case Studies in Chemical Biology. 191-206. DOI: 10.1002/9783527687503.ch13  1
2014 De Bruin G, Li N, Paniagua G, Willems L, Xin BT, Verdoes M, Geurink P, Van Der Linden W, Van Der Stelt M, Van Der Marel G, Overkleeft H, Florea B. Activity-Based Proteasome Profiling in Medicinal Chemistry and Chemical Biology Concepts and Case Studies in Chemical Biology. 177-190. DOI: 10.1002/9783527687503.ch12  1
2013 Baggelaar MP, Janssen FJ, van Esbroeck AC, den Dulk H, Allarà M, Hoogendoorn S, McGuire R, Florea BI, Meeuwenoord N, van den Elst H, van der Marel GA, Brouwer J, Di Marzo V, Overkleeft HS, van der Stelt M. Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-α in brain. Angewandte Chemie (International Ed. in English). 52: 12081-5. PMID 24173880 DOI: 10.1002/anie.201306295  0.56
2013 Rönnols J, Walvoort MT, van der Marel GA, Codée JD, Widmalm G. Chair interconversion and reactivity of mannuronic acid esters. Organic & Biomolecular Chemistry. 11: 8127-34. PMID 24173496 DOI: 10.1039/c3ob41747f  1
2013 Yu H, Segers F, Sliedregt-Bol K, Bot I, Woltman AM, Boross P, Verbeek S, Overkleeft H, van der Marel GA, van Kooten C, van Berkel TJ, Biessen EA. Identification of a novel CD40 ligand for targeted imaging of inflammatory plaques by phage display. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 27: 4136-46. PMID 23896727 DOI: 10.1096/fj.12-224667  1
2013 van Rijssel ER, Goumans TP, Lodder G, Overkleeft HS, van der Marel GA, Codée JD. Chiral pyrroline-based Ugi-three-component reactions are under kinetic control. Organic Letters. 15: 3026-9. PMID 23721351 DOI: 10.1021/ol4012053  1
2013 Kistemaker HA, van Noort GJ, Overkleeft HS, van der Marel GA, Filippov DV. Stereoselective ribosylation of amino acids. Organic Letters. 15: 2306-9. PMID 23614697 DOI: 10.1021/ol400929c  1
2013 Castelli R, Overkleeft HS, van der Marel GA, Codée JD. 2,2-Dimethyl-4-(4-methoxy-phenoxy) butanoate and 2,2-dimethyl-4-azido butanoate: two new pivaloate-ester-like protecting groups. Organic Letters. 15: 2270-3. PMID 23607790 DOI: 10.1021/ol4008475  1
2013 van der Heden van Noort GJ, Schein CH, Overkleeft HS, van der Marel GA, Filippov DV. A general synthetic method toward uridylylated picornavirus VPg proteins. Journal of Peptide Science : An Official Publication of the European Peptide Society. 19: 333-6. PMID 23606631 DOI: 10.1002/psc.2508  1
2013 Frihed TG, Walvoort MT, Codée JD, van der Marel GA, Bols M, Pedersen CM. Influence of O6 in mannosylations using benzylidene protected donors: stereoelectronic or conformational effects? The Journal of Organic Chemistry. 78: 2191-205. PMID 23336427 DOI: 10.1021/jo302455d  1
2013 Geurink PP, van der Linden WA, Mirabella AC, Gallastegui N, de Bruin G, Blom AE, Voges MJ, Mock ED, Florea BI, van der Marel GA, Driessen C, van der Stelt M, Groll M, Overkleeft HS, Kisselev AF. Incorporation of non-natural amino acids improves cell permeability and potency of specific inhibitors of proteasome trypsin-like sites. Journal of Medicinal Chemistry. 56: 1262-75. PMID 23320547 DOI: 10.1021/jm3016987  1
2013 Gold H, Mirzaian M, Dekker N, Joao Ferraz M, Lugtenburg J, Codée JD, van der Marel GA, Overkleeft HS, Linthorst GE, Groener JE, Aerts JM, Poorthuis BJ. Quantification of globotriaosylsphingosine in plasma and urine of fabry patients by stable isotope ultraperformance liquid chromatography-tandem mass spectrometry. Clinical Chemistry. 59: 547-56. PMID 23237761 DOI: 10.1373/clinchem.2012.192138  1
2013 Guisado-Barrios G, Muñoz BK, Kamer PC, Lastdrager B, van der Marel G, Overhand M, Vega-Vázquez M, Martin-Pastor M. Cyclic decapeptide gramicidin S derivatives containing phosphines: novel ligands for asymmetric catalysis. Dalton Transactions (Cambridge, England : 2003). 42: 1973-8. PMID 23235486 DOI: 10.1039/c2dt31782f  1
2013 Walvoort MTC, Van Der Marel GA, Overkleeft HS, Codée JDC. On the reactivity and selectivity of donor glycosides in glycochemistry and glycobiology: Trapped covalent intermediates Chemical Science. 4: 897-906. DOI: 10.1039/c2sc21610h  1
2013 Otero JM, Van Der Knaap M, Llamas-Saiz AL, Van Raaij MJ, Amorín M, Granja JR, Filippov DV, Van Der Marel GA, Overkleeft HS, Overhand M. Design, synthesis, and structural analysis of turn modified cyclo-(αβ3αβ2α)2 peptide derivatives toward crystalline hexagon-shaped cationic nanochannel assemblies Crystal Growth and Design. 13: 4355-4367. DOI: 10.1021/cg4007108  1
2013 De Jong AR, Volbeda AG, Hagen B, Van Den Elst H, Overkleeft HS, Van Der Marel GA, Codée JDC. A second-generation tandem ring-closing metathesis cleavable linker for solid-phase oligosaccharide synthesis European Journal of Organic Chemistry. 6644-6655. DOI: 10.1002/ejoc.201301055  1
2012 van der Knaap M, Basalan F, van de Mei HC, Busscher HJ, van der Marel GA, Overkleeft HS, Overhand M. Synthesis and biological evaluation of gramicidin S-inspired cyclic mixed α/β-peptides. Chemistry & Biodiversity. 9: 2494-506. PMID 23161631 DOI: 10.1002/cbdv.201200277  1
2012 Kallemeijn WW, Li KY, Witte MD, Marques AR, Aten J, Scheij S, Jiang J, Willems LI, Voorn-Brouwer TM, van Roomen CP, Ottenhoff R, Boot RG, van den Elst H, Walvoort MT, Florea BI, ... ... van der Marel GA, et al. Novel activity-based probes for broad-spectrum profiling of retaining β-exoglucosidases in situ and in vivo. Angewandte Chemie (International Ed. in English). 51: 12529-33. PMID 23139194 DOI: 10.1002/anie.201207771  1
2012 Barroso S, Castelli R, Baggelaar MP, Geerdink D, ter Horst B, Casas-Arce E, Overkleeft HS, van der Marel GA, Codée JD, Minnaard AJ. Total synthesis of the triglycosyl phenolic glycolipid PGL-tb1 from Mycobacterium tuberculosis. Angewandte Chemie (International Ed. in English). 51: 11774-7. PMID 23086739 DOI: 10.1002/anie.201206221  1
2012 Li J, Girard G, Florea BI, Geurink PP, Li N, van der Marel GA, Overhand M, Overkleeft HS, van Wezel GP. Identification and isolation of lantibiotics from culture: a bioorthogonal chemistry approach. Organic & Biomolecular Chemistry. 10: 8677-83. PMID 23033043 DOI: 10.1039/c2ob26050f  1
2012 Kapoerchan VV, Knijnenburg AD, Keizer P, Spalburg E, de Neeling AJ, Mars-Groenendijk RH, Noort D, Otero JM, Llamas-Saiz AL, van Raaij MJ, van der Marel GA, Overkleeft HS, Overhand M. 'Inverted' analogs of the antibiotic gramicidin S with an improved biological profile. Bioorganic & Medicinal Chemistry. 20: 6059-62. PMID 22989907 DOI: 10.1016/j.bmc.2012.08.038  1
2012 Walvoort MT, Kallemeijn WW, Willems LI, Witte MD, Aerts JM, van der Marel GA, Codée JD, Overkleeft HS. Tuning the leaving group in 2-deoxy-2-fluoroglucoside results in improved activity-based retaining β-glucosidase probes. Chemical Communications (Cambridge, England). 48: 10386-8. PMID 22932951 DOI: 10.1039/c2cc35653h  1
2012 van der Heden van Noort GJ, van Delft P, Meeuwenoord NJ, Overkleeft HS, van der Marel GA, Filippov DV. Fully automated sequential solid phase approach towards viral RNA-nucleopeptides. Chemical Communications (Cambridge, England). 48: 8093-5. PMID 22781550 DOI: 10.1039/c2cc33477a  1
2012 Walvoort MT, Volbeda AG, Reintjens NR, van den Elst H, Plante OJ, Overkleeft HS, van der Marel GA, Codée JD. Automated solid-phase synthesis of hyaluronan oligosaccharides. Organic Letters. 14: 3776-9. PMID 22780913 DOI: 10.1021/ol301666n  1
2012 Willems LI, Li N, Florea BI, Ruben M, van der Marel GA, Overkleeft HS. Triple bioorthogonal ligation strategy for simultaneous labeling of multiple enzymatic activities. Angewandte Chemie (International Ed. in English). 51: 4431-4. PMID 22438272 DOI: 10.1002/anie.201200923  1
2012 Hogendorf WF, Kropec A, Filippov DV, Overkleeft HS, Huebner J, van der Marel GA, Codée JD. Light fluorous synthesis of glucosylated glycerol teichoic acids. Carbohydrate Research. 356: 142-51. PMID 22429772 DOI: 10.1016/j.carres.2012.02.023  1
2012 Christina AE, Blas Ferrando VM, de Bordes F, Spruit WA, Overkleeft HS, Codée JD, van der Marel GA. Multigram-scale synthesis of an orthogonally protected 2-acetamido-4-amino-2,4,6-trideoxy-D-galactose (AAT) building block. Carbohydrate Research. 356: 282-7. PMID 22418093 DOI: 10.1016/j.carres.2012.02.015  1
2012 Theilacker C, Kropec A, Hammer F, Sava I, Wobser D, Sakinc T, Codée JD, Hogendorf WF, van der Marel GA, Huebner J. Protection against Staphylococcus aureus by antibody to the polyglycerolphosphate backbone of heterologous lipoteichoic acid. The Journal of Infectious Diseases. 205: 1076-85. PMID 22362863 DOI: 10.1093/infdis/jis022  1
2012 Walvoort MT, van den Elst H, Plante OJ, Kröck L, Seeberger PH, Overkleeft HS, van der Marel GA, Codée JD. Automated solid-phase synthesis of β-mannuronic acid alginates. Angewandte Chemie (International Ed. in English). 51: 4393-6. PMID 22334421 DOI: 10.1002/anie.201108744  1
2012 Christina AE, van der Es D, Dinkelaar J, Overkleeft HS, van der Marel GA, Codée JD. β-Rhamnosides from 6-thio mannosides. Chemical Communications (Cambridge, England). 48: 2686-8. PMID 22306867 DOI: 10.1039/c2cc17623h  0.56
2012 Hogendorf WF, Lameijer LN, Beenakker TJ, Overkleeft HS, Filippov DV, Codée JD, Van der Marel GA. Fluorous linker facilitated synthesis of teichoic acid fragments. Organic Letters. 14: 848-51. PMID 22264133 DOI: 10.1021/ol2033652  1
2012 de Jong AR, Hagen B, van der Ark V, Overkleeft HS, Codée JD, Van der Marel GA. Exploring and exploiting the reactivity of glucuronic acid donors. The Journal of Organic Chemistry. 77: 108-25. PMID 22126096 DOI: 10.1021/jo201586r  1
2012 Yu H, Bot I, Sliedregt K, Xu X, Bot M, van Heiningen SH, van der Marel GA, Bennett MR, Overkleeft H, van Berkel TJ, Biessen EA. Selective modulation of nuclear factor of activated T-cell function in restenosis by a potent bipartite peptide inhibitor. Circulation Research. 110: 200-10. PMID 22116820 DOI: 10.1161/CIRCRESAHA.111.240895  1
2012 van der Linden WA, Willems LI, Shabaneh TB, Li N, Ruben M, Florea BI, van der Marel GA, Kaiser M, Kisselev AF, Overkleeft HS. Discovery of a potent and highly β1 specific proteasome inhibitor from a focused library of urea-containing peptide vinyl sulfones and peptide epoxyketones. Organic & Biomolecular Chemistry. 10: 181-94. PMID 22105930 DOI: 10.1039/c1ob06554h  1
2012 Geurink PP, Prely LM, van der Marel GA, Bischoff R, Overkleeft HS. Photoaffinity labeling in activity-based protein profiling. Topics in Current Chemistry. 324: 85-113. PMID 22028098 DOI: 10.1007/128_2011_286  1
2012 van der Linden WA, Li N, Hoogendoorn S, Ruben M, Verdoes M, Guo J, Boons GJ, van der Marel GA, Florea BI, Overkleeft HS. Two-step bioorthogonal activity-based proteasome profiling using copper-free click reagents: a comparative study. Bioorganic & Medicinal Chemistry. 20: 662-6. PMID 21757357 DOI: 10.1016/j.bmc.2011.06.037  1
2012 Van Der Knaap M, Otero JM, Llamas-Saiz A, Van Raaij MJ, Lageveen LI, Busscher HJ, Grotenbreg GM, Van Der Marel GA, Overkleeft HS, Overhand M. Design, synthesis and structural analysis of mixed α/β-peptides that adopt stable cyclic hairpin-like conformations Tetrahedron. 68: 2391-2400. DOI: 10.1016/j.tet.2012.01.015  1
2012 Wennekes T, Bonger KM, Vogel K, Van Den Berg RJBHN, Strijland A, Donker-Koopman WE, Aerts JMFG, Van Der Marel GA, Overkleeft HS. The development of an aza-C-glycoside library based on a tandem staudinger/aza-wittig/ugi three-component reaction European Journal of Organic Chemistry. 6420-6454. DOI: 10.1002/ejoc.201200923  1
2012 Christina AE, Muns JA, Olivier JQA, Visser L, Hagen B, Van Den Bos LJ, Overkleeft HS, Codée JDC, Van Der Marel GA. On the reactivity and selectivity of galacturonic acid lactones European Journal of Organic Chemistry. 5729-5737. DOI: 10.1002/ejoc.201200717  1
2012 Van Den Nieuwendijk AMCH, Van Den Berg RJBHN, Ruben M, Witte MD, Brussee J, Boot RG, Van Der Marel GA, Aerts JMFG, Overkleeft HS. Synthesis of eight 1-deoxynojirimycin isomers from a single chiral cyanohydrin European Journal of Organic Chemistry. 3437-3446. DOI: 10.1002/ejoc.201200377  1
2011 van den Berg RJ, Wennekes T, Ghisaidoobe A, Donker-Koopman WE, Strijland A, Boot RG, van der Marel GA, Aerts JM, Overkleeft HS. Assessment of partially deoxygenated deoxynojirimycin derivatives as glucosylceramide synthase inhibitors. Acs Medicinal Chemistry Letters. 2: 519-22. PMID 24900342 DOI: 10.1021/ml200050s  1
2011 Bonger KM, Hoogendoorn S, van Koppen CJ, Timmers CM, van der Marel GA, Overkleeft HS. Development of Selective LH Receptor Agonists by Heterodimerization with a FSH Receptor Antagonist. Acs Medicinal Chemistry Letters. 2: 85-9. PMID 24900256 DOI: 10.1021/ml100229v  1
2011 Hoogendoorn S, Blom AE, Willems LI, van der Marel GA, Overkleeft HS. Synthesis of pH-activatable red fluorescent BODIPY dyes with distinct functionalities. Organic Letters. 13: 5656-9. PMID 21942639 DOI: 10.1021/ol202379w  1
2011 Willems LI, van der Linden WA, Li N, Li KY, Liu N, Hoogendoorn S, van der Marel GA, Florea BI, Overkleeft HS. Bioorthogonal chemistry: applications in activity-based protein profiling. Accounts of Chemical Research. 44: 718-29. PMID 21797256 DOI: 10.1021/ar200125k  1
2011 Walvoort MT, Moggré GJ, Lodder G, Overkleeft HS, Codée JD, van der Marel GA. Stereoselective synthesis of 2,3-diamino-2,3-dideoxy-β-D-mannopyranosyl uronates. The Journal of Organic Chemistry. 76: 7301-15. PMID 21793528 DOI: 10.1021/jo201179p  1
2011 Walvoort MT, de Witte W, van Dijk J, Dinkelaar J, Lodder G, Overkleeft HS, Codée JD, van der Marel GA. Mannopyranosyl uronic acid donor reactivity. Organic Letters. 13: 4360-3. PMID 21776974 DOI: 10.1021/ol2016862  1
2011 Witte MD, van der Marel GA, Aerts JM, Overkleeft HS. Irreversible inhibitors and activity-based probes as research tools in chemical glycobiology. Organic & Biomolecular Chemistry. 9: 5908-26. PMID 21769371 DOI: 10.1039/c1ob05531c  1
2011 Hoogendoorn S, Habets KL, Passemard S, Kuiper J, van der Marel GA, Florea BI, Overkleeft HS. Targeted pH-dependent fluorescent activity-based cathepsin probes. Chemical Communications (Cambridge, England). 47: 9363-5. PMID 21769329 DOI: 10.1039/c1cc12947c  1
2011 Hogendorf WF, Meeuwenoord N, Overkleeft HS, Filippov DV, Laverde D, Kropec A, Huebner J, Van der Marel GA, Codée JD. Automated solid phase synthesis of teichoic acids. Chemical Communications (Cambridge, England). 47: 8961-3. PMID 21734985 DOI: 10.1039/c1cc13132j  1
2011 Knijnenburg AD, Kapoerchan VV, Grotenbreg GM, Spalburg E, de Neeling AJ, Mars-Groenendijk RH, Noort D, Otero JM, Llamas-Saiz AL, van Raaij MJ, Ravensbergen B, Nibbering PH, van der Marel GA, Overkleeft HS, Overhand M. Synthesis and evaluation of strand and turn modified ring-extended gramicidin S derivatives. Bioorganic & Medicinal Chemistry. 19: 3402-9. PMID 21561781 DOI: 10.1016/j.bmc.2011.04.031  1
2011 van der Heden van Noort GJ, Overkleeft HS, van der Marel GA, Filippov DV. Ribosylation of adenosine: an orthogonally protected building block for the synthesis of ADP-ribosyl oligomers. Organic Letters. 13: 2920-3. PMID 21561136 DOI: 10.1021/ol200971z  1
2011 Witte MD, Walvoort MT, Li KY, Kallemeijn WW, Donker-Koopman WE, Boot RG, Aerts JM, Codée JD, van der Marel GA, Overkleeft HS. Activity-based profiling of retaining β-glucosidases: a comparative study. Chembiochem : a European Journal of Chemical Biology. 12: 1263-9. PMID 21538758 DOI: 10.1002/cbic.201000773  1
2011 Gold H, Munneke S, Dinkelaar J, Overkleeft HS, Aerts JM, Codée JD, van der Marel GA. A practical synthesis of capped 4-methylumbelliferyl hyaluronan disaccharides and tetrasaccharides as potential hyaluronidase substrates. Carbohydrate Research. 346: 1467-78. PMID 21536258 DOI: 10.1016/j.carres.2011.03.042  1
2011 Aerts JM, Kallemeijn WW, Wegdam W, Joao Ferraz M, van Breemen MJ, Dekker N, Kramer G, Poorthuis BJ, Groener JE, Cox-Brinkman J, Rombach SM, Hollak CE, Linthorst GE, Witte MD, Gold H, ... van der Marel GA, et al. Biomarkers in the diagnosis of lysosomal storage disorders: proteins, lipids, and inhibodies. Journal of Inherited Metabolic Disease. 34: 605-19. PMID 21445610 DOI: 10.1007/s10545-011-9308-6  1
2011 van der Knaap M, Lageveen LT, Busscher HJ, Mars-Groenendijk R, Noort D, Otero JM, Llamas-Saiz AL, van Raaij MJ, van der Marel GA, Overkleeft HS, Overhand M. Evaluation of readily accessible azoles as mimics of the aromatic ring of D-phenylalanine in the turn region of gramicidin S. Chemmedchem. 6: 840-7. PMID 21400662 DOI: 10.1002/cmdc.201000539  0.56
2011 Knijnenburg AD, Tuin AW, Spalburg E, de Neeling AJ, Mars-Groenendijk RH, Noort D, Otero JM, Llamas-Saiz AL, van Raaij MJ, van der Marel GA, Overkleeft HS, Overhand M. Exploring the conformational and biological versatility of β-turn-modified gramicidin S by using sugar amino acid homologues that vary in ring size. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 3995-4004. PMID 21365698 DOI: 10.1002/chem.201002895  1
2011 Christina AE, van den Bos LJ, Overkleeft HS, van der Marel GA, Codée JD. Galacturonic acid lactones in the synthesis of all trisaccharide repeating units of the zwitterionic polysaccharide Sp1. The Journal of Organic Chemistry. 76: 1692-706. PMID 21341806 DOI: 10.1021/jo102363d  1
2011 Codée JD, Christina AE, Walvoort MT, Overkleeft HS, van der Marel GA. Uronic acids in oligosaccharide and glycoconjugate synthesis. Topics in Current Chemistry. 301: 253-89. PMID 21222193 DOI: 10.1007/128_2010_111  1
2011 Codée JDC, Walvoort MTC, De Jong AR, Lodder G, Overkleeft HS, Van Der Marel GA. Mannuronic acids: Reactivity and selectivity Journal of Carbohydrate Chemistry. 30: 438-457. DOI: 10.1080/07328303.2011.624284  1
2011 Vandelft P, Vanschie E, Meeuwenoord NJ, Overkleeft HS, Van Der Marel GA, Filippov DV. Oligonucleotide conjugates by means of copper-free click chemistry - Expanding the repertoire of strained cyclooctyne phosphoramidites Synthesis. 2724-2732. DOI: 10.1055/s-0030-1260104  1
2011 Codée JDC, Ali A, Overkleeft HS, Van Der Marel GA. Novel protecting groups in carbohydrate chemistry Comptes Rendus Chimie. 14: 178-193. DOI: 10.1016/j.crci.2010.05.010  1
2011 Van Den Berg RJBHN, Van Den Elst H, Korevaar CGN, Aerts JMFG, Van Der Marel GA, Overkleeft HS. A rapid and efficient synthesis of D-erythro-sphingosine from D-ribo-phytosphingosine European Journal of Organic Chemistry. 6685-6689. DOI: 10.1002/ejoc.201100911  1
2011 Gold H, Boot RG, Aerts JMFG, Overkleeft HS, Codée JDC, Van Der Marel GA. A concise synthesis of globotriaosylsphingosine European Journal of Organic Chemistry. 1652-1663. DOI: 10.1002/ejoc.201001690  1
2010 Witte MD, Kallemeijn WW, Aten J, Li KY, Strijland A, Donker-Koopman WE, van den Nieuwendijk AM, Bleijlevens B, Kramer G, Florea BI, Hooibrink B, Hollak CE, Ottenhoff R, Boot RG, van der Marel GA, et al. Ultrasensitive in situ visualization of active glucocerebrosidase molecules. Nature Chemical Biology. 6: 907-13. PMID 21079602 DOI: 10.1038/nchembio.466  1
2010 Walvoort MT, Lodder G, Overkleeft HS, Codée JD, van der Marel GA. Mannosazide methyl uronate donors. Glycosylating properties and use in the construction of β-ManNAcA-containing oligosaccharides. The Journal of Organic Chemistry. 75: 7990-8002. PMID 21062001 DOI: 10.1021/jo101779v  1
2010 van Delft P, Meeuwenoord NJ, Hoogendoorn S, Dinkelaar J, Overkleeft HS, van der Marel GA, Filippov DV. Synthesis of oligoribonucleic acid conjugates using a cyclooctyne phosphoramidite. Organic Letters. 12: 5486-9. PMID 21049910 DOI: 10.1021/ol102357u  1
2010 Geurink PP, Florea BI, Van der Marel GA, Kessler BM, Overkleeft HS. Probing the proteasome cavity in three steps: bio-orthogonal photo-reactive suicide substrates. Chemical Communications (Cambridge, England). 46: 9052-4. PMID 20981375 DOI: 10.1039/c0cc03322g  1
2010 Knijnenburg AD, Kapoerchan VV, Spalburg E, de Neeling AJ, Mars-Groenendijk RH, Noort D, van der Marel GA, Overkleeft HS, Overhand M. Tuning hydrophobicity of highly cationic tetradecameric Gramicidin S analogues using adamantane amino acids. Bioorganic & Medicinal Chemistry. 18: 8403-9. PMID 20951594 DOI: 10.1016/j.bmc.2010.09.018  1
2010 Kapoerchan VV, Knijnenburg AD, Niamat M, Spalburg E, de Neeling AJ, Nibbering PH, Mars-Groenendijk RH, Noort D, Otero JM, Llamas-Saiz AL, van Raaij MJ, van der Marel GA, Overkleeft HS, Overhand M. An adamantyl amino acid containing gramicidin S analogue with broad spectrum antibacterial activity and reduced hemolytic activity. Chemistry (Weinheim An Der Bergstrasse, Germany). 16: 12174-81. PMID 20848624 DOI: 10.1002/chem.201001686  1
2010 Geurink PP, Florea BI, Li N, Witte MD, Verasdonck J, Kuo CL, van der Marel GA, Overkleeft HS. A cleavable linker based on the levulinoyl ester for activity-based protein profiling. Angewandte Chemie (International Ed. in English). 49: 6802-5. PMID 20715027 DOI: 10.1002/anie.201001767  1
2010 van der Heden van Noort GJ, Overkleeft HS, van der Marel GA, Filippov DV. Synthesis of nucleotidylated poliovirus VPg proteins. The Journal of Organic Chemistry. 75: 5733-6. PMID 20704445 DOI: 10.1021/jo100757t  1
2010 van den Nieuwendijk AM, Ruben M, Engelsma SE, Risseeuw MD, van den Berg RJ, Boot RG, Aerts JM, Brussee J, van der Marel GA, Overkleeft HS. Synthesis of L-altro-1-deoxynojirimycin, D-allo-1-deoxynojirimycin, and D-galacto-1-deoxynojirimycin from a single chiral cyanohydrin. Organic Letters. 12: 3957-9. PMID 20690611 DOI: 10.1021/ol101556k  1
2010 Willems LI, Verdoes M, Florea BI, van der Marel GA, Overkleeft HS. Two-step labeling of endogenous enzymatic activities by Diels-Alder ligation. Chembiochem : a European Journal of Chemical Biology. 11: 1769-81. PMID 20623570 DOI: 10.1002/cbic.201000280  1
2010 Risseeuw MD, Florea BI, van der Marel GA, Overkleeft HS, Overhand M. Sugar amino acid based peptide epoxyketones as potential proteasome inhibitors. Bioorganic Chemistry. 38: 202-9. PMID 20493511 DOI: 10.1016/j.bioorg.2010.04.004  1
2010 Verdoes M, Willems LI, van der Linden WA, Duivenvoorden BA, van der Marel GA, Florea BI, Kisselev AF, Overkleeft HS. A panel of subunit-selective activity-based proteasome probes. Organic & Biomolecular Chemistry. 8: 2719-27. PMID 20449511 DOI: 10.1039/c001036g  1
2010 van der Linden WA, Geurink PP, Oskam C, van der Marel GA, Florea BI, Overkleeft HS. Proteasome selectivity towards Michael acceptor containing oligopeptide-based inhibitors. Organic & Biomolecular Chemistry. 8: 1885-93. PMID 20449494 DOI: 10.1039/b924134e  1
2010 Bonger KM, Kapoerchan VV, Grotenbreg GM, van Koppen CJ, Timmers CM, van der Marel GA, Overkleeft HS. Oligoproline helices as structurally defined scaffolds for oligomeric G protein-coupled receptor ligands. Organic & Biomolecular Chemistry. 8: 1881-4. PMID 20449493 DOI: 10.1039/b923556f  1
2010 Walvoort MT, Dinkelaar J, van den Bos LJ, Lodder G, Overkleeft HS, Codée JD, van der Marel GA. The impact of oxacarbenium ion conformers on the stereochemical outcome of glycosylations. Carbohydrate Research. 345: 1252-63. PMID 20347068 DOI: 10.1016/j.carres.2010.02.027  1
2010 van der Heden van Noort GJ, van der Horst MG, Overkleeft HS, van der Marel GA, Filippov DV. Synthesis of mono-ADP-ribosylated oligopeptides using ribosylated amino acid building blocks. Journal of the American Chemical Society. 132: 5236-40. PMID 20232863 DOI: 10.1021/ja910940q  1
2010 Kapoerchan VV, Spalburg E, de Neeling AJ, Mars-Groenendijk RH, Noort D, Otero JM, Ferraces-Casais P, Llamas-Saiz AL, van Raaij MJ, van Doorn J, van der Marel GA, Overkleeft HS, Overhand M. Gramicidin S derivatives containing cis- and trans-morpholine amino acids (MAAs) as turn mimetics. Chemistry (Weinheim An Der Bergstrasse, Germany). 16: 4259-65. PMID 20209520 DOI: 10.1002/chem.200902984  1
2010 Geurink PP, Liu N, Spaans MP, Downey SL, van den Nieuwendijk AM, van der Marel GA, Kisselev AF, Florea BI, Overkleeft HS. Incorporation of fluorinated phenylalanine generates highly specific inhibitor of proteasome's chymotrypsin-like sites. Journal of Medicinal Chemistry. 53: 2319-23. PMID 20131905 DOI: 10.1021/jm9015685  1
2010 Wennekes T, Meijer AJ, Groen AK, Boot RG, Groener JE, van Eijk M, Ottenhoff R, Bijl N, Ghauharali K, Song H, O'Shea TJ, Liu H, Yew N, Copeland D, van den Berg RJ, ... van der Marel GA, et al. Dual-action lipophilic iminosugar improves glycemic control in obese rodents by reduction of visceral glycosphingolipids and buffering of carbohydrate assimilation. Journal of Medicinal Chemistry. 53: 689-98. PMID 20000679 DOI: 10.1021/jm901281m  1
2010 Kapoerchan VV, Wiesner M, Hillaert U, Drijfhout JW, Overhand M, Alard P, van der Marel GA, Overkleeft HS, Koning F. Design, synthesis and evaluation of high-affinity binders for the celiac disease associated HLA-DQ2 molecule. Molecular Immunology. 47: 1091-7. PMID 19962195 DOI: 10.1016/j.molimm.2009.10.036  1
2010 Ali A, Van Den Berg RJBHN, Overkleeft HS, Van Der Marel GA, Codée JDC. The methylsulfonylethoxymethyl (Msem) as a hydroxyl protecting group in oligosaccharide synthesis Tetrahedron. 66: 6121-6132. DOI: 10.1016/j.tet.2010.06.007  1
2010 Nuzzolo M, Grabulosa A, Slawin AMZ, Meeuwenoord NJ, Van Der Marel GA, Kamer PCJ. Functionalization of mono- and oligonucleotides with phosphane ligands by amide bond formation European Journal of Organic Chemistry. 3229-3236. DOI: 10.1002/ejoc.201000125  1
2010 Dinkelaar J, Duivenvoorden BA, Wennekes T, Overkleeft HS, Boot RG, Aerts JMFG, Codée JDC, Van Der Marel GA. A preparative synthesis of human chitinase fluorogenic substrate (4' -deoxychitobiosyl)-4-methylumbelliferone European Journal of Organic Chemistry. 2565-2570. DOI: 10.1002/ejoc.201000080  1
2010 Geurink PP, Klein T, Prèly L, Paal K, Leeuwenburgh MA, Van Der Marel GA, Kauffman HF, Overkleeft HS, Bischoff R. Design of peptide hydroxamate-based photoreactive activity-based probes of zinc-dependent metalloproteases European Journal of Organic Chemistry. 2100-2112. DOI: 10.1002/ejoc.200901385  1
2010 Wennekes T, Van Den Berg RJBHN, Boltje TJ, Donker-Koopman WE, Kuijper B, Van Der Marel GA, Strijland A, Verhagen CP, Aerts JMFG, Overkleeft HS. Synthesis and evaluation of lipophilic Aza-C-glycosides as inhibitors of glucosylceramide metabolism European Journal of Organic Chemistry. 1258-1283. DOI: 10.1002/ejoc.200901208  1
2010 Oualid FE, van der Marel GA, Overhand M. Inhibitors of protein: Geranylgeranyl transferases Frontiers in Medicinal Chemistry. 5: 167-233.  1
2009 Bonger KM, Hoogendoorn S, van Koppen CJ, Timmers CM, Overkleeft HS, van der Marel GA. Synthesis and pharmacological evaluation of dimeric follicle-stimulating hormone receptor antagonists. Chemmedchem. 4: 2098-102. PMID 19902448 DOI: 10.1002/cmdc.200900344  1
2009 Knijnenburg AD, Spalburg E, de Neeling AJ, Mars-Groenendijk RH, Noort D, Grotenbreg GM, van der Marel GA, Overkleeft HS, Overhand M. Ring-extended derivatives of gramicidin S with furanoid sugar amino acids in the turn region have enhanced antimicrobial activity. Chemmedchem. 4: 1976-9. PMID 19862783 DOI: 10.1002/cmdc.200900379  1
2009 Wennekes T, van den Berg RJ, Boot RG, van der Marel GA, Overkleeft HS, Aerts JM. Glycosphingolipids--nature, function, and pharmacological modulation. Angewandte Chemie (International Ed. in English). 48: 8848-69. PMID 19862781 DOI: 10.1002/anie.200902620  1
2009 Risseeuw MD, van den Berg RJ, Donker-Koopman WE, van der Marel GA, Aerts JM, Overhand M, Overkleeft HS. Synthesis and evaluation of D-gluco-pyranocyclopropyl amines as potential glucosidase inhibitors. Bioorganic & Medicinal Chemistry Letters. 19: 6600-3. PMID 19853441 DOI: 10.1016/j.bmcl.2009.10.022  1
2009 Tuin AW, Grotenbreg GM, Spalburg E, de Neeling AJ, Mars-Groenendijk RH, van der Marel GA, Noort D, Overkleeft HS, Overhand M. Structural and biological evaluation of some loloatin C analogues. Bioorganic & Medicinal Chemistry. 17: 6233-40. PMID 19679485 DOI: 10.1016/j.bmc.2009.07.049  1
2009 van der Knaap M, Engels E, Busscher HJ, Otero JM, Llamas-Saiz AL, van Raaij MJ, Mars-Groenendijk RH, Noort D, van der Marel GA, Overkleeft HS, Overhand M. Synthesis and biological evaluation of asymmetric gramicidin S analogues containing modified D-phenylalanine residues. Bioorganic & Medicinal Chemistry. 17: 6318-28. PMID 19674904 DOI: 10.1016/j.bmc.2009.07.042  1
2009 Walvoort MT, Lodder G, Mazurek J, Overkleeft HS, Codée JD, van der Marel GA. Equatorial anomeric triflates from mannuronic acid esters. Journal of the American Chemical Society. 131: 12080-1. PMID 19663422 DOI: 10.1021/ja905008p  1
2009 Witte MD, Florea BI, Verdoes M, Adeyanju O, Van Der Marel GA, Overkleeft HS. O-GlcNAc peptide epoxyketones are recognized by mammalian proteasomes Journal of the American Chemical Society. 131: 12064-12065. PMID 19658393 DOI: 10.1021/ja901231w  1
2009 Dinkelaar J, de Jong AR, van Meer R, Somers M, Lodder G, Overkleeft HS, Codée JD, van der Marel GA. Stereodirecting effect of the pyranosyl C-5 substituent in glycosylation reactions. The Journal of Organic Chemistry. 74: 4982-91. PMID 19489535 DOI: 10.1021/jo900662v  1
2009 Bonger KM, van den Berg RJ, Knijnenburg AD, Heitman LH, van Koppen CJ, Timmers CM, Overkleeft HS, van der Marel GA. Discovery of selective luteinizing hormone receptor agonists using the bivalent ligand method. Chemmedchem. 4: 1189-95. PMID 19475639 DOI: 10.1002/cmdc.200900058  1
2009 Dinkelaar J, Gold H, Overkleeft HS, Codée JD, van der Marel GA. Synthesis of hyaluronic acid oligomers using chemoselective and one-pot strategies. The Journal of Organic Chemistry. 74: 4208-16. PMID 19402694 DOI: 10.1021/jo9003713  1
2009 Weterings JJ, Khan S, Drijfhout JW, Ossendorp F, Overkleeft HS, van der Marel GA, Filippov DV. Synthesis of modified and hybrid protein derived biopolymers. Advances in Experimental Medicine and Biology. 611: 141-2. PMID 19400130 DOI: 10.1007/978-0-387-73657-0_63  1
2009 Weterings JJ, Khan S, van der Heden van Noort GJ, Melief CJ, Overkleeft HS, van der Burg SH, Ossendorp F, van der Marel GA, Filippov DV. 2-Azidoalkoxy-7-hydro-8-oxoadenine derivatives as TLR7 agonists inducing dendritic cell maturation. Bioorganic & Medicinal Chemistry Letters. 19: 2249-51. PMID 19299126 DOI: 10.1016/j.bmcl.2009.02.095  1
2009 Tuin AW, Mol MA, van den Berg RM, Fidder A, van der Marel GA, Overkleeft HS, Noort D. Activity-Based Protein Profiling Reveals Broad Reactivity of the Nerve Agent Sarin. Chemical Research in Toxicology. 22: 683-9. PMID 19226147 DOI: 10.1021/tx8004218  1
2009 Hillaert U, Verdoes M, Florea BI, Saragliadis A, Saragliadis A, Habets KL, Kuiper J, Van Calenbergh S, Ossendorp F, van der Marel GA, Driessen C, Overkleeft HS. Receptor-mediated targeting of cathepsins in professional antigen presenting cells. Angewandte Chemie (International Ed. in English). 48: 1629-32. PMID 19156780 DOI: 10.1002/anie.200805529  1
2009 Witte MD, Horst D, Wiertz EJ, van der Marel GA, Overkleeft HS. Synthesis and biological evaluation of a chitobiose-based peptide N-glycanase inhibitor library. The Journal of Organic Chemistry. 74: 605-16. PMID 19072094 DOI: 10.1021/jo801906s  1
2009 Codée JD, van den Bos LJ, de Jong AR, Dinkelaar J, Lodder G, Overkleeft HS, van der Marel GA. The stereodirecting effect of the glycosyl C5-carboxylate ester: stereoselective synthesis of beta-mannuronic acid alginates. The Journal of Organic Chemistry. 74: 38-47. PMID 19035740 DOI: 10.1021/jo8020192  1
2009 Ali A, van den Berg RJBHN, Overkleeft HS, Filippov DV, van der Marel GA, Codée JDC. Methylsulfonylethoxycarbonyl (Msc) and fluorous propylsulfonylethoxycarbonyl (FPsc) as hydroxy-protecting groups in carbohydrate chemistry Tetrahedron Letters. 50: 2185-2188. DOI: 10.1016/j.tetlet.2009.02.146  1
2009 Risseeuw MDP, van der Marel GA, Overkleeft HS, Overhand M. Pyranocyclopropanyl sugar amino acids, a new class of constrained (di)peptide isosteres Tetrahedron Asymmetry. 20: 945-951. DOI: 10.1016/j.tetasy.2009.03.009  1
2009 Wennekes T, van den Berg RJBHN, Bonger KM, Donker-Koopman WE, Ghisaidoobe A, van der Marel GA, Strijland A, Aerts JMFG, Overkleeft HS. Synthesis and evaluation of dimeric lipophilic iminosugars as inhibitors of glucosylceramide metabolism Tetrahedron Asymmetry. 20: 836-846. DOI: 10.1016/j.tetasy.2009.02.043  1
2009 Hogendorf WFJ, Verhagen CP, Malta E, Goosen N, Overkleeft HS, Filippov DV, Van der Marel GA. The synthesis of a menthol derivative of 2-aminopurine as a fluorescent DNA lesion Tetrahedron. 65: 10430-10435. DOI: 10.1016/j.tet.2009.10.023  1
2009 Codée JDC, de Jong AR, Dinkelaar J, Overkleeft HS, van der Marel GA. Stereoselectivity of glycosylations of conformationally restricted mannuronate esters Tetrahedron. 65: 3780-3788. DOI: 10.1016/j.tet.2009.02.067  1
2009 Tuin AW, Palachanis DK, Buizert A, Grotenbreg GM, Spalburg E, De Neeling AJ, Mars-Groenendijk RH, Noort D, Van Der Marel GA, Overkleeft HS, Overhand M. Synthesis and biological evaluation of novel gramicidin s analogues European Journal of Organic Chemistry. 4231-4241. DOI: 10.1002/ejoc.200900460  1
2009 Verdoes M, Florea BI, Van Der Marel GA, Overkleeft HS. Chemical tools to study the proteasome European Journal of Organic Chemistry. 3301-3313. DOI: 10.1002/ejoc.200900075  1
2008 Gold H, Van Delft P, Meeuwenoord N, Codée JDC, Filippov DV, Eggink G, Overkleeft HS, Van Der Marel GA. Synthesis of sugar nucleotides by application of phosphoramidites Journal of Organic Chemistry. 73: 9458-9460. PMID 18991380 DOI: 10.1021/jo802021t  1
2008 Abello N, Geurink PP, van der Toorn M, van Oosterhout AJ, Lugtenburg J, van der Marel GA, Kerstjens HA, Postma DS, Overkleeft HS, Bischoff R. Poly(ethylene glycol)-based stable isotope labeling reagents for the quantitative analysis of low molecular weight metabolites by LC-MS. Analytical Chemistry. 80: 9171-80. PMID 18954088 DOI: 10.1021/ac801215c  1
2008 van der Heden van Noort GJ, Verhagen CP, van der Horst MG, Overkleeft HS, van der Marel GA, Filippov DV. A versatile one-pot procedure to phosphate monoesters and pyrophosphates using di(p-methoxybenzyl)-N,N-diisopropylphosphoramidite. Organic Letters. 10: 4461-4. PMID 18800840 DOI: 10.1021/ol801608j  1
2008 Dinkelaar J, van den Bos LJ, Hogendorf WF, Lodder G, Overkleeft HS, Codée JD, van der Marel GA. Stereoselective synthesis of L-guluronic acid alginates. Chemistry (Weinheim An Der Bergstrasse, Germany). 14: 9400-11. PMID 18770512 DOI: 10.1002/chem.200800960  1
2008 Malta E, Verhagen CP, Moolenaar GF, Filippov DV, van der Marel GA, Goosen N. Functions of base flipping in E. coli nucleotide excision repair Dna Repair. 7: 1647-1658. PMID 18638572 DOI: 10.1016/j.dnarep.2008.06.011  1
2008 Verdoes M, Florea BI, Hillaert U, Willems LI, van der Linden WA, Sae-Heng M, Filippov DV, Kisselev AF, van der Marel GA, Overkleeft HS. Azido-BODIPY acid reveals quantitative Staudinger-Bertozzi ligation in two-step activity-based proteasome profiling. Chembiochem : a European Journal of Chemical Biology. 9: 1735-8. PMID 18600815 DOI: 10.1002/cbic.200800231  1
2008 Bonger KM, van den Berg RJ, Knijnenburg AD, Heitman LH, Ijzerman AP, Oosterom J, Timmers CM, Overkleeft HS, van der Marel GA. Synthesis and evaluation of homodimeric GnRHR antagonists having a rigid bis-propargylated benzene core. Bioorganic & Medicinal Chemistry. 16: 3744-58. PMID 18282756 DOI: 10.1016/j.bmc.2008.01.054  1
2008 Jawalekar AM, Meeuwenoord N, Cremers JS, Overkleeft HS, van der Marel GA, Rutjes FP, van Delft FL. Conjugation of nucleosides and oligonucleotides by [3+2] cycloaddition. The Journal of Organic Chemistry. 73: 287-90. PMID 18052191 DOI: 10.1021/jo702023s  1
2008 Kapoerchan VV, Wiesner M, Overhand M, van der Marel GA, Koning F, Overkleeft HS. Design of azidoproline containing gluten peptides to suppress CD4+ T-cell responses associated with celiac disease. Bioorganic & Medicinal Chemistry. 16: 2053-62. PMID 18037302 DOI: 10.1016/j.bmc.2007.10.091  1
2008 Wennekes T, Lang B, Leeman M, Van Der Marel GA, Smits E, Weber M, Van Wiltenburg J, Wolberg M, Aerts JMFG, Overkleeft HS. Large-scale synthesis of the glucosylceramide synthase inhibitor N-[5-(adamantan-1-yl-methoxy)-pentyl]-1-deoxynojirimycin Organic Process Research and Development. 12: 414-423. DOI: 10.1021/op700295x  1
2008 Ghisaidoobe ABT, de Koning MC, Duynstee HI, Ten Kortenaar PBW, Overkleeft HS, Filippov DV, van der Marel GA. A two-step sulfurization for efficient solution-phase synthesis of phosphorothioate oligonucleotides Tetrahedron Letters. 49: 3129-3132. DOI: 10.1016/j.tetlet.2008.03.025  1
2008 Bonger KM, Wennekes T, Filippov DV, Lodder G, Van Der Marel GA, Overkleeft HS. The effect of Lewis acids on the stereochemistry in the Ugi three-component reaction with D-lyxo-pyrroline European Journal of Organic Chemistry. 3678-3688. DOI: 10.1002/ejoc.200800340  1
2007 Witte MD, Descals CV, de Lavoir SV, Florea BI, van der Marel GA, Overkleeft HS. Bodipy-VAD-Fmk, a useful tool to study yeast peptide N-glycanase activity. Organic & Biomolecular Chemistry. 5: 3690-7. PMID 17971999 DOI: 10.1039/b711531h  1
2007 Verdoes M, Hillaert U, Florea BI, Sae-Heng M, Risseeuw MD, Filippov DV, van der Marel GA, Overkleeft HS. Acetylene functionalized BODIPY dyes and their application in the synthesis of activity based proteasome probes. Bioorganic & Medicinal Chemistry Letters. 17: 6169-71. PMID 17888658 DOI: 10.1016/j.bmcl.2007.09.025  1
2007 Risseeuw MD, Mazurek J, van Langenvelde A, van der Marel GA, Overkleeft HS, Overhand M. Synthesis of alkylated sugar amino acids: conformationally restricted L-Xaa-L-Ser/Thr mimics. Organic & Biomolecular Chemistry. 5: 2311-4. PMID 17609763 DOI: 10.1039/b705750d  1
2007 Dinkelaar J, Codée JD, van den Bos LJ, Overkleeft HS, van der Marel GA. Synthesis of hyaluronic acid oligomers using Ph2SO/Tf2O-mediated glycosylations. The Journal of Organic Chemistry. 72: 5737-42. PMID 17585821 DOI: 10.1021/jo070704s  1
2007 Bonger KM, van den Berg RJ, Heitman LH, IJzerman AP, Oosterom J, Timmers CM, Overkleeft HS, van der Marel GA. Synthesis and evaluation of homo-bivalent GnRHR ligands. Bioorganic & Medicinal Chemistry. 15: 4841-56. PMID 17517510 DOI: 10.1016/j.bmc.2007.04.065  1
2007 Verdoes M, Florea BI, Van Der Linden WA, Renou D, Van Den Nieuwendijk AMCH, Van Der Marel GA, Overkleeft HS. Mixing of peptides and electrophilic traps gives rise to potent, broad-spectrum proteasome inhibitors Organic and Biomolecular Chemistry. 5: 1416-1426. PMID 17464411 DOI: 10.1039/b702268a  1
2007 Khan S, Bijker MS, Weterings JJ, Tanke HJ, Adema GJ, van Hall T, Drijfhout JW, Melief CJ, Overkleeft HS, van der Marel GA, Filippov DV, van der Burg SH, Ossendorp F. Distinct uptake mechanisms but similar intracellular processing of two different toll-like receptor ligand-peptide conjugates in dendritic cells. The Journal of Biological Chemistry. 282: 21145-59. PMID 17462991 DOI: 10.1074/jbc.M701705200  1
2007 van Swieten PF, Samuel E, Hernández RO, van den Nieuwendijk AM, Leeuwenburgh MA, van der Marel GA, Kessler BM, Overkleeft HS, Kisselev AF. A cell-permeable inhibitor and activity-based probe for the caspase-like activity of the proteasome. Bioorganic & Medicinal Chemistry Letters. 17: 3402-5. PMID 17442566 DOI: 10.1016/j.bmcl.2007.03.092  1
2007 Ropartz L, Meeuwenoord NJ, van der Marel GA, van Leeuwen PW, Slawin AM, Kamer PC. Phosphine containing oligonucleotides for the development of metallodeoxyribozymes. Chemical Communications (Cambridge, England). 1556-8. PMID 17406706 DOI: 10.1039/b617871e  1
2007 Bussink AP, Van Swieten PF, Ghauharali K, Scheij S, Van Eijk M, Wennekes T, Van Der Marel GA, Boot RG, Aerts JMFG, Overkleeft HS. N-Azidoacetylmannosamine-mediated chemical tagging of gangliosides Journal of Lipid Research. 48: 1417-1421. PMID 17392268 DOI: 10.1194/jlr.C700006-JLR200  1
2007 Wennekes T, van den Berg RJ, Donker W, van der Marel GA, Strijland A, Aerts JM, Overkleeft HS. Development of adamantan-1-yl-methoxy-functionalized 1-deoxynojirimycin derivatives as selective inhibitors of glucosylceramide metabolism in man. The Journal of Organic Chemistry. 72: 1088-97. PMID 17243712 DOI: 10.1021/jo061280p  1
2007 Litjens REJN, van den Bos LJ, Codée JDC, Overkleeft HS, van der Marel GA. The use of cyclic bifunctional protecting groups in oligosaccharide synthesis-an overview Carbohydrate Research. 342: 419-429. PMID 17007825 DOI: 10.1016/j.carres.2006.09.002  1
2007 Lastdrager B, Timmer MSM, Van Der Marel GA, Overkleeft HS, Overhand M. Transformation of glucose into a novel carbasugar amino acid dipeptide isostere Journal of Carbohydrate Chemistry. 26: 41-59. DOI: 10.1080/07328300701252623  1
2007 van den Bos LJ, Boltje TJ, Provoost T, Mazurek J, Overkleeft HS, van der Marel GA. A synthetic study towards the PSA1 tetrasaccharide repeating unit Tetrahedron Letters. 48: 2697-2700. DOI: 10.1016/j.tetlet.2007.02.067  1
2007 Van Den Bos LJ, Codée JDC, Litjens REJN, Dinkelaar J, Overkleeft HS, Van Der Marel GA. Uronic acids in oligosaccharide synthesis European Journal of Organic Chemistry. 3963-3976. DOI: 10.1002/ejoc.200700101  1
2007 Van Den Bos LJ, Duivenvoorden BA, De Koning MC, Filippov DV, Overkleeft HS, Van Der Marel GA. Study of the glycosidation properties of 1-thiomannosazidopyranosides and 1-thiomannosaziduronic acid esters European Journal of Organic Chemistry. 116-124. DOI: 10.1002/ejoc.200600759  1
2007 Van Der Marel GA, Van Den Bos LJ, Overkleeft HS, Litjens REJN, Codée JDC. Sequential glycosylation strategies: A focus on thioglycosides as donors and acceptors Acs Symposium Series. 960: 190-203.  1
2006 Kriek NMAJ, Meeuwenoord NJ, Van Den Elst H, Heus HA, Van Der Marel GA, Filippov DV. Chemical synthesis of picornaviral protein primers of RNA replication Organic and Biomolecular Chemistry. 4: 3576-3586. PMID 16990933 DOI: 10.1039/b608544j  1
2006 El Oualid F, Cohen LH, van der Marel GA, Overhand M. Inhibitors of protein: geranylgeranyl transferases. Current Medicinal Chemistry. 13: 2385-427. PMID 16918362 DOI: 10.2174/092986706777935078  1
2006 Grotenbreg GM, Buizert AE, Llamas-Saiz AL, Spalburg E, van Hooft PA, de Neeling AJ, Noort D, van Raaij MJ, van der Marel GA, Overkleeft HS, Overhand M. Beta-turn modified gramicidin S analogues containing arylated sugar amino acids display antimicrobial and hemolytic activity comparable to the natural product. Journal of the American Chemical Society. 128: 7559-65. PMID 16756311 DOI: 10.1021/ja0588510  1
2006 Yu H, Sliedregt-Bol K, Overkleeft H, Van Der Marel GA, Van Berkel TJC, Biessen EAL. Therapeutic potential of a synthetic peptide inhibitor of nuclear factor of activated T cells as antirestenotic agent Arteriosclerosis, Thrombosis, and Vascular Biology. 26: 1531-1537. PMID 16675727 DOI: 10.1161/01.ATV.0000225286.30710.af  1
2006 Tuin AW, Siegal G, van der Marel GA, Overkleeft HS, Filippov DV. Facile synthesis and application of uniformly 13C, 15N-labeled phosphotyrosine for ligand binding studies Bioorganic and Medicinal Chemistry Letters. 16: 3806-3808. PMID 16650988 DOI: 10.1016/j.bmcl.2006.04.021  1
2006 Leeuwenburgh MA, Geurink PP, Klein T, Kauffman HF, Van Der Marel GA, Bischoff R, Overkleeft HS. Solid-phase synthesis of succinylhydroxamate peptides: Functionalized matrix metalloproteinase inhibitors Organic Letters. 8: 1705-1708. PMID 16597146 DOI: 10.1021/ol060409e  1
2006 Dinkelaar J, Witte MD, van den Bos LJ, Overkleeft HS, van der Marel GA. NIS/TFA: a general method for hydrolyzing thioglycosides Carbohydrate Research. 341: 1723-1729. PMID 16584717 DOI: 10.1016/j.carres.2006.03.009  1
2006 Weterings JJ, Khan S, van der Heden GJ, Drijfhout JW, Melief CJM, Overkleeft HS, van der Burg SH, Ossendorp F, van der Marel GA, Filippov DV. Synthesis of 2-alkoxy-8-hydroxyadenylpeptides: Towards synthetic epitope-based vaccines Bioorganic and Medicinal Chemistry Letters. 16: 3258-3261. PMID 16581248 DOI: 10.1016/j.bmcl.2006.03.034  1
2006 van den Berg RJ, Boltje TJ, Verhagen CP, Litjens RE, van der Marel GA, Overkleeft HS. An efficient synthesis of the natural tetrahydrofuran pachastrissamine starting from D-ribo-phytosphingosine. The Journal of Organic Chemistry. 71: 836-9. PMID 16409007 DOI: 10.1021/jo0520240  1
2006 Comuzzi C, Cogoi S, Overhand M, Van der Marel GA, Overkleeft HS, Xodo LE. Synthesis and biological evaluation of new pentaphyrin macrocycles for photodynamic therapy. Journal of Medicinal Chemistry. 49: 196-204. PMID 16392804 DOI: 10.1021/jm050831l  1
2006 De Koning MC, Ghisaidoobe ABT, Duynstee HI, Ten Kortenaar PBW, Filippov DV, Van Der Marel GA. Simple and efficient solution-phase synthesis of oligonucleotides using extractive work-up Organic Process Research and Development. 10: 1238-1245. DOI: 10.1021/op060133q  1
2006 Van Den Bos LJ, Dinkelaar J, Overkleeft HS, Van Der Marel GA. Stereocontrolled synthesis of β-D-mannuronic acid esters: Synthesis of an alginate trisaccharide Journal of the American Chemical Society. 128: 13066-13067. DOI: 10.1021/ja064787q  1
2006 Filippov DV, Welters MJP, Valentijn ARPM, Melief CJM, van der Marel GA, van der Burg SH, Overkleeft HS, Drijfhout JW. Chemical synthesis of the HPV16 E7 protein Tetrahedron Letters. 47: 9349-9352. DOI: 10.1016/j.tetlet.2006.10.119  1
2006 De Koning MC, Petersen L, Weterings JJ, Overhand M, Van Der Marel GA, Filippov DV. Synthesis of thiol-modified peptide nucleic acids designed for post-assembly conjugation reactions Tetrahedron. 62: 3248-3258. DOI: 10.1016/j.tet.2006.01.065  1
2006 Bonger KM, Wennekes T, De Lavoir SVP, Esposito D, Van Den Berg RJBHN, Litjens REJN, Van Der Marel GA, Overkleeft HS. Transformation of carbohydrate derived 4-azidopentanals into highly functionalized pyrrolidines via a tandem Staudinger/aza-Wittig/Ugi multicomponent reaction Qsar and Combinatorial Science. 25: 491-503. DOI: 10.1002/qsar.200540198  1
2006 Risseeuw MDP, Grotenbreg GM, Witte MD, Tuin AW, Leeuwenburgh MA, Van Der Marel GA, Overkleeft HS, Overhand M. The synthesis of cis- and trans-fused bicyclic sugar amino acids European Journal of Organic Chemistry. 3877-3886. DOI: 10.1002/ejoc.200600228  1
2005 El Oualid F, van den Elst H, Leroy IM, Pieterman E, Cohen LH, Burm BE, Overkleeft HS, van der Marel GA, Overhand M. A combinatorial approach toward the generation of ambiphilic peptide-based inhibitors of protein:geranylgeranyl transferase-1. Journal of Combinatorial Chemistry. 7: 703-13. PMID 16153065 DOI: 10.1021/cc0500203  1
2005 van Zutphen S, Stone EA, van Rijt S, Robillard MS, van der Marel GA, Overkleeft HS, den Dulk H, Brouwer J, Reedijk J. Combinatorial discovery of new asymmetric cis platinum anticancer complexes is made possible with solid-phase synthetic methods. Journal of Inorganic Biochemistry. 99: 2032-8. PMID 16099049 DOI: 10.1016/j.jinorgbio.2005.06.033  1
2005 Voerman G, Cavalli S, van der Marel GA, Pfleiderer W, van Boom JH, Filippov DV. 1,3-Dimethyllumazine derivatives from Limnatis nilotica. Journal of Natural Products. 68: 938-41. PMID 15974624 DOI: 10.1021/np049617a  1
2005 van Zutphen S, Kraus M, Driessen C, van der Marel GA, Overkleeft HS, Reedijk J. Probing the potential of platinum(II) complexes for the inhibition of thiol-dependent enzymatic activity. Journal of Inorganic Biochemistry. 99: 1384-9. PMID 15869797 DOI: 10.1016/j.jinorgbio.2005.03.014  0.6
2005 Codée JD, Stubba B, Schiattarella M, Overkleeft HS, van Boeckel CA, van Boom JH, van der Marel GA. A modular strategy toward the synthesis of heparin-like oligosaccharides using monomeric building blocks in a sequential glycosylation strategy. Journal of the American Chemical Society. 127: 3767-73. PMID 15771511 DOI: 10.1021/ja045613g  1
2005 Grotenbreg GM, Witte MD, van Hoof PA, Spalburg E, Reiss P, Noort D, de Neeling AJ, Koert U, van der Marel GA, Overkleeft HS, Overhand M. Synthesis and biological evaluation of gramicidin S dimers. Organic & Biomolecular Chemistry. 3: 233-8. PMID 15717418 DOI: 10.1039/b414618b  1
2005 El Oualid F, Baktawar J, Leroy IM, van den Elst H, Cohen LH, van der Marel GA, Overkleeft HS, Overhand M. Synthesis and biological evaluation of lipophilic Ca(1)a(2)L analogues as potential bisubstrate inhibitors of protein:geranylgeranyl transferase-1. Bioorganic & Medicinal Chemistry. 13: 1463-75. PMID 15698762 DOI: 10.1016/j.bmc.2004.12.035  1
2005 Litjens REJN, Hoogerhout P, Filippov DV, Codée JDC, Van Den Bos LJ, Van Den Berg RJBHN, Overkleeft HS, Van Der Marel GA. Synthesis of an α-Gal epitope α-D-Galp-(1 → 3)β-D-Galp-(1 → 4)-β-D-Glcp NAc-lipid conjugate Journal of Carbohydrate Chemistry. 24: 755-769. DOI: 10.1080/07328300500308113  1
2005 Timmer MSM, Chumillas MV, Donker-Koopman WE, Aerts JMFG, Van Der Marel GA, Overkleeft HS, Van Boom JH. Selective cross-metathesis of C-allyl-glycosides Journal of Carbohydrate Chemistry. 24: 335-351. DOI: 10.1080/07328300500174887  1
2004 Grotenbreg GM, Christina AE, Buizert AE, van der Marel GA, Overkleeft HS, Overhand M. Synthesis and application of carbohydrate-derived morpholine amino acids. The Journal of Organic Chemistry. 69: 8331-9. PMID 15549804 DOI: 10.1021/jo048630x  1
2004 Welters MJ, Filippov DV, van den Eeden SJ, Franken KL, Nouta J, Valentijn AR, van der Marel GA, Overkleeft HS, Lipford G, Offringa R, Melief CJ, van Boom JH, van der Burg SH, Drijfhout JW. Chemically synthesized protein as tumour-specific vaccine: immunogenicity and efficacy of synthetic HPV16 E7 in the TC-1 mouse tumour model. Vaccine. 23: 305-11. PMID 15530672 DOI: 10.1016/j.vaccine.2004.06.008  1
2004 Grotenbreg GM, Kronemeijer M, Timmer MS, El Oualid F, van Well RM, Verdoes M, Spalburg E, van Hooft PA, de Neeling AJ, Noort D, van Boom JH, van der Marel GA, Overkleeft HS, Overhand M. A practical synthesis of gramicidin s and sugar amino Acid containing analogues. The Journal of Organic Chemistry. 69: 7851-9. PMID 15527261 DOI: 10.1021/jo0487449  1
2004 Raunkjaer M, El Oualid F, van der Marel GA, Overkleeft HS, Overhand M. Alkylated sugar amino acids: a new entry toward highly functionalized dipeptide isosters. Organic Letters. 6: 3167-70. PMID 15330614 DOI: 10.1021/ol048750r  1
2004 van den Berg RJ, Korevaar CG, Overkleeft HS, van der Marel GA, van Boom JH. Effective, high-yielding, and stereospecific total synthesis of D-erythro-(2R,3S)-sphingosine from D-ribo-(2S,3S,4R)-phytosphingosine. The Journal of Organic Chemistry. 69: 5699-704. PMID 15307742 DOI: 10.1021/jo049277y  1
2004 El Oualid F, Burm BE, Leroy IM, Cohen LH, van Boom JH, van den Elst H, Overkleeft HS, van der Marel GA, Overhand M. Design, synthesis, and evaluation of sugar amino acid based inhibitors of protein prenyl transferases PFT and PGGT-1. Journal of Medicinal Chemistry. 47: 3920-3. PMID 15267228 DOI: 10.1021/jm049927q  1
2004 Tromp RA, van Boom SS, Marco Timmers C, van Zutphen S, van der Marel GA, Overkleeft HS, van Boom JH, Reedijk J. The beta-glucuronyl-based prodrug strategy allows for its application on beta-glucuronyl-platinum conjugates. Bioorganic & Medicinal Chemistry Letters. 14: 4273-6. PMID 15261285 DOI: 10.1016/j.bmcl.2004.06.015  1
2004 van Roon AM, Pannu NS, de Vrind JP, van der Marel GA, van Boom JH, Hokke CH, Deelder AM, Abrahams JP. Structure of an anti-Lewis X Fab fragment in complex with its Lewis X antigen. Structure (London, England : 1993). 12: 1227-36. PMID 15242599 DOI: 10.1016/j.str.2004.05.008  1
2004 Verhelst SH, Michiels PJ, van der Marel GA, van Boeckel CA, van Boom JH. Surface plasmon resonance evaluation of various aminoglycoside-RNA hairpin interactions reveals low degree of selectivity. Chembiochem : a European Journal of Chemical Biology. 5: 937-42. PMID 15239050 DOI: 10.1002/cbic.200300819  1
2004 van den Bos LJ, Codée JD, van der Toorn JC, Boltje TJ, van Boom JH, Overkleeft HS, van der Marel GA. Thioglycuronides: synthesis and application in the assembly of acidic oligosaccharides. Organic Letters. 6: 2165-8. PMID 15200311 DOI: 10.1021/ol049380+  1
2004 van Swieten PF, Maehr R, van den Nieuwendijk AM, Kessler BM, Reich M, Wong CS, Kalbacher H, Leeuwenburgh MA, Driessen C, van der Marel GA, Ploegh HL, Overkleeft HS. Development of an isotope-coded activity-based probe for the quantitative profiling of cysteine proteases. Bioorganic & Medicinal Chemistry Letters. 14: 3131-4. PMID 15149659 DOI: 10.1016/j.bmcl.2004.04.046  0.6
2004 Petersen L, de Koning MC, van Kuik-Romeijn P, Weterings J, Pol CJ, Platenburg G, Overhand M, van der Marel GA, van Boom JH. Synthesis and in vitro evaluation of PNA-peptide-DETA conjugates as potential cell penetrating artificial ribonucleases. Bioconjugate Chemistry. 15: 576-82. PMID 15149186 DOI: 10.1021/bc034219p  1
2004 van Hooft PA, El Oualid F, Overkleeft HS, van der Marel GA, van Boom JH, Leeuwenburgh MA. Synthesis and elaboration of functionalised carbohydrate-derived spiroketals. Organic & Biomolecular Chemistry. 2: 1395-403. PMID 15105932 DOI: 10.1039/b401699h  1
2004 Grotenbreg GM, Timmer MS, Llamas-Saiz AL, Verdoes M, van der Marel GA, van Raaij MJ, Overkleeft HS, Overhand M. An unusual reverse turn structure adopted by a furanoid sugar amino acid incorporated in gramicidin S. Journal of the American Chemical Society. 126: 3444-6. PMID 15025470 DOI: 10.1021/ja0397254  1
2003 van den Bos LJ, Codée JD, van Boom JH, Overkleeft HS, van der Marel GA. A novel strategy towards the synthesis of orthogonally functionalised 4-aminoglycosides. Organic & Biomolecular Chemistry. 1: 4160-5. PMID 14685319 DOI: 10.1039/b309823k  1
2003 Verhelst SH, Paez Martinez B, Timmer MS, Lodder G, van der Marel GA, Overkleeft HS, van Boom JH. A short route toward chiral, polyhydroxylated indolizidines and quinolizidines. The Journal of Organic Chemistry. 68: 9598-603. PMID 14656083 DOI: 10.1021/jo0350662  1
2003 Timmer MS, Verdoes M, Sliedregt LA, van der Marel GA, van Boom JH, Overkleeft HS. The use of a mannitol-derived fused oxacycle as a combinatorial scaffold. The Journal of Organic Chemistry. 68: 9406-11. PMID 14629165 DOI: 10.1021/jo0349429  1
2003 van Rossenberg SM, Sliedregt-Bol KM, Prince P, van Berkel TJ, van Boom JH, van der Marel GA, Biessen EA. A targeted peptide nucleic acid to down-regulate mouse microsomal triglyceride transfer protein expression in hepatocytes. Bioconjugate Chemistry. 14: 1077-82. PMID 14624620 DOI: 10.1021/bc0340417  1
2003 Robillard MS, Bacac M, van den Elst H, Flamigni A, van der Marel GA, van Boom JH, Reedijk J. Automated parallel solid-phase synthesis and anticancer screening of a library of peptide-tethered platinum(II) complexes. Journal of Combinatorial Chemistry. 5: 821-5. PMID 14606811 DOI: 10.1021/cc030011z  1
2003 Aguilera B, Ghauharali-van der Vlugt K, Helmond MT, Out JM, Donker-Koopman WE, Groener JE, Boot RG, Renkema GH, van der Marel GA, van Boom JH, Overkleeft HS, Aerts JM. Transglycosidase activity of chitotriosidase: improved enzymatic assay for the human macrophage chitinase. The Journal of Biological Chemistry. 278: 40911-6. PMID 12890686 DOI: 10.1074/jbc.M301804200  1
2003 Robillard MS, Davies NP, van der Marel GA, van Boom JH, Reedijk J, Murray V. The interaction of peptide-tethered platinum(II) complexes with DNA. Journal of Inorganic Biochemistry. 96: 331-8. PMID 12888268  1
2003 van Rossenberg SM, Sliedregt-Bol KM, Koning G, van den Elst H, van Berkel TJ, van Boom JH, van der Marel GA, Biessen EA. Improvement of hepatocyte-specific gene expression by a targeted colchicine prodrug. Chembiochem : a European Journal of Chemical Biology. 4: 633-9. PMID 12851933 DOI: 10.1002/cbic.200300582  1
2003 Grotenbreg GM, Spalburg E, de Neeling AJ, van der Marel GA, Overkleeft HS, van Boom JH, Overhand M. Synthesis and biological evaluation of novel turn-modified gramicidin S analogues. Bioorganic & Medicinal Chemistry. 11: 2835-41. PMID 12788356  1
2003 Codée JD, van den Bos LJ, Litjens RE, Overkleeft HS, van Boom JH, van der Marel GA. Sequential one-pot glycosylations using 1-hydroxyl and 1-thiodonors. Organic Letters. 5: 1947-50. PMID 12762693 DOI: 10.1021/ol034528v  1
2003 de Visser PC, Kriek NM, van Hooft PA, Van Schepdael A, Filippov DV, van der Marel GA, Overkleeft HS, van Boom JH, Noort D. Solid-phase synthesis of polymyxin B1 and analogues via a safety-catch approach. The Journal of Peptide Research : Official Journal of the American Peptide Society. 61: 298-306. PMID 12753377 DOI: 10.1034/j.1399-3011.2003.00061.x  1
2003 Codée JD, Litjens RE, den Heeten R, Overkleeft HS, van Boom JH, van der Marel GA. Ph2SO/Tf2O: a powerful promotor system in chemoselective glycosylations using thioglycosides. Organic Letters. 5: 1519-22. PMID 12713313 DOI: 10.1021/ol034312t  1
2003 Heetebrij RJ, de Kort M, Meeuwenoord NJ, den Dulk H, van der Marel GA, van Boom JH, Reedijk J. A versatile approach towards regioselective platinated DNA sequences. Chemistry (Weinheim An Der Bergstrasse, Germany). 9: 1823-7. PMID 12698440 DOI: 10.1002/chem.200390209  1
2003 van Zutphen S, Robillard MS, van der Marel GA, Overkleeft HS, den Dulk H, Brouwer J, Reedijk J. Extending solid-phase methods in inorganic synthesis: the first dinuclear platinum complex synthesised via the solid phase. Chemical Communications (Cambridge, England). 634-5. PMID 12669861  1
2003 van Well RM, Overkleeft HS, van der Marel GA, Bruss D, Thibault G, de Groot PG, van Boom JH, Overhand M. Solid-phase synthesis of cyclic RGD-furanoid sugar amino acid peptides as integrin inhibitors. Bioorganic & Medicinal Chemistry Letters. 13: 331-4. PMID 12565923  1
2002 Schmidt KS, Boudvillain M, Schwartz A, van der Marel GA, van Boom JH, Reedijk J, Lippert B. Monofunctionally trans-diammine platinum(II)-modified peptide nucleic acid oligomers: a new generation of potential antisense drugs. Chemistry (Weinheim An Der Bergstrasse, Germany). 8: 5566-70. PMID 12458496 DOI: 10.1002/1521-3765(20021216)8:24<5566::AID-CHEM5566>3.0.CO;2-#  1
2002 Van Rossenberg SM, Sliedregt-Bol KM, Meeuwenoord NJ, Van Berkel TJ, Van Boom JH, Van Der Marel GA, Biessen EA. Targeted lysosome disruptive elements for improvement of parenchymal liver cell-specific gene delivery. The Journal of Biological Chemistry. 277: 45803-10. PMID 12237290 DOI: 10.1074/jbc.M203510200  1
2002 Rapozzi V, Burm BE, Cogoi S, van der Marel GA, van Boom JH, Quadrifoglio F, Xodo LE. Antiproliferative effect in chronic myeloid leukaemia cells by antisense peptide nucleic acids. Nucleic Acids Research. 30: 3712-21. PMID 12202756  1
2002 Verhoeven EE, van Kesteren M, Turner JJ, van der Marel GA, van Boom JH, Moolenaar GF, Goosen N. The C-terminal region of Escherichia coli UvrC contributes to the flexibility of the UvrABC nucleotide excision repair system. Nucleic Acids Research. 30: 2492-500. PMID 12034838  1
2000 Verheijen JC, Chen L, Bayly SF, Torrence PF, van der Marel GA, van Boom JH. Synthesis and RNAse L binding and activation of a 2-5A-(5')-DNA-(3')-PNA chimera, a novel potential antisense molecule. Nucleosides, Nucleotides & Nucleic Acids. 19: 1821-30. PMID 11200276 DOI: 10.1080/15257770008045463  1
2000 Robillard MS, Valentijn AR, Meeuwenoord NJ, van Der Marel GA, van Boom JH, Reedijk J. The First Solid-Phase Synthesis of a Peptide-Tethered Platinum(II) Complex This research was supported by the Council for Chemical Sciences of The Netherlands Organization for Scientific Research (CW-NWO) and by The Netherlands Foundation for Technical Sciences (STW). Support and sponsorship by COST Action D8/00097 (biocoordination chemistry) is kindly acknowledged. The authors thank Johnson & Matthey (Reading, UK) for their generous loan of K(2)PtCl(4). Angewandte Chemie (International Ed. in English). 39: 3096-3099. PMID 11028044 DOI: 10.1002/1521-3773(20000901)39:17<3096::AID-ANIE3096>3.0.CO;2-D  1
2000 de Kort M, Regenbogen AD, Valentijn AR, Challiss RA, Iwata Y, Miyamoto S, van der Marel GA, van Boom JH. Spirophostins: conformationally restricted analogues of adenophostin A. Chemistry (Weinheim An Der Bergstrasse, Germany). 6: 2696-704. PMID 10985718 DOI: 10.1002/1521-3765(20000804)6:15<2696::AID-CHEM2696>3.0.CO;2-Y  1
2000 de Kort M, Correa V, Valentijn AR, van der Marel GA, Potter BV, Taylor CW, van Boom JH. Synthesis of potent agonists of the D-myo-inositol 1,4, 5-trisphosphate receptor based on clustered disaccharide polyphosphate analogues of adenophostin A. Journal of Medicinal Chemistry. 43: 3295-303. PMID 10966748 DOI: 10.1021/jm000957c  1
2000 Verheijen JC, van Roon AM, Meeuwenoord NJ, Stuivenberg HR, Bayly SF, Chen L, van der Marel GA, Torrence PF, van Boom JH. Incorporation of a 4-hydroxy-N-acetylprolinol nucleotide analogue improves the 3'-exonuclease stability of 2'-5'-oligoadenylate-antisense conjugates. Bioorganic & Medicinal Chemistry Letters. 10: 801-4. PMID 10782690 DOI: 10.1016/S0960-894X(00)00100-1  1
2000 Moolenaar GF, Herron MF, Monaco V, van der Marel GA, van Boom JH, Visse R, Goosen N. The role of ATP binding and hydrolysis by UvrB during nucleotide excision repair. The Journal of Biological Chemistry. 275: 8044-50. PMID 10713125 DOI: 10.1074/jbc.275.11.8044  1
2000 Moolenaar GF, Monaco V, van der Marel GA, van Boom JH, Visse R, Goosen N. The effect of the DNA flanking the lesion on formation of the UvrB-DNA preincision complex. Mechanism for the UvrA-mediated loading of UvrB onto a DNA damaged site. The Journal of Biological Chemistry. 275: 8038-43. PMID 10713124 DOI: 10.1074/jbc.275.11.8038  1
2000 Schmidt KS, Filippov DV, Meeuwenoord NJ, van Der Marel GA, van Boom JH, Lippert B, Reedijk J. Solid-Phase Synthesis of a Monofunctional trans-a(2)Pt(II) Complex Tethered to a Single-Stranded Oligonucleotide. Angewandte Chemie (International Ed. in English). 39: 375-377. PMID 10649415 DOI: 10.1002/(SICI)1521-3773(20000117)39:2<375::AID-ANIE375>3.0.CO;2-M  1
2000 Verheijen JC, Deiman BA, Yeheskiely E, van Der Marel GA, van Boom JH. Efficient Hydrolysis of RNA by a PNA - Diethylenetriamine Adduct. Angewandte Chemie (International Ed. in English). 39: 369-372. PMID 10649413 DOI: 10.1002/(SICI)1521-3773(20000117)39:2<369::AID-ANIE369>3.0.CO;2-A  1
1999 Buijsman RC, Basten JE, Dreef-Tromp CM, van der Marel GA, van Boeckel CA, van Boom JH. Synthesis of heparin-like antithrombotics having perphosphorylated thrombin binding domains. Bioorganic & Medicinal Chemistry. 7: 1881-90. PMID 10530936 DOI: 10.1016/S0968-0896(99)00139-X  1
1999 Buijsman RC, Basten JE, van Dinther TG, van der Marel GA, van Boeckel CA, van Boom JH. Design and synthesis of a novel synthetic NAPAP-penta-saccharide conjugate displaying a dual antithrombotic action. Bioorganic & Medicinal Chemistry Letters. 9: 2013-8. PMID 10450972 DOI: 10.1016/S0960-894X(99)00320-0  1
1999 Verheijen JC, van der Marel GA, van Boom JH, Bayly SF, Player MR, Torrence PF. 2,5-oligoadenylate-peptide nucleic acids (2-5A-PNAs) activate RNase L. Bioorganic & Medicinal Chemistry. 7: 449-55. PMID 10220031 DOI: 10.1016/S0968-0896(98)00258-2  1
1997 Slijper M, Boelens R, Davis AL, Konings RN, van der Marel GA, van Boom JH, Kaptein R. Backbone and side chain dynamics of lac repressor headpiece (1-56) and its complex with DNA. Biochemistry. 36: 249-54. PMID 8993340 DOI: 10.1021/bi961670d  1
1996 van Delft FL, de Kort M, van Der Marel GA, van Boom JH. Use of a Novel alpha-Hydroxyethylating Reagent in the Stereoselective Synthesis of Lincosamine. The Journal of Organic Chemistry. 61: 1883-1885. PMID 11667071  1
1996 Zegelaar-Jaarsveld K, Smits SA, van der Marel GA, van Boom JH. Synthesis of a pentasaccharide corresponding to the repeating unit of the exopolysaccharide from Cryptococcus neoformans serovar D. Bioorganic & Medicinal Chemistry. 4: 1819-32. PMID 9007267 DOI: 10.1016/S0968-0896(96)00164-2  1
1996 van Boom SS, Yang D, Reedijk J, van der Marel GA, Wang AH. Structural effect of intra-strand cisplatin-crosslink on palindromic DNA sequences. Journal of Biomolecular Structure & Dynamics. 13: 989-98. PMID 8832381 DOI: 10.1080/07391102.1996.10508913  0.36
1993 Zuurmond HM, Veeneman GH, van der Marel GA, van Boom JH. Iodonium ion-assisted synthesis of a haptenic tetrasaccharide fragment corresponding to the inner cell-wall glycopeptidolipid of Mycobacterium avium serotype 4. Carbohydrate Research. 241: 153-64. PMID 8472251  1
1992 Kellenbach ER, Remerowski ML, Eib D, Boelens R, van der Marel GA, van den Elst H, van Boom JH, Kaptein R. Synthesis of isotope labeled oligonucleotides and their use in an NMR study of a protein-DNA complex. Nucleic Acids Research. 20: 653-7. PMID 1542561  1
1992 Dreef-Tromp CM, van der Maarel JC, van den Elst H, van der Marel GA, van Boom JH. Solid-phase synthesis of the nucleopeptide fragment H-Asp-Ser[pAAAGTAAGCC]-Glu-OH from the nucleoprotein of Bacillus subtilis phage phi 29. Nucleic Acids Research. 20: 4015-20. PMID 1508685  1
1992 Dreef-Tromp CM, van den Elst H, van den Boogaart JE, van der Marel GA, van Boom JH. Solid-phase synthesis of an RNA nucleopeptide fragment from the nucleoprotein of poliovirus. Nucleic Acids Research. 20: 2435-9. PMID 1317954  1
1991 Roelen HC, Bijsterbosch MK, Bakkeren HF, van Berkel TJ, Kempen HJ, Buytenhek M, van der Marel GA, van Boom JH. Water-soluble cholesteryl-containing phosphorothioate monogalactosides: synthesis, properties, and use in lowering blood cholesterol by directing plasma lipoproteins to the liver. Journal of Medicinal Chemistry. 34: 1036-42. PMID 2002447 DOI: 10.1021/jm00107a024  1
1991 Roelen HC, Saris CP, Brugghe HF, van den Elst H, Westra JG, van der Marel GA, van Boom JH. Solid-phase synthesis of DNA fragments containing the modified base 7-hydro-8-oxo-2'-deoxyguanosine. Nucleic Acids Research. 19: 4361-9. PMID 1886763 DOI: 10.1093/nar/19.16.4361  1
1991 Koning TM, Boelens R, van der Marel GA, van Boom JH, Kaptein R. Structure determination of a DNA octamer in solution by NMR spectroscopy. Effect of fast local motions. Biochemistry. 30: 3787-97. PMID 1849738  1
1991 Remerowski ML, Kellenbach E, Boelens R, van der Marel GA, van Boom JH, Maler BA, Yamamoto KR, Kaptein R. 1H NMR studies of DNA recognition by the glucocorticoid receptor: complex of the DNA binding domain with a half-site response element. Biochemistry. 30: 11620-4. PMID 1751485  1
1990 Lamerichs RM, Boelens R, Van der Marel GA, Van Boom JH, Kaptein R. Assignment of the 1H-NMR spectrum of a lac repressor headpiece-operator complex in H2O and identification of NOEs. Consequences for protein-DNA interaction. European Journal of Biochemistry / Febs. 194: 629-37. PMID 2269288  1
1990 Pieters JM, de Vroom E, van der Marel GA, van Boom JH, Koning TM, Kaptein R, Altona C. Hairpin structures in DNA containing arabinofuranosylcytosine. A combination of nuclear magnetic resonance and molecular dynamics. Biochemistry. 29: 788-99. PMID 2159791  1
1990 Dreef-Tromp CM, van Dam EM, van den Elst H, van der Marel GA, van Boom JH. Solid-phase synthesis of H-Phe-Tyr-(pATAT)-NH2: a nucleopeptide fragment from the nucleoprotein of bacteriophage phi X174. Nucleic Acids Research. 18: 6491-5. PMID 2147473 DOI: 10.1093/nar/18.22.6491  1
1989 Pieters JM, de Vroom E, van der Marel GA, van Boom JH, Altona C. Conformational consequences of the incorporation of arabinofuranosylcytidine in DNA. An NMR study of the DNA fragments d(CGCTAGCG) and d(CGaCTAGCG) in solution. European Journal of Biochemistry / Febs. 184: 415-25. PMID 2792106  1
1989 Pieters JM, Mans RM, van den Elst H, van der Marel GA, van Boom JH, Altona C. Conformational and thermodynamic consequences of the introduction of a nick in duplexed DNA fragments: an NMR study augmented by biochemical experiments. Nucleic Acids Research. 17: 4551-65. PMID 2748334 DOI: 10.1093/nar/17.12.4551  1
1989 Lamerichs RM, Boelens R, van der Marel GA, van Boom JH, Kaptein R, Buck F, Fera B, Rüterjans H. H NMR study of a complex between the lac repressor headpiece and a 22 base pair symmetric lac operator. Biochemistry. 28: 2985-91. PMID 2742823  1
1989 Kuyl-Yeheskiely E, Dreef-Tromp CM, Geluk A, van der Marel GA, van Boom JH. Synthesis of the nucleopeptides H-Phe-Tyr(pGC)-NH2 and H-Phe-Ser(pGC)-Ala-OH via a phosphotriester approach. Nucleic Acids Research. 17: 2897-905. PMID 2726447 DOI: 10.1093/nar/17.8.2897  1
1989 Boons GJ, Overhand M, van der Marel GA, van Boom JH. Synthesis of a trisaccharide of the inner core region of Citrobacter PCM 187 lipopolysaccharide that contains L-glycero-alpha-D-manno-heptopyranosyl units. Carbohydrate Research. 192: C1-4. PMID 2611773 DOI: 10.1016/0008-6215(89)85198-5  1
1988 Roelen HC, de Vroom E, van der Marel GA, van Boom JH. Synthesis of nucleic acid methylphosphonothioates. Nucleic Acids Research. 16: 7633-45. PMID 3412896 DOI: 10.1093/nar/16.15.7633  1
1988 van den Hoogen YT, van Beuzekom AA, de Vroom E, van der Marel GA, van Boom JH, Altona C. Bulge-out structures in the single-stranded trimer AUA and in the duplex (CUGGUGCGG).(CCGCCCAG). A model-building and NMR study. Nucleic Acids Research. 16: 5013-30. PMID 3387215 DOI: 10.1093/nar/16.11.5013  1
1988 de Vroom E, Broxterman HJ, Sliedregt LA, van der Marel GA, van Boom JH. Synthesis of cyclic oligonucleotides by a modified phosphotriester approach. Nucleic Acids Research. 16: 4607-20. PMID 3380690 DOI: 10.1093/nar/16.10.4607  1
1988 van den Hoogen YT, van Beuzekom AA, van den Elst H, van der Marel GA, van Boom JH, Altona C. Extra thymidine stacks into the d(CTGGTGCGG).d(CCGCCCAG) duplex. An NMR and model-building study. Nucleic Acids Research. 16: 2971-86. PMID 3368313 DOI: 10.1093/nar/16.7.2971  1
1988 Kemmink J, Eker APM, van der Marel GA, van Boom JH, Kaptein R. Photoreactivation of the thymine dimer containing DNA octamer d(GCGT TGCG)·d(CGCAACGC) by the photoreactivating enzyme from Anacystis nidulans Journal of Photochemistry and Photobiology, B: Biology. 1: 323-328. PMID 3149667 DOI: 10.1016/1011-1344(88)85020-6  1
1988 van den Hoogen YT, Treurniet SJ, Roelen HC, de Vroom E, van der Marel GA, van Boom JH, Altona C. Conformational analysis of the tetranucleotides m6(2)A-m6(2)A-U-m6(2)A(m6(2)A = N6-dimethyladenosine) and U-m6(2)A-U-m6(2)A and of the hybrid dA-r(U-A). A one- and two-dimensional NMR study. European Journal of Biochemistry / Febs. 171: 155-62. PMID 3123229  1
1988 de Vroom E, Roelen HC, Saris CP, Budding TN, van der Marel GA, van Boom JH. Preparation of covalently linked DNA-RNA hybrids and arabinocytidine containing DNA fragments. Nucleic Acids Research. 16: 2987-3003. PMID 2453027 DOI: 10.1093/nar/16.7.2987  1
1988 van den Hoogen YT, Erkelens C, de Vroom E, van der Marel GA, van Boom JH, Altona C. Influence of uracil on the conformational behaviour of RNA oligonucleotides in solution. European Journal of Biochemistry / Febs. 173: 295-303. PMID 2452087  1
1987 de Vroom E, Fidder A, Saris CP, van der Marel GA, van Boom JH. Preparation of the individual diastereomers of adenylyl-(2'-5')-P-thioadenylyl-(2'-5')-adenosine and their 5'-phosphorylated derivatives. Nucleic Acids Research. 15: 9933-43. PMID 3697086 DOI: 10.1093/nar/15.23.9933  1
1987 Orbons LP, van der Marel GA, van Boom JH, Altona C. An NMR study of polymorphous behaviour of the mismatched DNA octamer d(m5C-G-m5C-G-A-G-m5C-G) in solution. The B-duplex and hairpin forms. European Journal of Biochemistry / Febs. 170: 225-39. PMID 3691520  0.72
1987 Kemmink J, Boelens R, Koning T, van der Marel GA, van Boom JH, Kaptein R. 1H NMR study of the exchangeable protons of the duplex d(GCGTTGCG).d(CGCAACGC) containing a thymine photodimer. Nucleic Acids Research. 15: 4645-53. PMID 3035498 DOI: 10.1093/nar/15.11.4645  1
1987 Kemmink J, Boelens R, Koning TM, Kaptein R, van der Marel GA, van Boom JH. Conformational changes in the oligonucleotide duplex d(GCGTTGCG) x d(CGCAACGC) induced by formation of a cis-syn thymine dimer. A two-dimensional NMR study. European Journal of Biochemistry / Febs. 162: 37-43. PMID 3028790  1
1987 Raap J, Dreef CE, van der Marel GA, van Boom JH, Hilbers CW. Synthesis and proton-NMR studies of oligonucleotides containing an apurinic (AP) site. Journal of Biomolecular Structure & Dynamics. 5: 219-47. PMID 2856028 DOI: 10.1080/07391102.1987.10506391  1
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