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K. Barry Sharpless - Publications

Affiliations: 
Massachusetts Institute of Technology, Cambridge, MA, United States 
 Scripps Research Institute, La Jolla, La Jolla, CA, United States 
Area:
Click chemistry
Website:
http://www.nobelprize.org/nobel_prizes/chemistry/laureates/2001/sharpless-bio.html
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437 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Brighty GJ, Botham RC, Li S, Nelson L, Mortenson DE, Li G, Morisseau C, Wang H, Hammock BD, Sharpless KB, Kelly JW. Using sulfuramidimidoyl fluorides that undergo sulfur(VI) fluoride exchange for inverse drug discovery. Nature Chemistry. PMID 32868886 DOI: 10.1038/s41557-020-0530-4  1
2020 Kitamura S, Zheng Q, Woehl JL, Solania A, Chen E, Dillon N, Hull MV, Kotaniguchi M, Cappiello JR, Kitamura S, Nizet V, Sharpless KB, Wolan DW. SuFEx-enabled high-throughput medicinal chemistry. Journal of the American Chemical Society. PMID 32479075 DOI: 10.1021/jacs.9b13652  1
2020 Lauwaet T, Miyamoto Y, Ihara S, Le C, Kalisiak J, Korthals K, Ghassemian M, Smith DK, Sharpless KB, Fokin VV, Eckmann L. Click chemistry-facilitated comprehensive identification of proteins adducted by antimicrobial 5-nitroimidazoles for discovery of alternative drug targets against giardiasis. Plos Neglected Tropical Diseases. 14: e0008224. PMID 32302296 DOI: 10.1371/journal.pntd.0008224  1
2020 Samskey N, Ho K, Momper J, Radic Z, Sit R, Sharpless KB, Taylor P. Pharmacokinetic Analysis of Ionizable Zwitterionic Oximes: Antidotes to Organophosphate Exposure. The Faseb Journal. 34: 1-1. DOI: 10.1096/fasebj.2020.34.s1.06319  0.8
2019 Maček Hrvat N, Kalisiak J, Šinko G, Radić Z, Sharpless KB, Taylor P, Kovarik Z. Evaluation of high-affinity phenyltetrahydroisoquinoline aldoximes, linked through anti-triazoles, as reactivators of phosphylated cholinesterases. Toxicology Letters. PMID 31863869 DOI: 10.1016/j.toxlet.2019.12.016  0.8
2019 Meng G, Guo T, Ma T, Zhang J, Shen Y, Sharpless KB, Dong J. Modular click chemistry libraries for functional screens using a diazotizing reagent. Nature. 574: 86-89. PMID 31578481 DOI: 10.1038/s41586-019-1589-1  1
2019 Zheng Q, Woehl JL, Kitamura S, Santos-Martins D, Smedley CJ, Li G, Forli S, Moses JE, Wolan DW, Sharpless KB. SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase. Proceedings of the National Academy of Sciences of the United States of America. PMID 31484779 DOI: 10.1073/pnas.1909972116  1
2019 Taylor P, Yan-Jye S, Momper J, Hou W, Camacho-Hernandez GA, Radic Z, Rosenberg Y, Kovarik Z, Sit R, Sharpless KB. Assessment of ionizable, zwitterionic oximes as reactivating antidotal agents for organophosphate exposure. Chemico-Biological Interactions. PMID 31100277 DOI: 10.1016/j.cbi.2019.05.015  0.8
2019 Liu F, Wang H, Li S, Bare GAL, Chen X, Wang C, Moses JE, Wu P, Sharpless KB. Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF4) Derived Connective Hubs For Bioconjugation to DNA and Proteins. Angewandte Chemie (International Ed. in English). PMID 30998840 DOI: 10.1002/anie.201902489  0.96
2019 Hong S, Shi Y, Wu NC, Grande G, Douthit L, Wang H, Zhou W, Sharpless KB, Wilson IA, Xie J, Wu P. Bacterial glycosyltransferase-mediated cell-surface chemoenzymatic glycan modification. Nature Communications. 10: 1799. PMID 30996301 DOI: 10.1038/s41467-019-09608-w  0.96
2019 Kovarik Z, Hrvat NM, Kalisiak J, Katalinić M, Sit RK, Zorbaz T, Radić Z, Fokin VV, Sharpless KB, Taylor P. Counteracting tabun inhibition by reactivation by pyridinium aldoximes that interact with active center gorge mutants of acetylcholinesterase. Toxicology and Applied Pharmacology. PMID 30978400 DOI: 10.1016/j.taap.2019.04.007  1
2019 Smedley CJ, Zheng Q, Gao B, Li S, Molino A, Duivenvoorden HM, Parker BS, Wilson DJD, Sharpless KB, Moses JE. Bifluoride Ion Mediated SuFEx Trifluoromethylation of Sulfonyl Fluorides and Iminosulfur Oxydifluorides. Angewandte Chemie (International Ed. in English). PMID 30740848 DOI: 10.1002/anie.201813761  1
2019 Liu F, Wang H, Li S, Bare GAL, Chen X, Wang C, Moses JE, Wu P, Sharpless KB. Back Cover: Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF 4 )‐Derived Connective Hubs for Bioconjugation to DNA and Proteins (Angew. Chem. Int. Ed. 24/2019) Angewandte Chemie International Edition. 58: 8242-8242. DOI: 10.1002/anie.201906154  0.96
2019 Liu F, Wang H, Li S, Bare GAL, Chen X, Wang C, Moses JE, Wu P, Sharpless KB. Rücktitelbild: Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF 4 )‐Derived Connective Hubs for Bioconjugation to DNA and Proteins (Angew. Chem. 24/2019) Angewandte Chemie. 131: 8328-8328. DOI: 10.1002/ange.201906154  0.96
2018 Kovarik Z, Kalisiak J, Hrvat NM, Katalinić M, Zorbaz T, Žunec S, Green C, Radić Z, Fokin VV, Sharpless KB, Taylor P. Reversal of tabun toxicity, enabled by a triazole annulated oxime library-reactivators of acetylcholinesterase. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 30458057 DOI: 10.1002/chem.201805051  1
2018 Sit R, Kovarik Z, Macek-Hrvat N, Zunec S, Green C, Fokin V, Sharpless KB, Radic' Z, Taylor P. Pharmacology, pharmacokinetics and tissue disposition of zwitterionic hydoxyiminoacetamido alkylamines as reactivating antidotes for organophosphate exposure. The Journal of Pharmacology and Experimental Therapeutics. PMID 30190337 DOI: 10.1124/jpet.118.249383  0.8
2018 Gahtory D, Sen R, Pujari S, Li S, Zheng Q, Moses JE, Sharpless KB, Zuilhof H. Quantitative and Orthogonal Formation and Reactivity of SuFEx Platforms. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29949211 DOI: 10.1002/chem.201802356  1
2018 Liu Z, Li J, Li S, Li G, Sharpless KB, Wu P. SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization. Journal of the American Chemical Society. PMID 29451783 DOI: 10.1021/jacs.7b12788  1
2018 Sharpless KB, Gao B, Li S, Wu P, Moses JE. SuFEx Chemistry of Thionyl Tetrafluoride (SOF4) with Organolithium Nucleophiles: Synthesis of Sulfonimidoyl Fluorides, Sulfoximines, Sulfonimidamides and Sulfonimidates. Angewandte Chemie (International Ed. in English). PMID 29314580 DOI: 10.1002/anie.201712145  0.96
2018 Guo T, Meng G, Zhan X, Yang Q, Ma T, Xu L, Sharpless KB, Dong J. Back Cover: A New Portal to SuFEx Click Chemistry: A Stable Fluorosulfuryl Imidazolium Salt Emerging as an “F−SO2 +” Donor of Unprecedented Reactivity, Selectivity, and Scope (Angew. Chem. Int. Ed. 10/2018) Angewandte Chemie International Edition. 57: 2728-2728. DOI: 10.1002/anie.201801651  1
2017 Guo T, Meng G, Zhan X, Yang Q, Ma T, Xu L, Sharpless KB, Dong J. A New Portal to SuFEx Click Chemistry: a Stable Fluorosulfuryl Imidazolium Salt Emerging as an "F-SO2+" Donor of Unprecedented Reactivity, Selectivity, and Scope. Angewandte Chemie (International Ed. in English). PMID 29276888 DOI: 10.1002/anie.201712429  1
2017 Mortenson DE, Brighty GJ, Plate L, Bare G, Chen W, Li S, Wang H, Cravatt BF, Forli S, Powers ET, Sharpless KB, Wilson IA, Kelly JW. "Inverse Drug Discovery" Strategy To Identify Proteins That Are Targeted by Latent Electrophiles As Exemplified by Aryl Fluorosulfates. Journal of the American Chemical Society. PMID 29265822 DOI: 10.1021/jacs.7b08366  0.96
2017 Gao B, Zhang L, Zheng Q, Zhou F, Klivansky LM, Lu J, Liu Y, Dong J, Wu P, Sharpless KB. Bifluoride-catalysed sulfur(VI) fluoride exchange reaction for the synthesis of polysulfates and polysulfonates. Nature Chemistry. 9: 1083-1088. PMID 29064495 DOI: 10.1038/nchem.2796  1
2017 Wang H, Zhou F, Ren G, Zheng Q, Chen H, Gao B, Klivansky L, Liu Y, Wu B, Xu Q, Lu J, Sharpless KB, Wu P. SuFEx-Based Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts. Angewandte Chemie (International Ed. in English). PMID 28792119 DOI: 10.1002/anie.201701160  1
2017 Kim WJ, Korthals K, Li S, Le C, Kalisiak J, Sharpless KB, Fokin VV, Miyamoto Y, Eckmann L. Click chemistry-facilitated structural diversification of nitrothiazoles, nitrofurans and nitropyrroles enhances antimicrobial activity against Giardia lamblia. Antimicrobial Agents and Chemotherapy. PMID 28396548 DOI: 10.1128/AAC.02397-16  1
2017 Zha GF, Zheng Q, Leng J, Wu P, Qin HL, Sharpless KB. Palladium-Catalyzed Fluorosulfonylvinylation of Organic Iodides. Angewandte Chemie (International Ed. in English). PMID 28370917 DOI: 10.1002/anie.201701162  1
2017 Li S, Wu P, Moses JE, Sharpless KB. Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride Exchange Connections of Diverse Modules Launched From An SOF4 Hub. Angewandte Chemie (International Ed. in English). PMID 28165188 DOI: 10.1002/anie.201611048  0.96
2017 Wang H, Zhou F, Ren G, Zheng Q, Chen H, Gao B, Klivansky L, Liu Y, Wu B, Xu Q, Lu J, Sharpless KB, Wu P. Back Cover: SuFEx-Based Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts (Angew. Chem. Int. Ed. 37/2017) Angewandte Chemie International Edition. 56: 11274-11274. DOI: 10.1002/anie.201706481  1
2017 Wang H, Zhou F, Ren G, Zheng Q, Chen H, Gao B, Klivansky L, Liu Y, Wu B, Xu Q, Lu J, Sharpless KB, Wu P. Rücktitelbild: SuFEx-Based Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts (Angew. Chem. 37/2017) Angewandte Chemie. 129: 11428-11428. DOI: 10.1002/ange.201706481  1
2016 Zheng Q, Dong J, Sharpless KB. Ethenesulfonyl Fluoride (ESF): An On-Water Procedure for the Kilogram-Scale Preparation. The Journal of Organic Chemistry. PMID 27764941 DOI: 10.1021/acs.joc.6b01423  1
2016 Qin HL, Zheng Q, Bare GA, Wu P, Sharpless KB. A Heck-Matsuda Process for the Synthesis of β-Arylethenesulfonyl Fluorides: Selectively Addressable Bis-electrophiles for SuFEx Click Chemistry. Angewandte Chemie (International Ed. in English). PMID 27723200 DOI: 10.1002/anie.201608807  1
2016 Chen W, Dong J, Plate L, Mortenson DE, Brighty GJ, Li S, Liu Y, Galmozzi A, Lee PS, Hulce JJ, Cravatt BF, Saez E, Powers ET, Wilson IA, Sharpless KB, et al. Arylfluorosulfates Inactivate Intracellular Lipid Binding Protein(s) through Chemoselective SuFEx Reaction with a Binding-site Tyr Residue. Journal of the American Chemical Society. PMID 27191344 DOI: 10.1021/jacs.6b02960  1
2016 Zhang E, Tang J, Li S, Wu P, Moses JE, Sharpless KB. Chemoselective Synthesis of Polysubstituted Pyridines from Heteroaryl Fluorosulfates. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26990693 DOI: 10.1002/chem.201600167  1
2016 Bourne Y, Sharpless KB, Taylor P, Marchot P. Steric and dynamic parameters influencing in situ cycloadditions to form triazole inhibitors with crystalline acetylcholinesterase. Journal of the American Chemical Society. PMID 26731630 DOI: 10.1021/jacs.5b11384  1
2015 Chen W, Dong J, Li S, Liu Y, Wang Y, Yoon L, Wu P, Sharpless KB, Kelly JW. Synthesis of Sulfotyrosine-Containing Peptides by Incorporating Fluorosulfated Tyrosine Using an Fmoc-Based Solid-Phase Strategy. Angewandte Chemie (International Ed. in English). PMID 26696445 DOI: 10.1002/anie.201509016  1
2015 Baranczak A, Liu Y, Connelly S, Du WG, Greiner ER, Genereux JC, Wiseman RL, Eisele YS, Bradbury NC, Dong J, Noodleman L, Sharpless KB, Wilson IA, Encalada SE, Kelly JW. A Fluorogenic Aryl Fluorosulfate for Intraorganellar Transthyretin Imaging in Living Cells and in Caenorhabditis elegans. Journal of the American Chemical Society. 137: 7404-14. PMID 26051248 DOI: 10.1021/jacs.5b03042  1
2015 Liang Q, Xing P, Huang Z, Dong J, Sharpless KB, Li X, Jiang B. Palladium-catalyzed, ligand-free Suzuki reaction in water using aryl fluorosulfates. Organic Letters. 17: 1942-5. PMID 25856416 DOI: 10.1021/acs.orglett.5b00654  1
2015 Sharpless KB, Finn MG, Martín VS. Tsutomu Katsuki (1946-2014). Angewandte Chemie (International Ed. in English). 54: 4708. PMID 25766459 DOI: 10.1002/anie.201501065  1
2015 Schantz MM, Benner BA, Heckert NA, Sander LC, Sharpless KE, Vander Pol SS, Vasquez Y, Villegas M, Wise SA, Alwis KU, Blount BC, Calafat AM, Li Z, Silva MJ, Ye X, et al. Development of urine standard reference materials for metabolites of organic chemicals including polycyclic aromatic hydrocarbons, phthalates, phenols, parabens, and volatile organic compounds. Analytical and Bioanalytical Chemistry. 407: 2945-54. PMID 25651899 DOI: 10.1007/s00216-014-8441-0  0.48
2015 Templeton DW, Wolfrum EJ, Yen JH, Sharpless KE. Compositional Analysis of Biomass Reference Materials: Results from an Interlaboratory Study Bioenergy Research. DOI: 10.1007/s12155-015-9675-1  0.48
2015 Sharpless KB. Building blocks for SuFEx, the next click reaction Aldrichimica Acta. 48: 41.  1
2014 Dong J, Krasnova L, Finn MG, Sharpless KB. Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry. Angewandte Chemie (International Ed. in English). 53: 9430-48. PMID 25112519 DOI: 10.1002/anie.201309399  0.88
2014 Dong J, Sharpless KB, Kwisnek L, Oakdale JS, Fokin VV. SuFEx-based synthesis of polysulfates. Angewandte Chemie (International Ed. in English). 53: 9466-70. PMID 25100330 DOI: 10.1002/anie.201403758  1
2014 Sit RK, Fokin VV, Amitai G, Sharpless KB, Taylor P, Radić Z. Imidazole aldoximes effective in assisting butyrylcholinesterase catalysis of organophosphate detoxification. Journal of Medicinal Chemistry. 57: 1378-89. PMID 24571195 DOI: 10.1021/jm401650z  1
2014 Dong J, Krasnova L, Finn MG, Sharpless KB. ChemInform Abstract: Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry Cheminform. 45: no-no. DOI: 10.1002/chin.201447274  1
2014 Dong J, Krasnova L, Finn MG, Sharpless KB. Cover Picture: Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry (Angew. Chem. Int. Ed. 36/2014) Angewandte Chemie International Edition. 53: 9391-9391. DOI: 10.1002/anie.201401157  1
2014 Dong J, Krasnova L, Finn MG, Sharpless KB. Titelbild: Schwefel(VI)-fluorid-Austausch (SuFEx): Eine weitere gute Anwendung für die Click-Chemie (Angew. Chem. 36/2014) Angewandte Chemie. 126: 9545-9545. DOI: 10.1002/ange.201401157  1
2014 Dong J, Krasnova L, Finn MG, Sharpless KB. Schwefel(VI)-fluorid-Austausch (SuFEx): Eine weitere gute Anwendung für die Click-Chemie Angewandte Chemie. 126: 9584-9603. DOI: 10.1002/ange.201309399  1
2013 Turk GC, Sharpless KE, Cleveland D, Jongsma C, Mackey EA, Marlow AF, Oflaz R, Paul RL, Sieber JR, Thompson RQ, Wood LJ, Yu LL, Zeisler R, Wise SA, Yen JH, et al. Certification of elements in and use of standard reference material 3280 multivitamin/multielement tablets. Journal of Aoac International. 96: 1281-7. PMID 24645505 DOI: 10.5740/jaoacint.13-135  0.48
2013 Phinney KW, Ballihaut G, Bedner M, Benford BS, Camara JE, Christopher SJ, Davis WC, Dodder NG, Eppe G, Lang BE, Long SE, Lowenthal MS, McGaw EA, Murphy KE, Nelson BC, ... ... Sharpless KE, et al. Development of a Standard Reference Material for metabolomics research. Analytical Chemistry. 85: 11732-8. PMID 24187941 DOI: 10.1021/ac402689t  0.48
2013 Miyamoto Y, Kalisiak J, Korthals K, Lauwaet T, Cheung DY, Lozano R, Cobo ER, Upcroft P, Upcroft JA, Berg DE, Gillin FD, Fokin VV, Sharpless KB, Eckmann L. Expanded therapeutic potential in activity space of next-generation 5-nitroimidazole antimicrobials with broad structural diversity. Proceedings of the National Academy of Sciences of the United States of America. 110: 17564-9. PMID 24101497 DOI: 10.1073/pnas.1302664110  1
2013 Hirose T, Maita N, Gouda H, Koseki J, Yamamoto T, Sugawara A, Nakano H, Hirono S, Shiomi K, Watanabe T, Taniguchi H, Sharpless KB, Omura S, Sunazuka T. Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor. Proceedings of the National Academy of Sciences of the United States of America. 110: 15892-7. PMID 24043811 DOI: 10.1073/pnas.1315049110  1
2013 Rimmer CA, Sharpless KE, Wise SA, Betz JM, Coates PM. Standard reference materials for dietary supplement analysis Analytical and Bioanalytical Chemistry. 405: 4337-4344. PMID 23575912 DOI: 10.1007/s00216-013-6942-x  0.48
2013 Sander LC, Bedner M, Duewer DL, Lippa KA, Phillips MM, Phinney KW, Rimmer CA, Schantz MM, Sharpless KE, Tai SS, Thomas JB, Wise SA, Wood LJ, Betz JM, Coates PM. The development and implementation of quality assurance programs to support nutritional measurements. Analytical and Bioanalytical Chemistry. 405: 4437-41. PMID 23552970 DOI: 10.1007/s00216-013-6864-7  0.48
2013 Thomas JB, Yen JH, Sharpless KE. Characterization of NIST food-matrix Standard Reference Materials for their vitamin C content. Analytical and Bioanalytical Chemistry. 405: 4539-48. PMID 23529413 DOI: 10.1007/s00216-013-6891-4  0.48
2013 Phillips MM, Sharpless KE, Wise SA. Standard reference materials for food analysis. Analytical and Bioanalytical Chemistry. 405: 4325-35. PMID 23515610 DOI: 10.1007/s00216-013-6890-5  0.48
2013 Morris GM, Green LG, Radić Z, Taylor P, Sharpless KB, Olson AJ, Grynszpan F. Automated docking with protein flexibility in the design of femtomolar "click chemistry" inhibitors of acetylcholinesterase. Journal of Chemical Information and Modeling. 53: 898-906. PMID 23451944 DOI: 10.1021/ci300545a  1
2013 Schantz MM, Sander LC, Sharpless KE, Wise SA, Yen JH, NguyenPho A, Betz JM. Development of botanical and fish oil standard reference materials for fatty acids. Analytical and Bioanalytical Chemistry. 405: 4531-8. PMID 23371533 DOI: 10.1007/s00216-013-6747-y  0.48
2013 Grimster NP, Connelly S, Baranczak A, Dong J, Krasnova LB, Sharpless KB, Powers ET, Wilson IA, Kelly JW. Aromatic sulfonyl fluorides covalently kinetically stabilize transthyretin to prevent amyloidogenesis while affording a fluorescent conjugate. Journal of the American Chemical Society. 135: 5656-68. PMID 23350654 DOI: 10.1021/ja311729d  1
2013 Schantz MM, Eppe G, Focant JF, Hamilton C, Heckert NA, Heltsley RM, Hoover D, Keller JM, Leigh SD, Patterson DG, Pintar AL, Sharpless KE, Sjödin A, Turner WE, Vander Pol SS, et al. Milk and serum standard reference materials for monitoring organic contaminants in human samples. Analytical and Bioanalytical Chemistry. 405: 1203-11. PMID 23132544 DOI: 10.1007/s00216-012-6524-3  0.48
2013 Fraser BH, Hamilton S, Krause-Heuer AM, Wright PJ, Greguric I, Tucker SP, Draffan AG, Fokin VV, Sharpless KB. Synthesis of 1,4-triazole linked zanamivir dimers as highly potent inhibitors of influenza A and B Medchemcomm. 4: 383-386. DOI: 10.1039/c2md20300f  1
2012 Yamauchi JG, Gomez K, Grimster N, Dufouil M, Nemecz A, Fotsing JR, Ho KY, Talley TT, Sharpless KB, Fokin VV, Taylor P. Synthesis of selective agonists for the α7 nicotinic acetylcholine receptor with in situ click-chemistry on acetylcholine-binding protein templates. Molecular Pharmacology. 82: 687-99. PMID 22784805 DOI: 10.1124/mol.112.080291  1
2012 Rimmer CA, Putzbach K, Sharpless KE, Sander LC, Yen JH. Preparation and certification of standard reference material 3278 tocopherols in edible oils. Journal of Agricultural and Food Chemistry. 60: 6794-8. PMID 22686411 DOI: 10.1021/jf2051619  0.48
2012 Grimster NP, Stump B, Fotsing JR, Weide T, Talley TT, Yamauchi JG, Nemecz Á, Kim C, Ho KY, Sharpless KB, Taylor P, Fokin VV. Generation of candidate ligands for nicotinic acetylcholine receptors via in situ click chemistry with a soluble acetylcholine binding protein template. Journal of the American Chemical Society. 134: 6732-40. PMID 22394239 DOI: 10.1021/ja3001858  1
2012 Radi? Z, Sit RK, Kovarik Z, Berend S, Garcia E, Zhang L, Amitai G, Green C, Radi? B, Fokin VV, Sharpless KB, Taylor P. Refinement of structural leads for centrally acting oxime reactivators of phosphylated cholinesterases. The Journal of Biological Chemistry. 287: 11798-809. PMID 22343626 DOI: 10.1074/jbc.M111.333732  1
2012 Phinney KW, Bedner M, Tai SS, Vamathevan VV, Sander LC, Sharpless KE, Wise SA, Yen JH, Schleicher RL, Chaudhary-Webb M, Pfeiffer CM, Betz JM, Coates PM, Picciano MF. Development and certification of a standard reference material for vitamin D metabolites in human serum. Analytical Chemistry. 84: 956-62. PMID 22141317 DOI: 10.1021/ac202047n  0.48
2012 Sander LC, Bedner M, Tims MC, Yen JH, Duewer DL, Porter B, Christopher SJ, Day RD, Long SE, Molloy JL, Murphy KE, Lang BE, Lieberman R, Wood LJ, Payne MJ, ... ... Sharpless KE, et al. Development and certification of green tea-containing standard reference materials. Analytical and Bioanalytical Chemistry. 402: 473-87. PMID 22127575 DOI: 10.1007/s00216-011-5472-7  0.48
2012 Thomas JB, Duewer DL, Mugenya IO, Phinney KW, Sander LC, Sharpless KE, Sniegoski LT, Tai SS, Welch MJ, Yen JH. Preparation and value assignment of standard reference material 968e fat-soluble vitamins, carotenoids, and cholesterol in human serum. Analytical and Bioanalytical Chemistry. 402: 749-62. PMID 22015475 DOI: 10.1007/s00216-011-5447-8  0.48
2012 Radi? Z, Sit RK, Kovarik Z, Berend S, Garcia E, Zhang L, Amitai G, Green C, Radi? B, Fokin VV, Sharpless KB, Taylor P. Refinement of structural leads for centrally acting oxime reactivators of phosphylated cholinesterases (Journal of Biological Chemistry (2012) 287, (11798-11809)) Journal of Biological Chemistry. 287: 19337. DOI: 10.1074/jbc.A111.333732  1
2012 Finn MG, Sharpless KB. On the Mechanism of Asymmetric Epoxidation with Titanium-Tartrate Catalysts Asymmetric Synthesis. 247-308. DOI: 10.1016/B978-0-08-092493-9.50013-X  1
2011 Millward SW, Henning RK, Kwong GA, Pitram S, Agnew HD, Deyle KM, Nag A, Hein J, Lee SS, Lim J, Pfeilsticker JA, Sharpless KB, Heath JR. Iterative in situ click chemistry assembles a branched capture agent and allosteric inhibitor for Akt1. Journal of the American Chemical Society. 133: 18280-8. PMID 21962254 DOI: 10.1021/ja2064389  1
2011 Thomas JB, Sharpless KE, Yen JH, Rimmer CA. Determination of fat-soluble vitamins and carotenoids in standard reference material 3280 multivitamin/multielement tablets by liquid chromatography with absorbance detection. Journal of Aoac International. 94: 815-22. PMID 21797009  0.48
2011 Phillips MM, Rimmer CA, Wood LJ, Lippa KA, Sharpless KE, Duewer DL, Sander LC, Betz JM. Dietary supplement laboratory quality assurance program: the first five exercises. Journal of Aoac International. 94: 803-14. PMID 21797008  0.48
2011 Cochran R, Kalisiak J, Küçükkilinç T, Radic Z, Garcia E, Zhang L, Ho KY, Amitai G, Kovarik Z, Fokin VV, Sharpless KB, Taylor P. Oxime-assisted acetylcholinesterase catalytic scavengers of organophosphates that resist aging. The Journal of Biological Chemistry. 286: 29718-24. PMID 21730071 DOI: 10.1074/jbc.M111.264739  1
2011 Wood LJ, Sharpless KE, Pichon M, Porter BJ, Yen JH, Ehling S. Characterization of three berry standard reference materials for nutrients. Journal of Agricultural and Food Chemistry. 59: 7246-52. PMID 21688777 DOI: 10.1021/jf200883e  0.48
2011 Sit RK, Radi? Z, Gerardi V, Zhang L, Garcia E, Katalini? M, Amitai G, Kovarik Z, Fokin VV, Sharpless KB, Taylor P. New structural scaffolds for centrally acting oxime reactivators of phosphylated cholinesterases. The Journal of Biological Chemistry. 286: 19422-30. PMID 21464125 DOI: 10.1074/jbc.M111.230656  1
2011 Gastaminza P, Pitram SM, Dreux M, Krasnova LB, Whitten-Bauer C, Dong J, Chung J, Fokin VV, Sharpless KB, Chisari FV. Antiviral stilbene 1,2-diamines prevent initiation of hepatitis C virus RNA replication at the outset of infection. Journal of Virology. 85: 5513-23. PMID 21430055 DOI: 10.1128/JVI.02116-10  1
2011 Sander LC, Sharpless KE, Wise SA, Nelson BC, Phinney KW, Porter BJ, Rimmer CA, Thomas JB, Wood LJ, Yen JH, Duewer DL, Atkinson R, Chen P, Goldschmidt R, Wolf WR, et al. Certification of vitamins and carotenoids in SRM 3280 multivitamin/multielement tablets. Analytical Chemistry. 83: 99-108. PMID 21128589 DOI: 10.1021/ac101953u  0.48
2011 Phinney KW, Rimmer CA, Thomas JB, Sander LC, Sharpless KE, Wise SA. Isotope dilution liquid chromatography - mass spectrometry methods for fat- and water-soluble vitamins in nutritional formulations. Analytical Chemistry. 83: 92-8. PMID 21117618 DOI: 10.1021/ac101950r  0.48
2010 Sharpless KE, Lindstrom RM, Nelson BC, Phinney KW, Rimmer CA, Sander LC, Schantz MM, Spatz RO, Thomas JB, Turk GC, Wise SA, Wood LJ, Yen JH. Preparation and characterization of standard reference material 1849 infant/adult nutritional formula. Journal of Aoac International. 93: 1262-74. PMID 20922961  0.48
2010 Weide T, Saldanha SA, Minond D, Spicer TP, Fotsing JR, Spaargaren M, Frère JM, Bebrone C, Sharpless KB, Hodder PS, Fokin VV. NH-1,2,3-Triazole-based Inhibitors of the VIM-2 Metallo-β-Lactamase: Synthesis and Structure-Activity Studies. Acs Medicinal Chemistry Letters. 1: 150-154. PMID 20625539 DOI: 10.1021/ml900022q  1
2010 Phillips MM, Case RJ, Rimmer CA, Sander LC, Sharpless KE, Wise SA, Yen JH. Determination of organic acids in Vaccinium berry standard reference materials. Analytical and Bioanalytical Chemistry. 398: 425-34. PMID 20582402 DOI: 10.1007/s00216-010-3916-0  0.48
2010 Bedner M, Sander LC, Sharpless KE. An LC-ESI/MS method for determining theanine in green tea dietary supplements Analytical and Bioanalytical Chemistry. 397: 1773-1777. PMID 20422160 DOI: 10.1007/s00216-010-3713-9  0.48
2010 Radi? Z, Kalisiak J, Fokin VV, Sharpless KB, Taylor P. Interaction kinetics of oximes with native, phosphylated and aged human acetylcholinesterase. Chemico-Biological Interactions. 187: 163-6. PMID 20412789 DOI: 10.1016/j.cbi.2010.04.014  1
2010 Berend S, Vrdoljak AL, Radic B, Kalisiak J, Radic Z, Taylor P, Fokin V, Sharpless K. Characterizing the therapeutic efficacy of novel oximes synthesized by click chemistry against organophosphorous compounds poisoning Toxicology Letters. 196: S254. DOI: 10.1016/j.toxlet.2010.03.849  0.8
2010 Hein JE, Tripp JC, Krasnova LB, Sharpless KB, Fokin VV. ChemInform Abstract: Copper(I)-Catalyzed Cycloaddition of Organic Azides and 1-Iodoalkynes. Cheminform. 41. DOI: 10.1002/chin.201007113  1
2010 Demko ZP, Sharpless KB. ChemInform Abstract: An Expedient Route to the Tetrazole Analogues of α-Amino Acids. Cheminform. 33: no-no. DOI: 10.1002/chin.200248140  0.92
2010 Dupau P, Epple R, Thomas AA, Fokin VV, Sharpless KB. ChemInform Abstract: Osmium-Catalyzed Dihydroxylation of Olefins in Acidic Media: Old Process, New Tricks. Cheminform. 33: no-no. DOI: 10.1002/chin.200244058  1
2010 Rostovtsev VV, Green LG, Fokin VV, Sharpless KB. ChemInform Abstract: A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes. Cheminform. 33: no-no. DOI: 10.1002/chin.200243045  1
2010 Demko ZP, Sharpless KB. ChemInform Abstract: A Click Chemistry Approach to Tetrazoles by Huisgen 1,3-Dipolar Cycloaddition: Synthesis of 5-Acyltetrazoles from Azides and Acyl Cyanides. Cheminform. 33: no-no. DOI: 10.1002/chin.200242151  0.92
2010 Andersson MA, Epple R, Fokin VV, Sharpless KB. ChemInform Abstract: A New Approach to Osmium-Catalyzed Asymmetric Dihydroxylation and Aminohydroxylation of Olefins. Cheminform. 33: no-no. DOI: 10.1002/chin.200228035  1
2010 Demko ZP, Sharpless KB. ChemInform Abstract: Preparation of 5-Substituted 1H-Tetrazoles from Nitriles in Water. Cheminform. 33: no-no. DOI: 10.1002/chin.200222135  0.92
2010 Demko ZP, Sharpless KB. ChemInform Abstract: An Intramolecular [2 + 3] Cycloaddition Route to Fused 5-Heterosubstituted Tetrazoles. Cheminform. 33: no-no. DOI: 10.1002/chin.200222134  0.92
2010 Kolb HC, Finn MG, Sharpless KB. ChemInform Abstract: Click Chemistry: Diverse Chemical Function from a Few Good Reactions Cheminform. 32: no-no. DOI: 10.1002/chin.200135279  1
2010 Johnson RA, Sharpless KB. ChemInform Abstract: Catalytic Asymmetric Dihydroxylation - Discovery and Development Cheminform. 32: no-no. DOI: 10.1002/chin.200129254  0.52
2010 Chuang T, Sharpless KB. ChemInform Abstract: Applications of Aziridinium Ions: Selective Syntheses of Pyrazolidin-3-ones and Pyrazolo[1,2-a]pyrazoles. Cheminform. 31: no-no. DOI: 10.1002/chin.200046142  0.48
2010 Chuang T, Sharpless KB. ChemInform Abstract: Applications of Aziridinium Ions. Selective Syntheses of β-Aryl-α,β-diamino Esters. Cheminform. 31: no-no. DOI: 10.1002/chin.200002111  0.48
2010 Gontcharov AV, Liu H, Sharpless KB. ChemInform Abstract: tert-Butylsulfonamide. A New Nitrogen Source for Catalytic Aminohydroxylation and Aziridination of Olefins. Cheminform. 30: no-no. DOI: 10.1002/chin.199949038  0.56
2010 Goossen LJ, Liu H, Dress KR, Sharpless KB. ChemInform Abstract: Catalytic Asymmetric Aminohydroxylation with Amino-Substituted Heterocycles as Nitrogen Sources. Cheminform. 30: no-no. DOI: 10.1002/chin.199933040  0.56
2010 DRESS KR, GOOSSEN LJ, LIU H, JERINA DM, SHARPLESS KB. ChemInform Abstract: Catalytic Aminohydroxylation Using Adenine-Derivatives as the Nitrogen Source. Cheminform. 29: no-no. DOI: 10.1002/chin.199852176  0.56
2010 TAO B, SCHLINGLOFF G, SHARPLESS KB. ChemInform Abstract: Reversal of Regioselection in the Asymmetric Aminohydroxylation of Cinnamates. Cheminform. 29: no-no. DOI: 10.1002/chin.199828042  0.48
2010 YUDIN AK, SHARPLESS KB. ChemInform Abstract: Bis(trimethylsilyl) Peroxide Extends the Range of Oxorhenium Catalysts for Olefin Epoxidation. Cheminform. 29: no-no. DOI: 10.1002/chin.199810117  1
2010 COPERET C, ADOLFSSON H, SHARPLESS KB. ChemInform Abstract: A Simple and Efficient Method for Epoxidation of Terminal Alkenes. Cheminform. 28: no-no. DOI: 10.1002/chin.199747120  0.8
2010 VANHESSCHE KPM, SHARPLESS KB. ChemInform Abstract: Ligand-Dependent Reversal of Facial Selectivity in the Asymmetric Dihydroxylation. Cheminform. 28: no-no. DOI: 10.1002/chin.199712063  0.76
2010 CHANG H, SHARPLESS KB. ChemInform Abstract: Molar Scale Synthesis of Enantiopure Stilbene Oxide. Cheminform. 28: no-no. DOI: 10.1002/chin.199704115  1
2010 CHANG H, SHARPLESS KB. ChemInform Abstract: A Practical Route to Enantiopure 1,2-Amino Alcohols. Cheminform. 27: no-no. DOI: 10.1002/chin.199633102  1
2010 JOHNSON RA, SHARPLESS KB. ChemInform Abstract: Catalytic Asymmetric Epoxidation of Allylic Alcohols Cheminform. 25: no-no. DOI: 10.1002/chin.199432281  0.52
2010 KOLB HC, ANDERSSON PG, SHARPLESS KB. ChemInform Abstract: Toward an Understanding of the High Enantioselectivity in the Osmium- Catalyzed Asymmetric Dihydroxylation (AD). Part 1. Kinetics. Cheminform. 25: no-no. DOI: 10.1002/chin.199426078  1
2010 WALSH PJ, SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation (AD) of α,β-Unsaturated Ketones. Cheminform. 25: no-no. DOI: 10.1002/chin.199411088  1
2010 WANG Z, SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation of α-Substituted Styrene Derivatives ( I), (III). Cheminform. 25: no-no. DOI: 10.1002/chin.199411087  1
2010 AMBERG W, BENNANI YL, CHADHA RK, CRISPINO GA, DAVIS WD, HARTUNG J, JEONG K, OGINO Y, SHIBATA T, SHARPLESS KB. ChemInform Abstract: Syntheses and Crystal Structures of the Cinchona Alkaloid Derivatives Used as Ligands in the Osmium-Catalyzed Asymmetric Dihydroxylation of Olefins, e.g. (I). Used as Ligands in the Osmium-Catalyzed Asymmetric Dihydroxylation of Olefi Cheminform. 25: no-no. DOI: 10.1002/chin.199404183  0.76
2010 WALSH PJ, BENNANI YL, SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation (AD)/Cyclization of N-DiBoc Allylic and Homoallylic Amines: Selective Differentiation of the Hydroxyl Groups. Cheminform. 24: no-no. DOI: 10.1002/chin.199352069  1
2010 KOLB HC, BENNANI YL, SHARPLESS KB. ChemInform Abstract: Short and Practical Syntheses of (R)-(-)-Carnitine and (R)-(-)-γ- Amino-β-hydroxybutyric Acid (GABOB). Cheminform. 24: no-no. DOI: 10.1002/chin.199321060  1
2010 CRISPINO GA, HO PT, SHARPLESS KB. ChemInform Abstract: Selective Perhydroxylation of Squalene: Taming the Arithmetic Demon. Cheminform. 24: no-no. DOI: 10.1002/chin.199316129  0.6
2010 KOLB HC, SHARPLESS KB. ChemInform Abstract: A Simplified Procedure for the Stereospecific Transformation of 1,2- Diols into Epoxides. Cheminform. 24: no-no. DOI: 10.1002/chin.199313174  1
2010 XU D, CRISPINO GA, SHARPLESS KB. ChemInform Abstract: Selective Asymmetric Dihydroxylation of Dienes. Cheminform. 24: no-no. DOI: 10.1002/chin.199301132  0.84
2010 WANG L, SHARPLESS KB. ChemInform Abstract: Catalytic Asymmetric Dihydroxylation of cis-Disubstituted Olefins. Cheminform. 24: no-no. DOI: 10.1002/chin.199301131  0.72
2010 JEONG K, SJOE P, SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation of Enynes. Cheminform. 23: no-no. DOI: 10.1002/chin.199252107  0.36
2010 SHARPLESS KB, AMBERG W, BENNANI YL, CRISPINO GA, HARTUNG J, JEONG K, KWONG H, MORIKAWA K, WANG Z, XU D, ZHANG X. ChemInform Abstract: The Osmium-Catalyzed Asymmetric Dihydroxylation: A New Ligand Class and a Process Improvement. Cheminform. 23: no-no. DOI: 10.1002/chin.199242058  1
2009 Hein JE, Tripp JC, Krasnova LB, Sharpless KB, Fokin VV. Copper(I)-catalyzed cycloaddition of organic azides and 1-iodoalkynes. Angewandte Chemie (International Ed. in English). 48: 8018-21. PMID 19774581 DOI: 10.1002/anie.200903558  1
2009 Duewer DL, Lippa KA, Long SE, Murphy KE, Sharpless KE, Sniegoski LT, Welch MJ, Tani W, Umemoto M. Demonstrating the comparability of certified reference materials. Analytical and Bioanalytical Chemistry. 395: 155-69. PMID 19629455 DOI: 10.1007/s00216-009-2949-8  0.48
2009 Minond D, Saldanha SA, Subramaniam P, Spaargaren M, Spicer T, Fotsing JR, Weide T, Fokin VV, Sharpless KB, Galleni M, Bebrone C, Lassaux P, Hodder P. Inhibitors of VIM-2 by screening pharmacologically active and click-chemistry compound libraries. Bioorganic & Medicinal Chemistry. 17: 5027-37. PMID 19553129 DOI: 10.1016/j.bmc.2009.05.070  1
2009 Valdez CA, Tripp JC, Miyamoto Y, Kalisiak J, Hruz P, Andersen YS, Brown SE, Kangas K, Arzu LV, Davids BJ, Gillin FD, Upcroft JA, Upcroft P, Fokin VV, Smith DK, ... Sharpless KB, et al. Synthesis and electrochemistry of 2-ethenyl and 2-ethanyl derivatives of 5-nitroimidazole and antimicrobial activity against Giardia lamblia. Journal of Medicinal Chemistry. 52: 4038-53. PMID 19480409 DOI: 10.1021/jm900356n  1
2009 Hirose T, Sunazuka T, Sugawara A, Endo A, Iguchi K, Yamamoto T, Ui H, Shiomi K, Watanabe T, Sharpless KB, Omura S. Chitinase inhibitors: extraction of the active framework from natural argifin and use of in situ click chemistry. The Journal of Antibiotics. 62: 277-82. PMID 19329983 DOI: 10.1038/ja.2009.28  1
2009 Agnew HD, Rohde RD, Millward SW, Nag A, Yeo WS, Hein JE, Pitram SM, Tariq AA, Burns VM, Krom RJ, Fokin VV, Sharpless KB, Heath JR. Iterative in situ click chemistry creates antibody-like protein-capture agents. Angewandte Chemie (International Ed. in English). 48: 4944-8. PMID 19301344 DOI: 10.1002/anie.200900488  1
2009 Kalisiak J, Trauger SA, Kalisiak E, Morita H, Fokin VV, Adams MW, Sharpless KB, Siuzdak G. Identification of a new endogenous metabolite and the characterization of its protein interactions through an immobilization approach. Journal of the American Chemical Society. 131: 378-86. PMID 19055353 DOI: 10.1021/ja808172n  1
2009 Sander L, Schantz M, Sharpless K, Wise S. Standard Reference Materials to support measurement of fatty acids Lipid Technology. 21: 7-12. DOI: 10.1002/lite.200800080  0.48
2009 Kwok SW, Hein JE, Fokin VV, Sharpless KB. ChemInform Abstract: Regioselective Synthesis of Either 1H- or 2H-1,2,3-Triazoles via Michael Addition to α,β-Unsaturated Ketones. Cheminform. 40. DOI: 10.1002/chin.200918132  1
2009 Schantz MM, Christopher SJ, Davis WC, Day RD, Keller JM, Kucklick JR, Long SE, Mackey EA, Point D, Porter BJ, Poster DL, Sharpless KE, Turk GC, Wise SA. Fish-Related: Standard reference materials American Laboratory. 41: 50-53.  0.48
2008 Dwyer JT, Picciano MF, Betz JM, Fisher KD, Saldanha LG, Yetley EA, Coates PM, Milner JA, Whitted J, Burt V, Radimer K, Wilger J, Sharpless KE, Holden JM, Andrews K, et al. Progress in developing analytical and label-based dietary supplement databases at the NIH Office of Dietary Supplements. Journal of Food Composition and Analysis : An Official Publication of the United Nations University, International Network of Food Data Systems. 21: S83-S93. PMID 25346570 DOI: 10.1016/j.jfca.2007.07.010  0.48
2008 Kwok SW, Hein JE, Fokin VV, Sharpless KB. REGIOSELECTIVE SYNTHESIS OF EITHER 1H- OR 2H-1,2,3- TRIAZOLES VIA MICHAEL ADDITION TO α,ß-UNSATURATED KETONES. Heterocycles. 76: 1141-1154. PMID 19802363 DOI: 10.3987/COM-08-S(N)73  1
2008 Sharpless KE, Duewer DL. Standard reference materials for analysis of dietary supplements Journal of Aoac International. 91: 1298-1302. PMID 19202789  0.48
2008 Schantz MM, Bedner M, Long SE, Molloy JL, Murphy KE, Porter BJ, Putzbach K, Rimmer CA, Sander LC, Sharpless KE, Thomas JB, Wise SA, Wood LJ, Yen JH, Yarita T, et al. Development of saw palmetto (Serenoa repens) fruit and extract standard reference materials. Analytical and Bioanalytical Chemistry. 392: 427-38. PMID 18677464 DOI: 10.1007/s00216-008-2297-0  0.48
2008 Kalisiak J, Sharpless KB, Fokin VV. Efficient synthesis of 2-substituted-1,2,3-triazoles. Organic Letters. 10: 3171-4. PMID 18597477 DOI: 10.1021/ol8006748  1
2008 Nelson BC, Pfeiffer CM, Zhang M, Duewer DL, Sharpless KE, Lippa KA. Commutability of NIST SRM 1955 Homocysteine and Folate in Frozen Human Serum with selected total homocysteine immunoassays and enzymatic assays Clinica Chimica Acta. 395: 99-105. PMID 18565331 DOI: 10.1016/j.cca.2008.05.016  0.48
2008 Yoo EJ, Ahlquist M, Bae I, Sharpless KB, Fokin VV, Chang S. Mechanistic studies on the Cu-catalyzed three-component reactions of sulfonyl azides, 1-alkynes and amines, alcohols, or water: dichotomy via a common pathway. The Journal of Organic Chemistry. 73: 5520-8. PMID 18557650 DOI: 10.1021/jo800733p  1
2008 Radi? Z, Manetsch R, Fournier D, Sharpless KB, Taylor P. Probing gorge dimensions of cholinesterases by freeze-frame click chemistry. Chemico-Biological Interactions. 175: 161-5. PMID 18555981 DOI: 10.1016/j.cbi.2008.04.048  1
2008 Sander LC, Putzbach K, Nelson BC, Rimmer CA, Bedner M, Thomas JB, Porter BJ, Wood LJ, Schantz MM, Murphy KE, Sharpless KE, Wise SA, Yen JH, Siitonen PH, Evans RL, et al. Certification of standard reference materials containing bitter orange. Analytical and Bioanalytical Chemistry. 391: 2023-34. PMID 18425642 DOI: 10.1007/s00216-008-2074-0  0.48
2008 Bedner M, Schantz MM, Sander LC, Sharpless KE. Development of liquid chromatographic methods for the determination of phytosterols in Standard Reference Materials containing saw palmetto Journal of Chromatography A. 1192: 74-80. PMID 18374927 DOI: 10.1016/j.chroma.2008.03.020  0.48
2008 Saupe SG, Sharpless KE. Solution to "doctrine of Signatures" challenge Analytical and Bioanalytical Chemistry. 390: 79-83. PMID 18074123 DOI: 10.1007/s00216-007-1743-8  0.48
2008 Roseland JM, Holden JM, Andrews KW, Zhao C, Schweitzer A, Harnly J, Wolf WR, Perry CR, Dwyer JT, Picciano MF, Betz JM, Saldanha LG, Yetley EA, Fisher KD, Sharpless KE. Dietary supplement ingredient database (DSID): Preliminary USDA studies on the composition of adult multivitamin/mineral supplements Journal of Food Composition and Analysis. 21: S69-S77. DOI: 10.1016/j.jfca.2007.07.009  0.48
2008 Santana J, Sharpless KE, Nelson BC. Determination of para-synephrine and meta-synephrine positional isomers in bitter orange-containing dietary supplements by LC/UV and LC/MS/MS Food Chemistry. 109: 675-682. DOI: 10.1016/j.foodchem.2007.12.076  0.48
2008 Finn MG, Kolb HC, Fokin VV, Sharpless KB. Click chemistry - Definition and aims Progress in Chemistry. 20: 1-4.  1
2007 Nelson BC, Putzbach K, Sharpless KE, Sander LC. Mass spectrometric determination of the predominant adrenergic protoalkaloids in bitter orange (Citrus aurantium) Journal of Agricultural and Food Chemistry. 55: 9769-9775. PMID 17966980 DOI: 10.1021/jf072030s  0.48
2007 Sugawara A, Sunazuka T, Hirose T, Nagai K, Yamaguchi Y, Hanaki H, Sharpless KB, Omura S. Design and synthesis via click chemistry of 8,9-anhydroerythromycin A 6,9-hemiketal analogues with anti-MRSA and -VRE activity. Bioorganic & Medicinal Chemistry Letters. 17: 6340-4. PMID 17869508 DOI: 10.1016/j.bmcl.2007.08.068  1
2007 Thomas JB, Sharpless KE, Mitvalsky S, Roman M, Yen J, Satterfield MB. Determination of caffeine and caffeine-related metabolites in ephedra-containing standard reference materials using liquid chromatography with absorbance detection and tandem mass spectrometry. Journal of Aoac International. 90: 934-40. PMID 17760330  0.48
2007 Schantz MM, Keller JM, Leigh S, Patterson DG, Sharpless KE, Sjödin A, Stapleton HM, Swarthout R, Turner WE, Wise SA. Certification of SRM 1589a PCBs, pesticides, PBDEs, and dioxins/furans in human serum Analytical and Bioanalytical Chemistry. 389: 1201-1208. PMID 17710387 DOI: 10.1007/s00216-007-1519-1  0.48
2007 Saupe SG, Sharpless KE. "doctrine of Signatures" challenge Analytical and Bioanalytical Chemistry. 389: 3-9. PMID 17646970 DOI: 10.1007/s00216-007-1465-y  0.48
2007 Dwyer JT, Holden J, Andrews K, Roseland J, Zhao C, Schweitzer A, Perry CR, Harnly J, Wolf WR, Picciano MF, Fisher KD, Saldanha LG, Yetley EA, Betz JM, Coates PM, ... ... Sharpless KE, et al. Measuring vitamins and minerals in dietary supplements for nutrition studies in the USA. Analytical and Bioanalytical Chemistry. 389: 37-46. PMID 17641882 DOI: 10.1007/s00216-007-1456-z  0.48
2007 Rimmer CA, Howerton SB, Sharpless KE, Sander LC, Long SE, Murphy KE, Porter BJ, Putzbach K, Rearick MS, Wise SA, Wood LJ, Zeisler R, Hancock DK, Yen JH, Betz JM, et al. Characterization of a suite of ginkgo-containing standard reference materials. Analytical and Bioanalytical Chemistry. 389: 179-96. PMID 17619180 DOI: 10.1007/s00216-007-1398-5  0.48
2007 Phillips KM, Wolf WR, Patterson KY, Sharpless KE, Holden JM. Reference materials to evaluate measurement systems for the nutrient composition of foods: Results from USDA's National Food and Nutrient Analysis Program (NFNAP) Analytical and Bioanalytical Chemistry. 389: 219-229. PMID 17583804 DOI: 10.1007/s00216-007-1366-0  0.48
2007 Putzbach K, Rimmer CA, Sharpless KE, Wise SA, Sander LC. Determination of bitter orange alkaloids in dietary supplement Standard Reference Materials by liquid chromatography with atmospheric-pressure ionization mass spectrometry Analytical and Bioanalytical Chemistry. 389: 197-205. PMID 17579842 DOI: 10.1007/s00216-007-1409-6  0.48
2007 Sharpless KE, Thomas JB, Christopher SJ, Greenberg RR, Sander LC, Schantz MM, Welch MJ, Wise SA. Standard reference materials for foods and dietary supplements. Analytical and Bioanalytical Chemistry. 389: 171-8. PMID 17534610 DOI: 10.1007/s00216-007-1315-y  0.48
2007 Putzbach K, Rimmer CA, Sharpless KE, Sander LC. Determination of Bitter Orange alkaloids in dietary supplements standard reference materials by liquid chromatography with ultraviolet absorbance and fluorescence detection Journal of Chromatography A. 1156: 304-311. PMID 17524413 DOI: 10.1016/j.chroma.2006.12.027  0.48
2007 Sharpless KE, Thomas JB, Duewer DL, Putzbach K, Rimmer CA, Sander LC, Schantz MM, Wise SA, Yarita T, Yen JH. Preparation and characterization of standard reference material 3276, carrot extract in oil. Analytical and Bioanalytical Chemistry. 389: 207-17. PMID 17440713 DOI: 10.1007/s00216-007-1278-z  0.48
2007 Yoo EJ, Ahlquist M, Kim SH, Bae I, Fokin VV, Sharpless KB, Chang S. Copper-catalyzed synthesis of N-sulfonyl-1,2,3-triazoles: controlling selectivity. Angewandte Chemie (International Ed. in English). 46: 1730-3. PMID 17397087 DOI: 10.1002/anie.200604241  1
2007 Hawker CJ, Fokin VV, Finn MG, Sharpless KB. Bringing efficiency to materials synthesis: The philosophy of click chemistry Australian Journal of Chemistry. 60: 381-383. DOI: 10.1071/CH07107  1
2007 Phillips KM, Wolf WR, Patterson KY, Sharpless KE, Amanna KR, Holden JM. Summary of reference materials for the determination of the nutrient composition of foods Accreditation and Quality Assurance. 12: 126-133. DOI: 10.1007/s00769-007-0257-6  0.48
2007 Sharpless KE, Ulberth F. Food and dietary supplements Analytical and Bioanalytical Chemistry. 389: 1-2. DOI: 10.1007/s00216-007-1473-y  0.48
2007 Liu Y, Díaz DD, Accurso AA, Sharpless KB, Fokin VV, Finn MG. Click chemistry in materials synthesis. III. Metal-adhesive polymers from Cu(I)-catalyzed azide-alkyne cycloaddition Journal of Polymer Science, Part a: Polymer Chemistry. 45: 5182-5189. DOI: 10.1002/pola.22262  1
2007 Vestberg R, Malkoch M, Kade M, Wu P, Fokin VV, Sharpless KB, Drockenmuller E, Hawker CJ. Role of architecture and molecular weight in the formation of tailor-made ultrathin multilayers using dendritic macromolecules and click chemistry Journal of Polymer Science, Part a: Polymer Chemistry. 45: 2835-2846. DOI: 10.1002/pola.22178  1
2007 Narayan S, Fokin VV, Sharpless KB. Chemistry 'On Water'-Organic Synthesis in Aqueous Suspension Organic Reactions in Water: Principles, Strategies and Applications. 350-365. DOI: 10.1002/9780470988817.ch11  1
2006 Dwyer JT, Picciano MF, Betz JM, Fisher KD, Saldanha LG, Yetley EA, Coates PM, Radimer K, Bindewald B, Sharpless KE, Holden J, Andrews K, Zhao C, Harnly J, Wolf WR, et al. Progress in development of an integrated dietary supplement ingredient database at the NIH Office of Dietary Supplements. Journal of Food Composition and Analysis : An Official Publication of the United Nations University, International Network of Food Data Systems. 19: S108-S114. PMID 25309034 DOI: 10.1016/j.jfca.2005.09.001  0.48
2006 Sharpless KB, Manetsch R. In situ click chemistry: a powerful means for lead discovery. Expert Opinion On Drug Discovery. 1: 525-38. PMID 23506064 DOI: 10.1517/17460441.1.6.525  1
2006 Díaz DD, Converso A, Sharpless KB, Finn MG. 2,6-Dichloro-9-thiabicyclo[3.3.1]nonane: multigram display of azide and cyanide components on a versatile scaffold. Molecules (Basel, Switzerland). 11: 212-8. PMID 17962753 DOI: 10.3390/11040212  1
2006 Sharpless KE, Anderson DL, Betz JM, Butler TA, Capar SG, Cheng J, Fraser CA, Gardner G, Gay ML, Howell DW, Ihara T, Khan MA, Lam JW, Long SE, McCooeye M, et al. Preparation and characterization of a suite of ephedra-containing standard reference materials. Journal of Aoac International. 89: 1483-95. PMID 17225593  0.48
2006 Whiting M, Tripp JC, Lin YC, Lindstrom W, Olson AJ, Elder JH, Sharpless KB, Fokin VV. Rapid discovery and structure-activity profiling of novel inhibitors of human immunodeficiency virus type 1 protease enabled by the copper(I)-catalyzed synthesis of 1,2,3-triazoles and their further functionalization. Journal of Medicinal Chemistry. 49: 7697-710. PMID 17181152 DOI: 10.1021/jm060754+  1
2006 Nelson BC, Sharpless KE, Sander LC. Improved liquid chromatography methods for the separation and quantification of biotin in NIST Standard Reference Material 3280: Multivitamin/multielement tablets Journal of Agricultural and Food Chemistry. 54: 8710-8716. PMID 17090111 DOI: 10.1021/jf062000+  0.48
2006 Nelson BC, Sharpless KE, Sander LC. Quantitative determination of folic acid in multivitamin/multielement tablets using liquid chromatography/tandem mass spectrometry Journal of Chromatography A. 1135: 203-211. PMID 17018234 DOI: 10.1016/j.chroma.2006.09.040  0.48
2006 Satterfield MB, Sniegoski LT, Sharpless KE, Welch MJ, Hornikova A, Zhang NF, Pfeiffer CM, Fazili Z, Zhang M, Nelson BC. Development of a new standard reference material: SRM 1955 (homocysteine and folate in human serum). Analytical and Bioanalytical Chemistry. 385: 612-22. PMID 16715281 DOI: 10.1007/s00216-006-0434-1  0.48
2006 Sander LC, Sharpless KE, Wise SA. Dietary supplement Standard Reference Materials Life Sciences. 78: 2044-2048. PMID 16457853 DOI: 10.1016/j.lfs.2005.12.037  0.48
2006 Whiting M, Muldoon J, Lin YC, Silverman SM, Lindstrom W, Olson AJ, Kolb HC, Finn MG, Sharpless KB, Elder JH, Fokin VV. Inhibitors of HIV-1 protease by using in situ click chemistry. Angewandte Chemie (International Ed. in English). 45: 1435-9. PMID 16425339 DOI: 10.1002/anie.200502161  1
2006 Hirose T, Sunazuka T, Noguchi Y, Yamaguchi Y, Hanaki H, Sharpless KB, Omura S. Rapid 'SAR' via click chemistry: An alkyne-bearing spiramycin is fused with diverse azides to yield new triazole-antibacterial candidates Heterocycles. 69: 55-61. DOI: 10.3987/com-06-s(o)7  1
2005 Wu P, Malkoch M, Hunt JN, Vestberg R, Kaltgrad E, Finn MG, Fokin VV, Sharpless KB, Hawker CJ. Multivalent, bifunctional dendrimers prepared by click chemistry. Chemical Communications (Cambridge, England). 5775-7. PMID 16307142 DOI: 10.1002/chin.200611077  1
2005 Radi? Z, Manetsch R, Krasi?ski A, Raushel J, Yamauchi J, Garcia C, Kolb H, Sharpless KB, Taylor P. Molecular basis of interactions of cholinesterases with tight binding inhibitors. Chemico-Biological Interactions. 157: 133-41. PMID 16289416 DOI: 10.1016/j.cbi.2005.10.020  1
2005 Zhang L, Chen X, Xue P, Sun HH, Williams ID, Sharpless KB, Fokin VV, Jia G. Ruthenium-catalyzed cycloaddition of alkynes and organic azides. Journal of the American Chemical Society. 127: 15998-9. PMID 16287266 DOI: 10.1002/chin.200612126  1
2005 Bourne Y, Radi? Z, Kolb HC, Sharpless KB, Taylor P, Marchot P. Structural insights into conformational flexibility at the peripheral site and within the active center gorge of AChE. Chemico-Biological Interactions. 157: 159-65. PMID 16259971 DOI: 10.1016/j.cbi.2005.10.018  1
2005 Feldman AK, Colasson B, Sharpless KB, Fokin VV. The allylic azide rearrangement: achieving selectivity. Journal of the American Chemical Society. 127: 13444-5. PMID 16190677 DOI: 10.1002/chin.200605124  1
2005 Sander LC, Sharpless KE, Satterfield MB, Ihara T, Phinney KW, Yen JH, Wise SA, Gay ML, Lam JW, McCooeye M, Gardner G, Fraser C, Sturgeon R, Roman M. Determination of ephedrine alkaloids in dietary supplement standard reference materials. Analytical Chemistry. 77: 3101-12. PMID 15889898 DOI: 10.1021/ac0484530  0.48
2005 Krasi?ski A, Radi? Z, Manetsch R, Raushel J, Taylor P, Sharpless KB, Kolb HC. In situ selection of lead compounds by click chemistry: target-guided optimization of acetylcholinesterase inhibitors. Journal of the American Chemical Society. 127: 6686-92. PMID 15869290 DOI: 10.1021/ja043031t  1
2005 Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. "On water": unique reactivity of organic compounds in aqueous suspension. Angewandte Chemie (International Ed. in English). 44: 3275-9. PMID 15844112 DOI: 10.1002/anie.200462883  1
2005 Woollard DC, Shoemaker DD, Ackman RG, Eitenmiller RR, Mossoba MM, Sharpless KE, Smith R, Wolf WR, Bonnin E, Phillips JG, Williams SM. Committee on Food Nutrition. Journal of Aoac International. 88: 371-2. PMID 15759763  0.48
2005 Johnson SM, Petrassi HM, Palaninathan SK, Mohamedmohaideen NN, Purkey HE, Nichols C, Chiang KP, Walkup T, Sacchettini JC, Sharpless KB, Kelly JW. Bisaryloxime ethers as potent inhibitors of transthyretin amyloid fibril formation. Journal of Medicinal Chemistry. 48: 1576-87. PMID 15743199 DOI: 10.1021/jm049274d  1
2005 Himo F, Lovell T, Hilgraf R, Rostovtsev VV, Noodleman L, Sharpless KB, Fokin VV. Copper(I)-catalyzed synthesis of azoles. DFT study predicts unprecedented reactivity and intermediates. Journal of the American Chemical Society. 127: 210-6. PMID 15631470 DOI: 10.1002/chin.200523127  1
2005 Loren JC, Krasiński A, Fokin VV, Sharpless KB. NH-1,2,3-triazoles from azidomethyl pivalate and carbamates: Base-labile N-protecting groups Synlett. 2847-2850. DOI: 10.1002/CHIN.200614133  1
2005 Loren JC, Sharpless KB. The Banert cascade: A synthetic sequence to polyfunctional NH-1,2,3-triazoles Synthesis. 1514-1520. DOI: 10.1002/chin.200541135  1
2005 Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. Cover Picture: “On Water”: Unique Reactivity of Organic Compounds in Aqueous Suspension (Angew. Chem. Int. Ed. 21/2005) Angewandte Chemie International Edition. 44: 3157-3157. DOI: 10.1002/anie.200590069  1
2005 Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. Titelbild: “On Water”: Unique Reactivity of Organic Compounds in Aqueous Suspension (Angew. Chem. 21/2005) Angewandte Chemie. 117: 3219-3219. DOI: 10.1002/ange.200590069  1
2004 Mocharla VP, Colasson B, Lee LV, Röper S, Sharpless KB, Wong CH, Kolb HC. In situ click chemistry: enzyme-generated inhibitors of carbonic anhydrase II. Angewandte Chemie (International Ed. in English). 44: 116-20. PMID 15599912 DOI: 10.1002/anie.200461580  1
2004 Converso A, Saaidi PL, Sharpless KB, Finn MG. Nucleophilic substitution by grignard reagents on sulfur mustards. The Journal of Organic Chemistry. 69: 7336-9. PMID 15471488 DOI: 10.1021/jo0489869  1
2004 Manetsch R, Krasi?ski A, Radi? Z, Raushel J, Taylor P, Sharpless KB, Kolb HC. In situ click chemistry: enzyme inhibitors made to their own specifications. Journal of the American Chemical Society. 126: 12809-18. PMID 15469276 DOI: 10.1021/ja046382g  1
2004 Chan TR, Hilgraf R, Sharpless KB, Fokin VV. Polytriazoles as copper(I)-stabilizing ligands in catalysis. Organic Letters. 6: 2853-5. PMID 15330631 DOI: 10.1021/ol0493094  1
2004 Wu P, Feldman AK, Nugent AK, Hawker CJ, Scheel A, Voit B, Pyun J, Fréchet JM, Sharpless KB, Fokin VV. Efficiency and fidelity in a click-chemistry route to triazole dendrimers by the copper(i)-catalyzed ligation of azides and alkynes. Angewandte Chemie (International Ed. in English). 43: 3928-32. PMID 15274216 DOI: 10.1002/anie.200454078  1
2004 Thomas JB, Yen JH, Schantz MM, Porter BJ, Sharpless KE. Determination of caffeine, theobromine, and theophylline in standard reference material 2384, baking chocolate, using reversed-phase liquid chromatography. Journal of Agricultural and Food Chemistry. 52: 3259-63. PMID 15161179 DOI: 10.1021/jf030817m  0.48
2004 Pearson CL, Xu K, Sharpless KE, Harris SD. MesA, a novel fungal protein required for the stabilization of polarity axes in Aspergillus nidulans. Molecular Biology of the Cell. 15: 3658-72. PMID 15155805 DOI: 10.1091/mbc.E03-11-0803  0.52
2004 Krasi?ski A, Fokin VV, Sharpless KB. Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited. Organic Letters. 6: 1237-40. PMID 15070306 DOI: 10.1002/chin.200434145  1
2004 Bourne Y, Kolb HC, Radi? Z, Sharpless KB, Taylor P, Marchot P. Freeze-frame inhibitor captures acetylcholinesterase in a unique conformation. Proceedings of the National Academy of Sciences of the United States of America. 101: 1449-54. PMID 14757816 DOI: 10.1073/pnas.0308206100  1
2004 Sharpless KE, Greenberg RR, Schantz MM, Welch MJ, Wise SA, Ihnat M. Filling the AOAC triangle with food-matrix standard reference materials Analytical and Bioanalytical Chemistry. 378: 1161-1167. PMID 14689156 DOI: 10.1007/s00216-003-2384-1  0.48
2004 Wise SA, Sharpless KE, Sander LC, May WE. Standard Reference Materials to support US regulations for nutrients and contaminants in food and dietary supplements Accreditation and Quality Assurance. 9: 543-550. DOI: 10.1007/s00769-004-0820-3  0.48
2004 Díaz DD, Punna S, Holzer P, Mcpherson AK, Sharpless KB, Fokin VV, Finn MG. Click chemistry in materials synthesis. 1. Adhesive polymers from copper-catalyzed azide-alkyne cycloaddition Journal of Polymer Science, Part a: Polymer Chemistry. 42: 4392-4403. DOI: 10.1002/pola.20330  1
2004 Wu P, Feldman AK, Nugent AK, Hawker CJ, Scheel A, Voit B, Pyun J, Fréchet JMJ, Sharpless KB, Fokin VV. Cover Picture: Efficiency and Fidelity in a Click-Chemistry Route to Triazole Dendrimers by the Copper(I)-Catalyzed Ligation of Azides and Alkynes (Angew. Chem. Int. Ed. 30/2004) Angewandte Chemie International Edition. 43: 3863-3863. DOI: 10.1002/anie.200490100  1
2004 Wu P, Feldman AK, Nugent AK, Hawker CJ, Scheel A, Voit B, Pyun J, Fréchet JMJ, Sharpless KB, Fokin VV. Titelbild: Efficiency and Fidelity in a Click-Chemistry Route to Triazole Dendrimers by the Copper(I)-Catalyzed Ligation of Azides and Alkynes (Angew. Chem. 30/2004) Angewandte Chemie. 116: 3951-3951. DOI: 10.1002/ange.200490100  1
2003 Kolb HC, Sharpless KB. The growing impact of click chemistry on drug discovery. Drug Discovery Today. 8: 1128-37. PMID 14678739 DOI: 10.1016/S1359-6446(03)02933-7  1
2003 Brik A, Muldoon J, Lin YC, Elder JH, Goodsell DS, Olson AJ, Fokin VV, Sharpless KB, Wong CH. Rapid diversity-oriented synthesis in microtiter plates for in situ screening of HIV protease inhibitors. Chembiochem : a European Journal of Chemical Biology. 4: 1246-8. PMID 14613121 DOI: 10.1002/cbic.200300724  1
2003 Sharpless KE, Phinney CS, Wood LJ, Yen JH, Howell DW. Value assignment of nutrient and aflatoxin concentrations in standard reference material 2387 peanut butter. Journal of Agricultural and Food Chemistry. 51: 6745-51. PMID 14582970 DOI: 10.1021/jf034637o  0.48
2003 Himo F, Demko ZP, Noodleman L, Sharpless KB. Why is tetrazole formation by addition of azide to organic nitriles catalyzed by zinc(II) salts? Journal of the American Chemical Society. 125: 9983-7. PMID 12914461 DOI: 10.1021/ja030204q  1
2003 Lee LV, Mitchell ML, Huang SJ, Fokin VV, Sharpless KB, Wong CH. A potent and highly selective inhibitor of human alpha-1,3-fucosyltransferase via click chemistry. Journal of the American Chemical Society. 125: 9588-9. PMID 12904015 DOI: 10.1021/ja0302836  1
2003 Ripka AS, Díaz DD, Sharpless KB, Finn MG. First practical synthesis of formamidine ureas and derivatives. Organic Letters. 5: 1531-3. PMID 12713316 DOI: 10.1002/chin.200335060  1
2003 Wang Q, Chan TR, Hilgraf R, Fokin VV, Sharpless KB, Finn MG. Bioconjugation by copper(I)-catalyzed azide-alkyne [3 + 2] cycloaddition. Journal of the American Chemical Society. 125: 3192-3. PMID 12630856 DOI: 10.1021/ja021381e  1
2003 Nelson BC, Sharpless KE. Quantification of the predominant monomeric catechins in baking chocolate standard reference material by LC/APCI-MS Journal of Agricultural and Food Chemistry. 51: 531-537. PMID 12537419 DOI: 10.1021/jf0207474  0.48
2003 Kitayama T, Yokoi T, Kawai Y, Hill RK, Morita M, Okamoto T, Yamamoto Y, Fokin VV, Sharpless KB, Sawada S. The chemistry of zerumbone. Part 5: Structural transformation of the dimethylamine derivatives Tetrahedron. 59: 4857-4866. DOI: 10.1016/S0040-4020(03)00667-7  1
2003 Beller M, Sharpless KB. Diols via Catalytic Dihydroxylation Cheminform. 34. DOI: 10.1002/chin.200327277  1
2002 Demko ZP, Sharpless KB. A click chemistry approach to tetrazoles by Huisgen 1,3-dipolar cycloaddition: synthesis of 5-acyltetrazoles from azides and acyl cyanides. Angewandte Chemie (International Ed. in English). 41: 2113-6. PMID 19746613 DOI: 10.1002/1521-3773(20020617)41:12<2113::AID-ANIE2113>3.0.CO;2-Q  1
2002 Demko ZP, Sharpless KB. A click chemistry approach to tetrazoles by Huisgen 1,3-dipolar cycloaddition: synthesis of 5-sulfonyl tetrazoles from azides and sulfonyl cyanides. Angewandte Chemie (International Ed. in English). 41: 2110-3. PMID 19746612 DOI: 10.1002/1521-3773(20020617)41:12<2110::AID-ANIE2110>3.0.CO;2-7  1
2002 Sharpless KB. Searching for new reactivity (Nobel lecture). Angewandte Chemie (International Ed. in English). 41: 2024-32. PMID 19746596 DOI: 10.1002/1521-3773(20020617)41:12<2024::AID-ANIE2024>3.0.CO;2-O  1
2002 Andersson MA, Epple R, Fokin VV, Sharpless KB. A new approach to osmium-catalyzed asymmetric dihydroxylation and aminohydroxylation of olefins. Angewandte Chemie (International Ed. in English). 41: 472-5. PMID 12491382 DOI: 10.1002/1521-3773(20020201)41:3<472::AID-ANIE472>3.0.CO;2-7  1
2002 Lewis WG, Green LG, Grynszpan F, Radi? Z, Carlier PR, Taylor P, Finn MG, Sharpless KB. Click chemistry in situ: acetylcholinesterase as a reaction vessel for the selective assembly of a femtomolar inhibitor from an array of building blocks. Angewandte Chemie (International Ed. in English). 41: 1053-7. PMID 12491310 DOI: 10.1002/1521-3757(20020315)114:6<1095::AID-ANGE1095>3.0.CO;2-3  1
2002 Sharpless KE, Brown Thomas J, Nelson BC, Phinney CS, Sieber JR, Wood LJ, Yen JH, Howell DW. Value assignment of nutrient concentrations in standard reference material 2384 baking chocolate. Journal of Agricultural and Food Chemistry. 50: 7069-75. PMID 12428961 DOI: 10.1021/jf020610d  0.48
2002 Himo F, Demko ZP, Noodleman L, Sharpless KB. Mechanisms of tetrazole formation by addition of azide to nitriles. Journal of the American Chemical Society. 124: 12210-6. PMID 12371861 DOI: 10.1021/ja0206644  1
2002 Rostovtsev VV, Green LG, Fokin VV, Sharpless KB. A stepwise huisgen cycloaddition process: copper(I)-catalyzed regioselective "ligation" of azides and terminal alkynes. Angewandte Chemie (International Ed. in English). 41: 2596-9. PMID 12203546 DOI: 10.1002/1521-3773(20020715)41:14<2596::AID-ANIE2596>3.0.CO;2-4  1
2002 Demko ZP, Sharpless KB. An expedient route to the tetrazole analogues of alpha-amino acids. Organic Letters. 4: 2525-7. PMID 12123367 DOI: 10.1021/ol020096x  1
2002 Sharpless KE, Harris SD. Functional characterization and localization of the Aspergillus nidulans formin SEPA Molecular Biology of the Cell. 13: 469-479. PMID 11854405 DOI: 10.1091/mbc.01-07-0356  0.52
2002 Dupau P, Epple R, Thomas AA, Fokin VV, Sharpless KB. Osmium-Catalyzed Dihydroxylation of Olefins in Acidic Media: Old Process, New Tricks Advanced Synthesis and Catalysis. 344: 421-433. DOI: 10.1002/1615-4169(200206)344:3/4<421::AID-ADSC421>3.0.CO;2-F  1
2002 Lewis WG, Green LG, Grynszpan F, Radić Z, Carlier PR, Taylor P, Finn MG, Sharpless KB. Cover Picture: Angew. Chem. Int. Ed. 6/2002 Angewandte Chemie International Edition. 41: 875-875. DOI: 10.1002/1521-3773(20020315)41:6<875::AID-ANIE875>3.0.CO;2-Y  1
2002 Demko ZP, Sharpless KB. A Click Chemistry Approach to Tetrazoles by Huisgen 1,3-Dipolar Cycloaddition: Synthesis of 5-Acyltetrazoles from Azides and Acyl Cyanides We thank the National Institute of General Medical Sciences, National Institutes of Health (GM-28384), the National Science Foundation (CHE-9985553), the Skaggs Institute for Chemical Biology for a Predoctoral Fellowship (Z.D.), and the W. M. Keck Foundation for financial support. Angewandte Chemie. 114: 2217. DOI: 10.1002/1521-3757(20020617)114:12<2217::aid-ange2217>3.0.co;2-x  0.92
2002 Lewis WG, Green LG, Grynszpan F, Radić Z, Carlier PR, Taylor P, Finn MG, Sharpless KB. Titelbild: 6/2002 Angewandte Chemie. 114: 915-915. DOI: 10.1002/1521-3757(20020315)114:6<915::AID-ANGE915>3.0.CO;2-3  1
2001 Demko ZP, Sharpless KB. An intramolecular [2 + 3] cycloaddition route to fused 5-heterosubstituted tetrazoles. Organic Letters. 3: 4091-4. PMID 11735592 DOI: 10.1021/ol010220x  1
2001 Demko ZP, Sharpless KB. Preparation of 5-substituted 1H-tetrazoles from nitriles in water. The Journal of Organic Chemistry. 66: 7945-50. PMID 11722189 DOI: 10.1021/jo010635w  1
2001 Fokin VV, Sharpless KB. A Practical and Highly Efficient Aminohydroxylation of Unsaturated Carboxylic Acids We thank the National Institute of General Medical Sciences, the National Institutes of Health (GM 28384), National Science Foundation (CHE-9985553), and the W. M. Keck Foundation for financial support. We are also grateful to Prof. M. G. Finn, Dr. Wallace Pringle, and Dr. A. Erik Rubin for many helpful discussions. Angewandte Chemie (International Ed. in English). 40: 3455-3457. PMID 11592169 DOI: 10.1002/1521-3773(20010917)40:18<3455::AID-ANIE3455>3.0.CO;2-I  1
2001 Sharpless KE, Colbert JC, Greenberg RR, Schantz MM, Welch MJ. Recent developments in food-matrix Reference Materials at NIST Analytical and Bioanalytical Chemistry. 370: 275-278. PMID 11451251  0.48
2001 Kolb HC, Finn MG, Sharpless KB. Click Chemistry: Diverse Chemical Function from a Few Good Reactions. Angewandte Chemie (International Ed. in English). 40: 2004-2021. PMID 11433435 DOI: 10.1002/1521-3773(20010601)40:11<2004::AID-ANIE2004>3.0.CO;2-5  1
2001 Petrassi HM, Sharpless KB, Kelly JW. The copper-mediated cross-coupling of phenylboronic acids and N-hydroxyphthalimide at room temperature: synthesis of aryloxyamines. Organic Letters. 3: 139-42. PMID 11429858 DOI: 10.1021/ol0003533  1
2001 Marzinzik AL, Sharpless KB. A simple method for the preparation of N-sulfonylsulfilimines from sulfides. The Journal of Organic Chemistry. 66: 594-6. PMID 11429835 DOI: 10.1021/jo0012039  1
2001 Converso A, Burow K, Marzinzik A, Sharpless KB, Finn MG. 2,6-Dichloro-9-thiabicyclo[3.3.1]nonane: a privileged, bivalent scaffold for the display of nucleophilic components. The Journal of Organic Chemistry. 66: 4386-92. PMID 11397181 DOI: 10.1021/jo015632y  1
2001 Welch MJ, Colbert JC, Gill LM, Phinney CS, Sharpless KE, Sniegoski LT, Wood LJ. The certification of SRM 1546--Meat Homogenate, a new reference material for nutrients in a high protein, high fat matrix. Fresenius' Journal of Analytical Chemistry. 370: 42-7. PMID 11393235  0.48
2001 Brown Thomas J, Kline MC, Gill LM, Yen JH, Duewer DL, Sniegoski LT, Sharpless KE. Preparation and value assignment of Standard Reference Material 968c Fat-Soluble Vitamins, Carotenoids, and Cholesterol in Human Serum. Clinica Chimica Acta; International Journal of Clinical Chemistry. 305: 141-55. PMID 11249933 DOI: 10.1016/S0009-8981(00)00429-0  0.48
2001 Chuang T, Sharpless KB. ChemInform Abstract: Applications of Aziridinium Ions. Selective Syntheses of α,β-Diamino Esters, α-Sulfanyl-β-amino Esters, β-Lactams, and 1,5-Benzodiazepin-2-one. Cheminform. 32: no-no. DOI: 10.1002/chin.200111049  0.48
2001 Kolb HC, Finn MG, Sharpless KB. Click-Chemie: diverse chemische Funktionalität mit einer Handvoll guter Reaktionen Angewandte Chemie. 113: 2056-2075. DOI: 10.1002/1521-3757(20010601)113:11<2056::AID-ANGE2056>3.0.CO;2-W  1
2001 Irurre J, Knowles WS, Noyori R, Sharpless KB. The nobel prizes in chemistry 2001 and his contribution. A hundred years of nobel prizes (1901-2001) | Los premios nobel de química 2001 y su aportación. Cien años de premios nobel (1901-2001) Afinidad. 58: 411-415.  1
2000 Chuang TH, Sharpless KB. Applications of aziridinium ions. Selective syntheses of alpha, beta-diamino esters, alpha-sulfanyl-beta-amino esters, beta-lactams, and 1,5-benzodiazepin-2-one. Organic Letters. 2: 3555-7. PMID 11073643  0.68
2000 Duewer DL, Kline MC, Sharpless KE, Thomas JB. NIST micronutrients measurement quality assurance program: characterizing the measurement community's performance over time. Analytical Chemistry. 72: 4163-70. PMID 10994979 DOI: 10.1021/ac991480j  0.48
2000 Duewer DL, Kline MC, Sharpless KE, Thomas JB, Stacewicz-Sapuntzakis M, Sowell AL. NIST micronutrients measurement quality assurance program: characterizing individual participant measurement performance over time. Analytical Chemistry. 72: 3611-9. PMID 10952550 DOI: 10.1021/ac991481b  0.48
2000 Demko ZP, Bartsch M, Sharpless KB. Primary amides. A general nitrogen source for catalytic asymmetric aminohydroxylation of olefins. Organic Letters. 2: 2221-3. PMID 10930248 DOI: 10.1021/ol000098m  1
2000 Sharpless KE, Margolis S, Thomas JB. Determination of vitamins in food-matrix Standard Reference Materials. Journal of Chromatography. A. 881: 171-81. PMID 10905701 DOI: 10.1016/S0021-9673(00)00260-0  0.48
2000 Sander LC, Sharpless KE, Pursch M. C30 Stationary phases for the analysis of food by liquid chromatography Journal of Chromatography A. 880: 189-202. PMID 10890520 DOI: 10.1016/S0021-9673(00)00121-7  0.48
2000 Sharpless KE, Gill LM. Value assignment of nutrient concentrations in five standard reference materials and six reference materials. Journal of Aoac International. 83: 413-23. PMID 10772181  0.48
2000 Demko ZP, Bartsch M, Sharpless KB. ChemInform Abstract: Primary Amides. A General Nitrogen Source for Catalytic Asymmetric Aminohydroxylation of Olefins. Cheminform. 31: no-no. DOI: 10.1002/chin.200045098  0.92
2000 Chuang TH, Sharpless KB. Applications of aziridinium ions: Selective syntheses of pyrazolidin-3-ones and pyrazolo[1,2-α]pyrazoles Helvetica Chimica Acta. 83: 1734-1743. DOI: 10.1002/1522-2675(20000809)83:8<1734::AID-HLCA1734>3.0.CO;2-E  1
2000 Chuang TH, Sharpless KB. Applications of aziridinium ions. Selective syntheses of α,β-diamino esters, α-sulfanyl-β-amino esters, β-lactams, and 1,5-benzodiazepin-2-one Organic Letters. 2: 3555-3557.  1
1999 Goossen LJ, Liu H, Dress KR, Sharpless KB. Catalytic asymmetric aminohydroxylation with amino-substituted heterocycles as nitrogen sources. Angewandte Chemie (International Ed. in English). 38: 1080-3. PMID 25138500 DOI: 10.1002/(SICI)1521-3773(19990419)38:8<1080::AID-ANIE1080>3.0.CO;2-D  1
1999 Thomas AA, Sharpless KB. The Catalytic Asymmetric Aminohydroxylation of Unsaturated Phosphonates. The Journal of Organic Chemistry. 64: 8379-8385. PMID 11674762 DOI: 10.1021/jo990060r  1
1999 Chuang TH, Sharpless KB. Applications of aziridinium ions. Selective syntheses of beta-aryl-alpha,beta-diamino esters. Organic Letters. 1: 1435-7. PMID 10825990  1
1999 Gontcharov AV, Liu H, Sharpless KB. Tert-butylsulfonamide. A new nitrogen source for catalytic aminohydroxylation and aziridination of olefins. Organic Letters. 1: 783-6. PMID 10823205 DOI: 10.1021/ol990761a  1
1999 Duewer DL, Kline MC, Sharpless KE, Thomas JB, Gary KT, Sowell AL. Micronutrients Measurement Quality Assurance Program: helping participants use interlaboratory comparison exercise results to improve their long-term measurement performance. Analytical Chemistry. 71: 1870-8. PMID 10330911 DOI: 10.1021/ac981074k  0.48
1999 Sharpless KE, Arce-Osuna M, Thomas JB, Gill LM. Value assignment of retinol, retinyl palmitate, tocopherol, and carotenoid concentrations in Standard Reference Material 2383 (Baby Food Composite). Journal of Aoac International. 82: 288-96. PMID 10191535  0.48
1999 Sharpless KE, Gill LM, Margolis SA, Wise SA, Elkins E. Preparation of Standard Reference Material 2383 (Baby Food Composite) and use of an interlaboratory comparison exercise for value assignment of its nutrient concentrations. Journal of Aoac International. 82: 276-87. PMID 10191534  0.48
1999 Pringle W, Sharpless KB. The osmium-catalyzed aminohydroxylation of Baylis-Hillman olefins Tetrahedron Letters. 40: 5151-5154. DOI: 10.1016/S0040-4039(99)00887-4  1
1999 Adolfsson H, Converso A, Sharpless KB. Comparison of amine additives most effective in the new methyltrioxorhenium-catalyzed epoxidation process Tetrahedron Letters. 40: 3991-3994. DOI: 10.1016/S0040-4039(99)00661-9  1
1999 Gooßen LJ, Liu H, Dress KR, Sharpless KB. Katalytische asymmetrische Aminohydroxylierung mit Amino-substituierten Heterocyclen als Stickstoffquelle Angewandte Chemie. 111: 1149-1152. DOI: 10.1002/(SICI)1521-3757(19990419)111:8<1149::AID-ANGE1149>3.0.CO;2-D  0.56
1998 Gypser A, Michel D, Nirschl DS, Sharpless KB. Dihydroxylation of Polyenes Using Narasaka's Modification of the Upjohn Procedure. The Journal of Organic Chemistry. 63: 7322-7327. PMID 11672379 DOI: 10.1021/jo980850l  0.84
1998 Brown Thomas J, Duewer DL, Kline MC, Sharpless KE. The stability of retinol, alpha-tocopherol, trans-lycopene, and trans-beta-carotene in liquid-frozen and lyophilized serum. Clinica Chimica Acta; International Journal of Clinical Chemistry. 276: 75-87. PMID 9760021 DOI: 10.1016/S0009-8981(98)00103-X  0.48
1998 Copéret C, Adolfsson H, Khuong TAV, Yudin AK, Sharpless KB. A simple and efficient method for the preparation of pyridine N-oxides Journal of Organic Chemistry. 63: 1740-1741. DOI: 10.1021/jo9723467  1
1998 Jeong JU, Tao B, Sagasser I, Henniges H, Sharpless KB. Bromine-catalyzed aziridination of olefins. A rare example of atom-transfer redox catalysis by a main group element Journal of the American Chemical Society. 120: 6844-6845. DOI: 10.1021/ja981419g  1
1998 Dress KR, Gooßen LJ, Liu H, Jerina DM, Sharpless KB. Catalytic aminohydroxylation using adenine-derivatives as the nitrogen source Tetrahedron Letters. 39: 7669-7672. DOI: 10.1016/S0040-4039(98)01716-X  1
1998 Reddy KL, Dress KR, Sharpless KB. N-chloro-N-sodio-2-trimethylsilyl ethyl carbamate: A new nitrogen source for the catalytic asymmetric aminohydroxylation Tetrahedron Letters. 39: 3667-3670. DOI: 10.1016/S0040-4039(98)00644-3  1
1998 Tao B, Schlingloff G, Sharpless KB. Reversal of regioselection in the asymmetric aminohydroxylation of cinnamates Tetrahedron Letters. 39: 2507-2510. DOI: 10.1016/S0040-4039(98)00350-5  1
1998 Copéret C, Adolfsson H, Chiang JP, Yudin AK, Sharpless KB. A simple and efficient method for the preparation of pyridine-N-oxides II Tetrahedron Letters. 39: 761-764. DOI: 10.1016/S0040-4039(97)10619-0  1
1998 Sharpless KE, Welch MJ, Greenberg RR, Iyengar GV, Colbert JC. Recent SRMs for organic and inorganic nutrients in food matrices Fresenius' Journal of Analytical Chemistry. 360: 456-458.  0.48
1997 Yudin AK, Sharpless KB. Bis(trimethylsilyl) peroxide extends the range of oxorhenium catalysts for olefin epoxidation [2] Journal of the American Chemical Society. 119: 11536-11537. DOI: 10.1021/ja973043x  1
1997 DelMonte AJ, Haller J, Houk KN, Sharpless KB, Singleton DA, Strassner T, Thomas AA. Experimental and theoretical kinetic isotope effects for asymmetric dihydroxylation. Evidence supporting a rate-limiting '(3+2)' cycloaddition Journal of the American Chemical Society. 119: 9907-9908. DOI: 10.1021/ja971650e  1
1997 Nelson DW, Gypser A, Ho PT, Kolb HC, Kondo T, Kwong HL, McGrath DV, Rubin AE, Norrby PO, Gable KP, Sharpless KB. Toward an understanding of the high enantioselectivity in the osmium-catalyzed asymmetric dihydroxylation. 4. Electronic effects in amine-accelerated osmylations Journal of the American Chemical Society. 119: 1840-1858. DOI: 10.1021/ja961464t  1
1997 Bruncko M, Schlingloff G, Sharpless KB. N-Bromoacetamide—A New Nitrogen Source for the Catalytic Asymmetric Aminohydroxylation of Olefins Angewandte Chemie International Edition in English. 36: 1483-1486. DOI: 10.1002/anie.199714831  0.48
1997 Bruncko M, Schlingloff G, Sharpless KB. N-Bromacetamid - eine neue Stickstoffquelle für die katalytische asymmetrische Aminohydroxylierung Angewandte Chemie. 109: 1580-1583. DOI: 10.1002/ange.19971091340  0.48
1996 Vanhessche KP, Sharpless KB. Ligand-Dependent Reversal of Facial Selectivity in the Asymmetric Dihydroxylation. The Journal of Organic Chemistry. 61: 7978-7979. PMID 11667767 DOI: 10.1021/jo961189t  1
1996 Chang HT, Sharpless KB. Molar Scale Synthesis of Enantiopure Stilbene Oxide. The Journal of Organic Chemistry. 61: 6456-6457. PMID 11667495 DOI: 10.1021/jo960718q  1
1996 Li G, Sharpless KB. Catalytic asymmetric aminohydroxylation provides a short taxol side-chain synthesis. Acta Chemica Scandinavica (Copenhagen, Denmark : 1989). 50: 649-51. PMID 8756354 DOI: 10.3891/acta.chem.scand.50-0649  1
1996 Norrby P, Becker H, Sharpless KB. Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation. 3. New Insights into Isomeric Forms of the Putative Osmaoxetane Intermediate Journal of the American Chemical Society. 118: 35-42. DOI: 10.1021/ja952470c  0.92
1996 Chang HT, Sharpless KB. A practical route to enantiopure 1,2-aminoalcohols Tetrahedron Letters. 37: 3219-3222. DOI: 10.1016/0040-4039(96)00534-5  1
1996 Li G, Angert HH, Sharpless KB. N-Halocarbamate Salts Lead to More Efficient Catalytic Asymmetric Aminohydroxylation Angewandte Chemie International Edition in English. 35: 2813-2817. DOI: 10.1002/anie.199628131  1
1996 Li G, Chang H, Sharpless KB. Catalytic Asymmetric Aminohydroxylation(AA) of Olefins Angewandte Chemie International Edition in English. 35: 451-454. DOI: 10.1002/anie.199604511  1
1996 Becker H, Sharpless KB. A New Ligand Class for the Asymmetric Dihydroxylation of Olefins Angewandte Chemie International Edition in English. 35: 448-451. DOI: 10.1002/anie.199604481  0.64
1996 Chang H, Chen C, Kondo T, Siuzdak G, Sharpless KB. Asymmetric Dihydroxylation Enables Rapid Construction of Chiral Dendrimers Based on 1,2-Diols Angewandte Chemie International Edition in English. 35: 182-186. DOI: 10.1002/anie.199601821  1
1996 Li G, Angert HH, Sharpless KB. Erhöhung der Effizienz der katalytischen asymmetrischen Aminohydroxylierung durchN-Halogencarbamat-Salze Angewandte Chemie. 108: 2995-2999. DOI: 10.1002/ange.19961082325  1
1996 Li G, Chang H, Sharpless KB. Katalytische asymmetrische Aminohydroxylierung (AA) von Olefinen Angewandte Chemie. 108: 449-452. DOI: 10.1002/ange.19961080409  1
1996 Becker H, Sharpless KB. Eine neue Ligandenklasse für die asymmetrische Dihydroxylierung von Olefinen Angewandte Chemie. 108: 447-449. DOI: 10.1002/ange.19961080408  0.64
1996 Chang H, Chen C, Kondo T, Siuzdak G, Sharpless KB. Asymmetrische Dihydroxylierung zum schnellen Aufbau von chiralen Dendrimeren aus 1,2-Diolen Angewandte Chemie. 108: 202-206. DOI: 10.1002/ange.19961080217  1
1995 Berrisford DJ, Bolm C, Sharpless KB. Ligand-Accelerated Catalysis Angewandte Chemie International Edition in English. 34: 1059-1070. DOI: 10.1002/anie.199510591  1
1994 Norrby PO, Kolb HC, Sharpless KB. Calculations on the reaction of ruthenium tetroxide with olefins using density functional theory (DFT). Implications for the possibility of intermediates in osmium-catalyzed asymmetric dihydroxylation Organometallics. 13: 344-347. DOI: 10.1021/om00013a050  1
1994 Wang Z, Sharpless KB. A Solid-to-Solid Asymmetric Dihydroxylation Procedure for Kilogram-Scale Preparation of Enantiopure Hydrobenzoin The Journal of Organic Chemistry. 59: 8302-8303. DOI: 10.1021/jo00105a065  1
1994 Wang Z, Kolb HC, Sharpless KB. Large-Scale and Highly Enantioselective Synthesis of the Taxol C-13 Side Chain through Asymmetric Dihydroxylation The Journal of Organic Chemistry. 59: 5104-5105. DOI: 10.1021/jo00096a072  1
1994 Norrby P, Kolb HC, Sharpless KB. Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation. 2. A Qualitative Molecular Mechanics Approach Journal of the American Chemical Society. 116: 8470-8478. DOI: 10.1021/ja00098a006  1
1994 Kolb HC, Andersson PG, Sharpless KB. Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation (AD). 1. Kinetics Journal of the American Chemical Society. 116: 1278-1291. DOI: 10.1021/ja00083a014  1
1994 Kolb HC, VanNieuwenhze MS, Sharpless KB. Catalytic Asymmetric Dihydroxylation Chemical Reviews. 94: 2483-2547. DOI: 10.1021/cr00032a009  1
1994 King SB, Sharpless KB. An efficient synthesis of enantiomerically pure trans-2-phenylcyclohexanol Tetrahedron Letters. 35: 5611-5612. DOI: 10.1016/S0040-4039(00)77259-5  1
1994 Xu D, Park CY, Sharpless KB. Study of the regio- and enantioselectivity of the reactions of osmium tetroxide with allylic alcohols and allylic sulfonamides Tetrahedron Letters. 35: 2495-2498. DOI: 10.1016/S0040-4039(00)77153-X  1
1994 VanNieuwenhze MS, Sharpless KB. The asymmetric dihydroxylation of cis-allylic and homoallylic alcohols Tetrahedron Letters. 35: 843-846. DOI: 10.1016/S0040-4039(00)75978-8  1
1994 Crispino GA, Makita A, Wang ZM, Sharpless KB. A comparison of ligands proposed for the asymmetric dihydroxylation Tetrahedron Letters. 35: 543-546. DOI: 10.1016/S0040-4039(00)75833-3  1
1994 Vanhessche KPM, Wang ZM, Sharpless KB. Asymmetric dihydroxylation of primary allylic halides and a concise synthesis of (-)-diepoxybutane Tetrahedron Letters. 35: 3469-3472. DOI: 10.1016/S0040-4039(00)73212-6  1
1994 Sharpless KB. Coelacanths and catalysis Tetrahedron. 50: 4235-4258. DOI: 10.1016/S0040-4020(01)89364-9  1
1994 Bennani YL, Vanhessche KPM, Sharpless KB. A short route to a moshe'rs acid precursor via catalytic asymmetric dihydroxylation (AD) Tetrahedron: Asymmetry. 5: 1473-1476. DOI: 10.1016/0957-4166(94)80116-9  1
1994 Becker H, Tong Ho P, Kolb HC, Loren S, Norrby PO, Sharpless KB. Comparing two models for the selectivity in the asymmetric dihydroxylation reaction (AD) Tetrahedron Letters. 35: 7315-7318. DOI: 10.1016/0040-4039(94)85302-9  1
1993 Kalantar TH, Sharpless KB. Transformations of hydroxy cyclic sulfates: stereospecific conversion into 2,3,5-trisubstituted tetrahydrofurans. Acta Chemica Scandinavica (Copenhagen, Denmark : 1989). 47: 307-13. PMID 8435231 DOI: 10.3891/acta.chem.scand.47-0307  1
1993 Crispino GA, Ho PT, Sharpless KB. Selective perhydroxylation of squalene: taming the arithmetic demon. Science (New York, N.Y.). 259: 64-6. PMID 8418495 DOI: 10.1126/science.8418495  1
1993 Walsh PJ, Sharpless KB. Asymmetric Dihydroxylation (AD) of α,β-Unsaturated Ketones Synlett. 1993: 605-606. DOI: 10.1055/s-1993-22548  1
1993 Wang Z, Sharpless KB. Asymmetric Dihydroxylation of α-Substituted Styrene Derivatives Synlett. 1993: 603-604. DOI: 10.1055/s-1993-22547  1
1993 Crispino GA, Sharpless KB. Enantioselective Synthesis of Both Enantiomers of 7,7-Dimethyl-6,8-dioxa-bicyclo[3.2.1]octane via Regioselective Asymmetric Dihydroxylation Synlett. 1993: 47-48. DOI: 10.1055/s-1993-22343  0.6
1993 Amberg W, Bennani YL, Chadha RK, Crispino GA, Davis WD, Hartung J, Jeong KS, Ogino Y, Shibata T, Sharpless KB. Syntheses and crystal structures of the cinchona alkaloid derivatives used as ligands in the osmium-catalyzed asymmetric dihydroxylation of olefins The Journal of Organic Chemistry. 58: 844-849. DOI: 10.1021/jo00056a015  0.76
1993 Kolb HC, Andersson PG, Bennani YL, Crispino GA, Jeong KS, Kwong HL, Sharpless KB. On "The origin of high enantioselectivity in the dihydroxylation of olefins using osmium tetraoxide and cinchona alkaloid catalysts" Journal of the American Chemical Society. 115: 12226-12227. DOI: 10.1021/ja00078a096  1
1993 VanNieuwenhze MS, Sharpless KB. Kinetic resolution of racemic olefins via asymmetric dihydroxylation Journal of the American Chemical Society. 115: 7864-7865. DOI: 10.1021/ja00070a037  0.92
1993 Andersson PG, Sharpless KB. A dramatic ligand effect on the relative reactivities of substituted alkenes with osmium tetroxide Journal of the American Chemical Society. 115: 7047-7048. DOI: 10.1021/ja00068a102  1
1993 McGrath DV, Brabson GD, Sharpless KB, Andrews L. Reinvestigation of the infrared spectra of oxoosmium(VI) esters by isotopic labeling Inorganic Chemistry. 32: 4164-4165. DOI: 10.1021/ic00071a035  0.68
1993 Kolb HC, Bennani YL, Sharpless KB. Short and practical syntheses of(R)-(-)-carnitine and (R)-(-)-γ-amino-β-hydroxybutyric acid (GABOB) Tetrahedron: Asymmetry. 4: 133-141. DOI: 10.1016/S0957-4166(00)86023-1  1
1993 Wang ZM, Zhang XL, Sharpless KB. Asymmetric dihydroxylation of aryl allyl ethers Tetrahedron Letters. 34: 2267-2270. DOI: 10.1016/S0040-4039(00)77590-3  1
1993 Xu D, Sharpless KB. A simple route to enantiomerically enriched oxazolidin-2-ones Tetrahedron Letters. 34: 951-952. DOI: 10.1016/S0040-4039(00)77462-4  1
1993 Morikawa K, Sharpless KB. Double diastereoselection in asymmetric dihydroxylation Tetrahedron Letters. 34: 5575-5578. DOI: 10.1016/S0040-4039(00)73885-8  1
1993 Walsh PJ, Bennani YL, Sharpless KB. Asymmetric dihydroxylation (AD)/cyclization of N-diBoc allylic and homoallylic amines: Selective differentiation of the hydroxyl groups Tetrahedron Letters. 34: 5545-5548. DOI: 10.1016/S0040-4039(00)73877-9  1
1993 Wang ZM, Sharpless KB. Asymmetric dihydroxylation of tertiary allylic alcohols Tetrahedron Letters. 34: 8225-8228. DOI: 10.1016/S0040-4039(00)61396-5  1
1993 Bennani YL, Sharpless KB. Asymmetric Synthesis of γ-Hydroxy α,β-Unsaturated Amides via an AD-elimination Process; Synthesis of (+)-Coriolic Acid Tetrahedron Letters. 34: 2083-2086. DOI: 10.1016/S0040-4039(00)60351-9  1
1993 Bennani YL, Sharpless KB. Asymmetric dihydroxylation (AD) of N,N-dialkyl and N-methoxy-N-methyl α,β- and β,γ-unsaturated amides Tetrahedron Letters. 34: 2079-2082. DOI: 10.1016/S0040-4039(00)60350-7  1
1993 Arrington MP, Bennani YL, Göbel T, Walsh P, Zhao SH, Sharpless KB. Modified cinchona alkaloid ligands: Improved selectivities in the osmium tetroxide catalyzed asymmetric dihydroxylation (AD) of terminal olefins Tetrahedron Letters. 34: 7375-7378. DOI: 10.1016/S0040-4039(00)60129-6  1
1992 Sharpless KB, Amberg W, Bennani YL, Crispino GA, Hartung J, Jeong KS, Kwong HL, Morikawa K, Wang ZM. The osmium-catalyzed asymmetric dihydroxylation: a new ligand class and a process improvement The Journal of Organic Chemistry. 57: 2768-2771. DOI: 10.1021/jo00036a003  0.92
1992 Xu D, Crispino GA, Sharpless KB. Selective asymmetric dihydroxylation (AD) of dienes Journal of the American Chemical Society. 114: 7570-7571. DOI: 10.1021/ja00045a043  0.84
1992 Jeong KS, Sjö P, Sharpless KB. Asymmetric dihydroxylation of enynes Tetrahedron Letters. 33: 3833-3836. DOI: 10.1016/S0040-4039(00)74797-6  1
1992 Crispino GA, Sharpless KB. Asymmetric dihydroxylation of squalene Tetrahedron Letters. 33: 4273-4274. DOI: 10.1016/S0040-4039(00)74236-5  1
1992 Kolb HC, Sharpless KB. A simplified procedure for the stereospecific transformation of 1,2-diols into epoxides Tetrahedron. 48: 10515-10530. DOI: 10.1016/S0040-4020(01)88349-6  1
1992 Oi R, Sharpless KB. Asymmetric dihydroxylation of acrolein acetals: synthesis of stable equivalents of Enantiopure glyceraldehyde and glycidaldehyde Tetrahedron Letters. 33: 2095-2098. DOI: 10.1016/0040-4039(92)88149-Y  1
1991 McKee BH, Kalantar TH, Sharpless KB. Subtle effects in the asymmetric epoxidation: dependence of kinetic resolution efficiency on the monodentate alkoxide ligands of the bystander titanium center The Journal of Organic Chemistry. 56: 6966-6968. DOI: 10.1021/jo00025a003  0.44
1991 Finn MG, Sharpless KB. Mechanism of asymmetric epoxidation. 2. Catalyst structure Journal of the American Chemical Society. 113: 113-126. DOI: 10.1021/ja00001a019  1
1991 Woodard SS, Finn MG, Sharpless KB. Mechanism of asymmetric epoxidation. 1. Kinetics Journal of the American Chemical Society. 113: 106-113. DOI: 10.1021/ja00001a018  1
1991 Park CY, Kim BM, Sharpless KB. Catalytic osmylation of conjugated dienes: a one-pot stereoselective synthesis of polyols Tetrahedron Letters. 32: 1003-1006. DOI: 10.1016/S0040-4039(00)74472-8  1
1991 Oi R, Sharpless KB. Stereospecific conversion of chiral 1,2-cyclic sulfates to chiral imidazolines Tetrahedron Letters. 32: 999-1002. DOI: 10.1016/S0040-4039(00)74471-6  1
1991 Ogino Y, Chen H, Kwong HL, Sharpless KB. On the timing of hydrolysis / reoxidation in the osmium-catalyzed asymmetric dihydroxylation of olefins using potassium ferricyanide as the reoxidant Tetrahedron Letters. 32: 3965-3968. DOI: 10.1016/0040-4039(91)80601-2  1
1990 Shibata T, Gilheany DG, Blackburn BK, Sharpless KB. Ligand-based improvement of enantioselectivity in the catalytic asymmetric dihydroxylation of dialkyl substituted olefins Tetrahedron Letters. 31: 3817-3820. DOI: 10.1016/S0040-4039(00)97477-X  1
1990 Moon Kim B, Sharpless KB. Heterogeneous catalytic asymmetric dihydroxylation: Use of a polymer-bound alkaloid Tetrahedron Letters. 31: 3003-3006. DOI: 10.1016/S0040-4039(00)89009-7  1
1990 DIJKSTRA GDH, KELLOGG RM, WYNBERG H, SVENDSEN JS, MARKO I, SHARPLESS KB. ChemInform Abstract: Conformational Study of Cinchona Alkaloids. A Combined NMR, Molecular Mechanics, and X-Ray Approach. Cheminform. 21. DOI: 10.1002/chin.199005282  0.64
1990 Pearlstein RM, Blackburn BK, Davis WM, Sharpless KB. Structural Characterization of the Pseudoenantiomericcis-Dioxo Osmium(VI) Esters of Chiral Diols with Cinchona Alkaloid Ligands Angewandte Chemie International Edition in English. 29: 639-641. DOI: 10.1002/anie.199006391  0.44
1990 Pearlstein RM, Blackburn BK, Davis WM, Sharpless KB. Strukturelle Charakterisierung pseudoenantiomerercis-Dioxoosmium(VI)-Komplexe mit chiralen Diolen und Cinchona-Alkaloid-Liganden Angewandte Chemie. 102: 710-712. DOI: 10.1002/ange.19901020630  0.44
1989 Carlier PR, Sharpless KB. Studies on the mechanism of the asymmetric epoxidation: a ligand variation approach The Journal of Organic Chemistry. 54: 4016-4018. DOI: 10.1021/jo00278a004  1
1989 Svendsen JS, Marko I, Jacobsen EN, Rao CP, Bott S, Sharpless KB. The structure of osmium tetraoxide-cinchona alkaloid complexes The Journal of Organic Chemistry. 54: 2263-2264. DOI: 10.1021/jo00271a002  0.64
1989 Klunder JM, Onami T, Sharpless KB. Arenesulfonate derivatives of homochiral glycidol: versatile chiral building blocks for organic synthesis The Journal of Organic Chemistry. 54: 1295-1304. DOI: 10.1021/jo00267a014  0.68
1989 Wai JSM, Marko I, Svendsen JS, Finn MG, Jacobsen EN, Sharpless KB. A mechanistic insight leads to a greatly improved osmium-catalyzed asymmetric dihydroxylation process Journal of the American Chemical Society. 111: 1123-1125. DOI: 10.1021/ja00185a050  1
1989 Jacobsen EN, Marko I, France MB, Svendsen JS, Sharpless KB. Kinetic role of the alkaloid ligands in asymmetric catalytic dihydroxylation Journal of the American Chemical Society. 111: 737-739. DOI: 10.1021/ja00184a055  0.64
1989 Kim BM, Sharpless KB. Cyclic sulfates containing acid-sensitive groups and chemoselective hydrolysis of sulfate esters Tetrahedron Letters. 30: 655-658. DOI: 10.1016/S0040-4039(01)80274-4  1
1989 Lohray BB, Gao Y, Sharpless KB. One pot synthesis of homochiral aziridines and aminoalcohols from homochiral 1,2-cyclic sulfates Tetrahedron Letters. 30: 2623-2626. DOI: 10.1016/S0040-4039(00)99081-6  1
1989 LOHRAY BB, KALANTAR TH, KIM BM, PARK CY, SHIBATA T, WAI JSM, SHARPLESS KB. ChemInform Abstract: Documenting the Scope of the Catalytic Asymmetric Dihydroxylation. Cheminform. 20. DOI: 10.1002/chin.198948090  0.64
1989 SVENDSEN JS, SHARPLESS KB. ChemInform Abstract: Type I Intramolecular Cycloadditions of Vinylketenes Cheminform. 20. DOI: 10.1002/chin.198943295  0.64
1989 GAO Y, SHARPLESS KB. ChemInform Abstract: Ti(O-i-Pr)4-Mediated Formation of 2,3-Epithio Alcohols from 2,3-Epoxy Alcohols. Cheminform. 20. DOI: 10.1002/chin.198905175  0.8
1988 Caron M, Carlier PR, Sharpless KB. Regioselective azide opening of 2,3-epoxy alcohols by [Ti(O-i-Pr)2(N3)2]: synthesis of .alpha.-amino acids The Journal of Organic Chemistry. 53: 5185-5187. DOI: 10.1021/jo00256a063  1
1988 Gao Y, Sharpless KB. Titanium isopropoxide mediated formation of 2,3-epithio alcohols from 2,3-epoxy alcohols The Journal of Organic Chemistry. 53: 4114-4116. DOI: 10.1021/jo00252a046  0.8
1988 Gao Y, Sharpless KB. Asymmetric synthesis of both enantiomers of tomoxetine and fluoxetine. Selective reduction of 2,3-epoxycinnamyl alcohol with Red-Al The Journal of Organic Chemistry. 53: 4081-4084. DOI: 10.1021/jo00252a036  0.8
1988 Gao Y, Sharpless KB. Vicinal diol cyclic sulfates. Like epoxides only more reactive Journal of the American Chemical Society. 110: 7538-7539. DOI: 10.1021/ja00230a045  0.8
1988 Carlier PR, Mungall WS, Schroder G, Sharpless KB. Enhanced kinetic resolution and enzyme-like shape selectivity Journal of the American Chemical Society. 110: 2978-2979. DOI: 10.1021/ja00217a052  1
1988 Jacobsen EN, Marko I, Mungall WS, Schroeder G, Sharpless KB. Asymmetric dihydroxylation via ligand-accelerated catalysis Journal of the American Chemical Society. 110: 1968-1970. DOI: 10.1021/ja00214a053  0.64
1988 Bolm C, Sharpless KB. Synthesis of a C3-symmetric phospha[2.2.2]cyclophane Tetrahedron Letters. 29: 5101-5104. DOI: 10.1016/S0040-4039(00)80690-5  1
1988 BOLM C, DAVIS WM, HALTERMAN RL, SHARPLESS KB. ChemInform Abstract: Synthesis and Structure of a Chiral, C3-Symmetric Monophosphane. Cheminform. 19. DOI: 10.1002/chin.198841254  1
1988 Bolm C, Davis WM, Halterman RL, Sharpless KB. Synthesis and Crystal Structure of a ChiralC3-Symmetric Monophosphane Angewandte Chemie International Edition in English. 27: 835-837. DOI: 10.1002/anie.198808351  1
1988 Bolm C, Davis WM, Halterman RL, Barry Sharpless K. Synthese und Struktur eines chiralen,C3-symmetrischen Monophosphans Angewandte Chemie. 100: 882-883. DOI: 10.1002/ange.19881000625  0.4
1987 Klunder JM, Sharpless KB. Convenient synthesis of sulfinate esters from sulfonyl chlorides The Journal of Organic Chemistry. 52: 2598-2602. DOI: 10.1021/jo00388a051  0.68
1987 Ko SY, Masamune H, Sharpless KB. p-Nitrobenzoate esters of epoxy alcohols: convenient synthons for water-soluble epoxy alcohols The Journal of Organic Chemistry. 52: 667-671. DOI: 10.1021/jo00380a032  0.6
1987 Gao Y, Klunder JM, Hanson RM, Masamune H, Ko SY, Sharpless KB. Catalytic asymmetric epoxidation and kinetic resolution: modified procedures including in situ derivatization Journal of the American Chemical Society. 109: 5765-5780. DOI: 10.1021/ja00253a032  0.8
1987 Hawkins JM, Sharpless KB. Asymmetric epoxidation models: An alkyl hydroperoxide dependent change in mehanism Tetrahedron Letters. 28: 2825-2828. DOI: 10.1016/S0040-4039(00)96219-1  1
1986 Ko SY, Sharpless KB. In situ opening of epoxy alcohols: a convenient alternative to the isolation of unstable epoxy alcohols The Journal of Organic Chemistry. 51: 5413-5415. DOI: 10.1021/jo00376a068  0.6
1986 Klunder JM, Ko SY, Sharpless KB. Asymmetric epoxidation of allyl alcohol: efficient routes to homochiral .beta.-adrenergic blocking agents The Journal of Organic Chemistry. 51: 3710-3712. DOI: 10.1021/jo00369a032  0.68
1986 Hanson RM, Sharpless KB. Procedure for the catalytic asymmetric epoxidation of allylic alcohols in the presence of molecular sieves The Journal of Organic Chemistry. 51: 1922-1925. DOI: 10.1021/jo00360a058  0.36
1986 FINN MG, SHARPLESS KB. ChemInform Abstract: On the Mechanism of Asymmetric Epoxidation with Titanium-Tartrate Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198635340  1
1986 BEHRENS CH, KO SY, SHARPLESS KB, WALKER FJ. ChemInform Abstract: Selective Transformation of 2,3-Epoxy Alcohols and Related Derivatives. Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198628137  0.6
1985 Behrens CH, Sharpless KB. Selective transformations of 2,3-epoxy alcohols and related derivatives. Strategies for nucleophilic attack at carbon-3 or carbon-2 The Journal of Organic Chemistry. 50: 5696-5704. DOI: 10.1021/jo00350a051  0.44
1985 Behrens CH, Ko SY, Sharpless KB, Walker FJ. Selective transformation of 2,3-epoxy alcohols and related derivatives. Strategies for nucleophilic attack at carbon-1 The Journal of Organic Chemistry. 50: 5687-5696. DOI: 10.1021/jo00350a050  0.6
1985 Miyano S, Lu LDL, Viti SM, Sharpless KB. Kinetic resolution of racemic .beta.-hydroxy amines by enantioselective N-oxide formation The Journal of Organic Chemistry. 50: 4350-4360. DOI: 10.1021/jo00222a030  0.52
1985 Caron M, Sharpless KB. Titanium isopropoxide-mediated nucleophilic openings of 2,3-epoxy alcohols. A mild procedure for regioselective ring-opening The Journal of Organic Chemistry. 50: 1557-1560. DOI: 10.1021/jo00209a047  0.52
1985 Klunder JM, Caron M, Uchiyama M, Sharpless KB. Chlorohydroxylation of olefins with peroxides and titanium tetrachloride The Journal of Organic Chemistry. 50: 912-915. DOI: 10.1021/jo00206a048  0.68
1985 Adams CE, Walker FJ, Sharpless KB. Enantioselective synthesis of swainsonine, a trihydroxylated indolizidine alkaloid The Journal of Organic Chemistry. 50: 420-422. DOI: 10.1021/jo00203a039  0.44
1985 Chong J, Sharpless K. Regioselective openings of 2,3-epoxy acids with organocuprates Tetrahedron Letters. 26: 4683-4686. DOI: 10.1016/S0040-4039(00)94923-2  0.68
1985 KLUNDER JM, CARON M, UCHIYAMA M, SHARPLESS KB. ChemInform Abstract: CHLOROHYDROXYLATION OF OLEFINS WITH PEROXIDES AND TITANIUM TETRACHLORIDE Chemischer Informationsdienst. 16. DOI: 10.1002/chin.198534155  0.68
1984 Rossiter BE, Sharpless KB. Asymmetric epoxidation of homoallylic alcohols. Synthesis of (-)-.gamma.-amino-.beta.-(R)-hydroxybutyric acid (GABOB) The Journal of Organic Chemistry. 49: 3707-3711. DOI: 10.1021/jo00194a007  0.52
1984 Lu LDL, Johnson RA, Finn MG, Sharpless KB. Two new asymmetric epoxidation catalysts. Unusual stoichiometry and inverse enantiofacial selection The Journal of Organic Chemistry. 49: 728-731. DOI: 10.1021/jo00178a039  1
1984 Williams ID, Pedersen SF, Sharpless KB, Lippard SJ. Crystal structures of two titanium tartrate asymmetric epoxidation catalysts Journal of the American Chemical Society. 106: 6430-6431. DOI: 10.1021/ja00333a060  0.88
1984 BEHRENS CH, SHARPLESS KB. ChemInform Abstract: NEW TRANSFORMATIONS OF 2,3-EPOXY ALCOHOLS AND RELATED DERIVATIVES. EASY ROUTES TO HOMOCHIRAL SUBSTANCES Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198441351  0.44
1984 MIYANO S, LU LD, VITI SM, SHARPLESS KB. ChemInform Abstract: KINETIC RESOLUTION OF RACEMIC β-HYDROXY AMINES BY ENANTIOSELECTIVE N-OXIDE FORMATION Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198412105  0.36
1983 Ko SY, Lee AW, Masamune S, Reed LA, Sharpless KB, Walker FJ. Total synthesis of the L-hexoses. Science (New York, N.Y.). 220: 949-51. PMID 17816019 DOI: 10.1016/S0040-4020(01)97596-9  0.6
1983 Sharpless KB, Woodard SS. On the mechanism of titanium-tartrate catalyzed asymmetric epoxidation Pure and Applied Chemistry. 55: 1823-1836. DOI: 10.1351/pac198355111823  0.48
1983 Miyano S, Lu LDL, Viti SM, Sharpless KB. Kinetic resolution of racemic .beta.-hydroxy amines by enantioselective N-oxide formation The Journal of Organic Chemistry. 48: 3608-3611. DOI: 10.1021/jo00168a064  0.52
1983 Hill JG, Rossiter BE, Sharpless KB. Anhydrous tert-butyl hydroperoxide in toluene: the preferred reagent for applications requiring dry TBHP The Journal of Organic Chemistry. 48: 3607-3608. DOI: 10.1021/jo00168a063  0.52
1982 Katsuki T, Lee AWM, Ma P, Martin VS, Masamune S, Sharpless KB, Tuddenham D, Walker FJ. Synthesis of saccharides and related polyhydroxylated natural products. 1. Simple alditols The Journal of Organic Chemistry. 47: 1373-1378. DOI: 10.1021/jo00346a051  0.44
1982 Warpehoski MA, Chabaud B, Sharpless KB. Selenium dioxide oxidation of endocyclic olefins. Evidence for a dissociation-recombination pathway The Journal of Organic Chemistry. 47: 2897-2900. DOI: 10.1021/jo00136a017  0.32
1982 LEE AWM, MARTIN VS, MASAMUNE S, SHARPLESS KB, WALKER FJ. ChemInform Abstract: SYNTHESIS OF SACCHARIDES AND RELATED POLYHYDROXYLATED NATURAL PRODUCTS. 3. EFFICIENT CONVERSION OF 2,3-ERYTHRO-ALDOSES TO 2,3-THREO-ALDOSES Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198239354  0.44
1982 MA P, MARTIN VS, MASAMUNE S, SHARPLESS KB, VITI SM. ChemInform Abstract: SYNTHESIS OF SACCHARIDES AND RELATED POLYHYDROXYLATED NATURAL PRODUCTS. 2. SIMPLE DEOXYALDITOLS Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198237319  0.36
1981 Martin VS, Woodard SS, Katsuki T, Yamada Y, Ikeda M, Sharpless KB. Kinetic resolution of racemic allylic alcohols by enantioselective epoxidation. A route to substances of absolute enantiomeric purity? Journal of the American Chemical Society. 103: 6237-6240. DOI: 10.1021/ja00410a053  0.48
1981 Rossiter BE, Katsuki T, Sharpless KB. Asymmetric epoxidation provides shortest routes to four chiral epoxy alcohols which are key intermediates in syntheses of methymycin, erythromycin, leukotriene C-1, and disparlure Journal of the American Chemical Society. 103: 464-465. DOI: 10.1021/ja00392a038  0.52
1979 Chabaud B, Sharpless KB. Oxidation of acetylenes with tert-butyl hydroperoxide catalyzed by selenium dioxide. .alpha.,.alpha.'-Dioxygenation of internal alkynes The Journal of Organic Chemistry. 44: 4202-4204. DOI: 10.1021/jo01337a045  0.32
1979 Baeckvall JE, Oshima K, Palermo RE, Sharpless KB. Some reactions of N-(2-hydroxyalkyl)-p-toluenesulfonamides and N-allyl-p-toluenesulfonamides The Journal of Organic Chemistry. 44: 1953-1957. DOI: 10.1021/jo01326a013  0.92
1979 BAECKVALL J, OSHIMA K, PALERMO RE, SHARPLESS KB. ChemInform Abstract: SOME REACTIONS OF N-(2-HYDROXYALKYL)-P-TOLUENESULFONAMIDES AND N-ALLYL-P-TOLUENESULFONAMIDES Chemischer Informationsdienst. 10. DOI: 10.1002/chin.197943206  0.92
1979 LIESBESKIND LS, SHARPLESS KB, WILSON RD, IBERS JA. ChemInform Abstract: THE FIRST D0 METALLOOXAZIRIDINES. AMINATION OF OLEFINS Chemischer Informationsdienst. 10. DOI: 10.1002/chin.197905268  0.48
1978 Patrick DW, Truesdale LK, Biller SA, Sharpless KB. Stereospecific vicinal oxyamination of olefins by alkylimidoosmium compounds The Journal of Organic Chemistry. 43: 2628-2638. DOI: 10.1021/jo00407a016  0.44
1978 Akashi K, Palermo RE, Sharpless KB. A major improvement in the osmium catalyzed vicinal hydroxylation of olefins by tert-butyl hydroperoxide The Journal of Organic Chemistry. 43: 2063-2066. DOI: 10.1021/jo00404a052  0.88
1978 Liebeskind LS, Sharpless KB, Wilson RD, Ibers JA. The first d0 metallooxaziridines. Amination of olefins Journal of the American Chemical Society. 100: 7061-7063. DOI: 10.1021/ja00490a047  0.48
1978 Herranz E, Biller SA, Sharpless KB. Osmium-catalyzed vicinal oxyamination of olefins by N-chloro-N-argentocarbamates Journal of the American Chemical Society. 100: 3596-3598. DOI: 10.1021/ja00479a051  0.44
1978 Current S, Sharpless K. Carbonyl participation in the addition of p-chlorophenylselenenyl bromide to ()-4-hexenal: A new route to 2,6-dideoxylgycosides Tetrahedron Letters. 19: 5075-5078. DOI: 10.1016/S0040-4039(01)85816-0  0.44
1978 HERRANZ E, BILLER SA, SHARPLESS KB. ChemInform Abstract: OSMIUM-CATALYZED VICINAL OXYAMINATION OF OLEFINS BY N-CHLORO-N-ARGENTOCARBAMATES Chemischer Informationsdienst. 9. DOI: 10.1002/chin.197836123  0.44
1977 Chong AO, Sharpless KB. Mechanism of the molybdenum and vanadium catalyzed epoxidation of olefins by alkyl hydroperoxides The Journal of Organic Chemistry. 42: 1587-1590. DOI: 10.1021/jo00429a024  0.92
1977 Chong AO, Oshima K, Sharpless KB. Synthesis of dioxobis(tert-alkylimido)osmium(VIII) and oxotris(tert-alkylimido)osmium(VIII) complexes. Stereospecific vicinal diamination of olefins Journal of the American Chemical Society. 99: 3420-3426. DOI: 10.1021/ja00452a039  0.92
1977 Sharpless KB, Teranishi AY, Backvall JE. Chromyl chloride oxidations of olefins. Possible role of organometallic intermediates in the oxidations of olefins by oxo transition metal species Journal of the American Chemical Society. 99: 3120-3128. DOI: 10.1021/ja00451a043  0.68
1977 Michaelson RC, Palermo RE, Sharpless KB. Chiral hydroxamic acids as ligands in the vanadium catalyzed asymmetric epoxidation of allylic alcohols by tert-butyl hydroperoxide Journal of the American Chemical Society. 99: 1990-1992. DOI: 10.1021/ja00448a059  0.88
1977 Backvall JE, Young MW, Sharpless KB. Vicinal acetoxychlorination of olefins by chromyl chloride in acetyl chloride Tetrahedron Letters. 18: 3523-3526. DOI: 10.1016/S0040-4039(01)83282-2  1
1976 Sharpless KB, Chong AO, Oshima K. Osmium-catalyzed vicinal oxyamination of olefins by Chloramine-T The Journal of Organic Chemistry. 41: 177-179. DOI: 10.1021/jo00863a052  0.92
1976 Sharpless KB, Akashi K. Osmium catalyzed vicinal hydroxylation of olefins by tert-butyl hydroperoxide under alkaline conditions Journal of the American Chemical Society. 98: 1986-1987. DOI: 10.1021/ja00423a067  0.56
1976 Sharpless KB, Hori T, Truesdale LK, Dietrich CO. Allylic amination of olefins and acetylenes by imido selenium compounds Journal of the American Chemical Society. 98: 269-271. DOI: 10.1021/ja00417a062  0.44
1976 Sharpless K, Akashi K, Oshima K. Ruthenium catalyzed oxidation of alcohols to aldehydes and ketones by amine-n-oxides Tetrahedron Letters. 17: 2503-2506. DOI: 10.1016/S0040-4039(00)78130-5  0.92
1975 Sharpless KB, Chong AO, Scott JA. Rapid separation of organic mixtures by formation of metal complexes The Journal of Organic Chemistry. 40: 1252-1257. DOI: 10.1021/jo00897a015  0.92
1975 Sharpless KB, Young MW. Olefin synthesis. Rate enhancement of the elimination of alkyl aryl selenoxides by electron-withdrawing substituents The Journal of Organic Chemistry. 40: 947-949. DOI: 10.1021/jo00895a030  0.68
1975 Jensen HP, Sharpless KB. Selenium dioxide oxidation of d-limonene. Reinvestigation The Journal of Organic Chemistry. 40: 264-265. DOI: 10.1021/jo00890a030  0.4
1975 Sharpless KB, Akashi K. Oxidation of alcohols to aldehydes by reagents derived from chromyl chloride Journal of the American Chemical Society. 97: 5927-5928. DOI: 10.1021/ja00853a055  0.56
1975 Sharpless KB, Patrick DW, Truesdale LK, Biller SA. New reaction. Stereospecific vicinal oxyamination of olefins by alkyl imido osmium compounds Journal of the American Chemical Society. 97: 2305-2307. DOI: 10.1021/ja00841a071  0.44
1975 Nelson JA, Kahn S, Spencer TA, Sharpless KB, Clayton RB. Some aspects of substrate specificity in biological demethylation at C4 of steroids Bioorganic Chemistry. 4: 363-376. DOI: 10.1016/0045-2068(75)90047-4  1
1974 Sharpless KB, Jensen HP. Synthesis of a novel pentacoordinate glyoxime-based ligand and preparation of its chlorocobalt(III) complex Inorganic Chemistry. 13: 2617-2620. DOI: 10.1021/ic50141a017  0.4
1973 Sharpless KB, Teranishi AY. Chromyl chloride in acetone. .alpha.-Chloro ketones and ketones directly from olefins The Journal of Organic Chemistry. 38: 185-186. DOI: 10.1021/jo00941a054  0.4
1973 Arigoni D, Vasella A, Sharpless KB, Jensen HP. Selenium dioxide oxidations of olefins. Trapping of the allylic seleninic acid intermediate as a seleninolactone Journal of the American Chemical Society. 95: 7917-7919. DOI: 10.1021/ja00804a087  0.4
1973 Sharpless KB, Lauer RF, Teranishi AY. Electrophilic and nucleophilic organoselenium reagents. New routes to .alpha.,.beta.-unsaturated carbonyl compounds Journal of the American Chemical Society. 95: 6137-6139. DOI: 10.1021/ja00799a062  0.4
1973 Sharpless KB, Young MW, Lauer RF. Reactions of selenoxides: Thermal syn-elimination and H218O exchange Tetrahedron Letters. 14: 1979-1982. DOI: 10.1016/S0040-4039(01)96098-8  1
1973 SHARPLESS KB, YOUNG MW, LAUER RF. ChemInform Abstract: RK. VON SELENOXIDEN, THERMISCHE SYN-ELIMINIERUNG UND H2 (18)O-AUSTAUSCH Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/chin.197334142  0.68
1973 SHARPLESS KB, TERANISHI AY. ChemInform Abstract: CHROMYLCHLORID IN ACETON, ALPHA-CHLOR-KETONE UND KETONE AUS OLEFINEN Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/chin.197318200  0.4
1972 Sharpless KB, Flood TC. Direct deoxygenation of vicinal diols with tungsten(IV). A new olefin synthesis Journal of the Chemical Society, Chemical Communications. 370-371. DOI: 10.1039/C39720000370  1
1971 Sharpless KB, Lauer RF, Repic O, Teranishi AY, Williams DR. Permanganate in acetic anhydride. .alpha.-Diketones directly from olefins Journal of the American Chemical Society. 93: 3303-3304. DOI: 10.1021/ja00742a045  0.4
1971 SHARPLESS KB, LAUER RF, REPIC O, TERANISHI AY, WILLIAMS DR. ChemInform Abstract: PERMANGANAT IN ACETANHYDRID, BLDG. VON ALPHA-DIKETONEN DIREKT AUS OLEFINEN Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/chin.197138134  0.4
1970 Rahman R, Sharpless KB, Spencer TA, Clayton RB. Removal of the 4,4-dimethyl carbons in the enzymic conversion of lanosterol to cholesterol. Initial loss of the 4-alpha-methyl group. The Journal of Biological Chemistry. 245: 2667-71. PMID 5445804  1
1969 Sharpless KB, Snyder TE, Spencer TA, Maheshwari KK, Nelson JA. Biological demethylation of 4,4-dimethyl sterols, Evidence for enzymic epimerization of the 4beta-methyl group prior to its oxidative removal. Journal of the American Chemical Society. 91: 3394-6. PMID 5791927 DOI: 10.1021/ja01040a065  1
1969 Anderson RJ, Hanzlik RP, Sharpless KB, Van Tamelen EE, Clayton RB. Enzymic transformation of an acyclic sesterterpene terminal epoxide into a lanosterol analogue Journal of the Chemical Society D: Chemical Communications. 53-54. DOI: 10.1039/C29690000053  1
1969 Sharpless KB, Van Tamelen EE. Terpene terminal epoxides. Skeletal rearrangement accompanying bicyclization of squalene 2,3-oxide Journal of the American Chemical Society. 91: 1848-1849. DOI: 10.1021/ja01035a043  0.84
1969 Van Tamelen EE, Akermark B, Sharpless KB. Mechanism of the titanium-promoted deoxygenative coupling of allyl and benzyl alcohols to hydrocarbons Journal of the American Chemical Society. 91: 1552-1554. DOI: 10.1021/ja01034a058  0.84
1968 Sharpless KB, Snyder TE, Spencer TA, Maheshwari KK, Guhn G, Clayton RB. Biological demethylation of 4,4-dimethyl sterols. Initial removal of the 4.alpha.-methyl group Journal of the American Chemical Society. 90: 6874-6875. DOI: 10.1021/ja01026a073  0.88
1968 Van Tamelen EE, Hanzlik RP, Sharpless KB, Clayton RB, Richter WJ, Burlingame AL. Enzymic cyclization of 15-norsqualene 2,3-oxide Journal of the American Chemical Society. 90: 3284-3286. DOI: 10.1021/ja01014a081  0.84
1968 Sharpless KB, Hanzlik RP, Van Tamelen EE. One-step synthesis of 1,5-dienes involving reductive coupling of allyl alcohols Journal of the American Chemical Society. 90: 209-210. DOI: 10.1021/ja01003a037  0.84
1967 van Tamelen EE, Sharpless KB, Hanzlik R, Clayton RB, Burlingame AL, Wszolek PC. Enzymic cyclization of trans,trans,trans-18,19-dihydrosqualene 2,3-oxide. Journal of the American Chemical Society. 89: 7150-1. PMID 6064361 DOI: 10.1021/ja01002a077  0.64
1967 Willett JD, Sharpless KB, Lord KE, van Tamelen EE, Clayton RB. Squalene-2,3oxide, an intermediate in the enzymatic conversion of squalene to lanosterol and cholesterol. The Journal of Biological Chemistry. 242: 4182-91. PMID 6061706  1
1967 Van Tamelen EE, Sharpless KB, Willett JD, Clayton RB, Burlingame AL. Biological activities of some terminally modified squalene and squalene 2,3-oxide analogs Journal of the American Chemical Society. 89: 3920-3922. DOI: 10.1021/ja00991a055  0.84
1967 van Tamelen E, Sharpless K. Positional selectivity during controlled oxidation of polyolefins Tetrahedron Letters. 8: 2655-2659. DOI: 10.1016/S0040-4039(01)89969-X  0.84
1964 Spencer TA, Schwartz MA, Sharpless KB. Synthesis of Resin Acid Intermediates. 8α,10β-Dimethyl-8β-carbomethoxy-Δ1,9,3,4-hexahydronaphthalone-2 and 8α,10β-Dimethyl-8β-carbomethoxy-Δ1,9-octalone-2 The Journal of Organic Chemistry. 29: 782-786. DOI: 10.1021/jo01027a003  0.88
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