| Year |
Citation |
Score |
| 2024 |
McFadden WM, Casey-Moore MC, Bare GAL, Kirby KA, Wen X, Li G, Wang H, Slack RL, Snyder AA, Lorson ZC, Kaufman IL, Cilento ME, Tedbury PR, Gembicky M, Olson AJ, ... ... Sharpless KB, et al. Identification of clickable HIV-1 capsid-targeting probes for viral replication inhibition. Cell Chemical Biology. 31: 477-486.e7. PMID 38518746 DOI: 10.1016/j.chembiol.2024.02.012 |
0.647 |
|
| 2023 |
Yang B, Sukheja P, Qin B, Li G, Bare GAL, Cascioferro A, Love MS, Petrassi HM, Sharpless KB, McNamara CW, Chatterjee AK. Synthesis and structure-activity relationships of aryl fluorosulfate-based inhibitors as novel antitubercular agents. Bioorganic & Medicinal Chemistry Letters. 98: 129596. PMID 38142914 DOI: 10.1016/j.bmcl.2023.129596 |
0.652 |
|
| 2023 |
Li H, Chang BS, Kim H, Xie Z, Lainé A, Ma L, Xu T, Yang C, Kwon J, Shelton SW, Klivansky LM, Altoé V, Gao B, Schwartzberg AM, Peng Z, ... ... Sharpless KB, et al. High-performing polysulfate dielectrics for electrostatic energy storage under harsh conditions. Joule. 7: 95-111. PMID 37034575 DOI: 10.1016/j.joule.2022.12.010 |
0.37 |
|
| 2023 |
Xin Y, Liu S, Liu Y, Qian Z, Liu H, Zhang B, Guo T, Thompson GJ, Stevens RC, Sharpless KB, Dong J, Shui W. Affinity selection of double-click triazole libraries for rapid discovery of allosteric modulators for GLP-1 receptor. Proceedings of the National Academy of Sciences of the United States of America. 120: e2220767120. PMID 36893261 DOI: 10.1073/pnas.2220767120 |
0.556 |
|
| 2022 |
Cheng Y, Li G, Smedley CJ, Giel MC, Kitamura S, Woehl JL, Bianco G, Forli S, Homer JA, Cappiello JR, Wolan DW, Moses JE, Sharpless KB. Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors. Proceedings of the National Academy of Sciences of the United States of America. 119: e2208540119. PMID 36070343 DOI: 10.1073/pnas.2208540119 |
0.708 |
|
| 2021 |
Kim H, Zhao J, Bae J, Klivansky LM, Dailing EA, Liu Y, Cappiello JR, Sharpless KB, Wu P. Chain-Growth Sulfur(VI) Fluoride Exchange Polycondensation: Molecular Weight Control and Synthesis of Degradable Polysulfates. Acs Central Science. 7: 1919-1928. PMID 34841062 DOI: 10.1021/acscentsci.1c01015 |
0.418 |
|
| 2021 |
Li S, Li G, Gao B, Pujari SP, Chen X, Kim H, Zhou F, Klivansky LM, Liu Y, Driss H, Liang DD, Lu J, Wu P, Zuilhof H, Moses J, ... Sharpless KB, et al. SuFExable polymers with helical structures derived from thionyl tetrafluoride. Nature Chemistry. PMID 34400816 DOI: 10.1038/s41557-021-00726-x |
0.758 |
|
| 2021 |
Dong J, Sharpless KB, Gao B, Sun S, Chen J. Fluorosulfuryl Isocyanate Enabled SuFEx Ligation of Alcohols and Amines. Angewandte Chemie (International Ed. in English). PMID 34259368 DOI: 10.1002/anie.202105583 |
0.485 |
|
| 2021 |
Zhang J, Zhao X, Cappiello JR, Yang Y, Cheng Y, Liu G, Fang W, Luo Y, Zhang Y, Dong J, Zhang L, Sharpless KB. Identification of simple arylfluorosulfates as potent agents against resistant bacteria. Proceedings of the National Academy of Sciences of the United States of America. 118. PMID 34244433 DOI: 10.1073/pnas.2103513118 |
0.523 |
|
| 2021 |
Garnar-Wortzel L, Bishop TR, Kitamura S, Milosevich N, Asiaban JN, Zhang X, Zheng Q, Chen E, Ramos AR, Ackerman CJ, Hampton EN, Chatterjee AK, Young TS, Hull MV, Sharpless KB, et al. Chemical Inhibition of ENL/AF9 YEATS Domains in Acute Leukemia. Acs Central Science. 7: 815-830. PMID 34079898 DOI: 10.1021/acscentsci.0c01550 |
0.406 |
|
| 2021 |
Zheng Q, Xu H, Wang H, Du WH, Wang N, Xiong H, Gu Y, Noodleman L, Sharpless KB, Yang G, Wu P. Sulfur [F]Fluoride Exchange Click Chemistry Enabled Ultrafast Late-Stage Radiosynthesis. Journal of the American Chemical Society. PMID 33630577 DOI: 10.1021/jacs.0c09306 |
0.547 |
|
| 2020 |
Brighty GJ, Botham RC, Li S, Nelson L, Mortenson DE, Li G, Morisseau C, Wang H, Hammock BD, Sharpless KB, Kelly JW. Using sulfuramidimidoyl fluorides that undergo sulfur(VI) fluoride exchange for inverse drug discovery. Nature Chemistry. PMID 32868886 DOI: 10.1038/S41557-020-0530-4 |
0.747 |
|
| 2020 |
Kitamura S, Zheng Q, Woehl JL, Solania A, Chen E, Dillon N, Hull MV, Kotaniguchi M, Cappiello JR, Kitamura S, Nizet V, Sharpless KB, Wolan DW. SuFEx-enabled high-throughput medicinal chemistry. Journal of the American Chemical Society. PMID 32479075 DOI: 10.1021/Jacs.9B13652 |
0.52 |
|
| 2020 |
Lauwaet T, Miyamoto Y, Ihara S, Le C, Kalisiak J, Korthals K, Ghassemian M, Smith DK, Sharpless KB, Fokin VV, Eckmann L. Click chemistry-facilitated comprehensive identification of proteins adducted by antimicrobial 5-nitroimidazoles for discovery of alternative drug targets against giardiasis. Plos Neglected Tropical Diseases. 14: e0008224. PMID 32302296 DOI: 10.1371/Journal.Pntd.0008224 |
0.668 |
|
| 2020 |
Smedley CJ, Li G, Barrow AS, Gialelis TL, Giel MC, Ottonello A, Cheng Y, Kitamura S, Wolan DW, Sharpless KB, Moses JE. Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores From 2-Substituted-Alkynyl-1-Sulfonyl Fluoride (SASF) Hubs. Angewandte Chemie (International Ed. in English). PMID 32301265 DOI: 10.1002/Anie.202003219 |
0.725 |
|
| 2019 |
Meng G, Guo T, Ma T, Zhang J, Shen Y, Sharpless KB, Dong J. Modular click chemistry libraries for functional screens using a diazotizing reagent. Nature. 574: 86-89. PMID 31578481 DOI: 10.1038/S41586-019-1589-1 |
0.604 |
|
| 2019 |
Zheng Q, Woehl JL, Kitamura S, Santos-Martins D, Smedley CJ, Li G, Forli S, Moses JE, Wolan DW, Sharpless KB. SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase. Proceedings of the National Academy of Sciences of the United States of America. PMID 31484779 DOI: 10.1073/Pnas.1909972116 |
0.738 |
|
| 2019 |
Liu F, Wang H, Li S, Bare GAL, Chen X, Wang C, Moses JE, Wu P, Sharpless KB. Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF4) Derived Connective Hubs For Bioconjugation to DNA and Proteins. Angewandte Chemie (International Ed. in English). PMID 30998840 DOI: 10.1002/Anie.201902489 |
0.658 |
|
| 2019 |
Hong S, Shi Y, Wu NC, Grande G, Douthit L, Wang H, Zhou W, Sharpless KB, Wilson IA, Xie J, Wu P. Bacterial glycosyltransferase-mediated cell-surface chemoenzymatic glycan modification. Nature Communications. 10: 1799. PMID 30996301 DOI: 10.1038/S41467-019-09608-W |
0.621 |
|
| 2019 |
Kovarik Z, Hrvat NM, Kalisiak J, Katalinić M, Sit RK, Zorbaz T, Radić Z, Fokin VV, Sharpless KB, Taylor P. Counteracting tabun inhibition by reactivation by pyridinium aldoximes that interact with active center gorge mutants of acetylcholinesterase. Toxicology and Applied Pharmacology. PMID 30978400 DOI: 10.1016/J.Taap.2019.04.007 |
0.688 |
|
| 2019 |
Smedley CJ, Zheng Q, Gao B, Li S, Molino A, Duivenvoorden HM, Parker BS, Wilson DJD, Sharpless KB, Moses JE. Bifluoride Ion Mediated SuFEx Trifluoromethylation of Sulfonyl Fluorides and Iminosulfur Oxydifluorides. Angewandte Chemie (International Ed. in English). PMID 30740848 DOI: 10.1002/Anie.201813761 |
0.681 |
|
| 2019 |
Liu F, Wang H, Li S, Bare GAL, Chen X, Wang C, Moses JE, Wu P, Sharpless KB. Back Cover: Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF
4
)‐Derived Connective Hubs for Bioconjugation to DNA and Proteins (Angew. Chem. Int. Ed. 24/2019) Angewandte Chemie International Edition. 58: 8242-8242. DOI: 10.1002/Anie.201906154 |
0.429 |
|
| 2019 |
Liu F, Wang H, Li S, Bare GAL, Chen X, Wang C, Moses JE, Wu P, Sharpless KB. Rücktitelbild: Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF
4
)‐Derived Connective Hubs for Bioconjugation to DNA and Proteins (Angew. Chem. 24/2019) Angewandte Chemie. 131: 8328-8328. DOI: 10.1002/Ange.201906154 |
0.428 |
|
| 2018 |
Kovarik Z, Kalisiak J, Hrvat NM, Katalinić M, Zorbaz T, Žunec S, Green C, Radić Z, Fokin VV, Sharpless KB, Taylor P. Reversal of tabun toxicity, enabled by a triazole annulated oxime library-reactivators of acetylcholinesterase. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 30458057 DOI: 10.1002/Chem.201805051 |
0.687 |
|
| 2018 |
Sit R, Kovarik Z, Macek-Hrvat N, Zunec S, Green C, Fokin V, Sharpless KB, Radic' Z, Taylor P. Pharmacology, pharmacokinetics and tissue disposition of zwitterionic hydoxyiminoacetamido alkylamines as reactivating antidotes for organophosphate exposure. The Journal of Pharmacology and Experimental Therapeutics. PMID 30190337 DOI: 10.1124/Jpet.118.249383 |
0.658 |
|
| 2018 |
Gahtory D, Sen R, Pujari S, Li S, Zheng Q, Moses JE, Sharpless KB, Zuilhof H. Quantitative and Orthogonal Formation and Reactivity of SuFEx Platforms. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29949211 DOI: 10.1002/Chem.201802356 |
0.656 |
|
| 2018 |
Liu Z, Li J, Li S, Li G, Sharpless KB, Wu P. SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization. Journal of the American Chemical Society. PMID 29451783 DOI: 10.1021/Jacs.7B12788 |
0.773 |
|
| 2018 |
Sharpless KB, Gao B, Li S, Wu P, Moses JE. SuFEx Chemistry of Thionyl Tetrafluoride (SOF4) with Organolithium Nucleophiles: Synthesis of Sulfonimidoyl Fluorides, Sulfoximines, Sulfonimidamides and Sulfonimidates. Angewandte Chemie (International Ed. in English). PMID 29314580 DOI: 10.1002/Anie.201712145 |
0.65 |
|
| 2018 |
Guo T, Meng G, Zhan X, Yang Q, Ma T, Xu L, Sharpless KB, Dong J. Back Cover: A New Portal to SuFEx Click Chemistry: A Stable Fluorosulfuryl Imidazolium Salt Emerging as an “F−SO2
+” Donor of Unprecedented Reactivity, Selectivity, and Scope (Angew. Chem. Int. Ed. 10/2018) Angewandte Chemie International Edition. 57: 2728-2728. DOI: 10.1002/Anie.201801651 |
0.583 |
|
| 2017 |
Guo T, Meng G, Zhan X, Yang Q, Ma T, Xu L, Sharpless KB, Dong J. A New Portal to SuFEx Click Chemistry: a Stable Fluorosulfuryl Imidazolium Salt Emerging as an "F-SO2+" Donor of Unprecedented Reactivity, Selectivity, and Scope. Angewandte Chemie (International Ed. in English). PMID 29276888 DOI: 10.1002/Anie.201712429 |
0.611 |
|
| 2017 |
Mortenson DE, Brighty GJ, Plate L, Bare G, Chen W, Li S, Wang H, Cravatt BF, Forli S, Powers ET, Sharpless KB, Wilson IA, Kelly JW. "Inverse Drug Discovery" Strategy To Identify Proteins That Are Targeted by Latent Electrophiles As Exemplified by Aryl Fluorosulfates. Journal of the American Chemical Society. PMID 29265822 DOI: 10.1021/Jacs.7B08366 |
0.562 |
|
| 2017 |
Gao B, Zhang L, Zheng Q, Zhou F, Klivansky LM, Lu J, Liu Y, Dong J, Wu P, Sharpless KB. Bifluoride-catalysed sulfur(VI) fluoride exchange reaction for the synthesis of polysulfates and polysulfonates. Nature Chemistry. 9: 1083-1088. PMID 29064495 DOI: 10.1038/Nchem.2796 |
0.74 |
|
| 2017 |
Wang H, Zhou F, Ren G, Zheng Q, Chen H, Gao B, Klivansky L, Liu Y, Wu B, Xu Q, Lu J, Sharpless KB, Wu P. SuFEx-Based Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts. Angewandte Chemie (International Ed. in English). PMID 28792119 DOI: 10.1002/Anie.201701160 |
0.65 |
|
| 2017 |
Kim WJ, Korthals K, Li S, Le C, Kalisiak J, Sharpless KB, Fokin VV, Miyamoto Y, Eckmann L. Click chemistry-facilitated structural diversification of nitrothiazoles, nitrofurans and nitropyrroles enhances antimicrobial activity against Giardia lamblia. Antimicrobial Agents and Chemotherapy. PMID 28396548 DOI: 10.1128/Aac.02397-16 |
0.747 |
|
| 2017 |
Zha GF, Zheng Q, Leng J, Wu P, Qin HL, Sharpless KB. Palladium-Catalyzed Fluorosulfonylvinylation of Organic Iodides. Angewandte Chemie (International Ed. in English). PMID 28370917 DOI: 10.1002/Anie.201701162 |
0.722 |
|
| 2017 |
Li S, Wu P, Moses JE, Sharpless KB. Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride Exchange Connections of Diverse Modules Launched From An SOF4 Hub. Angewandte Chemie (International Ed. in English). PMID 28165188 DOI: 10.1002/Anie.201611048 |
0.629 |
|
| 2017 |
Wang H, Zhou F, Ren G, Zheng Q, Chen H, Gao B, Klivansky L, Liu Y, Wu B, Xu Q, Lu J, Sharpless KB, Wu P. Back Cover: SuFEx-Based Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts (Angew. Chem. Int. Ed. 37/2017) Angewandte Chemie International Edition. 56: 11274-11274. DOI: 10.1002/Anie.201706481 |
0.602 |
|
| 2017 |
Wang H, Zhou F, Ren G, Zheng Q, Chen H, Gao B, Klivansky L, Liu Y, Wu B, Xu Q, Lu J, Sharpless KB, Wu P. Rücktitelbild: SuFEx-Based Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts (Angew. Chem. 37/2017) Angewandte Chemie. 129: 11428-11428. DOI: 10.1002/Ange.201706481 |
0.613 |
|
| 2016 |
Zheng Q, Dong J, Sharpless KB. Ethenesulfonyl Fluoride (ESF): An On-Water Procedure for the Kilogram-Scale Preparation. The Journal of Organic Chemistry. PMID 27764941 DOI: 10.1021/Acs.Joc.6B01423 |
0.674 |
|
| 2016 |
Silverman S, Moses J, Sharpless KB. Reengineering Antibiotics to Combat Bacterial Resistance: Click Chemistry [1,2,3]-Triazole Vancomycin Dimers with Potent Activity Against MRSA and VRE. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27747932 DOI: 10.1002/Chem.201604765 |
0.587 |
|
| 2016 |
Qin HL, Zheng Q, Bare GA, Wu P, Sharpless KB. A Heck-Matsuda Process for the Synthesis of β-Arylethenesulfonyl Fluorides: Selectively Addressable Bis-electrophiles for SuFEx Click Chemistry. Angewandte Chemie (International Ed. in English). PMID 27723200 DOI: 10.1002/Anie.201608807 |
0.715 |
|
| 2016 |
Chen W, Dong J, Plate L, Mortenson DE, Brighty GJ, Li S, Liu Y, Galmozzi A, Lee PS, Hulce JJ, Cravatt BF, Saez E, Powers ET, Wilson IA, Sharpless KB, et al. Arylfluorosulfates Inactivate Intracellular Lipid Binding Protein(s) through Chemoselective SuFEx Reaction with a Binding-site Tyr Residue. Journal of the American Chemical Society. PMID 27191344 DOI: 10.1021/Jacs.6B02960 |
0.688 |
|
| 2016 |
Zhang E, Tang J, Li S, Wu P, Moses JE, Sharpless KB. Chemoselective Synthesis of Polysubstituted Pyridines from Heteroaryl Fluorosulfates. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26990693 DOI: 10.1002/Chem.201600167 |
0.668 |
|
| 2016 |
Bourne Y, Sharpless KB, Taylor P, Marchot P. Steric and dynamic parameters influencing in situ cycloadditions to form triazole inhibitors with crystalline acetylcholinesterase. Journal of the American Chemical Society. PMID 26731630 DOI: 10.1021/Jacs.5B11384 |
0.33 |
|
| 2015 |
Chen W, Dong J, Li S, Liu Y, Wang Y, Yoon L, Wu P, Sharpless KB, Kelly JW. Synthesis of Sulfotyrosine-Containing Peptides by Incorporating Fluorosulfated Tyrosine Using an Fmoc-Based Solid-Phase Strategy. Angewandte Chemie (International Ed. in English). PMID 26696445 DOI: 10.1002/Anie.201509016 |
0.708 |
|
| 2015 |
Toguchi S, Hirose T, Yorita K, Fukui K, Sharpless KB, Ōmura S, Sunazuka T. In situ Click Chemistry for the Identification of a Potent D-Amino Acid Oxidase Inhibitor. Chemical & Pharmaceutical Bulletin. PMID 26686243 DOI: 10.1248/Cpb.C15-00867 |
0.326 |
|
| 2015 |
Baranczak A, Liu Y, Connelly S, Du WG, Greiner ER, Genereux JC, Wiseman RL, Eisele YS, Bradbury NC, Dong J, Noodleman L, Sharpless KB, Wilson IA, Encalada SE, Kelly JW. A Fluorogenic Aryl Fluorosulfate for Intraorganellar Transthyretin Imaging in Living Cells and in Caenorhabditis elegans. Journal of the American Chemical Society. 137: 7404-14. PMID 26051248 DOI: 10.1021/Jacs.5B03042 |
0.554 |
|
| 2015 |
Liang Q, Xing P, Huang Z, Dong J, Sharpless KB, Li X, Jiang B. Palladium-catalyzed, ligand-free Suzuki reaction in water using aryl fluorosulfates. Organic Letters. 17: 1942-5. PMID 25856416 DOI: 10.1021/Acs.Orglett.5B00654 |
0.614 |
|
| 2015 |
Sharpless KB, Finn MG, Martín VS. Tsutomu Katsuki (1946-2014). Angewandte Chemie (International Ed. in English). 54: 4708. PMID 25766459 DOI: 10.1002/Anie.201501065 |
0.582 |
|
| 2014 |
Dong J, Krasnova L, Finn MG, Sharpless KB. Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry. Angewandte Chemie (International Ed. in English). 53: 9430-48. PMID 25112519 DOI: 10.1002/Anie.201309399 |
0.711 |
|
| 2014 |
Dong J, Sharpless KB, Kwisnek L, Oakdale JS, Fokin VV. SuFEx-based synthesis of polysulfates. Angewandte Chemie (International Ed. in English). 53: 9466-70. PMID 25100330 DOI: 10.1002/Anie.201403758 |
0.773 |
|
| 2014 |
Sit RK, Fokin VV, Amitai G, Sharpless KB, Taylor P, Radić Z. Imidazole aldoximes effective in assisting butyrylcholinesterase catalysis of organophosphate detoxification. Journal of Medicinal Chemistry. 57: 1378-89. PMID 24571195 DOI: 10.1021/Jm401650Z |
0.699 |
|
| 2014 |
Dong J, Krasnova L, Finn MG, Sharpless KB. ChemInform Abstract: Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry Cheminform. 45: no-no. DOI: 10.1002/chin.201447274 |
0.574 |
|
| 2014 |
Dong J, Krasnova L, Finn MG, Sharpless KB. Cover Picture: Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry (Angew. Chem. Int. Ed. 36/2014) Angewandte Chemie International Edition. 53: 9391-9391. DOI: 10.1002/Anie.201401157 |
0.726 |
|
| 2014 |
Dong J, Krasnova L, Finn MG, Sharpless KB. Titelbild: Schwefel(VI)-fluorid-Austausch (SuFEx): Eine weitere gute Anwendung für die Click-Chemie (Angew. Chem. 36/2014) Angewandte Chemie. 126: 9545-9545. DOI: 10.1002/Ange.201401157 |
0.683 |
|
| 2014 |
Dong J, Krasnova L, Finn MG, Sharpless KB. Schwefel(VI)-fluorid-Austausch (SuFEx): Eine weitere gute Anwendung für die Click-Chemie Angewandte Chemie. 126: 9584-9603. DOI: 10.1002/Ange.201309399 |
0.68 |
|
| 2013 |
Miyamoto Y, Kalisiak J, Korthals K, Lauwaet T, Cheung DY, Lozano R, Cobo ER, Upcroft P, Upcroft JA, Berg DE, Gillin FD, Fokin VV, Sharpless KB, Eckmann L. Expanded therapeutic potential in activity space of next-generation 5-nitroimidazole antimicrobials with broad structural diversity. Proceedings of the National Academy of Sciences of the United States of America. 110: 17564-9. PMID 24101497 DOI: 10.1073/Pnas.1302664110 |
0.671 |
|
| 2013 |
Morris GM, Green LG, Radić Z, Taylor P, Sharpless KB, Olson AJ, Grynszpan F. Automated docking with protein flexibility in the design of femtomolar "click chemistry" inhibitors of acetylcholinesterase. Journal of Chemical Information and Modeling. 53: 898-906. PMID 23451944 DOI: 10.1021/Ci300545A |
0.662 |
|
| 2013 |
Grimster NP, Connelly S, Baranczak A, Dong J, Krasnova LB, Sharpless KB, Powers ET, Wilson IA, Kelly JW. Aromatic sulfonyl fluorides covalently kinetically stabilize transthyretin to prevent amyloidogenesis while affording a fluorescent conjugate. Journal of the American Chemical Society. 135: 5656-68. PMID 23350654 DOI: 10.1021/Ja311729D |
0.608 |
|
| 2013 |
Fraser BH, Hamilton S, Krause-Heuer AM, Wright PJ, Greguric I, Tucker SP, Draffan AG, Fokin VV, Sharpless KB. Synthesis of 1,4-triazole linked zanamivir dimers as highly potent inhibitors of influenza A and B Medchemcomm. 4: 383-386. DOI: 10.1039/C2Md20300F |
0.708 |
|
| 2012 |
Yamauchi JG, Gomez K, Grimster N, Dufouil M, Nemecz A, Fotsing JR, Ho KY, Talley TT, Sharpless KB, Fokin VV, Taylor P. Synthesis of selective agonists for the α7 nicotinic acetylcholine receptor with in situ click-chemistry on acetylcholine-binding protein templates. Molecular Pharmacology. 82: 687-99. PMID 22784805 DOI: 10.1124/Mol.112.080291 |
0.713 |
|
| 2012 |
Grimster NP, Stump B, Fotsing JR, Weide T, Talley TT, Yamauchi JG, Nemecz Á, Kim C, Ho KY, Sharpless KB, Taylor P, Fokin VV. Generation of candidate ligands for nicotinic acetylcholine receptors via in situ click chemistry with a soluble acetylcholine binding protein template. Journal of the American Chemical Society. 134: 6732-40. PMID 22394239 DOI: 10.1021/Ja3001858 |
0.689 |
|
| 2012 |
Radi? Z, Sit RK, Kovarik Z, Berend S, Garcia E, Zhang L, Amitai G, Green C, Radi? B, Fokin VV, Sharpless KB, Taylor P. Refinement of structural leads for centrally acting oxime reactivators of phosphylated cholinesterases. The Journal of Biological Chemistry. 287: 11798-809. PMID 22343626 DOI: 10.1074/Jbc.M111.333732 |
0.694 |
|
| 2012 |
Radi? Z, Sit RK, Kovarik Z, Berend S, Garcia E, Zhang L, Amitai G, Green C, Radi? B, Fokin VV, Sharpless KB, Taylor P. Refinement of structural leads for centrally acting oxime reactivators of phosphylated cholinesterases (Journal of Biological Chemistry (2012) 287, (11798-11809)) Journal of Biological Chemistry. 287: 19337. DOI: 10.1074/jbc.A111.333732 |
0.652 |
|
| 2012 |
Finn MG, Sharpless KB. On the Mechanism of Asymmetric Epoxidation with Titanium-Tartrate Catalysts Asymmetric Synthesis. 247-308. DOI: 10.1016/B978-0-08-092493-9.50013-X |
0.541 |
|
| 2011 |
Millward SW, Henning RK, Kwong GA, Pitram S, Agnew HD, Deyle KM, Nag A, Hein J, Lee SS, Lim J, Pfeilsticker JA, Sharpless KB, Heath JR. Iterative in situ click chemistry assembles a branched capture agent and allosteric inhibitor for Akt1. Journal of the American Chemical Society. 133: 18280-8. PMID 21962254 DOI: 10.1021/Ja2064389 |
0.755 |
|
| 2011 |
Cochran R, Kalisiak J, Küçükkilinç T, Radic Z, Garcia E, Zhang L, Ho KY, Amitai G, Kovarik Z, Fokin VV, Sharpless KB, Taylor P. Oxime-assisted acetylcholinesterase catalytic scavengers of organophosphates that resist aging. The Journal of Biological Chemistry. 286: 29718-24. PMID 21730071 DOI: 10.1074/Jbc.M111.264739 |
0.683 |
|
| 2011 |
Sit RK, Radi? Z, Gerardi V, Zhang L, Garcia E, Katalini? M, Amitai G, Kovarik Z, Fokin VV, Sharpless KB, Taylor P. New structural scaffolds for centrally acting oxime reactivators of phosphylated cholinesterases. The Journal of Biological Chemistry. 286: 19422-30. PMID 21464125 DOI: 10.1074/Jbc.M111.230656 |
0.696 |
|
| 2011 |
Gastaminza P, Pitram SM, Dreux M, Krasnova LB, Whitten-Bauer C, Dong J, Chung J, Fokin VV, Sharpless KB, Chisari FV. Antiviral stilbene 1,2-diamines prevent initiation of hepatitis C virus RNA replication at the outset of infection. Journal of Virology. 85: 5513-23. PMID 21430055 DOI: 10.1128/Jvi.02116-10 |
0.733 |
|
| 2010 |
Weide T, Saldanha SA, Minond D, Spicer TP, Fotsing JR, Spaargaren M, Frère JM, Bebrone C, Sharpless KB, Hodder PS, Fokin VV. NH-1,2,3-Triazole-based Inhibitors of the VIM-2 Metallo-β-Lactamase: Synthesis and Structure-Activity Studies. Acs Medicinal Chemistry Letters. 1: 150-154. PMID 20625539 DOI: 10.1021/Ml900022Q |
0.676 |
|
| 2010 |
Radi? Z, Kalisiak J, Fokin VV, Sharpless KB, Taylor P. Interaction kinetics of oximes with native, phosphylated and aged human acetylcholinesterase. Chemico-Biological Interactions. 187: 163-6. PMID 20412789 DOI: 10.1016/J.Cbi.2010.04.014 |
0.678 |
|
| 2010 |
Berend S, Vrdoljak AL, Radic B, Kalisiak J, Radic Z, Taylor P, Fokin V, Sharpless K. Characterizing the therapeutic efficacy of novel oximes synthesized by click chemistry against organophosphorous compounds poisoning Toxicology Letters. 196: S254. DOI: 10.1016/J.Toxlet.2010.03.849 |
0.663 |
|
| 2010 |
Hein JE, Tripp JC, Krasnova LB, Sharpless KB, Fokin VV. ChemInform Abstract: Copper(I)-Catalyzed Cycloaddition of Organic Azides and 1-Iodoalkynes. Cheminform. 41. DOI: 10.1002/chin.201007113 |
0.789 |
|
| 2010 |
Dupau P, Epple R, Thomas AA, Fokin VV, Sharpless KB. ChemInform Abstract: Osmium-Catalyzed Dihydroxylation of Olefins in Acidic Media: Old Process, New Tricks. Cheminform. 33: no-no. DOI: 10.1002/chin.200244058 |
0.725 |
|
| 2010 |
Rostovtsev VV, Green LG, Fokin VV, Sharpless KB. ChemInform Abstract: A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes. Cheminform. 33: no-no. DOI: 10.1002/chin.200243045 |
0.693 |
|
| 2010 |
Andersson MA, Epple R, Fokin VV, Sharpless KB. ChemInform Abstract: A New Approach to Osmium-Catalyzed Asymmetric Dihydroxylation and Aminohydroxylation of Olefins. Cheminform. 33: no-no. DOI: 10.1002/chin.200228035 |
0.675 |
|
| 2010 |
Kolb HC, Finn MG, Sharpless KB. ChemInform Abstract: Click Chemistry: Diverse Chemical Function from a Few Good Reactions Cheminform. 32: no-no. DOI: 10.1002/chin.200135279 |
0.569 |
|
| 2010 |
YUDIN AK, SHARPLESS KB. ChemInform Abstract: Bis(trimethylsilyl) Peroxide Extends the Range of Oxorhenium Catalysts for Olefin Epoxidation. Cheminform. 29: no-no. DOI: 10.1002/chin.199810117 |
0.494 |
|
| 2010 |
COPERET C, ADOLFSSON H, SHARPLESS KB. ChemInform Abstract: A Simple and Efficient Method for Epoxidation of Terminal Alkenes. Cheminform. 28: no-no. DOI: 10.1002/chin.199747120 |
0.419 |
|
| 2010 |
KOLB HC, ANDERSSON PG, SHARPLESS KB. ChemInform Abstract: Toward an Understanding of the High Enantioselectivity in the Osmium- Catalyzed Asymmetric Dihydroxylation (AD). Part 1. Kinetics. Cheminform. 25: no-no. DOI: 10.1002/chin.199426078 |
0.713 |
|
| 2010 |
WALSH PJ, SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation (AD) of α,β-Unsaturated Ketones. Cheminform. 25: no-no. DOI: 10.1002/chin.199411088 |
0.364 |
|
| 2010 |
AMBERG W, BENNANI YL, CHADHA RK, CRISPINO GA, DAVIS WD, HARTUNG J, JEONG K, OGINO Y, SHIBATA T, SHARPLESS KB. ChemInform Abstract: Syntheses and Crystal Structures of the Cinchona Alkaloid Derivatives Used as Ligands in the Osmium-Catalyzed Asymmetric Dihydroxylation of Olefins, e.g. (I). Used as Ligands in the Osmium-Catalyzed Asymmetric Dihydroxylation of Olefi Cheminform. 25: no-no. DOI: 10.1002/chin.199404183 |
0.51 |
|
| 2010 |
WALSH PJ, BENNANI YL, SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation (AD)/Cyclization of N-DiBoc Allylic and Homoallylic Amines: Selective Differentiation of the Hydroxyl Groups. Cheminform. 24: no-no. DOI: 10.1002/chin.199352069 |
0.416 |
|
| 2010 |
KOLB HC, BENNANI YL, SHARPLESS KB. ChemInform Abstract: Short and Practical Syntheses of (R)-(-)-Carnitine and (R)-(-)-γ- Amino-β-hydroxybutyric Acid (GABOB). Cheminform. 24: no-no. DOI: 10.1002/chin.199321060 |
0.488 |
|
| 2010 |
KOLB HC, SHARPLESS KB. ChemInform Abstract: A Simplified Procedure for the Stereospecific Transformation of 1,2- Diols into Epoxides. Cheminform. 24: no-no. DOI: 10.1002/chin.199313174 |
0.503 |
|
| 2010 |
SHARPLESS KB, AMBERG W, BENNANI YL, CRISPINO GA, HARTUNG J, JEONG K, KWONG H, MORIKAWA K, WANG Z, XU D, ZHANG X. ChemInform Abstract: The Osmium-Catalyzed Asymmetric Dihydroxylation: A New Ligand Class and a Process Improvement. Cheminform. 23: no-no. DOI: 10.1002/chin.199242058 |
0.501 |
|
| 2009 |
Hein JE, Tripp JC, Krasnova LB, Sharpless KB, Fokin VV. Copper(I)-catalyzed cycloaddition of organic azides and 1-iodoalkynes. Angewandte Chemie (International Ed. in English). 48: 8018-21. PMID 19774581 DOI: 10.1002/anie.200903558 |
0.788 |
|
| 2009 |
Minond D, Saldanha SA, Subramaniam P, Spaargaren M, Spicer T, Fotsing JR, Weide T, Fokin VV, Sharpless KB, Galleni M, Bebrone C, Lassaux P, Hodder P. Inhibitors of VIM-2 by screening pharmacologically active and click-chemistry compound libraries. Bioorganic & Medicinal Chemistry. 17: 5027-37. PMID 19553129 DOI: 10.1016/J.Bmc.2009.05.070 |
0.686 |
|
| 2009 |
Valdez CA, Tripp JC, Miyamoto Y, Kalisiak J, Hruz P, Andersen YS, Brown SE, Kangas K, Arzu LV, Davids BJ, Gillin FD, Upcroft JA, Upcroft P, Fokin VV, Smith DK, Sharpless KB, et al. Synthesis and electrochemistry of 2-ethenyl and 2-ethanyl derivatives of 5-nitroimidazole and antimicrobial activity against Giardia lamblia. Journal of Medicinal Chemistry. 52: 4038-53. PMID 19480409 DOI: 10.1021/Jm900356N |
0.777 |
|
| 2009 |
Agnew HD, Rohde RD, Millward SW, Nag A, Yeo WS, Hein JE, Pitram SM, Tariq AA, Burns VM, Krom RJ, Fokin VV, Sharpless KB, Heath JR. Iterative in situ click chemistry creates antibody-like protein-capture agents. Angewandte Chemie (International Ed. in English). 48: 4944-8. PMID 19301344 DOI: 10.1002/Anie.200900488 |
0.788 |
|
| 2009 |
Kalisiak J, Trauger SA, Kalisiak E, Morita H, Fokin VV, Adams MW, Sharpless KB, Siuzdak G. Identification of a new endogenous metabolite and the characterization of its protein interactions through an immobilization approach. Journal of the American Chemical Society. 131: 378-86. PMID 19055353 DOI: 10.1021/Ja808172N |
0.678 |
|
| 2009 |
Kwok SW, Hein JE, Fokin VV, Sharpless KB. ChemInform Abstract: Regioselective Synthesis of Either 1H- or 2H-1,2,3-Triazoles via Michael Addition to α,β-Unsaturated Ketones. Cheminform. 40. DOI: 10.1002/chin.200918132 |
0.774 |
|
| 2008 |
Kwok SW, Hein JE, Fokin VV, Sharpless KB. REGIOSELECTIVE SYNTHESIS OF EITHER 1H- OR 2H-1,2,3- TRIAZOLES VIA MICHAEL ADDITION TO α,ß-UNSATURATED KETONES. Heterocycles. 76: 1141-1154. PMID 19802363 DOI: 10.3987/Com-08-S(N)73 |
0.792 |
|
| 2008 |
Kalisiak J, Sharpless KB, Fokin VV. Efficient synthesis of 2-substituted-1,2,3-triazoles. Organic Letters. 10: 3171-4. PMID 18597477 DOI: 10.1021/Ol8006748 |
0.733 |
|
| 2008 |
Yoo EJ, Ahlquist M, Bae I, Sharpless KB, Fokin VV, Chang S. Mechanistic studies on the Cu-catalyzed three-component reactions of sulfonyl azides, 1-alkynes and amines, alcohols, or water: dichotomy via a common pathway. The Journal of Organic Chemistry. 73: 5520-8. PMID 18557650 DOI: 10.1021/Jo800733P |
0.806 |
|
| 2008 |
Radi? Z, Manetsch R, Fournier D, Sharpless KB, Taylor P. Probing gorge dimensions of cholinesterases by freeze-frame click chemistry. Chemico-Biological Interactions. 175: 161-5. PMID 18555981 DOI: 10.1016/J.Cbi.2008.04.048 |
0.677 |
|
| 2008 |
Finn MG, Kolb HC, Fokin VV, Sharpless KB. Click chemistry - Definition and aims Progress in Chemistry. 20: 1-4. |
0.759 |
|
| 2007 |
Sugawara A, Sunazuka T, Hirose T, Nagai K, Yamaguchi Y, Hanaki H, Sharpless KB, Omura S. Design and synthesis via click chemistry of 8,9-anhydroerythromycin A 6,9-hemiketal analogues with anti-MRSA and -VRE activity. Bioorganic & Medicinal Chemistry Letters. 17: 6340-4. PMID 17869508 DOI: 10.1016/J.Bmcl.2007.08.068 |
0.3 |
|
| 2007 |
Yoo EJ, Ahlquist M, Kim SH, Bae I, Fokin VV, Sharpless KB, Chang S. Copper-catalyzed synthesis of N-sulfonyl-1,2,3-triazoles: controlling selectivity. Angewandte Chemie (International Ed. in English). 46: 1730-3. PMID 17397087 DOI: 10.1002/CHIN.200724118 |
0.81 |
|
| 2007 |
Hawker CJ, Fokin VV, Finn MG, Sharpless KB. Bringing efficiency to materials synthesis: The philosophy of click chemistry Australian Journal of Chemistry. 60: 381-383. DOI: 10.1071/Ch07107 |
0.772 |
|
| 2007 |
Liu Y, Díaz DD, Accurso AA, Sharpless KB, Fokin VV, Finn MG. Click chemistry in materials synthesis. III. Metal-adhesive polymers from Cu(I)-catalyzed azide-alkyne cycloaddition Journal of Polymer Science, Part a: Polymer Chemistry. 45: 5182-5189. DOI: 10.1002/Pola.22262 |
0.783 |
|
| 2007 |
Vestberg R, Malkoch M, Kade M, Wu P, Fokin VV, Sharpless KB, Drockenmuller E, Hawker CJ. Role of architecture and molecular weight in the formation of tailor-made ultrathin multilayers using dendritic macromolecules and click chemistry Journal of Polymer Science, Part a: Polymer Chemistry. 45: 2835-2846. DOI: 10.1002/Pola.22178 |
0.709 |
|
| 2007 |
Narayan S, Fokin VV, Sharpless KB. Chemistry 'On Water'-Organic Synthesis in Aqueous Suspension Organic Reactions in Water: Principles, Strategies and Applications. 350-365. DOI: 10.1002/9780470988817.ch11 |
0.656 |
|
| 2006 |
Sharpless KB, Manetsch R. In situ click chemistry: a powerful means for lead discovery. Expert Opinion On Drug Discovery. 1: 525-38. PMID 23506064 DOI: 10.1517/17460441.1.6.525 |
0.68 |
|
| 2006 |
Díaz DD, Converso A, Sharpless KB, Finn MG. 2,6-Dichloro-9-thiabicyclo[3.3.1]nonane: multigram display of azide and cyanide components on a versatile scaffold. Molecules (Basel, Switzerland). 11: 212-8. PMID 17962753 DOI: 10.3390/11040212 |
0.786 |
|
| 2006 |
Whiting M, Tripp JC, Lin YC, Lindstrom W, Olson AJ, Elder JH, Sharpless KB, Fokin VV. Rapid discovery and structure-activity profiling of novel inhibitors of human immunodeficiency virus type 1 protease enabled by the copper(I)-catalyzed synthesis of 1,2,3-triazoles and their further functionalization. Journal of Medicinal Chemistry. 49: 7697-710. PMID 17181152 DOI: 10.1021/Jm060754+ |
0.805 |
|
| 2006 |
Whiting M, Muldoon J, Lin YC, Silverman SM, Lindstrom W, Olson AJ, Kolb HC, Finn MG, Sharpless KB, Elder JH, Fokin VV. Inhibitors of HIV-1 protease by using in situ click chemistry. Angewandte Chemie (International Ed. in English). 45: 1435-9. PMID 16425339 DOI: 10.1002/Anie.200502161 |
0.758 |
|
| 2006 |
Hirose T, Sunazuka T, Noguchi Y, Yamaguchi Y, Hanaki H, Sharpless KB, Omura S. Rapid 'SAR' via click chemistry: An alkyne-bearing spiramycin is fused with diverse azides to yield new triazole-antibacterial candidates Heterocycles. 69: 55-61. DOI: 10.3987/Com-06-S(O)7 |
0.363 |
|
| 2005 |
Wu P, Malkoch M, Hunt JN, Vestberg R, Kaltgrad E, Finn MG, Fokin VV, Sharpless KB, Hawker CJ. Multivalent, bifunctional dendrimers prepared by click chemistry. Chemical Communications (Cambridge, England). 5775-7. PMID 16307142 DOI: 10.1039/B512021G |
0.783 |
|
| 2005 |
Radi? Z, Manetsch R, Krasi?ski A, Raushel J, Yamauchi J, Garcia C, Kolb H, Sharpless KB, Taylor P. Molecular basis of interactions of cholinesterases with tight binding inhibitors. Chemico-Biological Interactions. 157: 133-41. PMID 16289416 DOI: 10.1016/J.Cbi.2005.10.020 |
0.73 |
|
| 2005 |
Zhang L, Chen X, Xue P, Sun HH, Williams ID, Sharpless KB, Fokin VV, Jia G. Ruthenium-catalyzed cycloaddition of alkynes and organic azides. Journal of the American Chemical Society. 127: 15998-9. PMID 16287266 DOI: 10.1002/chin.200612126 |
0.689 |
|
| 2005 |
Bourne Y, Radi? Z, Kolb HC, Sharpless KB, Taylor P, Marchot P. Structural insights into conformational flexibility at the peripheral site and within the active center gorge of AChE. Chemico-Biological Interactions. 157: 159-65. PMID 16259971 DOI: 10.1016/J.Cbi.2005.10.018 |
0.567 |
|
| 2005 |
Feldman AK, Colasson B, Sharpless KB, Fokin VV. The allylic azide rearrangement: achieving selectivity. Journal of the American Chemical Society. 127: 13444-5. PMID 16190677 DOI: 10.1021/Ja050622Q |
0.803 |
|
| 2005 |
Krasi?ski A, Radi? Z, Manetsch R, Raushel J, Taylor P, Sharpless KB, Kolb HC. In situ selection of lead compounds by click chemistry: target-guided optimization of acetylcholinesterase inhibitors. Journal of the American Chemical Society. 127: 6686-92. PMID 15869290 DOI: 10.1021/Ja043031T |
0.755 |
|
| 2005 |
Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. "On water": unique reactivity of organic compounds in aqueous suspension. Angewandte Chemie (International Ed. in English). 44: 3275-9. PMID 15844112 DOI: 10.1002/Anie.200462883 |
0.77 |
|
| 2005 |
Himo F, Lovell T, Hilgraf R, Rostovtsev VV, Noodleman L, Sharpless KB, Fokin VV. Copper(I)-catalyzed synthesis of azoles. DFT study predicts unprecedented reactivity and intermediates. Journal of the American Chemical Society. 127: 210-6. PMID 15631470 DOI: 10.1021/Ja0471525 |
0.805 |
|
| 2005 |
Loren JC, Krasiński A, Fokin VV, Sharpless KB. NH-1,2,3-triazoles from azidomethyl pivalate and carbamates: Base-labile N-protecting groups Synlett. 2847-2850. DOI: 10.1055/S-2005-918944 |
0.679 |
|
| 2005 |
Loren JC, Sharpless KB. The Banert cascade: A synthetic sequence to polyfunctional NH-1,2,3-triazoles Synthesis. 1514-1520. DOI: 10.1055/S-2005-869892 |
0.336 |
|
| 2005 |
Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. Cover Picture: “On Water”: Unique Reactivity of Organic Compounds in Aqueous Suspension (Angew. Chem. Int. Ed. 21/2005) Angewandte Chemie International Edition. 44: 3157-3157. DOI: 10.1002/Anie.200590069 |
0.775 |
|
| 2005 |
Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. Titelbild: “On Water”: Unique Reactivity of Organic Compounds in Aqueous Suspension (Angew. Chem. 21/2005) Angewandte Chemie. 117: 3219-3219. DOI: 10.1002/Ange.200590069 |
0.775 |
|
| 2004 |
Mocharla VP, Colasson B, Lee LV, Röper S, Sharpless KB, Wong CH, Kolb HC. In situ click chemistry: enzyme-generated inhibitors of carbonic anhydrase II. Angewandte Chemie (International Ed. in English). 44: 116-20. PMID 15599912 DOI: 10.1002/Anie.200461580 |
0.719 |
|
| 2004 |
Converso A, Saaidi PL, Sharpless KB, Finn MG. Nucleophilic substitution by grignard reagents on sulfur mustards. The Journal of Organic Chemistry. 69: 7336-9. PMID 15471488 DOI: 10.1021/Jo0489869 |
0.785 |
|
| 2004 |
Manetsch R, Krasi?ski A, Radi? Z, Raushel J, Taylor P, Sharpless KB, Kolb HC. In situ click chemistry: enzyme inhibitors made to their own specifications. Journal of the American Chemical Society. 126: 12809-18. PMID 15469276 DOI: 10.1021/Ja046382G |
0.754 |
|
| 2004 |
Chan TR, Hilgraf R, Sharpless KB, Fokin VV. Polytriazoles as copper(I)-stabilizing ligands in catalysis. Organic Letters. 6: 2853-5. PMID 15330631 DOI: 10.1021/Ol0493094 |
0.79 |
|
| 2004 |
Wu P, Feldman AK, Nugent AK, Hawker CJ, Scheel A, Voit B, Pyun J, Fréchet JM, Sharpless KB, Fokin VV. Efficiency and fidelity in a click-chemistry route to triazole dendrimers by the copper(i)-catalyzed ligation of azides and alkynes. Angewandte Chemie (International Ed. in English). 43: 3928-32. PMID 15274216 DOI: 10.1002/Anie.200454078 |
0.805 |
|
| 2004 |
Krasi?ski A, Fokin VV, Sharpless KB. Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited. Organic Letters. 6: 1237-40. PMID 15070306 DOI: 10.1021/Ol0499203 |
0.729 |
|
| 2004 |
Bourne Y, Kolb HC, Radi? Z, Sharpless KB, Taylor P, Marchot P. Freeze-frame inhibitor captures acetylcholinesterase in a unique conformation. Proceedings of the National Academy of Sciences of the United States of America. 101: 1449-54. PMID 14757816 DOI: 10.1073/Pnas.0308206100 |
0.619 |
|
| 2004 |
Díaz DD, Punna S, Holzer P, Mcpherson AK, Sharpless KB, Fokin VV, Finn MG. Click chemistry in materials synthesis. 1. Adhesive polymers from copper-catalyzed azide-alkyne cycloaddition Journal of Polymer Science, Part a: Polymer Chemistry. 42: 4392-4403. DOI: 10.1002/Pola.20330 |
0.796 |
|
| 2004 |
Wu P, Feldman AK, Nugent AK, Hawker CJ, Scheel A, Voit B, Pyun J, Fréchet JMJ, Sharpless KB, Fokin VV. Cover Picture: Efficiency and Fidelity in a Click-Chemistry Route to Triazole Dendrimers by the Copper(I)-Catalyzed Ligation of Azides and Alkynes (Angew. Chem. Int. Ed. 30/2004) Angewandte Chemie International Edition. 43: 3863-3863. DOI: 10.1002/Anie.200490100 |
0.802 |
|
| 2004 |
Wu P, Feldman AK, Nugent AK, Hawker CJ, Scheel A, Voit B, Pyun J, Fréchet JMJ, Sharpless KB, Fokin VV. Titelbild: Efficiency and Fidelity in a Click-Chemistry Route to Triazole Dendrimers by the Copper(I)-Catalyzed Ligation of Azides and Alkynes (Angew. Chem. 30/2004) Angewandte Chemie. 116: 3951-3951. DOI: 10.1002/Ange.200490100 |
0.805 |
|
| 2003 |
Kolb HC, Sharpless KB. The growing impact of click chemistry on drug discovery. Drug Discovery Today. 8: 1128-37. PMID 14678739 DOI: 10.1016/S1359-6446(03)02933-7 |
0.613 |
|
| 2003 |
Brik A, Muldoon J, Lin YC, Elder JH, Goodsell DS, Olson AJ, Fokin VV, Sharpless KB, Wong CH. Rapid diversity-oriented synthesis in microtiter plates for in situ screening of HIV protease inhibitors. Chembiochem : a European Journal of Chemical Biology. 4: 1246-8. PMID 14613121 DOI: 10.1002/Cbic.200300724 |
0.678 |
|
| 2003 |
Himo F, Demko ZP, Noodleman L, Sharpless KB. Why is tetrazole formation by addition of azide to organic nitriles catalyzed by zinc(II) salts? Journal of the American Chemical Society. 125: 9983-7. PMID 12914461 DOI: 10.1021/Ja030204Q |
0.61 |
|
| 2003 |
Lee LV, Mitchell ML, Huang SJ, Fokin VV, Sharpless KB, Wong CH. A potent and highly selective inhibitor of human alpha-1,3-fucosyltransferase via click chemistry. Journal of the American Chemical Society. 125: 9588-9. PMID 12904015 DOI: 10.1021/Ja0302836 |
0.714 |
|
| 2003 |
Ripka AS, Díaz DD, Sharpless KB, Finn MG. First practical synthesis of formamidine ureas and derivatives. Organic Letters. 5: 1531-3. PMID 12713316 DOI: 10.1021/Ol034287R |
0.716 |
|
| 2003 |
Wang Q, Chan TR, Hilgraf R, Fokin VV, Sharpless KB, Finn MG. Bioconjugation by copper(I)-catalyzed azide-alkyne [3 + 2] cycloaddition. Journal of the American Chemical Society. 125: 3192-3. PMID 12630856 DOI: 10.1021/Ja021381E |
0.796 |
|
| 2003 |
Kitayama T, Yokoi T, Kawai Y, Hill RK, Morita M, Okamoto T, Yamamoto Y, Fokin VV, Sharpless KB, Sawada S. The chemistry of zerumbone. Part 5: Structural transformation of the dimethylamine derivatives Tetrahedron. 59: 4857-4866. DOI: 10.1016/S0040-4020(03)00667-7 |
0.711 |
|
| 2003 |
Oi R, Sharpless KB. 3‐[(1S)‐1,2‐Dihydroxyethyl]‐1,5‐Dihydro‐3H‐2,4‐Benzodioxepine Organic Syntheses. 1-1. DOI: 10.1002/0471264180.Os073.01 |
0.351 |
|
| 2003 |
Herranz E, Sharpless KB. Osmium‐catalyzed vicinal oxyamination of olefins by N‐chloro‐N‐argentocarbamates: ethyl threo‐[1‐(2‐hydroxy‐1,2‐diphenylethyl)]carbamate Organic Syntheses. 93-93. DOI: 10.1002/0471264180.Os061.21 |
0.324 |
|
| 2002 |
Demko ZP, Sharpless KB. A click chemistry approach to tetrazoles by Huisgen 1,3-dipolar cycloaddition: synthesis of 5-acyltetrazoles from azides and acyl cyanides. Angewandte Chemie (International Ed. in English). 41: 2113-6. PMID 19746613 DOI: 10.1002/1521-3773(20020617)41:12<2113::AID-ANIE2113>3.0.CO;2-Q |
0.629 |
|
| 2002 |
Demko ZP, Sharpless KB. A click chemistry approach to tetrazoles by Huisgen 1,3-dipolar cycloaddition: synthesis of 5-sulfonyl tetrazoles from azides and sulfonyl cyanides. Angewandte Chemie (International Ed. in English). 41: 2110-3. PMID 19746612 DOI: 10.1002/1521-3773(20020617)41:12<2110::Aid-Anie2110>3.0.Co;2-7 |
0.66 |
|
| 2002 |
Sharpless KB. Searching for new reactivity (Nobel lecture). Angewandte Chemie (International Ed. in English). 41: 2024-32. PMID 19746596 DOI: 10.1002/1521-3773(20020617)41:12<2024::Aid-Anie2024>3.0.Co;2-O |
0.399 |
|
| 2002 |
Andersson MA, Epple R, Fokin VV, Sharpless KB. A new approach to osmium-catalyzed asymmetric dihydroxylation and aminohydroxylation of olefins. Angewandte Chemie (International Ed. in English). 41: 472-5. PMID 12491382 DOI: 10.1002/1521-3773(20020201)41:3<472::Aid-Anie472>3.0.Co;2-7 |
0.693 |
|
| 2002 |
Lewis WG, Green LG, Grynszpan F, Radi? Z, Carlier PR, Taylor P, Finn MG, Sharpless KB. Click chemistry in situ: acetylcholinesterase as a reaction vessel for the selective assembly of a femtomolar inhibitor from an array of building blocks. Angewandte Chemie (International Ed. in English). 41: 1053-7. PMID 12491310 DOI: 10.1002/1521-3773(20020315)41:6<1053::Aid-Anie1053>3.0.Co;2-4 |
0.788 |
|
| 2002 |
Himo F, Demko ZP, Noodleman L, Sharpless KB. Mechanisms of tetrazole formation by addition of azide to nitriles. Journal of the American Chemical Society. 124: 12210-6. PMID 12371861 DOI: 10.1021/Ja0206644 |
0.645 |
|
| 2002 |
Rostovtsev VV, Green LG, Fokin VV, Sharpless KB. A stepwise huisgen cycloaddition process: copper(I)-catalyzed regioselective "ligation" of azides and terminal alkynes. Angewandte Chemie (International Ed. in English). 41: 2596-9. PMID 12203546 DOI: 10.1002/1521-3773(20020715)41:14<2596::Aid-Anie2596>3.0.Co;2-4 |
0.714 |
|
| 2002 |
Demko ZP, Sharpless KB. An expedient route to the tetrazole analogues of alpha-amino acids. Organic Letters. 4: 2525-7. PMID 12123367 DOI: 10.1021/Ol020096X |
0.626 |
|
| 2002 |
Dupau P, Epple R, Thomas AA, Fokin VV, Sharpless KB. Osmium-Catalyzed Dihydroxylation of Olefins in Acidic Media: Old Process, New Tricks Advanced Synthesis and Catalysis. 344: 421-433. DOI: 10.1002/1615-4169(200206)344:3/4<421::Aid-Adsc421>3.0.Co;2-F |
0.762 |
|
| 2002 |
Lewis WG, Green LG, Grynszpan F, Radić Z, Carlier PR, Taylor P, Finn MG, Sharpless KB. Cover Picture: Angew. Chem. Int. Ed. 6/2002 Angewandte Chemie International Edition. 41: 875-875. DOI: 10.1002/1521-3773(20020315)41:6<875::Aid-Anie875>3.0.Co;2-Y |
0.783 |
|
| 2002 |
Demko ZP, Sharpless KB. A Click Chemistry Approach to Tetrazoles by Huisgen 1,3-Dipolar Cycloaddition: Synthesis of 5-Acyltetrazoles from Azides and Acyl Cyanides We thank the National Institute of General Medical Sciences, National Institutes of Health (GM-28384), the National Science Foundation (CHE-9985553), the Skaggs Institute for Chemical Biology for a Predoctoral Fellowship (Z.D.), and the W. M. Keck Foundation for financial support. Angewandte Chemie. 114: 2217. DOI: 10.1002/1521-3757(20020617)114:12<2217::Aid-Ange2217>3.0.Co;2-X |
0.602 |
|
| 2002 |
Lewis WG, Green LG, Grynszpan F, Radić Z, Carlier PR, Taylor P, Finn MG, Sharpless KB. Titelbild: 6/2002 Angewandte Chemie. 114: 915-915. DOI: 10.1002/1521-3757(20020315)114:6<915::Aid-Ange915>3.0.Co;2-3 |
0.763 |
|
| 2001 |
Demko ZP, Sharpless KB. An intramolecular [2 + 3] cycloaddition route to fused 5-heterosubstituted tetrazoles. Organic Letters. 3: 4091-4. PMID 11735592 DOI: 10.1021/Ol010220X |
0.669 |
|
| 2001 |
Demko ZP, Sharpless KB. Preparation of 5-substituted 1H-tetrazoles from nitriles in water. The Journal of Organic Chemistry. 66: 7945-50. PMID 11722189 DOI: 10.1021/Jo010635W |
0.665 |
|
| 2001 |
Fokin VV, Sharpless KB. A Practical and Highly Efficient Aminohydroxylation of Unsaturated Carboxylic Acids We thank the National Institute of General Medical Sciences, the National Institutes of Health (GM 28384), National Science Foundation (CHE-9985553), and the W. M. Keck Foundation for financial support. We are also grateful to Prof. M. G. Finn, Dr. Wallace Pringle, and Dr. A. Erik Rubin for many helpful discussions. Angewandte Chemie (International Ed. in English). 40: 3455-3457. PMID 11592169 DOI: 10.1002/1521-3773(20010917)40:18<3455::Aid-Anie3455>3.0.Co;2-I |
0.646 |
|
| 2001 |
Kolb HC, Finn MG, Sharpless KB. Click Chemistry: Diverse Chemical Function from a Few Good Reactions. Angewandte Chemie (International Ed. in English). 40: 2004-2021. PMID 11433435 DOI: 10.1002/1521-3773(20010601)40:11<2004::Aid-Anie2004>3.3.Co;2-X |
0.724 |
|
| 2001 |
Marzinzik AL, Sharpless KB. A simple method for the preparation of N-sulfonylsulfilimines from sulfides. The Journal of Organic Chemistry. 66: 594-6. PMID 11429835 DOI: 10.1021/Jo0012039 |
0.335 |
|
| 2001 |
Converso A, Burow K, Marzinzik A, Sharpless KB, Finn MG. 2,6-Dichloro-9-thiabicyclo[3.3.1]nonane: a privileged, bivalent scaffold for the display of nucleophilic components. The Journal of Organic Chemistry. 66: 4386-92. PMID 11397181 DOI: 10.1021/Jo015632Y |
0.784 |
|
| 2001 |
Kolb HC, Finn MG, Sharpless KB. Click-Chemie: diverse chemische Funktionalität mit einer Handvoll guter Reaktionen Angewandte Chemie. 113: 2056-2075. DOI: 10.1002/1521-3757(20010601)113:11<2056::Aid-Ange2056>3.0.Co;2-W |
0.674 |
|
| 2000 |
Demko ZP, Bartsch M, Sharpless KB. Primary amides. A general nitrogen source for catalytic asymmetric aminohydroxylation of olefins. Organic Letters. 2: 2221-3. PMID 10930248 DOI: 10.1021/Ol000098M |
0.638 |
|
| 2000 |
Demko ZP, Bartsch M, Sharpless KB. ChemInform Abstract: Primary Amides. A General Nitrogen Source for Catalytic Asymmetric Aminohydroxylation of Olefins. Cheminform. 31: no-no. DOI: 10.1002/chin.200045098 |
0.598 |
|
| 2000 |
Chuang TH, Sharpless KB. Applications of aziridinium ions: Selective syntheses of pyrazolidin-3-ones and pyrazolo[1,2-α]pyrazoles Helvetica Chimica Acta. 83: 1734-1743. DOI: 10.1002/1522-2675(20000809)83:8<1734::Aid-Hlca1734>3.0.Co;2-E |
0.35 |
|
| 1999 |
Goossen LJ, Liu H, Dress KR, Sharpless KB. Catalytic asymmetric aminohydroxylation with amino-substituted heterocycles as nitrogen sources. Angewandte Chemie (International Ed. in English). 38: 1080-3. PMID 25138500 DOI: 10.1002/(Sici)1521-3773(19990419)38:8<1080::Aid-Anie1080>3.0.Co;2-D |
0.333 |
|
| 1999 |
Thomas AA, Sharpless KB. The Catalytic Asymmetric Aminohydroxylation of Unsaturated Phosphonates. The Journal of Organic Chemistry. 64: 8379-8385. PMID 11674762 DOI: 10.1021/Jo990060R |
0.582 |
|
| 1999 |
Gontcharov AV, Liu H, Sharpless KB. Tert-butylsulfonamide. A new nitrogen source for catalytic aminohydroxylation and aziridination of olefins. Organic Letters. 1: 783-6. PMID 10823205 DOI: 10.1021/Ol990761A |
0.378 |
|
| 1999 |
Pringle W, Sharpless KB. The osmium-catalyzed aminohydroxylation of Baylis-Hillman olefins Tetrahedron Letters. 40: 5151-5154. DOI: 10.1016/S0040-4039(99)00887-4 |
0.389 |
|
| 1999 |
Adolfsson H, Converso A, Sharpless KB. Comparison of amine additives most effective in the new methyltrioxorhenium-catalyzed epoxidation process Tetrahedron Letters. 40: 3991-3994. DOI: 10.1016/S0040-4039(99)00661-9 |
0.764 |
|
| 1998 |
Gypser A, Michel D, Nirschl DS, Sharpless KB. Dihydroxylation of Polyenes Using Narasaka's Modification of the Upjohn Procedure. The Journal of Organic Chemistry. 63: 7322-7327. PMID 11672379 DOI: 10.1021/jo980850l |
0.713 |
|
| 1998 |
Copéret C, Adolfsson H, Khuong TAV, Yudin AK, Sharpless KB. A simple and efficient method for the preparation of pyridine N-oxides Journal of Organic Chemistry. 63: 1740-1741. DOI: 10.1021/Jo9723467 |
0.626 |
|
| 1998 |
and KLR, Sharpless KB. From Styrenes to Enantiopure α-Arylglycines in Two Steps Journal of the American Chemical Society. 120: 1207-1217. DOI: 10.1021/Ja9728177 |
0.323 |
|
| 1998 |
Dress KR, Gooßen LJ, Liu H, Jerina DM, Sharpless KB. Catalytic aminohydroxylation using adenine-derivatives as the nitrogen source Tetrahedron Letters. 39: 7669-7672. DOI: 10.1016/S0040-4039(98)01716-X |
0.333 |
|
| 1998 |
Tao B, Schlingloff G, Sharpless KB. Reversal of regioselection in the asymmetric aminohydroxylation of cinnamates Tetrahedron Letters. 39: 2507-2510. DOI: 10.1016/S0040-4039(98)00350-5 |
0.316 |
|
| 1998 |
Copéret C, Adolfsson H, Chiang JP, Yudin AK, Sharpless KB. A simple and efficient method for the preparation of pyridine-N-oxides II Tetrahedron Letters. 39: 761-764. DOI: 10.1016/S0040-4039(97)10619-0 |
0.786 |
|
| 1997 |
Copéret C, Adolfsson H, Sharpless KB. A Simple And Efficient Method For Epoxidation Of Terminal Alkenes Chemical Communications. 1565-1566. DOI: 10.1039/A703542J |
0.517 |
|
| 1997 |
Yudin AK, Sharpless KB. Bis(trimethylsilyl) peroxide extends the range of oxorhenium catalysts for olefin epoxidation [2] Journal of the American Chemical Society. 119: 11536-11537. DOI: 10.1021/Ja973043X |
0.542 |
|
| 1997 |
DelMonte AJ, Haller J, Houk KN, Sharpless KB, Singleton DA, Strassner T, Thomas AA. Experimental and theoretical kinetic isotope effects for asymmetric dihydroxylation. Evidence supporting a rate-limiting '(3+2)' cycloaddition Journal of the American Chemical Society. 119: 9907-9908. DOI: 10.1021/Ja971650E |
0.459 |
|
| 1997 |
Nelson DW, Gypser A, Ho PT, Kolb HC, Kondo T, Kwong HL, McGrath DV, Rubin AE, Norrby PO, Gable KP, Sharpless KB. Toward an understanding of the high enantioselectivity in the osmium-catalyzed asymmetric dihydroxylation. 4. Electronic effects in amine-accelerated osmylations Journal of the American Chemical Society. 119: 1840-1858. DOI: 10.1021/Ja961464T |
0.777 |
|
| 1996 |
Li G, Sharpless KB. Catalytic asymmetric aminohydroxylation provides a short taxol side-chain synthesis. Acta Chemica Scandinavica (Copenhagen, Denmark : 1989). 50: 649-51. PMID 8756354 DOI: 10.3891/acta.chem.scand.50-0649 |
0.686 |
|
| 1996 |
Norrby P, Becker H, Sharpless KB. Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation. 3. New Insights into Isomeric Forms of the Putative Osmaoxetane Intermediate Journal of the American Chemical Society. 118: 35-42. DOI: 10.1021/Ja952470C |
0.596 |
|
| 1996 |
Li G, Angert HH, Sharpless KB. N-Halocarbamate Salts Lead to More Efficient Catalytic Asymmetric Aminohydroxylation Angewandte Chemie International Edition in English. 35: 2813-2817. DOI: 10.1002/Anie.199628131 |
0.487 |
|
| 1996 |
Rudolph J, Sennhenn PC, Vlaar CP, Sharpless KB. Smaller Substituents on Nitrogen Facilitate the Osmium-Catalyzed Asymmetric Aminohydroxylation Angewandte Chemie International Edition in English. 35: 2810-2813. DOI: 10.1002/Anie.199628101 |
0.389 |
|
| 1996 |
Bruncko M, Khuong TV, Sharpless KB. Allylic Amination and 1,2-Diamination with a Modified Diimidoselenium Reagent Angewandte Chemie International Edition in English. 35: 454-456. DOI: 10.1002/Anie.199604541 |
0.389 |
|
| 1996 |
Li G, Chang H, Sharpless KB. Catalytic Asymmetric Aminohydroxylation(AA) of Olefins Angewandte Chemie International Edition in English. 35: 451-454. DOI: 10.1002/Anie.199604511 |
0.498 |
|
| 1996 |
Chang H, Chen C, Kondo T, Siuzdak G, Sharpless KB. Asymmetric Dihydroxylation Enables Rapid Construction of Chiral Dendrimers Based on 1,2-Diols Angewandte Chemie International Edition in English. 35: 182-186. DOI: 10.1002/Anie.199601821 |
0.303 |
|
| 1996 |
Li G, Angert HH, Sharpless KB. Erhöhung der Effizienz der katalytischen asymmetrischen Aminohydroxylierung durchN-Halogencarbamat-Salze Angewandte Chemie. 108: 2995-2999. DOI: 10.1002/Ange.19961082325 |
0.388 |
|
| 1996 |
Li G, Chang H, Sharpless KB. Katalytische asymmetrische Aminohydroxylierung (AA) von Olefinen Angewandte Chemie. 108: 449-452. DOI: 10.1002/Ange.19961080409 |
0.378 |
|
| 1995 |
Becker H, King SB, Taniguchi M, Vanhessche KPM, Sharpless KB. New Ligands and Improved Enantioselectivities for the Asymmetric Dihydroxylation of Olefins Journal of Organic Chemistry. 60: 3940-3941. DOI: 10.1021/Jo00118A005 |
0.415 |
|
| 1995 |
Richardson PF, Nelson LTJ, Sharpless KB. Synthesis of vicinal diamines from cyclic sulfates Tetrahedron Letters. 36: 9241-9244. DOI: 10.1016/0040-4039(95)02014-G |
0.347 |
|
| 1995 |
Berrisford DJ, Bolm C, Sharpless KB. Ligand-Accelerated Catalysis Angewandte Chemie International Edition in English. 34: 1059-1070. DOI: 10.1002/Anie.199510591 |
0.776 |
|
| 1994 |
Norrby PO, Kolb HC, Sharpless KB. Calculations on the reaction of ruthenium tetroxide with olefins using density functional theory (DFT). Implications for the possibility of intermediates in osmium-catalyzed asymmetric dihydroxylation Organometallics. 13: 344-347. DOI: 10.1021/Om00013A050 |
0.682 |
|
| 1994 |
Wang Z, Kolb HC, Sharpless KB. Large-Scale and Highly Enantioselective Synthesis of the Taxol C-13 Side Chain through Asymmetric Dihydroxylation The Journal of Organic Chemistry. 59: 5104-5105. DOI: 10.1021/Jo00096A072 |
0.579 |
|
| 1994 |
Norrby P, Kolb HC, Sharpless KB. Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation. 2. A Qualitative Molecular Mechanics Approach Journal of the American Chemical Society. 116: 8470-8478. DOI: 10.1021/Ja00098A006 |
0.677 |
|
| 1994 |
Kolb HC, Andersson PG, Sharpless KB. Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation (AD). 1. Kinetics Journal of the American Chemical Society. 116: 1278-1291. DOI: 10.1021/Ja00083A014 |
0.726 |
|
| 1994 |
Kolb HC, VanNieuwenhze MS, Sharpless KB. Catalytic Asymmetric Dihydroxylation Chemical Reviews. 94: 2483-2547. DOI: 10.1021/Cr00032A009 |
0.724 |
|
| 1994 |
King SB, Sharpless KB. An efficient synthesis of enantiomerically pure trans-2-phenylcyclohexanol Tetrahedron Letters. 35: 5611-5612. DOI: 10.1016/S0040-4039(00)77259-5 |
0.358 |
|
| 1994 |
Xu D, Park CY, Sharpless KB. Study of the regio- and enantioselectivity of the reactions of osmium tetroxide with allylic alcohols and allylic sulfonamides Tetrahedron Letters. 35: 2495-2498. DOI: 10.1016/S0040-4039(00)77153-X |
0.31 |
|
| 1994 |
Walsh PJ, Tong Ho P, King SB, Sharpless KB. Asymmetric dihydroxylation of olefins containing sulfur: Chemoselective oxidation of CC double bonds in the presence of sulfides, 1,3-dithianes, and disulfides Tetrahedron Letters. 35: 5129-5132. DOI: 10.1016/S0040-4039(00)77045-6 |
0.498 |
|
| 1994 |
VanNieuwenhze MS, Sharpless KB. The asymmetric dihydroxylation of cis-allylic and homoallylic alcohols Tetrahedron Letters. 35: 843-846. DOI: 10.1016/S0040-4039(00)75978-8 |
0.597 |
|
| 1994 |
Vanhessche KPM, Wang ZM, Sharpless KB. Asymmetric dihydroxylation of primary allylic halides and a concise synthesis of (-)-diepoxybutane Tetrahedron Letters. 35: 3469-3472. DOI: 10.1016/S0040-4039(00)73212-6 |
0.344 |
|
| 1994 |
Sharpless KB. Coelacanths and catalysis Tetrahedron. 50: 4235-4258. DOI: 10.1016/S0040-4020(01)89364-9 |
0.334 |
|
| 1994 |
Bennani YL, Vanhessche KPM, Sharpless KB. A short route to a moshe'rs acid precursor via catalytic asymmetric dihydroxylation (AD) Tetrahedron: Asymmetry. 5: 1473-1476. DOI: 10.1016/0957-4166(94)80116-9 |
0.336 |
|
| 1994 |
Becker H, Tong Ho P, Kolb HC, Loren S, Norrby PO, Sharpless KB. Comparing two models for the selectivity in the asymmetric dihydroxylation reaction (AD) Tetrahedron Letters. 35: 7315-7318. DOI: 10.1016/0040-4039(94)85302-9 |
0.787 |
|
| 1993 |
Walsh PJ, Sharpless KB. Asymmetric Dihydroxylation (AD) of α,β-Unsaturated Ketones Synlett. 1993: 605-606. DOI: 10.1055/S-1993-22548 |
0.436 |
|
| 1993 |
Crispino GA, Sharpless KB. Enantioselective Synthesis of Both Enantiomers of 7,7-Dimethyl-6,8-dioxa-bicyclo[3.2.1]octane via Regioselective Asymmetric Dihydroxylation Synlett. 1993: 47-48. DOI: 10.1055/S-1993-22343 |
0.349 |
|
| 1993 |
Crispino GA, Jeong KS, Kolb HC, Wang ZM, Xu D, Sharpless KB. Improved enantioselectivity in asymmetric dihydroxylations of terminal olefins using pyrimidine ligands Journal of Organic Chemistry. 58: 3785-3786. DOI: 10.1021/Jo00067A002 |
0.335 |
|
| 1993 |
Amberg W, Bennani YL, Chadha RK, Crispino GA, Davis WD, Hartung J, Jeong KS, Ogino Y, Shibata T, Sharpless KB. Syntheses and crystal structures of the cinchona alkaloid derivatives used as ligands in the osmium-catalyzed asymmetric dihydroxylation of olefins The Journal of Organic Chemistry. 58: 844-849. DOI: 10.1021/Jo00056A015 |
0.571 |
|
| 1993 |
Kolb HC, Andersson PG, Bennani YL, Crispino GA, Jeong KS, Kwong HL, Sharpless KB. On "The origin of high enantioselectivity in the dihydroxylation of olefins using osmium tetraoxide and cinchona alkaloid catalysts" Journal of the American Chemical Society. 115: 12226-12227. DOI: 10.1021/Ja00078A096 |
0.721 |
|
| 1993 |
VanNieuwenhze MS, Sharpless KB. Kinetic resolution of racemic olefins via asymmetric dihydroxylation Journal of the American Chemical Society. 115: 7864-7865. DOI: 10.1021/Ja00070A037 |
0.609 |
|
| 1993 |
Andersson PG, Sharpless KB. A dramatic ligand effect on the relative reactivities of substituted alkenes with osmium tetroxide Journal of the American Chemical Society. 115: 7047-7048. DOI: 10.1021/Ja00068A102 |
0.638 |
|
| 1993 |
McGrath DV, Brabson GD, Sharpless KB, Andrews L. Reinvestigation of the infrared spectra of oxoosmium(VI) esters by isotopic labeling Inorganic Chemistry. 32: 4164-4165. DOI: 10.1021/Ic00071A035 |
0.554 |
|
| 1993 |
Kolb HC, Bennani YL, Sharpless KB. Short and practical syntheses of(R)-(-)-carnitine and (R)-(-)-γ-amino-β-hydroxybutyric acid (GABOB) Tetrahedron: Asymmetry. 4: 133-141. DOI: 10.1016/S0957-4166(00)86023-1 |
0.549 |
|
| 1993 |
Wang ZM, Zhang XL, Sharpless KB. Asymmetric dihydroxylation of aryl allyl ethers Tetrahedron Letters. 34: 2267-2270. DOI: 10.1016/S0040-4039(00)77590-3 |
0.351 |
|
| 1993 |
Xu D, Sharpless KB. A simple route to enantiomerically enriched oxazolidin-2-ones Tetrahedron Letters. 34: 951-952. DOI: 10.1016/S0040-4039(00)77462-4 |
0.357 |
|
| 1993 |
Morikawa K, Sharpless KB. Double diastereoselection in asymmetric dihydroxylation Tetrahedron Letters. 34: 5575-5578. DOI: 10.1016/S0040-4039(00)73885-8 |
0.322 |
|
| 1993 |
Walsh PJ, Bennani YL, Sharpless KB. Asymmetric dihydroxylation (AD)/cyclization of N-diBoc allylic and homoallylic amines: Selective differentiation of the hydroxyl groups Tetrahedron Letters. 34: 5545-5548. DOI: 10.1016/S0040-4039(00)73877-9 |
0.521 |
|
| 1993 |
Bennani YL, Sharpless KB. Asymmetric Synthesis of γ-Hydroxy α,β-Unsaturated Amides via an AD-elimination Process; Synthesis of (+)-Coriolic Acid Tetrahedron Letters. 34: 2083-2086. DOI: 10.1016/S0040-4039(00)60351-9 |
0.314 |
|
| 1993 |
Arrington MP, Bennani YL, Göbel T, Walsh P, Zhao SH, Sharpless KB. Modified cinchona alkaloid ligands: Improved selectivities in the osmium tetroxide catalyzed asymmetric dihydroxylation (AD) of terminal olefins Tetrahedron Letters. 34: 7375-7378. DOI: 10.1016/S0040-4039(00)60129-6 |
0.529 |
|
| 1992 |
Hashiyama T, Morikawa K, Sharpless KB. .alpha.-Hydroxy ketones in high enantiomeric purity from asymmetric dihydroxylation of enol ethers Journal of Organic Chemistry. 57: 5067-5068. DOI: 10.1021/Jo00045A011 |
0.338 |
|
| 1992 |
Sharpless KB, Amberg W, Bennani YL, Crispino GA, Hartung J, Jeong KS, Kwong HL, Morikawa K, Wang ZM. The osmium-catalyzed asymmetric dihydroxylation: a new ligand class and a process improvement The Journal of Organic Chemistry. 57: 2768-2771. DOI: 10.1021/Jo00036A003 |
0.572 |
|
| 1992 |
Morikawa K, Park J, Andersson PG, Hashiyama T, Sharpless KB. Catalytic asymmetric dihydroxylation of tetrasubstituted olefins Journal of the American Chemical Society. 114: 8463-8464. DOI: 10.1021/Ja00071A072 |
0.653 |
|
| 1992 |
Keinan E, Sinha SC, Sinha-Bagchi A, Zhi-Min W, Xiu-Lian Z, Sharpless KB. Synthesis of all four isomers of disparlure using osmium-catalyzed asymmetric dihydroxylation Tetrahedron Letters. 33: 6411-6414. DOI: 10.1016/S0040-4039(00)79002-2 |
0.37 |
|
| 1992 |
Wang ZM, Zhang XL, Sharpless KB, Sinha SC, Sinha-Bagchi A, Keinan E. A general approach to γ-lactones via osmium-catalyzed asymmetric dihydroxylation. Synthesis of (-)- and (+)-muricatacin Tetrahedron Letters. 33: 6407-6410. DOI: 10.1016/S0040-4039(00)79001-0 |
0.316 |
|
| 1992 |
Crispino GA, Sharpless KB. Asymmetric dihydroxylation of squalene Tetrahedron Letters. 33: 4273-4274. DOI: 10.1016/S0040-4039(00)74236-5 |
0.333 |
|
| 1992 |
Kolb HC, Sharpless KB. A simplified procedure for the stereospecific transformation of 1,2-diols into epoxides Tetrahedron. 48: 10515-10530. DOI: 10.1016/S0040-4020(01)88349-6 |
0.63 |
|
| 1992 |
Oi R, Sharpless KB. Asymmetric dihydroxylation of acrolein acetals: synthesis of stable equivalents of Enantiopure glyceraldehyde and glycidaldehyde Tetrahedron Letters. 33: 2095-2098. DOI: 10.1016/0040-4039(92)88149-Y |
0.318 |
|
| 1991 |
McKee BH, Kalantar TH, Sharpless KB. Subtle effects in the asymmetric epoxidation: dependence of kinetic resolution efficiency on the monodentate alkoxide ligands of the bystander titanium center The Journal of Organic Chemistry. 56: 6966-6968. DOI: 10.1021/Jo00025A003 |
0.323 |
|
| 1991 |
Sharpless KB, Amberg W, Beller M, Chen H, Hartung J, Kawanami Y, Lubben D, Manoury E, Ogino Y, Shibata T, Ukita T. New ligands double the scope of the catalytic asymmetric dihydroxylation of olefins Journal of Organic Chemistry. 56: 4585-4588. DOI: 10.1021/Jo00015A001 |
0.575 |
|
| 1991 |
Finn MG, Sharpless KB. Mechanism of asymmetric epoxidation. 2. Catalyst structure Journal of the American Chemical Society. 113: 113-126. DOI: 10.1021/Ja00001A019 |
0.612 |
|
| 1991 |
Woodard SS, Finn MG, Sharpless KB. Mechanism of asymmetric epoxidation. 1. Kinetics Journal of the American Chemical Society. 113: 106-113. DOI: 10.1021/Ja00001A018 |
0.615 |
|
| 1991 |
Ogino Y, Chen H, Manoury E, Shibata T, Beller M, Lübben D, Sharpless KB. A ligand structure-enantioselectivity relationship for the osmium-catalyzed asymmetric dihydroxylation of olefins Tetrahedron Letters. 32: 5761-5764. DOI: 10.1016/S0040-4039(00)93549-4 |
0.323 |
|
| 1991 |
Oi R, Sharpless KB. Facile synthesis of enantiopure trans-2,3-diphenyl-1,4-diazabicyclo[2.2.2]octane Tetrahedron Letters. 32: 4853-4854. DOI: 10.1016/S0040-4039(00)93478-6 |
0.358 |
|
| 1991 |
Park CY, Kim BM, Sharpless KB. Catalytic osmylation of conjugated dienes: a one-pot stereoselective synthesis of polyols Tetrahedron Letters. 32: 1003-1006. DOI: 10.1016/S0040-4039(00)74472-8 |
0.416 |
|
| 1991 |
Oi R, Sharpless KB. Stereospecific conversion of chiral 1,2-cyclic sulfates to chiral imidazolines Tetrahedron Letters. 32: 999-1002. DOI: 10.1016/S0040-4039(00)74471-6 |
0.363 |
|
| 1991 |
Ogino Y, Chen H, Kwong HL, Sharpless KB. On the timing of hydrolysis / reoxidation in the osmium-catalyzed asymmetric dihydroxylation of olefins using potassium ferricyanide as the reoxidant Tetrahedron Letters. 32: 3965-3968. DOI: 10.1016/0040-4039(91)80601-2 |
0.342 |
|
| 1990 |
Kim BM, Sharpless KB. A short route to β-lactams: Use of cyclic sulfites from syn-2,3-dihydroxy esters Tetrahedron Letters. 31: 4317-4320. DOI: 10.1016/S0040-4039(00)97610-X |
0.316 |
|
| 1990 |
Shibata T, Gilheany DG, Blackburn BK, Sharpless KB. Ligand-based improvement of enantioselectivity in the catalytic asymmetric dihydroxylation of dialkyl substituted olefins Tetrahedron Letters. 31: 3817-3820. DOI: 10.1016/S0040-4039(00)97477-X |
0.343 |
|
| 1990 |
Pearlstein RM, Blackburn BK, Davis WM, Sharpless KB. Structural Characterization of the Pseudoenantiomericcis-Dioxo Osmium(VI) Esters of Chiral Diols with Cinchona Alkaloid Ligands Angewandte Chemie International Edition in English. 29: 639-641. DOI: 10.1002/Anie.199006391 |
0.302 |
|
| 1989 |
Carlier PR, Sharpless KB. Studies on the mechanism of the asymmetric epoxidation: a ligand variation approach The Journal of Organic Chemistry. 54: 4016-4018. DOI: 10.1021/Jo00278A004 |
0.577 |
|
| 1989 |
Svendsen JS, Marko I, Jacobsen EN, Rao CP, Bott S, Sharpless KB. The structure of osmium tetraoxide-cinchona alkaloid complexes The Journal of Organic Chemistry. 54: 2263-2264. DOI: 10.1021/Jo00271A002 |
0.561 |
|
| 1989 |
Klunder JM, Onami T, Sharpless KB. Arenesulfonate derivatives of homochiral glycidol: versatile chiral building blocks for organic synthesis The Journal of Organic Chemistry. 54: 1295-1304. DOI: 10.1021/Jo00267A014 |
0.323 |
|
| 1989 |
Dijkstra GDH, Kellogg RM, Wynberg H, Svendsen JS, Marko I, Sharpless KB. Conformational Study Of Cinchona Alkaloids - A Combined Nmr, Molecular Mechanics, And X-Ray Approach Journal of the American Chemical Society. 111: 8069-8076. DOI: 10.1021/Ja00203A001 |
0.483 |
|
| 1989 |
Wai JSM, Marko I, Svendsen JS, Finn MG, Jacobsen EN, Sharpless KB. A mechanistic insight leads to a greatly improved osmium-catalyzed asymmetric dihydroxylation process Journal of the American Chemical Society. 111: 1123-1125. DOI: 10.1021/Ja00185A050 |
0.739 |
|
| 1989 |
Jacobsen EN, Marko I, France MB, Svendsen JS, Sharpless KB. Kinetic role of the alkaloid ligands in asymmetric catalytic dihydroxylation Journal of the American Chemical Society. 111: 737-739. DOI: 10.1021/Ja00184A055 |
0.647 |
|
| 1989 |
Kim BM, Sharpless KB. Cyclic sulfates containing acid-sensitive groups and chemoselective hydrolysis of sulfate esters Tetrahedron Letters. 30: 655-658. DOI: 10.1016/S0040-4039(01)80274-4 |
0.348 |
|
| 1989 |
Lohray BB, Gao Y, Sharpless KB. One pot synthesis of homochiral aziridines and aminoalcohols from homochiral 1,2-cyclic sulfates Tetrahedron Letters. 30: 2623-2626. DOI: 10.1016/S0040-4039(00)99081-6 |
0.381 |
|
| 1988 |
Caron M, Carlier PR, Sharpless KB. Regioselective azide opening of 2,3-epoxy alcohols by [Ti(O-i-Pr)2(N3)2]: synthesis of .alpha.-amino acids The Journal of Organic Chemistry. 53: 5185-5187. DOI: 10.1021/Jo00256A063 |
0.57 |
|
| 1988 |
Carlier PR, Mungall WS, Schroder G, Sharpless KB. Enhanced kinetic resolution and enzyme-like shape selectivity Journal of the American Chemical Society. 110: 2978-2979. DOI: 10.1021/Ja00217A052 |
0.563 |
|
| 1988 |
Jacobsen EN, Marko I, Mungall WS, Schroeder G, Sharpless KB. Asymmetric dihydroxylation via ligand-accelerated catalysis Journal of the American Chemical Society. 110: 1968-1970. DOI: 10.1021/Ja00214A053 |
0.595 |
|
| 1988 |
Bolm C, Sharpless KB. Synthesis of a C3-symmetric phospha[2.2.2]cyclophane Tetrahedron Letters. 29: 5101-5104. DOI: 10.1016/S0040-4039(00)80690-5 |
0.436 |
|
| 1988 |
BOLM C, DAVIS WM, HALTERMAN RL, SHARPLESS KB. ChemInform Abstract: Synthesis and Structure of a Chiral, C3-Symmetric Monophosphane. Cheminform. 19. DOI: 10.1002/chin.198841254 |
0.38 |
|
| 1988 |
Bolm C, Davis WM, Halterman RL, Sharpless KB. Synthesis and Crystal Structure of a ChiralC3-Symmetric Monophosphane Angewandte Chemie International Edition in English. 27: 835-837. DOI: 10.1002/Anie.198808351 |
0.42 |
|
| 1987 |
Klunder JM, Sharpless KB. Convenient synthesis of sulfinate esters from sulfonyl chlorides The Journal of Organic Chemistry. 52: 2598-2602. DOI: 10.1021/Jo00388A051 |
0.367 |
|
| 1987 |
Pedersen SF, Dewan JC, Eckman RR, Sharpless KB. Unexpected diversity in the coordination chemistry of tartrate esters with titanium(IV) Journal of the American Chemical Society. 109: 1279-1282. DOI: 10.1021/Ja00238A065 |
0.31 |
|
| 1987 |
Hawkins JM, Sharpless KB. Asymmetric epoxidation models: An alkyl hydroperoxide dependent change in mehanism Tetrahedron Letters. 28: 2825-2828. DOI: 10.1016/S0040-4039(00)96219-1 |
0.314 |
|
| 1986 |
FINN MG, SHARPLESS KB. ChemInform Abstract: On the Mechanism of Asymmetric Epoxidation with Titanium-Tartrate Chemischer Informationsdienst. 17. DOI: 10.1002/Chin.198635340 |
0.552 |
|
| 1985 |
Adams CE, Walker FJ, Sharpless KB. Enantioselective synthesis of swainsonine, a trihydroxylated indolizidine alkaloid The Journal of Organic Chemistry. 50: 420-422. DOI: 10.1021/Jo00203A039 |
0.304 |
|
| 1985 |
Schweiter M, Sharpless K. The asymmetric epoxidation of -butyl substituted allylic alcohols Tetrahedron Letters. 26: 2543-2546. DOI: 10.1016/S0040-4039(00)98832-4 |
0.303 |
|
| 1984 |
Lu LDL, Johnson RA, Finn MG, Sharpless KB. Two new asymmetric epoxidation catalysts. Unusual stoichiometry and inverse enantiofacial selection The Journal of Organic Chemistry. 49: 728-731. DOI: 10.1021/Jo00178A039 |
0.595 |
|
| 1983 |
Ko SY, Lee AW, Masamune S, Reed LA, Sharpless KB, Walker FJ. Total synthesis of the L-hexoses. Science (New York, N.Y.). 220: 949-51. PMID 17816019 DOI: 10.1016/S0040-4020(01)97596-9 |
0.517 |
|
| 1982 |
Lee AWM, Martin VS, Masamune S, Sharpless KB, Walker FJ. Synthesis of saccharides and related polyhydroxylated natural products. 3. Efficient conversion of 2,3-erythro-aldoses to 2,3-threo-aldoses Journal of the American Chemical Society. 104: 3515-3516. DOI: 10.1021/Ja00376A050 |
0.31 |
|
| 1980 |
Hentges SG, Sharpless KB. Asymmetric induction in the reaction of osmium tetroxide with olefins Journal of the American Chemical Society. 102: 4263-4265. DOI: 10.1021/Ja00532A050 |
0.346 |
|
| 1979 |
Baeckvall JE, Oshima K, Palermo RE, Sharpless KB. Some reactions of N-(2-hydroxyalkyl)-p-toluenesulfonamides and N-allyl-p-toluenesulfonamides The Journal of Organic Chemistry. 44: 1953-1957. DOI: 10.1021/Jo01326A013 |
0.43 |
|
| 1978 |
Akashi K, Palermo RE, Sharpless KB. A major improvement in the osmium catalyzed vicinal hydroxylation of olefins by tert-butyl hydroperoxide The Journal of Organic Chemistry. 43: 2063-2066. DOI: 10.1021/Jo00404A052 |
0.366 |
|
| 1978 |
Liebeskind LS, Sharpless KB, Wilson RD, Ibers JA. The first d0 metallooxaziridines. Amination of olefins Journal of the American Chemical Society. 100: 7061-7063. DOI: 10.1002/Chin.197905268 |
0.501 |
|
| 1977 |
Chong AO, Oshima K, Sharpless KB. Synthesis of dioxobis(tert-alkylimido)osmium(VIII) and oxotris(tert-alkylimido)osmium(VIII) complexes. Stereospecific vicinal diamination of olefins Journal of the American Chemical Society. 99: 3420-3426. DOI: 10.1021/Ja00452A039 |
0.489 |
|
| 1977 |
Sharpless KB, Teranishi AY, Backvall JE. Chromyl chloride oxidations of olefins. Possible role of organometallic intermediates in the oxidations of olefins by oxo transition metal species Journal of the American Chemical Society. 99: 3120-3128. DOI: 10.1021/Ja00451A043 |
0.563 |
|
| 1977 |
Backvall JE, Young MW, Sharpless KB. Vicinal acetoxychlorination of olefins by chromyl chloride in acetyl chloride Tetrahedron Letters. 18: 3523-3526. DOI: 10.1016/S0040-4039(01)83282-2 |
0.549 |
|
| 1976 |
Sharpless KB, Chong AO, Oshima K. Osmium-catalyzed vicinal oxyamination of olefins by Chloramine-T The Journal of Organic Chemistry. 41: 177-179. DOI: 10.1021/Jo00863A052 |
0.334 |
|
| 1976 |
Sharpless KB, Akashi K. Osmium catalyzed vicinal hydroxylation of olefins by tert-butyl hydroperoxide under alkaline conditions Journal of the American Chemical Society. 98: 1986-1987. DOI: 10.1021/Ja00423A067 |
0.335 |
|
| 1976 |
Sharpless K, Akashi K, Oshima K. Ruthenium catalyzed oxidation of alcohols to aldehydes and ketones by amine-n-oxides Tetrahedron Letters. 17: 2503-2506. DOI: 10.1016/S0040-4039(00)78130-5 |
0.362 |
|
| 1975 |
Sharpless KB, Young MW. Olefin synthesis. Rate enhancement of the elimination of alkyl aryl selenoxides by electron-withdrawing substituents The Journal of Organic Chemistry. 40: 947-949. DOI: 10.1021/Jo00895A030 |
0.314 |
|
| 1975 |
Sharpless KB, Patrick DW, Truesdale LK, Biller SA. New reaction. Stereospecific vicinal oxyamination of olefins by alkyl imido osmium compounds Journal of the American Chemical Society. 97: 2305-2307. DOI: 10.1021/Ja00841A071 |
0.357 |
|
| 1975 |
Sharpless K, Williams DR. The reactions of olefins with permanganate, ruthenium tetroxide, and osmium tetroxide; dependence of rate on degree of substitution Tetrahedron Letters. 16: 3045-3046. DOI: 10.1016/S0040-4039(00)75068-4 |
0.329 |
|
| 1975 |
Nelson JA, Kahn S, Spencer TA, Sharpless KB, Clayton RB. Some aspects of substrate specificity in biological demethylation at C4 of steroids Bioorganic Chemistry. 4: 363-376. DOI: 10.1016/0045-2068(75)90047-4 |
0.551 |
|
| 1974 |
Tanaka S, Yamamoto H, Nozaki H, Sharpless KB, Michaelson RC, Cutting JD. Stereoselective epoxidations of acyclic allylic alcohols by transition metal--hydroperoxide reagents. Synthesis of dl-C18 Cecropia juvenile hormone from farnesol. Journal of the American Chemical Society. 96: 5254-5. PMID 4854400 DOI: 10.1002/Chin.197442454 |
0.34 |
|
| 1974 |
Sharpless KB, Jensen HP. Synthesis of a novel pentacoordinate glyoxime-based ligand and preparation of its chlorocobalt(III) complex Inorganic Chemistry. 13: 2617-2620. DOI: 10.1021/Ic50141A017 |
0.315 |
|
| 1972 |
Sharpless KB, Flood TC. Direct deoxygenation of vicinal diols with tungsten(IV). A new olefin synthesis Journal of the Chemical Society, Chemical Communications. 370-371. DOI: 10.1039/C39720000370 |
0.349 |
|
| 1970 |
Rahman R, Sharpless KB, Spencer TA, Clayton RB. Removal of the 4,4-dimethyl carbons in the enzymic conversion of lanosterol to cholesterol. Initial loss of the 4-alpha-methyl group. The Journal of Biological Chemistry. 245: 2667-71. PMID 5445804 |
0.548 |
|
| 1970 |
Sharpless KB. Synthesis of erythro-18,19-dihydroxysqualene 2,3-oxide and other internally oxidized squalene derivatives Journal of the Chemical Society D: Chemical Communications. 1450-1451. DOI: 10.1039/C29700001450 |
0.331 |
|
| 1969 |
Sharpless KB, Snyder TE, Spencer TA, Maheshwari KK, Nelson JA. Biological demethylation of 4,4-dimethyl sterols, Evidence for enzymic epimerization of the 4beta-methyl group prior to its oxidative removal. Journal of the American Chemical Society. 91: 3394-6. PMID 5791927 DOI: 10.1021/Ja01040A065 |
0.549 |
|
| 1969 |
Anderson RJ, Hanzlik RP, Sharpless KB, Van Tamelen EE, Clayton RB. Enzymic transformation of an acyclic sesterterpene terminal epoxide into a lanosterol analogue Journal of the Chemical Society D: Chemical Communications. 53-54. DOI: 10.1039/C29690000053 |
0.631 |
|
| 1969 |
Van Tamelen EE, Akermark B, Sharpless KB. Mechanism of the titanium-promoted deoxygenative coupling of allyl and benzyl alcohols to hydrocarbons Journal of the American Chemical Society. 91: 1552-1554. DOI: 10.1021/Ja01034A058 |
0.389 |
|
| 1968 |
Sharpless KB, Snyder TE, Spencer TA, Maheshwari KK, Guhn G, Clayton RB. Biological demethylation of 4,4-dimethyl sterols. Initial removal of the 4.alpha.-methyl group Journal of the American Chemical Society. 90: 6874-6875. DOI: 10.1021/Ja01026A073 |
0.542 |
|
| 1968 |
Van Tamelen EE, Hanzlik RP, Sharpless KB, Clayton RB, Richter WJ, Burlingame AL. Enzymic cyclization of 15-norsqualene 2,3-oxide Journal of the American Chemical Society. 90: 3284-3286. DOI: 10.1021/Ja01014A081 |
0.483 |
|
| 1968 |
Sharpless KB, Hanzlik RP, Van Tamelen EE. One-step synthesis of 1,5-dienes involving reductive coupling of allyl alcohols Journal of the American Chemical Society. 90: 209-210. DOI: 10.1021/ja01003a037 |
0.51 |
|
| 1967 |
van Tamelen EE, Sharpless KB, Hanzlik R, Clayton RB, Burlingame AL, Wszolek PC. Enzymic cyclization of trans,trans,trans-18,19-dihydrosqualene 2,3-oxide. Journal of the American Chemical Society. 89: 7150-1. PMID 6064361 DOI: 10.1021/Ja01002A077 |
0.637 |
|
| 1967 |
Willett JD, Sharpless KB, Lord KE, van Tamelen EE, Clayton RB. Squalene-2,3oxide, an intermediate in the enzymatic conversion of squalene to lanosterol and cholesterol. The Journal of Biological Chemistry. 242: 4182-91. PMID 6061706 |
0.464 |
|
| 1964 |
Spencer TA, Schwartz MA, Sharpless KB. Synthesis of Resin Acid Intermediates. 8α,10β-Dimethyl-8β-carbomethoxy-Δ1,9,3,4-hexahydronaphthalone-2 and 8α,10β-Dimethyl-8β-carbomethoxy-Δ1,9-octalone-2 The Journal of Organic Chemistry. 29: 782-786. DOI: 10.1021/Jo01027A003 |
0.543 |
|
| Low-probability matches (unlikely to be authored by this person) |
| 2019 |
Maček Hrvat N, Kalisiak J, Šinko G, Radić Z, Sharpless KB, Taylor P, Kovarik Z. Evaluation of high-affinity phenyltetrahydroisoquinoline aldoximes, linked through anti-triazoles, as reactivators of phosphylated cholinesterases. Toxicology Letters. PMID 31863869 DOI: 10.1016/J.Toxlet.2019.12.016 |
0.3 |
|
| 1981 |
Carlsen PHJ, Katsuki T, Martin VS, Sharpless KB. A greatly improved procedure for ruthenium tetroxide catalyzed oxidations of organic compounds Journal of Organic Chemistry. 46: 3936-3938. DOI: 10.1021/Jo00332A045 |
0.299 |
|
| 1979 |
Hori T, Sharpless KB. Conversion of allylic phenylselenides to the rearranged allylic chlorides by N-chlorosuccinimide. Mechanism of selenium-catalyzed allylic chlorination of .beta.-pinene The Journal of Organic Chemistry. 44: 4208-4210. DOI: 10.1021/Jo01337A047 |
0.297 |
|
| 1979 |
Hori T, Sharpless KB. Selenium-catalyzed nonradical chlorination of olefins with N-chlorosuccinimide The Journal of Organic Chemistry. 44: 4204-4208. DOI: 10.1021/Jo01337A046 |
0.297 |
|
| 2005 |
Johnson SM, Petrassi HM, Palaninathan SK, Mohamedmohaideen NN, Purkey HE, Nichols C, Chiang KP, Walkup T, Sacchettini JC, Sharpless KB, Kelly JW. Bisaryloxime ethers as potent inhibitors of transthyretin amyloid fibril formation. Journal of Medicinal Chemistry. 48: 1576-87. PMID 15743199 DOI: 10.1021/Jm049274D |
0.297 |
|
| 1991 |
Fleming PR, Sharpless KB. Selective transformations of threo-2,3-dihydroxy esters Journal of Organic Chemistry. 56: 2869-2875. DOI: 10.1021/Jo00008A051 |
0.295 |
|
| 2003 |
Umbreit MA, Sharpless KB. Deoxygenation of Epoxides with Lower Valent Tungsten Halides: trans‐Cyclododecene Organic Syntheses. 29-29. DOI: 10.1002/0471264180.Os060.08 |
0.294 |
|
| 1992 |
Jeong KS, Sjö P, Sharpless KB. Asymmetric dihydroxylation of enynes Tetrahedron Letters. 33: 3833-3836. DOI: 10.1016/S0040-4039(00)74797-6 |
0.294 |
|
| 1994 |
Crispino GA, Makita A, Wang ZM, Sharpless KB. A comparison of ligands proposed for the asymmetric dihydroxylation Tetrahedron Letters. 35: 543-546. DOI: 10.1016/S0040-4039(00)75833-3 |
0.29 |
|
| 1981 |
Rossiter BE, Katsuki T, Sharpless KB. Asymmetric epoxidation provides shortest routes to four chiral epoxy alcohols which are key intermediates in syntheses of methymycin, erythromycin, leukotriene C-1, and disparlure Journal of the American Chemical Society. 103: 464-465. DOI: 10.1021/Ja00392A038 |
0.289 |
|
| 1989 |
Burns CJ, Martin CA, Sharpless KB. Tartrate-like ligands in the asymmetric epoxidation The Journal of Organic Chemistry. 54: 2826-2834. DOI: 10.1021/Jo00273A010 |
0.288 |
|
| 1998 |
Reddy KL, Dress KR, Sharpless KB. N-chloro-N-sodio-2-trimethylsilyl ethyl carbamate: A new nitrogen source for the catalytic asymmetric aminohydroxylation Tetrahedron Letters. 39: 3667-3670. DOI: 10.1016/S0040-4039(98)00644-3 |
0.288 |
|
| 1997 |
Bruncko M, Schlingloff G, Sharpless KB. N-Bromoacetamide—A New Nitrogen Source for the Catalytic Asymmetric Aminohydroxylation of Olefins Angewandte Chemie International Edition in English. 36: 1483-1486. DOI: 10.1002/Anie.199714831 |
0.285 |
|
| 1993 |
Wang Z, Sharpless KB. Asymmetric Dihydroxylation of α-Substituted Styrene Derivatives Synlett. 1993: 603-604. DOI: 10.1055/S-1993-22547 |
0.283 |
|
| 1990 |
Moon Kim B, Sharpless KB. Heterogeneous catalytic asymmetric dihydroxylation: Use of a polymer-bound alkaloid Tetrahedron Letters. 31: 3003-3006. DOI: 10.1016/S0040-4039(00)89009-7 |
0.28 |
|
| 1985 |
Chong J, Sharpless K. Regioselective openings of 2,3-epoxy acids with organocuprates Tetrahedron Letters. 26: 4683-4686. DOI: 10.1016/S0040-4039(00)94923-2 |
0.279 |
|
| 1996 |
Becker H, Sharpless KB. A New Ligand Class for the Asymmetric Dihydroxylation of Olefins Angewandte Chemie International Edition in English. 35: 448-451. DOI: 10.1002/Anie.199604481 |
0.279 |
|
| 1987 |
Kirshenbaum KS, Sharpless KB. Regioselective Nucleophilic Opening oferythro-andthreo-2,3-Epoxy Alcohols Chemistry Letters. 16: 11-14. DOI: 10.1246/Cl.1987.11 |
0.279 |
|
| 1996 |
Chang HT, Sharpless KB. A practical route to enantiopure 1,2-aminoalcohols Tetrahedron Letters. 37: 3219-3222. DOI: 10.1016/0040-4039(96)00534-5 |
0.278 |
|
| 1993 |
Crispino GA, Sharpless KB. Enantioselective Synthesis of Juvenile Hormone III in Three Steps from Methyl Farnesoate Synthesis. 1993: 777-779. DOI: 10.1055/S-1993-25939 |
0.274 |
|
| 1993 |
Wang ZM, Sharpless KB. Asymmetric dihydroxylation of tertiary allylic alcohols Tetrahedron Letters. 34: 8225-8228. DOI: 10.1016/S0040-4039(00)61396-5 |
0.274 |
|
| 1981 |
Martin VS, Woodard SS, Katsuki T, Yamada Y, Ikeda M, Sharpless KB. Kinetic resolution of racemic allylic alcohols by enantioselective epoxidation. A route to substances of absolute enantiomeric purity? Journal of the American Chemical Society. 103: 6237-6240. DOI: 10.1021/Ja00410A053 |
0.274 |
|
| 1995 |
Hugger U, Sharpless KB. Asymmetric dihydroxylation affords enantiomerically pure C12 building blocks from traps, traps, cis-1,5,9-cyclododecatriene Tetrahedron Letters. 36: 6603-6606. DOI: 10.1016/00404-0399(50)1365-O |
0.273 |
|
| 1986 |
SHARPLESS KB. ChemInform Abstract: The Discovery of Titanium-Catalyzed Asymmetric Epoxidation Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198611389 |
0.271 |
|
| 2003 |
Hill JG, Sharpless KB, Exon CM, Regenye R. Enantioselective Epoxidation of Allylic Alcohols: (2S,3S)‐3‐Propyloxiranemethanol Organic Syntheses. 66-66. DOI: 10.1002/0471264180.Os063.08 |
0.271 |
|
| 1976 |
Sharpless KB, Singer SP. 1,2-Diamination of 1,3-dienes by imido selenium compounds The Journal of Organic Chemistry. 41: 2504-2506. DOI: 10.1021/Jo00876A040 |
0.271 |
|
| 1990 |
Pearlstein RM, Blackburn BK, Davis WM, Sharpless KB. Strukturelle Charakterisierung pseudoenantiomerercis-Dioxoosmium(VI)-Komplexe mit chiralen Diolen und Cinchona-Alkaloid-Liganden Angewandte Chemie. 102: 710-712. DOI: 10.1002/Ange.19901020630 |
0.27 |
|
| 1983 |
Hill JG, Rossiter BE, Sharpless KB. Anhydrous tert-butyl hydroperoxide in toluene: the preferred reagent for applications requiring dry TBHP The Journal of Organic Chemistry. 48: 3607-3608. DOI: 10.1021/Jo00168A063 |
0.27 |
|
| 1978 |
Patrick DW, Truesdale LK, Biller SA, Sharpless KB. Stereospecific vicinal oxyamination of olefins by alkylimidoosmium compounds The Journal of Organic Chemistry. 43: 2628-2638. DOI: 10.1021/Jo00407A016 |
0.267 |
|
| 1978 |
Frejd T, Sharpless K. A new rearrangement of N-arylhydroxamic acids catalyzed by seleninic acids and phenylselenenyl chloride Tetrahedron Letters. 19: 2239-2242. DOI: 10.1016/S0040-4039(01)91501-1 |
0.266 |
|
| 1998 |
Jeong JU, Tao B, Sagasser I, Henniges H, Sharpless KB. Bromine-catalyzed aziridination of olefins. A rare example of atom-transfer redox catalysis by a main group element Journal of the American Chemical Society. 120: 6844-6845. DOI: 10.1021/Ja981419G |
0.262 |
|
| 1972 |
SHARPLESS KB, UMBREIT MA, NIEH MT, FLOOD TC. ChemInform Abstract: NIEDERWERTIGE WOLFRAMHALOGENIDE, NEUE KLASSE VON REAGENTIEN FUER DIE DESOX. ORGANISCHER MOLEKUELE Chemischer Informationsdienst. 3: no-no. DOI: 10.1002/Chin.197247187 |
0.262 |
|
| 2019 |
Taylor P, Yan-Jye S, Momper J, Hou W, Camacho-Hernandez GA, Radic Z, Rosenberg Y, Kovarik Z, Sit R, Sharpless KB. Assessment of ionizable, zwitterionic oximes as reactivating antidotal agents for organophosphate exposure. Chemico-Biological Interactions. PMID 31100277 DOI: 10.1016/J.Cbi.2019.05.015 |
0.261 |
|
| 1973 |
Sharpless KB, Teranishi AY. Chromyl chloride in acetone. .alpha.-Chloro ketones and ketones directly from olefins The Journal of Organic Chemistry. 38: 185-186. DOI: 10.1021/Jo00941A054 |
0.261 |
|
| 2003 |
McKee BH, Gilheany DG, Sharpless KB. (R,R)‐1,2‐Diphenyl‐1,2‐Ethanediol (Stilbene Diol) Organic Syntheses. 47-47. DOI: 10.1002/0471264180.Os070.06 |
0.26 |
|
| 2010 |
Pringle W, Sharpless KB. ChemInform Abstract: The Osmium-Catalyzed Aminohydroxylation of Baylis-Hillman Olefins. Cheminform. 30: no-no. DOI: 10.1002/chin.199941058 |
0.259 |
|
| 1978 |
Hori T, Singer SP, Sharpless KB. Allylic deuteration and tritiation of olefins with N-sulfinylsulfonamides The Journal of Organic Chemistry. 43: 1456-1459. DOI: 10.1021/Jo00401A035 |
0.259 |
|
| 1993 |
Bennani YL, Sharpless KB. Asymmetric dihydroxylation (AD) of N,N-dialkyl and N-methoxy-N-methyl α,β- and β,γ-unsaturated amides Tetrahedron Letters. 34: 2079-2082. DOI: 10.1016/S0040-4039(00)60350-7 |
0.258 |
|
| 1984 |
Williams ID, Pedersen SF, Sharpless KB, Lippard SJ. Crystal structures of two titanium tartrate asymmetric epoxidation catalysts Journal of the American Chemical Society. 106: 6430-6431. DOI: 10.1002/Chin.198506283 |
0.256 |
|
| 1975 |
Sharpless KB, Akashi K. Oxidation of alcohols to aldehydes by reagents derived from chromyl chloride Journal of the American Chemical Society. 97: 5927-5928. DOI: 10.1021/Ja00853A055 |
0.256 |
|
| 1987 |
Ko SY, Masamune H, Sharpless KB. p-Nitrobenzoate esters of epoxy alcohols: convenient synthons for water-soluble epoxy alcohols The Journal of Organic Chemistry. 52: 667-671. DOI: 10.1021/Jo00380A032 |
0.256 |
|
| 1997 |
Rubin AE, Sharpless KB. A Highly Efficient Aminohydroxylation Process Angewandte Chemie International Edition in English. 36: 2637-2640. DOI: 10.1002/Anie.199726371 |
0.253 |
|
| 1972 |
Sharpless KB, Umbreit MA, Nieh MT, Flood TC. Lower valent tungsten halides. New class of reagents for deoxygenation of organic molecules Journal of the American Chemical Society. 94: 6538-6540. DOI: 10.1021/Ja00773A045 |
0.252 |
|
| 1980 |
Herranz E, Sharpless KB. Osmium-catalyzed vicinal oxyamination of olefins by N-chloro-N-metallocarbamates The Journal of Organic Chemistry. 45: 2710-2713. DOI: 10.1021/Jo01301A033 |
0.252 |
|
| 1978 |
Herranz E, Biller SA, Sharpless KB. Osmium-catalyzed vicinal oxyamination of olefins by N-chloro-N-argentocarbamates Journal of the American Chemical Society. 100: 3596-3598. DOI: 10.1021/Ja00479A051 |
0.252 |
|
| 1978 |
Current S, Sharpless K. Carbonyl participation in the addition of p-chlorophenylselenenyl bromide to ()-4-hexenal: A new route to 2,6-dideoxylgycosides Tetrahedron Letters. 19: 5075-5078. DOI: 10.1016/S0040-4039(01)85816-0 |
0.251 |
|
| 1983 |
Miyano S, Lu LDL, Viti SM, Sharpless KB. Kinetic resolution of racemic .beta.-hydroxy amines by enantioselective N-oxide formation The Journal of Organic Chemistry. 48: 3608-3611. DOI: 10.1021/Jo00168A064 |
0.251 |
|
| 1994 |
Wang Z, Sharpless KB. A Solid-to-Solid Asymmetric Dihydroxylation Procedure for Kilogram-Scale Preparation of Enantiopure Hydrobenzoin The Journal of Organic Chemistry. 59: 8302-8303. DOI: 10.1021/Jo00105A065 |
0.251 |
|
| 1986 |
Hawkins JM, Dewan JC, Sharpless KB. Dioxomolybdenum(VI)-substituted 2,6-pyridinedimethanol complexes: new five-coordinate species Inorganic Chemistry. 25: 1501-1503. DOI: 10.1021/Ic00229A041 |
0.249 |
|
| 1999 |
Chuang TH, Sharpless KB. Applications of aziridinium ions. Selective syntheses of beta-aryl-alpha,beta-diamino esters. Organic Letters. 1: 1435-7. PMID 10825990 DOI: 10.1021/Ol990256D |
0.249 |
|
| 1986 |
Klunder JM, Ko SY, Sharpless KB. Asymmetric epoxidation of allyl alcohol: efficient routes to homochiral .beta.-adrenergic blocking agents The Journal of Organic Chemistry. 51: 3710-3712. DOI: 10.1021/Jo00369A032 |
0.248 |
|
| 1985 |
Behrens CH, Sharpless KB. Selective transformations of 2,3-epoxy alcohols and related derivatives. Strategies for nucleophilic attack at carbon-3 or carbon-2 The Journal of Organic Chemistry. 50: 5696-5704. DOI: 10.1021/Jo00350A051 |
0.248 |
|
| 2007 |
Hirose T, Sunazuka T, Noguchi Y, Yamaguchi Y, Hanaki H, Sharpless KB, Omura S. Rapid “SAR” via Click Chemistry: An Alkyne-Bearing Spiramycin Is Fused with Diverse Azides to Yield New Triazole-Antibacterial Candidates. Cheminform. 38. DOI: 10.1002/chin.200722209 |
0.245 |
|
| 1978 |
Herranz E, Sharpless KB. Improvements in the osmium-catalyzed oxyamination of olefins by chloramine-T The Journal of Organic Chemistry. 43: 2544-2548. DOI: 10.1021/Jo00406A057 |
0.245 |
|
| 1988 |
Gao Y, Sharpless KB. Vicinal diol cyclic sulfates. Like epoxides only more reactive Journal of the American Chemical Society. 110: 7538-7539. DOI: 10.1021/Ja00230A045 |
0.244 |
|
| 1992 |
Xu D, Crispino GA, Sharpless KB. Selective asymmetric dihydroxylation (AD) of dienes Journal of the American Chemical Society. 114: 7570-7571. DOI: 10.1021/Ja00045A043 |
0.244 |
|
| 1975 |
Sharpless KB, Chong AO, Scott JA. Rapid separation of organic mixtures by formation of metal complexes The Journal of Organic Chemistry. 40: 1252-1257. DOI: 10.1021/Jo00897A015 |
0.243 |
|
| 2010 |
Demko ZP, Sharpless KB. ChemInform Abstract: A Click Chemistry Approach to Tetrazoles by Huisgen 1,3-Dipolar Cycloaddition: Synthesis of 5-Acyltetrazoles from Azides and Acyl Cyanides. Cheminform. 33: no-no. DOI: 10.1002/chin.200242151 |
0.243 |
|
| 1993 |
Crispino GA, Ho PT, Sharpless KB. Selective perhydroxylation of squalene: taming the arithmetic demon. Science (New York, N.Y.). 259: 64-6. PMID 8418495 DOI: 10.1126/science.8418495 |
0.241 |
|
| 1978 |
Singer SP, Sharpless KB. Synthesis of dl-gabaculine utilizing direct allylic amination as the key step The Journal of Organic Chemistry. 43: 1448-1455. DOI: 10.1021/jo00401a034 |
0.24 |
|
| 1979 |
Chabaud B, Sharpless KB. Oxidation of acetylenes with tert-butyl hydroperoxide catalyzed by selenium dioxide. .alpha.,.alpha.'-Dioxygenation of internal alkynes The Journal of Organic Chemistry. 44: 4202-4204. DOI: 10.1021/Jo01337A045 |
0.239 |
|
| 1982 |
Reed LA, Ito Y, Masamune S, Sharpless KB. Synthesis of saccharides and related polyhydroxylated natural products. 4. .alpha.-D- and .beta.-D-C-Glycopyranosides (2,6-dialkyl-substituted tetrahydropyrans) Journal of the American Chemical Society. 104: 6468-6470. DOI: 10.1021/Ja00387A062 |
0.238 |
|
| 1980 |
Hentges SG, Sharpless KB. Improved procedure for the oxyamination of olefins with trioxo(tert-butylimido)osmium(VIII) The Journal of Organic Chemistry. 45: 2257-2259. DOI: 10.1021/Jo01299A045 |
0.237 |
|
| 1985 |
Sharpless KB, Hawkins JM. New pathways for organic synthesis: Practical applications of transition metals. By H. M. Colquhoun, J. Holton, D. J. Thompson, and M. V. Twigg. Plenum Press, 233 Spring Street, New York, NY 10013. 1984. 454 pp. 16 × 2. cm. $59.50 Journal of Pharmaceutical Sciences. 74: 362-363. DOI: 10.1002/Jps.2600740336 |
0.237 |
|
| 1985 |
Kirshenbaum KS, Sharpless KB. Improved procedure for the tungstate-catalyzed epoxidation of .alpha.,.beta.-unsaturated acids The Journal of Organic Chemistry. 50: 1979-1982. DOI: 10.1021/Jo00211A040 |
0.236 |
|
| 1986 |
Hanson RM, Sharpless KB. Procedure for the catalytic asymmetric epoxidation of allylic alcohols in the presence of molecular sieves The Journal of Organic Chemistry. 51: 1922-1925. DOI: 10.1021/Jo00360A058 |
0.236 |
|
| 1985 |
Behrens CH, Ko SY, Sharpless KB, Walker FJ. Selective transformation of 2,3-epoxy alcohols and related derivatives. Strategies for nucleophilic attack at carbon-1 The Journal of Organic Chemistry. 50: 5687-5696. DOI: 10.1021/Jo00350A050 |
0.236 |
|
| 1977 |
Chong AO, Sharpless KB. Mechanism of the molybdenum and vanadium catalyzed epoxidation of olefins by alkyl hydroperoxides The Journal of Organic Chemistry. 42: 1587-1590. DOI: 10.1021/jo00429a024 |
0.236 |
|
| 2009 |
Vanacore R, Ham AJ, Voehler M, Sanders CR, Conrads TP, Veenstra TD, Sharpless KB, Dawson PE, Hudson BG. A sulfilimine bond identified in collagen IV. Science (New York, N.Y.). 325: 1230-4. PMID 19729652 DOI: 10.1126/Science.1176811 |
0.234 |
|
| 1984 |
Rossiter BE, Sharpless KB. Asymmetric epoxidation of homoallylic alcohols. Synthesis of (-)-.gamma.-amino-.beta.-(R)-hydroxybutyric acid (GABOB) The Journal of Organic Chemistry. 49: 3707-3711. DOI: 10.1021/Jo00194A007 |
0.233 |
|
| 1972 |
Townsend JM, Sharpless K. Mechanism of decomposition of sulfonium betaines to epoxides Tetrahedron Letters. 13: 3313-3316. DOI: 10.1016/S0040-4039(01)94031-6 |
0.231 |
|
| 2009 |
Hirose T, Sunazuka T, Sugawara A, Endo A, Iguchi K, Yamamoto T, Ui H, Shiomi K, Watanabe T, Sharpless KB, Omura S. Chitinase inhibitors: extraction of the active framework from natural argifin and use of in situ click chemistry. The Journal of Antibiotics. 62: 277-82. PMID 19329983 DOI: 10.1038/ja.2009.28 |
0.23 |
|
| 1976 |
Sharpless KB, Gordon KM. Selenium dioxide oxidation of ketones and aldehydes. Evidence for the intermediacy of .beta.-ketoseleninic Journal of the American Chemical Society. 98: 300-301. DOI: 10.1021/Ja00417A083 |
0.229 |
|
| 2003 |
Herranz E, Sharpless KB. Osmium‐Catalyzed Vicinal Oxyamination of Olefins by Chloramine‐T: cis‐2‐(p‐Toluenesulfonamido)Cyclohexanol and 2‐Methyl‐3‐(p‐Toluenesulfonamido)‐2‐Pentanol Organic Syntheses. 85-85. DOI: 10.1002/0471264180.Os061.20 |
0.226 |
|
| 1982 |
Gonnella NC, Nakanishi K, Martin VS, Sharpless KB. General method for determining absolute configuration of acyclic allylic alcohols Journal of the American Chemical Society. 104: 3775-3776. DOI: 10.1021/Ja00377A063 |
0.224 |
|
| 2001 |
Petrassi HM, Sharpless KB, Kelly JW. The copper-mediated cross-coupling of phenylboronic acids and N-hydroxyphthalimide at room temperature: synthesis of aryloxyamines. Organic Letters. 3: 139-42. PMID 11429858 DOI: 10.1021/Ol0003533 |
0.222 |
|
| 1986 |
Ko SY, Sharpless KB. In situ opening of epoxy alcohols: a convenient alternative to the isolation of unstable epoxy alcohols The Journal of Organic Chemistry. 51: 5413-5415. DOI: 10.1021/Jo00376A068 |
0.219 |
|
| 1997 |
Bruncko M, Schlingloff G, Sharpless KB. N-Bromacetamid - eine neue Stickstoffquelle für die katalytische asymmetrische Aminohydroxylierung Angewandte Chemie. 109: 1580-1583. DOI: 10.1002/Ange.19971091340 |
0.208 |
|
| 1993 |
Göbel T, Sharpless KB. Temperature Effects in Asymmetric Dihydroxylation: Evidence for a Stepwise Mechanism Angewandte Chemie International Edition in English. 32: 1329-1331. DOI: 10.1002/Anie.199313291 |
0.208 |
|
| 1974 |
Sharpless KB, Lauer RF. Electrophilic organoselenium reagents. New route to allylic acetates and ethers The Journal of Organic Chemistry. 39: 429-430. DOI: 10.1021/jo00917a038 |
0.206 |
|
| 1975 |
Jensen HP, Sharpless KB. Selenium dioxide oxidation of d-limonene. Reinvestigation The Journal of Organic Chemistry. 40: 264-265. DOI: 10.1021/Jo00890A030 |
0.206 |
|
| 2013 |
Hirose T, Maita N, Gouda H, Koseki J, Yamamoto T, Sugawara A, Nakano H, Hirono S, Shiomi K, Watanabe T, Taniguchi H, Sharpless KB, Omura S, Sunazuka T. Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor. Proceedings of the National Academy of Sciences of the United States of America. 110: 15892-7. PMID 24043811 DOI: 10.1073/Pnas.1315049110 |
0.204 |
|
| 2010 |
TAO B, SCHLINGLOFF G, SHARPLESS KB. ChemInform Abstract: Reversal of Regioselection in the Asymmetric Aminohydroxylation of Cinnamates. Cheminform. 29: no-no. DOI: 10.1002/chin.199828042 |
0.203 |
|
| 1989 |
LOHRAY BB, KALANTAR TH, KIM BM, PARK CY, SHIBATA T, WAI JSM, SHARPLESS KB. ChemInform Abstract: Documenting the Scope of the Catalytic Asymmetric Dihydroxylation. Cheminform. 20. DOI: 10.1002/chin.198948090 |
0.201 |
|
| 1971 |
SHARPLESS KB, FLOOD TC. ChemInform Abstract: OXO-UEBERGANGSMETALL-OXIDANTIEN ALS MODELLE FUER DIE WIRKUNG VON OXYGENASEN MIT GEMISCHTEN FUNKTIONEN, ′NIH-VERSCHIEBUNG′ BEI CHROMYLREAGENTIEN Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197131117 |
0.201 |
|
| 1983 |
Sharpless KB, Woodard SS. On the mechanism of titanium-tartrate catalyzed asymmetric epoxidation Pure and Applied Chemistry. 55: 1823-1836. DOI: 10.1351/pac198355111823 |
0.2 |
|
| 2008 |
Sharpless KB. The secret life of enzymes Journal of Biotechnology. 136: S3. DOI: 10.1016/J.Jbiotec.2008.07.1845 |
0.2 |
|
| 2010 |
Goossen LJ, Liu H, Dress KR, Sharpless KB. ChemInform Abstract: Catalytic Asymmetric Aminohydroxylation with Amino-Substituted Heterocycles as Nitrogen Sources. Cheminform. 30: no-no. DOI: 10.1002/chin.199933040 |
0.197 |
|
| 1976 |
Sharpless KB, Hori T. Allylic amination of olefins and acetylenes by imido sulfur compounds The Journal of Organic Chemistry. 41: 176-177. DOI: 10.1021/jo00863a051 |
0.197 |
|
| 2010 |
Johnson RA, Sharpless KB. ChemInform Abstract: Catalytic Asymmetric Dihydroxylation - Discovery and Development Cheminform. 32: no-no. DOI: 10.1002/chin.200129254 |
0.195 |
|
| 2020 |
Samskey N, Ho K, Momper J, Radic Z, Sit R, Sharpless KB, Taylor P. Pharmacokinetic Analysis of Ionizable Zwitterionic Oximes: Antidotes to Organophosphate Exposure. The Faseb Journal. 34: 1-1. DOI: 10.1096/Fasebj.2020.34.S1.06319 |
0.194 |
|
| 2002 |
Sharpless KB. Auf der Suche nach neuer Reaktivität (Nobel-Vortrag) Copyright© The Nobel Foundation 2002. – Wir danken der Nobel-Stiftung, Stockholm, für die Genehmigung zum Druck einer deutschen Fassung des Vortrags. Abdruck in veränderter Fassung mit freundlicher Genehmigung aus „Coelacanths and Catalysis“: K. B. Sharpless, Tetrahedron 1994, 50, 4235. Angewandte Chemie. 114: 2126. DOI: 10.1002/1521-3757(20020617)114:12<2126::Aid-Ange2126>3.0.Co;2-6 |
0.193 |
|
| 2010 |
Demko ZP, Sharpless KB. ChemInform Abstract: An Intramolecular [2 + 3] Cycloaddition Route to Fused 5-Heterosubstituted Tetrazoles. Cheminform. 33: no-no. DOI: 10.1002/chin.200222134 |
0.192 |
|
| 1999 |
Gooßen LJ, Liu H, Dress KR, Sharpless KB. Katalytische asymmetrische Aminohydroxylierung mit Amino-substituierten Heterocyclen als Stickstoffquelle Angewandte Chemie. 111: 1149-1152. DOI: 10.1002/(Sici)1521-3757(19990419)111:8<1149::Aid-Ange1149>3.0.Co;2-D |
0.191 |
|
| 1976 |
Sharpless KB, Hori T, Truesdale LK, Dietrich CO. Allylic amination of olefins and acetylenes by imido selenium compounds Journal of the American Chemical Society. 98: 269-271. DOI: 10.1021/ja00417a062 |
0.19 |
|
| 1987 |
PEDERSEN SF, DEWAN JC, ECKMAN RR, SHARPLESS KB. ChemInform Abstract: Unexpected Diversity in the Coordination Chemistry of Tartrate Esters with Titanium(IV). Cheminform. 18. DOI: 10.1002/chin.198727244 |
0.189 |
|
| 1993 |
Kalantar TH, Sharpless KB. Transformations of hydroxy cyclic sulfates: stereospecific conversion into 2,3,5-trisubstituted tetrahydrofurans. Acta Chemica Scandinavica (Copenhagen, Denmark : 1989). 47: 307-13. PMID 8435231 DOI: 10.3891/acta.chem.scand.47-0307 |
0.188 |
|
| 1982 |
LEE AWM, MARTIN VS, MASAMUNE S, SHARPLESS KB, WALKER FJ. ChemInform Abstract: SYNTHESIS OF SACCHARIDES AND RELATED POLYHYDROXYLATED NATURAL PRODUCTS. 3. EFFICIENT CONVERSION OF 2,3-ERYTHRO-ALDOSES TO 2,3-THREO-ALDOSES Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198239354 |
0.187 |
|
| 1996 |
Chang H, Chen C, Kondo T, Siuzdak G, Sharpless KB. Asymmetrische Dihydroxylierung zum schnellen Aufbau von chiralen Dendrimeren aus 1,2-Diolen Angewandte Chemie. 108: 202-206. DOI: 10.1002/Ange.19961080217 |
0.186 |
|
| 2003 |
Beller M, Sharpless KB. Diols via Catalytic Dihydroxylation Cheminform. 34. DOI: 10.1002/chin.200327277 |
0.184 |
|
| 1996 |
Becker H, Sharpless KB. Eine neue Ligandenklasse für die asymmetrische Dihydroxylierung von Olefinen Angewandte Chemie. 108: 447-449. DOI: 10.1002/Ange.19961080408 |
0.181 |
|
| 1997 |
Rubin AE, Sharpless KB. Ein effizientes Verfahren zur asymmetrischen Aminohydroxylierung Angewandte Chemie. 109: 2751-2754. DOI: 10.1002/Ange.19971092324 |
0.18 |
|
| 1996 |
Bruncko M, Khuong TV, Sharpless KB. Allylische Aminierung und 1,2-Diaminierung mit einem modifizierten Diimidoselen-Reagens Angewandte Chemie. 108: 453-455. DOI: 10.1002/Ange.19961080410 |
0.179 |
|
| 1996 |
Rudolph J, Sennhenn PC, Vlaar CP, Sharpless KB. Osmiumkatalysierte asymmetrische Aminohydroxylierung: kleinere Substituenten am Stickstoffatom erleichtern die Reaktion Angewandte Chemie. 108: 2991-2995. DOI: 10.1002/Ange.19961082324 |
0.178 |
|
| 1982 |
Lee A, Martin V, Masamune S, Sharpless K, Walker F. Additions and Corrections - Synthesis of Saccharides and Related Polyhydroxylated Natural Products. 3. Efficient Conversion of 2,3-erythro-Aldoses to 2,3-threo-Aldoses Journal of the American Chemical Society. 104: 6167-6167. DOI: 10.1021/Ja00386A607 |
0.178 |
|
| 1987 |
Gao Y, Klunder JM, Hanson RM, Masamune H, Ko SY, Sharpless KB. Catalytic asymmetric epoxidation and kinetic resolution: modified procedures including in situ derivatization Journal of the American Chemical Society. 109: 5765-5780. DOI: 10.1021/ja00253a032 |
0.172 |
|
| 1977 |
Michaelson RC, Palermo RE, Sharpless KB. Chiral hydroxamic acids as ligands in the vanadium catalyzed asymmetric epoxidation of allylic alcohols by tert-butyl hydroperoxide Journal of the American Chemical Society. 99: 1990-1992. DOI: 10.1021/ja00448a059 |
0.171 |
|
| 2010 |
JEONG K, SJOE P, SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation of Enynes. Cheminform. 23: no-no. DOI: 10.1002/chin.199252107 |
0.17 |
|
| 1977 |
Umbreit MA, Sharpless KB. Allylic oxidation of olefins by catalytic and stoichiometric selenium dioxide with tert-butyl hydroperoxide Journal of the American Chemical Society. 99: 5526-5528. DOI: 10.1021/ja00458a072 |
0.167 |
|
| 2007 |
Sharpless KB. A 60th Birthday! Advanced Synthesis & Catalysis. 349: 2533-2534. DOI: 10.1002/Adsc.200700454 |
0.166 |
|
| 2010 |
Gontcharov AV, Liu H, Sharpless KB. ChemInform Abstract: tert-Butylsulfonamide. A New Nitrogen Source for Catalytic Aminohydroxylation and Aziridination of Olefins. Cheminform. 30: no-no. DOI: 10.1002/chin.199949038 |
0.165 |
|
| 1984 |
MIYANO S, LU LD, VITI SM, SHARPLESS KB. ChemInform Abstract: KINETIC RESOLUTION OF RACEMIC β-HYDROXY AMINES BY ENANTIOSELECTIVE N-OXIDE FORMATION Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198412105 |
0.165 |
|
| 2020 |
Sharpless KB. Eric Jacobsen@60, a Personal Statement Advanced Synthesis & Catalysis. 362: 281-284. DOI: 10.1002/Adsc.201901658 |
0.163 |
|
| 2008 |
Sugawara A, Sunazuka T, Hirose T, Nagai K, Yamaguchi Y, Hanaki H, Sharpless KB, Omura S. ChemInform Abstract: Design and Synthesis via Click Chemistry of 8,9-Anhydroerythromycin A 6,9-Hemiketal Analogues with anti-MRSA and -VRE Activity. Cheminform. 39. DOI: 10.1002/chin.200810222 |
0.162 |
|
| 2015 |
Sharpless KB. Building blocks for SuFEx, the next click reaction Aldrichimica Acta. 48: 41. |
0.162 |
|
| 1982 |
MA P, MARTIN VS, MASAMUNE S, SHARPLESS KB, VITI SM. ChemInform Abstract: SYNTHESIS OF SACCHARIDES AND RELATED POLYHYDROXYLATED NATURAL PRODUCTS. 2. SIMPLE DEOXYALDITOLS Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198237319 |
0.162 |
|
| 2010 |
XU D, CRISPINO GA, SHARPLESS KB. ChemInform Abstract: Selective Asymmetric Dihydroxylation of Dienes. Cheminform. 24: no-no. DOI: 10.1002/chin.199301132 |
0.152 |
|
| 1982 |
Katsuki T, Lee AWM, Ma P, Martin VS, Masamune S, Sharpless KB, Tuddenham D, Walker FJ. Synthesis of saccharides and related polyhydroxylated natural products. 1. Simple alditols The Journal of Organic Chemistry. 47: 1373-1378. DOI: 10.1021/jo00346a051 |
0.147 |
|
| 1984 |
Hawkins JM, Sharpless KB. Threo-N,N'-Bis(.alpha.-methylbenzyl)sulfamide: a readily available chiral ligand for asymmetric lithium aluminum hydride reductions The Journal of Organic Chemistry. 49: 3861-3862. DOI: 10.1021/jo00194a048 |
0.147 |
|
| 2010 |
DRESS KR, GOOSSEN LJ, LIU H, JERINA DM, SHARPLESS KB. ChemInform Abstract: Catalytic Aminohydroxylation Using Adenine-Derivatives as the Nitrogen Source. Cheminform. 29: no-no. DOI: 10.1002/chin.199852176 |
0.147 |
|
| 1989 |
Wink D, Anderson A, Byon C, Collet T, Hickman A, Miller A, Salifoglou T, Sharpless K, Orme-Johnson W. Homocitrate complexes: Role in MoFe cofactor synthesis and function in nitrogenase Journal of Inorganic Biochemistry. 36: 171. DOI: 10.1016/0162-0134(89)84080-2 |
0.146 |
|
| 2010 |
WANG Z, SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation of α-Substituted Styrene Derivatives ( I), (III). Cheminform. 25: no-no. DOI: 10.1002/chin.199411087 |
0.146 |
|
| 2010 |
VANHESSCHE KPM, SHARPLESS KB. ChemInform Abstract: Ligand-Dependent Reversal of Facial Selectivity in the Asymmetric Dihydroxylation. Cheminform. 28: no-no. DOI: 10.1002/chin.199712063 |
0.146 |
|
| 1973 |
Sharpless KB, Young MW, Lauer RF. Reactions of selenoxides: Thermal syn-elimination and H218O exchange Tetrahedron Letters. 14: 1979-1982. DOI: 10.1016/S0040-4039(01)96098-8 |
0.146 |
|
| 1985 |
KLUNDER JM, CARON M, UCHIYAMA M, SHARPLESS KB. ChemInform Abstract: CHLOROHYDROXYLATION OF OLEFINS WITH PEROXIDES AND TITANIUM TETRACHLORIDE Chemischer Informationsdienst. 16. DOI: 10.1002/chin.198534155 |
0.142 |
|
| 2010 |
WANG L, SHARPLESS KB. ChemInform Abstract: Catalytic Asymmetric Dihydroxylation of cis-Disubstituted Olefins. Cheminform. 24: no-no. DOI: 10.1002/chin.199301131 |
0.141 |
|
| 2010 |
CHANG H, SHARPLESS KB. ChemInform Abstract: Molar Scale Synthesis of Enantiopure Stilbene Oxide. Cheminform. 28: no-no. DOI: 10.1002/chin.199704115 |
0.139 |
|
| 2010 |
SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation (AD) and Drug Synthesis. Cheminform. 24: no-no. DOI: 10.1002/chin.199326089 |
0.138 |
|
| 1996 |
Vanhessche KP, Sharpless KB. Ligand-Dependent Reversal of Facial Selectivity in the Asymmetric Dihydroxylation. The Journal of Organic Chemistry. 61: 7978-7979. PMID 11667767 DOI: 10.1021/jo961189t |
0.131 |
|
| 1989 |
SVENDSEN JS, SHARPLESS KB. ChemInform Abstract: Type I Intramolecular Cycloadditions of Vinylketenes Cheminform. 20. DOI: 10.1002/chin.198943295 |
0.13 |
|
| 1985 |
Miyano S, Lu LDL, Viti SM, Sharpless KB. Kinetic resolution of racemic .beta.-hydroxy amines by enantioselective N-oxide formation The Journal of Organic Chemistry. 50: 4350-4360. DOI: 10.1021/jo00222a030 |
0.13 |
|
| 2000 |
Chuang TH, Sharpless KB. Applications of aziridinium ions. Selective syntheses of alpha, beta-diamino esters, alpha-sulfanyl-beta-amino esters, beta-lactams, and 1,5-benzodiazepin-2-one. Organic Letters. 2: 3555-7. PMID 11073643 |
0.13 |
|
| 1972 |
Sharpless KB, Townsend JM, Williams DR. Mechanism of epoxidation of olefins by covalent peroxides of molybdenum(VI) Journal of the American Chemical Society. 94: 295-296. DOI: 10.1021/ja00756a062 |
0.129 |
|
| 1973 |
Arigoni D, Vasella A, Sharpless KB, Jensen HP. Selenium dioxide oxidations of olefins. Trapping of the allylic seleninic acid intermediate as a seleninolactone Journal of the American Chemical Society. 95: 7917-7919. DOI: 10.1021/ja00804a087 |
0.129 |
|
| 1988 |
Gao Y, Sharpless KB. Asymmetric synthesis of both enantiomers of tomoxetine and fluoxetine. Selective reduction of 2,3-epoxycinnamyl alcohol with Red-Al The Journal of Organic Chemistry. 53: 4081-4084. DOI: 10.1021/jo00252a036 |
0.125 |
|
| 1985 |
Chong JM, Sharpless KB. Nucleophilic opening of 2,3-epoxy acids and amides mediated by titanium isopropoxide. Highly enhanced C-3 selectivity The Journal of Organic Chemistry. 50: 1560-1563. DOI: 10.1021/jo00209a048 |
0.125 |
|
| 1996 |
Chang HT, Sharpless KB. Molar Scale Synthesis of Enantiopure Stilbene Oxide. The Journal of Organic Chemistry. 61: 6456-6457. PMID 11667495 DOI: 10.1021/jo960718q |
0.123 |
|
| 2010 |
JOHNSON RA, SHARPLESS KB. ChemInform Abstract: Catalytic Asymmetric Epoxidation of Allylic Alcohols Cheminform. 25: no-no. DOI: 10.1002/chin.199432281 |
0.122 |
|
| 2012 |
Sharpless KB. Foreword Efficient Preparations of Fluorine Compounds. xi. DOI: 10.1002/9781118409466 |
0.12 |
|
| 1973 |
Sharpless KB, Lauer RF, Teranishi AY. Electrophilic and nucleophilic organoselenium reagents. New routes to .alpha.,.beta.-unsaturated carbonyl compounds Journal of the American Chemical Society. 95: 6137-6139. DOI: 10.1021/ja00799a062 |
0.12 |
|
| 1979 |
BAECKVALL J, OSHIMA K, PALERMO RE, SHARPLESS KB. ChemInform Abstract: SOME REACTIONS OF N-(2-HYDROXYALKYL)-P-TOLUENESULFONAMIDES AND N-ALLYL-P-TOLUENESULFONAMIDES Chemischer Informationsdienst. 10. DOI: 10.1002/chin.197943206 |
0.119 |
|
| 1985 |
Klunder JM, Caron M, Uchiyama M, Sharpless KB. Chlorohydroxylation of olefins with peroxides and titanium tetrachloride The Journal of Organic Chemistry. 50: 912-915. DOI: 10.1021/jo00206a048 |
0.118 |
|
| 1973 |
Sharpless KB, Michaelson RC. High stereo- and regioselectivities in the transition metal catalyzed epoxidations of olefinic alcohols by tert-butyl hydroperoxide Journal of the American Chemical Society. 95: 6136-6137. DOI: 10.1021/ja00799a061 |
0.116 |
|
| 1978 |
HERRANZ E, BILLER SA, SHARPLESS KB. ChemInform Abstract: OSMIUM-CATALYZED VICINAL OXYAMINATION OF OLEFINS BY N-CHLORO-N-ARGENTOCARBAMATES Chemischer Informationsdienst. 9. DOI: 10.1002/chin.197836123 |
0.115 |
|
| 2021 |
Taylor P, Shong YJ, Samskey N, Ho KY, Radic' Z, Fenical W, Sharpless KB, Kovarik Z, Andrea Camacho-Hernandez G. Ligand design for human acetylcholinesterase and nicotinic acetylcholine receptors, extending beyond the conventional and canonical. Journal of Neurochemistry. PMID 33638151 DOI: 10.1111/jnc.15335 |
0.115 |
|
| 2010 |
Demko ZP, Sharpless KB. ChemInform Abstract: Preparation of 5-Substituted 1H-Tetrazoles from Nitriles in Water. Cheminform. 33: no-no. DOI: 10.1002/chin.200222135 |
0.114 |
|
| 1978 |
Hori T, Sharpless KB. Synthetic applications of arylselenenic and arylseleninic acids. Conversion of olefins to allylic alcohols and epoxides The Journal of Organic Chemistry. 43: 1689-1697. DOI: 10.1021/jo00403a015 |
0.114 |
|
| 1986 |
HAWKINS JM, DEWAN JC, SHARPLESS KB. ChemInform Abstract: Dioxomolybdenum(VI)-Substituted 2,6-Pyridinedimethanol Complexes: New Five- Coordinate Species. Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198635268 |
0.114 |
|
| 1978 |
HERRANZ E, SHARPLESS KB. ChemInform Abstract: IMPROVEMENTS IN THE OSMIUM-CATALYZED OXYAMINATION OF OLEFINS BY CHLORAMINE-T Chemischer Informationsdienst. 9. DOI: 10.1002/chin.197844081 |
0.113 |
|
| 1972 |
SHARPLESS KB, FLOOD TC. ChemInform Abstract: DIREKTE DESOXYGENIERUNG VICINALER DIOLE MIT WOLFRAM(IV), EINE NEUE SYNTH. VON OLEFINEN Chemischer Informationsdienst. 3: no-no. DOI: 10.1002/chin.197228236 |
0.11 |
|
| 1967 |
Van Tamelen EE, Sharpless KB, Willett JD, Clayton RB, Burlingame AL. Biological activities of some terminally modified squalene and squalene 2,3-oxide analogs Journal of the American Chemical Society. 89: 3920-3922. DOI: 10.1021/Ja00991A055 |
0.109 |
|
| 2010 |
Chuang T, Sharpless KB. ChemInform Abstract: Applications of Aziridinium Ions: Selective Syntheses of Pyrazolidin-3-ones and Pyrazolo[1,2-a]pyrazoles. Cheminform. 31: no-no. DOI: 10.1002/chin.200046142 |
0.109 |
|
| 1980 |
HENTGES SG, SHARPLESS KB. ChemInform Abstract: IMPROVED PROCEDURE FOR THE OXYAMINATION OF OLEFINS WITH TRIOXO(TERT-BUTYLIMIDO)OSMIUM(VIII) Chemischer Informationsdienst. 11. DOI: 10.1002/chin.198050140 |
0.109 |
|
| 2010 |
HUGGER U, SHARPLESS KB. ChemInform Abstract: Asymmetric Dihydroxylation Affords Enantiomerically Pure C12 Building Blocks from trans,trans,cis-1,5,9-Cyclododecatriene. Cheminform. 26: no-no. DOI: 10.1002/chin.199551094 |
0.106 |
|
| 1985 |
Caron M, Sharpless KB. Titanium isopropoxide-mediated nucleophilic openings of 2,3-epoxy alcohols. A mild procedure for regioselective ring-opening The Journal of Organic Chemistry. 50: 1557-1560. DOI: 10.1021/jo00209a047 |
0.105 |
|
| 2000 |
Sander LC, Sharpless KE, Pursch M. C30 Stationary phases for the analysis of food by liquid chromatography Journal of Chromatography A. 880: 189-202. PMID 10890520 DOI: 10.1016/S0021-9673(00)00121-7 |
0.105 |
|
| 2010 |
Chuang T, Sharpless KB. ChemInform Abstract: Applications of Aziridinium Ions. Selective Syntheses of β-Aryl-α,β-diamino Esters. Cheminform. 31: no-no. DOI: 10.1002/chin.200002111 |
0.103 |
|
| 2010 |
Sharpless KB. ChemInform Abstract: Searching for New Reactivity (Nobel Lecture) Cheminform. 33: no-no. DOI: 10.1002/chin.200240288 |
0.103 |
|
| 1973 |
Sharpless KB, Lauer RF. Mild procedure for the conversion of epoxides to allylic alcohols. First organoselenium reagent Journal of the American Chemical Society. 95: 2697-2699. DOI: 10.1021/ja00789a055 |
0.102 |
|
| 1984 |
BEHRENS CH, SHARPLESS KB. ChemInform Abstract: NEW TRANSFORMATIONS OF 2,3-EPOXY ALCOHOLS AND RELATED DERIVATIVES. EASY ROUTES TO HOMOCHIRAL SUBSTANCES Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198441351 |
0.101 |
|
| 1969 |
Sharpless KB, Van Tamelen EE. Terpene terminal epoxides. Skeletal rearrangement accompanying bicyclization of squalene 2,3-oxide Journal of the American Chemical Society. 91: 1848-1849. DOI: 10.1021/ja01035a043 |
0.1 |
|
| 2010 |
Demko ZP, Sharpless KB. ChemInform Abstract: An Expedient Route to the Tetrazole Analogues of α-Amino Acids. Cheminform. 33: no-no. DOI: 10.1002/chin.200248140 |
0.099 |
|
| 2015 |
Schantz MM, Benner BA, Heckert NA, Sander LC, Sharpless KE, Vander Pol SS, Vasquez Y, Villegas M, Wise SA, Alwis KU, Blount BC, Calafat AM, Li Z, Silva MJ, Ye X, et al. Development of urine standard reference materials for metabolites of organic chemicals including polycyclic aromatic hydrocarbons, phthalates, phenols, parabens, and volatile organic compounds. Analytical and Bioanalytical Chemistry. 407: 2945-54. PMID 25651899 DOI: 10.1007/s00216-014-8441-0 |
0.098 |
|
| 1980 |
KATSUKI T, SHARPLESS KB. ChemInform Abstract: THE FIRST PRACTICAL METHOD FOR ASYMMETRIC EPOXIDATION Chemischer Informationsdienst. 11. DOI: 10.1002/chin.198048174 |
0.098 |
|
| 1973 |
SHARPLESS KB, TERANISHI AY. ChemInform Abstract: CHROMYLCHLORID IN ACETON, ALPHA-CHLOR-KETONE UND KETONE AUS OLEFINEN Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/chin.197318200 |
0.096 |
|
| 2010 |
CRISPINO GA, HO PT, SHARPLESS KB. ChemInform Abstract: Selective Perhydroxylation of Squalene: Taming the Arithmetic Demon. Cheminform. 24: no-no. DOI: 10.1002/chin.199316129 |
0.094 |
|
| 1979 |
LIESBESKIND LS, SHARPLESS KB, WILSON RD, IBERS JA. ChemInform Abstract: THE FIRST D0 METALLOOXAZIRIDINES. AMINATION OF OLEFINS Chemischer Informationsdienst. 10. DOI: 10.1002/chin.197905268 |
0.094 |
|
| 1986 |
BEHRENS CH, KO SY, SHARPLESS KB, WALKER FJ. ChemInform Abstract: Selective Transformation of 2,3-Epoxy Alcohols and Related Derivatives. Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198628137 |
0.09 |
|
| 1972 |
Sharpless KB, Lauer RF. Selenium dioxide oxidation of olefins. Evidence for the intermediacy of allylseleninic acids Journal of the American Chemical Society. 94: 7154-7155. DOI: 10.1021/ja00775a050 |
0.086 |
|
| 2001 |
Chuang T, Sharpless KB. ChemInform Abstract: Applications of Aziridinium Ions. Selective Syntheses of α,β-Diamino Esters, α-Sulfanyl-β-amino Esters, β-Lactams, and 1,5-Benzodiazepin-2-one. Cheminform. 32: no-no. DOI: 10.1002/chin.200111049 |
0.086 |
|
| 2010 |
Phillips MM, Case RJ, Rimmer CA, Sander LC, Sharpless KE, Wise SA, Yen JH. Determination of organic acids in Vaccinium berry standard reference materials. Analytical and Bioanalytical Chemistry. 398: 425-34. PMID 20582402 DOI: 10.1007/S00216-010-3916-0 |
0.085 |
|
| 1972 |
TOWNSEND JM, SHARPLESS KB. ChemInform Abstract: MECHANISMEN DER ZERS. VON SULFONIUMBETAINEN ZU EPOXIDEN Chemischer Informationsdienst. 3: no-no. DOI: 10.1002/chin.197247314 |
0.084 |
|
| 1982 |
Warpehoski MA, Chabaud B, Sharpless KB. Selenium dioxide oxidation of endocyclic olefins. Evidence for a dissociation-recombination pathway The Journal of Organic Chemistry. 47: 2897-2900. DOI: 10.1021/jo00136a017 |
0.083 |
|
| 1982 |
GONNELLA NC, NAKANISHI K, MARTIN VS, SHARPLESS KB. ChemInform Abstract: GENERAL METHOD FOR DETERMINING ABSOLUTE CONFIGURATION OF ACYCLIC ALLYLIC ALCOHOLS Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198242070 |
0.082 |
|
| 2000 |
Chuang TH, Sharpless KB. Applications of aziridinium ions. Selective syntheses of α,β-diamino esters, α-sulfanyl-β-amino esters, β-lactams, and 1,5-benzodiazepin-2-one Organic Letters. 2: 3555-3557. |
0.082 |
|
| 2021 |
Shyong YJ, Sepulveda Y, Garcia A, Samskey NM, Radic' Z, Sit R, Sharpless KB, Momper JD, Taylor PW.
The Journal of Pharmacology and Experimental Therapeutics. PMID 34145064 DOI: 10.1124/jpet.121.000715 |
0.081 |
|
| 1973 |
SHARPLESS KB, LAUER RF. ChemInform Abstract: MILDE METHODE DER UMWANDLUNG VON EPOXIDEN ZU ALLYLALKOHOLEN, ERSTES ORGANOSELEN-REAGENZ Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/chin.197326207 |
0.081 |
|
| 1970 |
Sharpless KB. d,1-Malabaricanediol. First cyclic natural product derived from squalene in a nonenzymic process Journal of the American Chemical Society. 92: 6999-7001. DOI: 10.1021/ja00726a064 |
0.079 |
|
| 1972 |
Sharpless KB, Lauer RF. Facile thermal rearrangements of allyl selenides and diselenides. [1,3] and [2,3] Shifts The Journal of Organic Chemistry. 37: 3973-3974. DOI: 10.1021/jo00797a058 |
0.078 |
|
| 1973 |
SHARPLESS KB, LAUER RF. ChemInform Abstract: GLATTE THERMISCHE UMLAGERUNGEN VON ALLYLSELENIDEN UND DISELENIDEN, (1,3)- UND (2,3)-VERSCHIEBUNGEN Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/chin.197312131 |
0.078 |
|
| 1979 |
Rossiter B, Verhoeven T, Sharpless K. Stereoselective epoxidation of acyclic allylic alcohols. A correction of our previous work. Tetrahedron Letters. 20: 4733-4736. DOI: 10.1016/S0040-4039(01)86696-X |
0.076 |
|
| 1971 |
Sharpless KB, Flood TC. Oxotransition metal oxidants as mimics for the action of mixed-function oxygenases. "NIH shift" with chromyl reagents. Journal of the American Chemical Society. 93: 2316-8. PMID 5553075 DOI: 10.1021/Ja00738A039 |
0.074 |
|
| 2013 |
Schantz MM, Eppe G, Focant JF, Hamilton C, Heckert NA, Heltsley RM, Hoover D, Keller JM, Leigh SD, Patterson DG, Pintar AL, Sharpless KE, Sjödin A, Turner WE, Vander Pol SS, et al. Milk and serum standard reference materials for monitoring organic contaminants in human samples. Analytical and Bioanalytical Chemistry. 405: 1203-11. PMID 23132544 DOI: 10.1007/S00216-012-6524-3 |
0.074 |
|
| 1981 |
Morgans DJ, Sharpless KB, Traynor SG. Epoxy alcohol rearrangements: hydroxyl-mediated delivery of Lewis acid promoters Journal of the American Chemical Society. 103: 462-464. DOI: 10.1021/ja00392a037 |
0.074 |
|
| 2001 |
Welch MJ, Colbert JC, Gill LM, Phinney CS, Sharpless KE, Sniegoski LT, Wood LJ. The certification of SRM 1546--Meat Homogenate, a new reference material for nutrients in a high protein, high fat matrix. Fresenius' Journal of Analytical Chemistry. 370: 42-7. PMID 11393235 |
0.074 |
|
| 2013 |
Phinney KW, Ballihaut G, Bedner M, Benford BS, Camara JE, Christopher SJ, Davis WC, Dodder NG, Eppe G, Lang BE, Long SE, Lowenthal MS, McGaw EA, Murphy KE, Nelson BC, ... ... Sharpless KE, et al. Development of a Standard Reference Material for metabolomics research. Analytical Chemistry. 85: 11732-8. PMID 24187941 DOI: 10.1021/Ac402689T |
0.073 |
|
| 1980 |
Katsuki T, Sharpless KB. The first practical method for asymmetric epoxidation Journal of the American Chemical Society. 102: 5974-5976. DOI: 10.1021/ja00538a077 |
0.072 |
|
| 1987 |
Elbein AD, Szumilo T, Sanford BA, Sharpless KB, Adams C. Effect of isomers of swainsonine on glycosidase activity and glycoprotein processing. Biochemistry. 26: 2502-10. PMID 3111529 DOI: 10.1021/bi00383a015 |
0.071 |
|
| 1990 |
DIJKSTRA GDH, KELLOGG RM, WYNBERG H, SVENDSEN JS, MARKO I, SHARPLESS KB. ChemInform Abstract: Conformational Study of Cinchona Alkaloids. A Combined NMR, Molecular Mechanics, and X-Ray Approach. Cheminform. 21. DOI: 10.1002/chin.199005282 |
0.071 |
|
| 2006 |
Sander LC, Sharpless KE, Wise SA. Dietary supplement Standard Reference Materials Life Sciences. 78: 2044-2048. PMID 16457853 DOI: 10.1016/j.lfs.2005.12.037 |
0.069 |
|
| 2003 |
Nelson BC, Sharpless KE. Quantification of the predominant monomeric catechins in baking chocolate standard reference material by LC/APCI-MS Journal of Agricultural and Food Chemistry. 51: 531-537. PMID 12537419 DOI: 10.1021/jf0207474 |
0.069 |
|
| 2004 |
Pearson CL, Xu K, Sharpless KE, Harris SD. MesA, a novel fungal protein required for the stabilization of polarity axes in Aspergillus nidulans. Molecular Biology of the Cell. 15: 3658-72. PMID 15155805 DOI: 10.1091/mbc.E03-11-0803 |
0.069 |
|
| 2010 |
CHANG H, SHARPLESS KB. ChemInform Abstract: A Practical Route to Enantiopure 1,2-Amino Alcohols. Cheminform. 27: no-no. DOI: 10.1002/chin.199633102 |
0.069 |
|
| 1999 |
Sharpless KE, Gill LM, Margolis SA, Wise SA, Elkins E. Preparation of Standard Reference Material 2383 (Baby Food Composite) and use of an interlaboratory comparison exercise for value assignment of its nutrient concentrations. Journal of Aoac International. 82: 276-87. PMID 10191534 |
0.069 |
|
| 1967 |
van Tamelen E, Sharpless K. Positional selectivity during controlled oxidation of polyolefins Tetrahedron Letters. 8: 2655-2659. DOI: 10.1016/S0040-4039(01)89969-X |
0.069 |
|
| 2012 |
Sander LC, Bedner M, Tims MC, Yen JH, Duewer DL, Porter B, Christopher SJ, Day RD, Long SE, Molloy JL, Murphy KE, Lang BE, Lieberman R, Wood LJ, Payne MJ, ... ... Sharpless KE, et al. Development and certification of green tea-containing standard reference materials. Analytical and Bioanalytical Chemistry. 402: 473-87. PMID 22127575 DOI: 10.1007/S00216-011-5472-7 |
0.068 |
|
| 2007 |
Thomas JB, Sharpless KE, Mitvalsky S, Roman M, Yen J, Satterfield MB. Determination of caffeine and caffeine-related metabolites in ephedra-containing standard reference materials using liquid chromatography with absorbance detection and tandem mass spectrometry. Journal of Aoac International. 90: 934-40. PMID 17760330 |
0.067 |
|
| 2002 |
Sharpless KE, Harris SD. Functional characterization and localization of the Aspergillus nidulans formin SEPA Molecular Biology of the Cell. 13: 469-479. PMID 11854405 DOI: 10.1091/mbc.01-07-0356 |
0.067 |
|
| 2010 |
Bedner M, Sander LC, Sharpless KE. An LC-ESI/MS method for determining theanine in green tea dietary supplements Analytical and Bioanalytical Chemistry. 397: 1773-1777. PMID 20422160 DOI: 10.1007/s00216-010-3713-9 |
0.066 |
|
| 2003 |
Sharpless KE, Phinney CS, Wood LJ, Yen JH, Howell DW. Value assignment of nutrient and aflatoxin concentrations in standard reference material 2387 peanut butter. Journal of Agricultural and Food Chemistry. 51: 6745-51. PMID 14582970 DOI: 10.1021/jf034637o |
0.066 |
|
| 2008 |
Nelson BC, Pfeiffer CM, Zhang M, Duewer DL, Sharpless KE, Lippa KA. Commutability of NIST SRM 1955 Homocysteine and Folate in Frozen Human Serum with selected total homocysteine immunoassays and enzymatic assays Clinica Chimica Acta. 395: 99-105. PMID 18565331 DOI: 10.1016/J.Cca.2008.05.016 |
0.063 |
|
| 1971 |
Sharpless KB, Lauer RF, Repic O, Teranishi AY, Williams DR. Permanganate in acetic anhydride. .alpha.-Diketones directly from olefins Journal of the American Chemical Society. 93: 3303-3304. DOI: 10.1021/ja00742a045 |
0.062 |
|
| 2009 |
Duewer DL, Lippa KA, Long SE, Murphy KE, Sharpless KE, Sniegoski LT, Welch MJ, Tani W, Umemoto M. Demonstrating the comparability of certified reference materials. Analytical and Bioanalytical Chemistry. 395: 155-69. PMID 19629455 DOI: 10.1007/S00216-009-2949-8 |
0.062 |
|
| 2012 |
Thomas JB, Duewer DL, Mugenya IO, Phinney KW, Sander LC, Sharpless KE, Sniegoski LT, Tai SS, Welch MJ, Yen JH. Preparation and value assignment of standard reference material 968e fat-soluble vitamins, carotenoids, and cholesterol in human serum. Analytical and Bioanalytical Chemistry. 402: 749-62. PMID 22015475 DOI: 10.1007/S00216-011-5447-8 |
0.062 |
|
| 2006 |
Sharpless KE, Anderson DL, Betz JM, Butler TA, Capar SG, Cheng J, Fraser CA, Gardner G, Gay ML, Howell DW, Ihara T, Khan MA, Lam JW, Long SE, McCooeye M, et al. Preparation and characterization of a suite of ephedra-containing standard reference materials. Journal of Aoac International. 89: 1483-95. PMID 17225593 DOI: 10.1093/Jaoac/89.6.1483 |
0.062 |
|
| 2007 |
Putzbach K, Rimmer CA, Sharpless KE, Sander LC. Determination of Bitter Orange alkaloids in dietary supplements standard reference materials by liquid chromatography with ultraviolet absorbance and fluorescence detection Journal of Chromatography A. 1156: 304-311. PMID 17524413 DOI: 10.1016/J.Chroma.2006.12.027 |
0.061 |
|
| 2006 |
Nelson BC, Sharpless KE, Sander LC. Improved liquid chromatography methods for the separation and quantification of biotin in NIST Standard Reference Material 3280: Multivitamin/multielement tablets Journal of Agricultural and Food Chemistry. 54: 8710-8716. PMID 17090111 DOI: 10.1021/jf062000+ |
0.06 |
|
| 1972 |
SHARPLESS KB, TOWNSEND JM, WILLIAMS DR. ChemInform Abstract: MECHANISMUS DER EPOX. VON OLEFINEN DURCH KOVALENTE PEROXIDE DES MOLYBDAEN(VI) Chemischer Informationsdienst. 3. DOI: 10.1002/chin.197212098 |
0.06 |
|
| 2006 |
Dwyer JT, Picciano MF, Betz JM, Fisher KD, Saldanha LG, Yetley EA, Coates PM, Radimer K, Bindewald B, Sharpless KE, Holden J, Andrews K, Zhao C, Harnly J, Wolf WR, et al. Progress in development of an integrated dietary supplement ingredient database at the NIH Office of Dietary Supplements. Journal of Food Composition and Analysis : An Official Publication of the United Nations University, International Network of Food Data Systems. 19: S108-S114. PMID 25309034 DOI: 10.1016/J.Jfca.2005.09.001 |
0.06 |
|
| 2005 |
Sander LC, Sharpless KE, Satterfield MB, Ihara T, Phinney KW, Yen JH, Wise SA, Gay ML, Lam JW, McCooeye M, Gardner G, Fraser C, Sturgeon R, Roman M. Determination of ephedrine alkaloids in dietary supplement standard reference materials. Analytical Chemistry. 77: 3101-12. PMID 15889898 DOI: 10.1021/Ac0484530 |
0.059 |
|
| 2013 |
Rimmer CA, Sharpless KE, Wise SA, Betz JM, Coates PM. Standard reference materials for dietary supplement analysis Analytical and Bioanalytical Chemistry. 405: 4337-4344. PMID 23575912 DOI: 10.1007/S00216-013-6942-X |
0.058 |
|
| 2008 |
Sander LC, Putzbach K, Nelson BC, Rimmer CA, Bedner M, Thomas JB, Porter BJ, Wood LJ, Schantz MM, Murphy KE, Sharpless KE, Wise SA, Yen JH, Siitonen PH, Evans RL, et al. Certification of standard reference materials containing bitter orange. Analytical and Bioanalytical Chemistry. 391: 2023-34. PMID 18425642 DOI: 10.1007/S00216-008-2074-0 |
0.058 |
|
| 2006 |
Satterfield MB, Sniegoski LT, Sharpless KE, Welch MJ, Hornikova A, Zhang NF, Pfeiffer CM, Fazili Z, Zhang M, Nelson BC. Development of a new standard reference material: SRM 1955 (homocysteine and folate in human serum). Analytical and Bioanalytical Chemistry. 385: 612-22. PMID 16715281 DOI: 10.1007/s00216-006-0434-1 |
0.058 |
|
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