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Samuel J. Danishefsky - Publications

Affiliations: 
Columbia University, New York, NY 
 Memorial Sloan-Kettering Cancer Center, Rockville Centre, NY, United States 
Area:
synthetic organic chemistry
Website:
http://www.mskcc.org/research/lab/samuel-danishefsky

449 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2019 Li Y, Tran AH, Danishefsky SJ, Tan Z. Chemical biology of glycoproteins: From chemical synthesis to biological impact. Methods in Enzymology. 621: 213-229. PMID 31128780 DOI: 10.1016/Bs.Mie.2019.02.030  0.486
2018 Brailsford JA, Stockdill JL, Axelrod AJ, Peterson MT, Vadola PA, Johnston EV, Danishefsky SJ. Total Chemical Synthesis of Human Thyroid-Stimulating Hormone (hTSH) -Subunit: Application of Arginine-tagged Acetamidomethyl (Acm) Protecting Groups. Tetrahedron. 74: 1951-1956. PMID 30853725 DOI: 10.1016/J.Tet.2018.02.067  0.785
2017 Rao TD, Fernández-Tejada A, Axelrod A, Rosales N, Yan X, Thapi S, Wang A, Park KJ, Nemieboka B, Xiang J, Lewis JS, Olvera N, Levine DA, Danishefsky SJ, Spriggs D. Antibodies Against Specific MUC16 Glycosylation Sites Inhibit Ovarian Cancer Growth. Acs Chemical Biology. PMID 28617578 DOI: 10.1021/Acschembio.7B00305  0.768
2017 Levinson AM, McGee JH, Roberts AG, Creech G, Wang T, Peterson MT, Hendrickson RC, Verdine GL, Danishefsky SJ. Total Chemical Synthesis and Folding of All-L and All-D Variants of Oncogenic KRas(G12V). Journal of the American Chemical Society. PMID 28448128 DOI: 10.1021/Jacs.7B02988  0.783
2016 O'Cearbhaill RE, Ragupathi G, Zhu J, Wan Q, Mironov S, Yang G, Spassova MK, Iasonos A, Kravetz S, Ouerfelli O, Spriggs DR, Danishefsky SJ, Sabbatini PJ. A Phase I Study of Unimolecular Pentavalent (Globo-H-GM2-sTn-TF-Tn) Immunization of Patients with Epithelial Ovarian, Fallopian Tube, or Peritoneal Cancer in First Remission. Cancers. 8. PMID 27110823 DOI: 10.3390/Cancers8040046  0.528
2015 Roberts AG, Johnston EV, Shieh JH, Sondey JP, Hendrickson RC, Moore MA, Danishefsky SJ. Fully Synthetic Granulocyte Colony-Stimulating Factor Enabled by Isonitrile-Mediated Coupling of Large, Side-Chain-Unprotected Peptides. Journal of the American Chemical Society. 137: 13167-75. PMID 26401918 DOI: 10.1021/Jacs.5B08754  0.598
2015 Fernández-Tejada A, Brailsford J, Zhang Q, Shieh JH, Moore MA, Danishefsky SJ. Total synthesis of glycosylated proteins. Topics in Current Chemistry. 362: 1-26. PMID 25805144 DOI: 10.1007/128_2014_622  0.425
2014 Hartung J, J D Wright B, Danishefsky SJ. Studies toward the total synthesis of pluraflavin A. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 8731-6. PMID 24919792 DOI: 10.1002/Chem.201402254  0.536
2014 Townsend SD, Ross AG, Liu K, Danishefsky SJ. Stereospecific cis- and trans-ring fusions arising from common intermediates. Proceedings of the National Academy of Sciences of the United States of America. 111: 7931-5. PMID 24843125 DOI: 10.1073/Pnas.1407613111  0.774
2014 Fernández-Tejada A, Vadola PA, Danishefsky SJ. Chemical synthesis of the β-subunit of human luteinizing (hLH) and chorionic gonadotropin (hCG) glycoprotein hormones. Journal of the American Chemical Society. 136: 8450-8. PMID 24806200 DOI: 10.1021/Ja503545R  0.785
2014 Creech GS, Paresi C, Li YM, Danishefsky SJ. Chemical synthesis of the ATAD2 bromodomain. Proceedings of the National Academy of Sciences of the United States of America. 111: 2891-6. PMID 24516155 DOI: 10.1073/Pnas.1400556111  0.802
2014 Zhang Q, Johnston EV, Shieh JH, Moore MA, Danishefsky SJ. Synthesis of granulocyte-macrophage colony-stimulating factor as homogeneous glycoforms and early comparisons with yeast cell-derived material. Proceedings of the National Academy of Sciences of the United States of America. 111: 2885-90. PMID 24516138 DOI: 10.1073/Pnas.1400140111  0.379
2014 Pham HV, Paton RS, Ross AG, Danishefsky SJ, Houk KN. Intramolecular Diels-Alder reactions of cycloalkenones: stereoselectivity, Lewis acid acceleration, and halogen substituent effects. Journal of the American Chemical Society. 136: 2397-403. PMID 24410341 DOI: 10.1021/Ja410220W  0.624
2013 Wang P, Dong S, Shieh JH, Peguero E, Hendrickson R, Moore MA, Danishefsky SJ. Erythropoietin derived by chemical synthesis. Science (New York, N.Y.). 342: 1357-60. PMID 24337294 DOI: 10.1126/Science.1245095  0.498
2013 Alam SM, Dennison SM, Aussedat B, Vohra Y, Park PK, Fernández-Tejada A, Stewart S, Jaeger FH, Anasti K, Blinn JH, Kepler TB, Bonsignori M, Liao HX, Sodroski JG, Danishefsky SJ, et al. Recognition of synthetic glycopeptides by HIV-1 broadly neutralizing antibodies and their unmutated ancestors. Proceedings of the National Academy of Sciences of the United States of America. 110: 18214-9. PMID 24145434 DOI: 10.1073/Pnas.1317855110  0.646
2013 Aussedat B, Vohra Y, Park PK, Fernández-Tejada A, Alam SM, Dennison SM, Jaeger FH, Anasti K, Stewart S, Blinn JH, Liao HX, Sodroski JG, Haynes BF, Danishefsky SJ. Chemical synthesis of highly congested gp120 V1V2 N-glycopeptide antigens for potential HIV-1-directed vaccines. Journal of the American Chemical Society. 135: 13113-20. PMID 23915436 DOI: 10.1021/Ja405990Z  0.657
2013 Wang T, Danishefsky SJ. Solid-phase peptide synthesis and solid-phase fragment coupling mediated by isonitriles. Proceedings of the National Academy of Sciences of the United States of America. 110: 11708-13. PMID 23821753 DOI: 10.1073/Pnas.1310431110  0.406
2013 Peng F, Grote RE, Wilson RM, Danishefsky SJ. Pattern recognition analysis in complex molecule synthesis and the preparation of iso-Diels-Alder motifs. Proceedings of the National Academy of Sciences of the United States of America. 110: 10904-9. PMID 23784777 DOI: 10.1073/Pnas.1309795110  0.789
2013 Wilson RM, Dong S, Wang P, Danishefsky SJ. The winding pathway to erythropoietin along the chemistry-biology frontier: a success at last. Angewandte Chemie (International Ed. in English). 52: 7646-65. PMID 23775885 DOI: 10.1002/Anie.201301666  0.384
2013 Walczak MA, Hayashida J, Danishefsky SJ. Building biologics by chemical synthesis: practical preparation of di- and triantennary N-linked glycoconjugates. Journal of the American Chemical Society. 135: 4700-3. PMID 23461434 DOI: 10.1021/Ja401385V  0.564
2013 Ross AG, Townsend SD, Danishefsky SJ. Halocycloalkenones as Diels-Alder dienophiles. Applications to generating useful structural patterns. The Journal of Organic Chemistry. 78: 204-10. PMID 23151095 DOI: 10.1021/Jo302230M  0.79
2013 Wilson RM, Dong S, Wang P, Danishefsky SJ. Der gewundene Pfad zum Erythropoietin entlang der Grenze von Chemie und Biologie Angewandte Chemie. 125: 7798-7818. DOI: 10.1002/Ange.201301666  0.374
2012 Peng F, Dai M, Angeles AR, Danishefsky SJ. Permuting Diels-Alder and Robinson Annulation Stereopatterns. Chemical Science (Royal Society of Chemistry : 2010). 3: 3076-3080. PMID 23139855 DOI: 10.1039/C2Sc20868G  0.795
2012 Peng F, Danishefsky SJ. Total synthesis of (±)-maoecrystal V. Journal of the American Chemical Society. 134: 18860-7. PMID 23126440 DOI: 10.1021/Ja309905J  0.522
2012 Li J, Dong S, Townsend SD, Dean T, Gardella TJ, Danishefsky SJ. Chemistry as an expanding resource in protein science: fully synthetic and fully active human parathyroid hormone-related protein (1-141). Angewandte Chemie (International Ed. in English). 51: 12263-7. PMID 23124999 DOI: 10.1002/Anie.201207603  0.788
2012 Wang P, Dong S, Brailsford JA, Iyer K, Townsend SD, Zhang Q, Hendrickson RC, Shieh J, Moore MA, Danishefsky SJ. At last: erythropoietin as a single glycoform. Angewandte Chemie (International Ed. in English). 51: 11576-84. PMID 23012228 DOI: 10.1002/Anie.201206090  0.81
2012 Wang P, Aussedat B, Vohra Y, Danishefsky SJ. An advance in the chemical synthesis of homogeneous N-linked glycopolypeptides by convergent aspartylation. Angewandte Chemie (International Ed. in English). 51: 11571-5. PMID 23011954 DOI: 10.1002/Anie.201205038  0.496
2012 Walczak MA, Danishefsky SJ. Solving the convergence problem in the synthesis of triantennary N-glycan relevant to prostate-specific membrane antigen (PSMA). Journal of the American Chemical Society. 134: 16430-3. PMID 22954207 DOI: 10.1021/Ja307628W  0.516
2012 Ross AG, Li X, Danishefsky SJ. Intramolecular Diels-Alder reactions of cycloalkenones: translation of high endo selectivity to trans junctions. Journal of the American Chemical Society. 134: 16080-4. PMID 22950514 DOI: 10.1021/Ja307708Q  0.629
2012 Dong S, Shang S, Li J, Tan Z, Dean T, Maeda A, Gardella TJ, Danishefsky SJ. Engineering of therapeutic polypeptides through chemical synthesis: early lessons from human parathyroid hormone and analogues. Journal of the American Chemical Society. 134: 15122-9. PMID 22891619 DOI: 10.1021/Ja306637U  0.548
2012 Wang T, Danishefsky SJ. Revisiting oxytocin through the medium of isonitriles. Journal of the American Chemical Society. 134: 13244-7. PMID 22830449 DOI: 10.1021/Ja3063452  0.421
2012 Townsend SD, Wu X, Danishefsky SJ. Enhancing the scope of the Diels-Alder reaction through isonitrile chemistry: emergence of a new class of acyl-activated dienophiles. Journal of the American Chemical Society. 134: 10659-63. PMID 22708980 DOI: 10.1021/Ja303876E  0.778
2012 Brailsford JA, Danishefsky SJ. Probing the stability of nonglycosylated wild-type erythropoietin protein via reiterative alanine ligations. Proceedings of the National Academy of Sciences of the United States of America. 109: 7196-201. PMID 22499784 DOI: 10.1073/Pnas.1202762109  0.363
2012 Wilson RM, Stockdill JL, Wu X, Li X, Vadola PA, Park PK, Wang P, Danishefsky SJ. A fascinating journey into history: exploration of the world of isonitriles en route to complex amides. Angewandte Chemie (International Ed. in English). 51: 2834-48. PMID 22368033 DOI: 10.1002/Anie.201106628  0.779
2012 Townsend SD, Tan Z, Dong S, Shang S, Brailsford JA, Danishefsky SJ. Advances in proline ligation. Journal of the American Chemical Society. 134: 3912-6. PMID 22332757 DOI: 10.1021/Ja212182Q  0.785
2012 Aussedat B, Fasching B, Johnston E, Sane N, Nagorny P, Danishefsky SJ. Total synthesis of the α-subunit of human glycoprotein hormones: toward fully synthetic homogeneous human follicle-stimulating hormone. Journal of the American Chemical Society. 134: 3532-41. PMID 22280541 DOI: 10.1021/Ja2111459  0.656
2012 Wu X, Stockdill JL, Park PK, Danishefsky SJ. Expanding the limits of isonitrile-mediated amidations: on the remarkable stereosubtleties of macrolactam formation from synthetic seco-cyclosporins. Journal of the American Chemical Society. 134: 2378-84. PMID 22280518 DOI: 10.1021/Ja2103372  0.736
2012 Danishefsky S, Hungate R. The total synthesis of octosyl acid A: a new departure in organostannylene chemistry. Journal of the American Chemical Society. 108: 2486-7. PMID 22175627 DOI: 10.1021/Ja00269A080  0.352
2012 Nagorny P, Sane N, Fasching B, Aussedat B, Danishefsky SJ. Probing the frontiers of glycoprotein synthesis: the fully elaborated β-subunit of the human follicle-stimulating hormone. Angewandte Chemie (International Ed. in English). 51: 975-9. PMID 22162182 DOI: 10.1002/Anie.201107482  0.611
2012 Wang P, Dong S, Brailsford JA, Iyer K, Townsend SD, Zhang Q, Hendrickson RC, Shieh J, Moore MAS, Danishefsky SJ. Cover Picture: At Last: Erythropoietin as a Single Glycoform (Angew. Chem. Int. Ed. 46/2012) Angewandte Chemie International Edition. 51: 11391-11391. DOI: 10.1002/Anie.201208087  0.759
2012 Wang P, Dong S, Brailsford JA, Iyer K, Townsend SD, Zhang Q, Hendrickson RC, Shieh J, Moore MAS, Danishefsky SJ. Titelbild: At Last: Erythropoietin as a Single Glycoform (Angew. Chem. 46/2012) Angewandte Chemie. 124: 11555-11555. DOI: 10.1002/Ange.201208087  0.756
2012 Wilson RM, Stockdill JL, Wu X, Li X, Vadola PA, Park PK, Wang P, Danishefsky SJ. Eine faszinierende Reise in die Geschichte: Isonitrile als Ausgangsverbindungen für komplexe Amide Angewandte Chemie. 124: 2888-2902. DOI: 10.1002/Ange.201106628  0.761
2012 Yu B, Wang LX, Danishefsky S, Crich D. Carbohydrate Synthesis towards Glycobiology Organic Chemistry - Breakthroughs and Perspectives. 181-219. DOI: 10.1002/9783527664801.ch5  0.306
2012 Ross AG, Li X, Danishefsky SJ. Preparation of cyclobutenone Organic Syntheses. 89: 491-500. DOI: 10.1002/0471264229.Os089.47  0.589
2011 Dong S, Shang S, Tan Z, Danishefsky SJ. Toward Homogeneous Erythropoietin: Application of Metal Free Dethiylation in the Chemical Synthesis of the Ala79-Arg166 Glycopeptide Domain. Israel Journal of Chemistry. 51: 968-976. PMID 23585694 DOI: 10.1002/Ijch.201100077  0.547
2011 Wang Z, Dai M, Park PK, Danishefsky SJ. Synthetic studies toward (+)-cortistatin A. Tetrahedron. 67: 10249-10260. PMID 22879684 DOI: 10.1016/J.Tet.2011.10.026  0.711
2011 Paton RS, Kim S, Ross AG, Danishefsky SJ, Houk KN. Experimental Diels-Alder reactivities of cycloalkenones and cyclic dienes explained through transition-state distortion energies. Angewandte Chemie (International Ed. in English). 50: 10366-8. PMID 21910195 DOI: 10.1002/Anie.201103998  0.567
2011 Chou TC, Dong H, Zhang X, Lei X, Hartung J, Zhang Y, Lee JH, Wilson RM, Danishefsky SJ. Multifaceted cytoprotection by synthetic polyacetylenes inspired by the ginseng-derived natural product, panaxytriol. Proceedings of the National Academy of Sciences of the United States of America. 108: 14336-41. PMID 21844359 DOI: 10.1073/Pnas.1111332108  0.714
2011 Peng F, Grote RE, Danishefsky SJ. Further Expansion of the trans-Diels-Alder Paradigm: Reductive Alkylation of α-Cyanoketones. Tetrahedron Letters. 52: 3957-3959. PMID 21808427 DOI: 10.1016/J.Tetlet.2011.05.110  0.789
2011 Lecomte N, Njardarson JT, Nagorny P, Yang G, Downey R, Ouerfelli O, Moore MA, Danishefsky SJ. Emergence of potent inhibitors of metastasis in lung cancer via syntheses based on migrastatin. Proceedings of the National Academy of Sciences of the United States of America. 108: 15074-8. PMID 21808037 DOI: 10.1073/Pnas.1015247108  0.737
2011 Shang S, Tan Z, Dong S, Danishefsky SJ. An advance in proline ligation. Journal of the American Chemical Society. 133: 10784-6. PMID 21696220 DOI: 10.1021/Ja204277B  0.509
2011 Wu X, Park PK, Danishefsky SJ. On the synthesis of conformationally modified peptides through isonitrile chemistry: implications for dealing with polypeptide aggregation. Journal of the American Chemical Society. 133: 7700-3. PMID 21539308 DOI: 10.1021/Ja2023898  0.317
2011 Peng F, Danishefsky SJ. Toward the total synthesis of maoecrystal V: an intramolecular Diels-Alder route to the maoecrystal V pentacyclic core with the appropriate relative stereochemistry. Tetrahedron Letters. 52: 2104-2106. PMID 21516211 DOI: 10.1016/J.Tetlet.2010.11.029  0.503
2011 Shang S, Tan Z, Danishefsky SJ. Application of the logic of cysteine-free native chemical ligation to the synthesis of Human Parathyroid Hormone (hPTH). Proceedings of the National Academy of Sciences of the United States of America. 108: 5986-9. PMID 21444787 DOI: 10.1073/Pnas.1103118108  0.531
2011 Tan Z, Shang S, Danishefsky SJ. Rational development of a strategy for modifying the aggregatibility of proteins. Proceedings of the National Academy of Sciences of the United States of America. 108: 4297-302. PMID 21368182 DOI: 10.1073/Pnas.1100195108  0.527
2011 Wang P, Li X, Zhu J, Chen J, Yuan Y, Wu X, Danishefsky SJ. Encouraging progress in the ω-aspartylation of complex oligosaccharides as a general route to β-N-linked glycopolypeptides. Journal of the American Chemical Society. 133: 1597-602. PMID 21207981 DOI: 10.1021/Ja110115A  0.575
2011 Zhang Y, Lee JH, Danishefsky SJ. Antarafacial mediation of oxygen delivery by a phenylsulfinyl group in the epoxidation of proximal double bonds: intramolecular trapping of an early Pummerer intermediate with stereoelectronic control. Journal of the American Chemical Society. 133: 752-5. PMID 21182300 DOI: 10.1021/Ja1107707  0.678
2010 Tan Z, Shang S, Danishefsky SJ. Insights into the finer issues of native chemical ligation: an approach to cascade ligations. Angewandte Chemie (International Ed. in English). 49: 9500-3. PMID 21053233 DOI: 10.1002/Anie.201005513  0.551
2010 Wang P, Danishefsky SJ. Promising general solution to the problem of ligating peptides and glycopeptides. Journal of the American Chemical Society. 132: 17045-51. PMID 21049949 DOI: 10.1021/Ja1084628  0.476
2010 Lee JH, Zhang Y, Danishefsky SJ. A straightforward route to functionalized trans-Diels-Alder motifs. Journal of the American Chemical Society. 132: 14330-3. PMID 20863105 DOI: 10.1021/Ja1073855  0.66
2010 Lee JH, Danishefsky SJ. Diels-Alder routes to angularly halogenated cis-fused bicyclic ketones: Readily accessible cyclynone intermediates. Tetrahedron Letters. 51: 4653-4654. PMID 20835369 DOI: 10.1016/j.tetlet.2010.06.135  0.431
2010 Chen J, Wang P, Zhu J, Wan Q, Danishefsky SJ. A program for ligation at threonine sites: application to the controlled total synthesis of glycopeptides. Tetrahedron. 66: 2277-2283. PMID 20798898 DOI: 10.1016/J.Tet.2010.01.067  0.623
2010 Kim WH, Lee JH, Aussedat B, Danishefsky SJ. A Diels-Alder Route to Angularly Functionalized Bicyclic Structures. Tetrahedron. 66: 6391-6398. PMID 20717474 DOI: 10.1016/j.tet.2010.04.094  0.39
2010 Trzupek JD, Li C, Chan C, Crowley BM, Heimann AC, Danishefsky SJ. Lessons from the Total Synthesis of (±) Phalarine: Insights Into the Mechanism of the Pictet-Spengler Reaction. Pure and Applied Chemistry. Chimie Pure Et Appliquee. 82: 1735-1748. PMID 20711493 DOI: 10.1351/Pac-Con-09-11-14  0.73
2010 Nagorny P, Krauss I, Njardarson JT, Perez L, Gaul C, Yang G, Ouerfelli O, Danishefsky SJ. Confirmation of the Structures of Synthetic Derivatives of Migrastatin in the Light of Recently Disclosed Crystallographically Based Claims. Tetrahedron Letters. 51: 3873-3875. PMID 20676392 DOI: 10.1016/J.Tetlet.2010.05.056  0.773
2010 Wilson RM, Danishefsky SJ. On the reach of chemical synthesis: creation of a mini-pipeline from an academic laboratory. Angewandte Chemie (International Ed. in English). 49: 6032-56. PMID 20661969 DOI: 10.1002/Anie.201000775  0.336
2010 Yuan Y, Chen J, Wan Q, Wilson RM, Danishefsky SJ. Toward fully synthetic, homogeneous glycoproteins: advances in chemical ligation. Biopolymers. 94: 373-84. PMID 20593459 DOI: 10.1002/Bip.21374  0.477
2010 Paton RS, Mackey JL, Kim WH, Lee JH, Danishefsky SJ, Houk KN. Origins of stereoselectivity in the trans Diels-Alder paradigm. Journal of the American Chemical Society. 132: 9335-40. PMID 20557046 DOI: 10.1021/Ja1009162  0.467
2010 Zhang Y, Danishefsky SJ. Total synthesis of (+/-)-aplykurodinone-1: traceless stereochemical guidance. Journal of the American Chemical Society. 132: 9567-9. PMID 20513158 DOI: 10.1021/Ja1035495  0.604
2010 Wu X, Stockdill JL, Wang P, Danishefsky SJ. Total synthesis of cyclosporine: access to N-methylated peptides via isonitrile coupling reactions. Journal of the American Chemical Society. 132: 4098-100. PMID 20199071 DOI: 10.1021/Ja100517V  0.775
2010 Lee JH, Kim WH, Danishefsky SJ. An Ionic Diels-Alder Route to cis-Fused Octalins Containing an All-Carbon Quaternary Stereocenter in an Angular Position. Tetrahedron Letters. 51: 1252. PMID 20174450 DOI: 10.1016/j.tetlet.2009.12.127  0.353
2010 Oskarsson T, Nagorny P, Krauss IJ, Perez L, Mandal M, Yang G, Ouerfelli O, Xiao D, Moore MA, Massagué J, Danishefsky SJ. Diverted total synthesis leads to the generation of promising cell-migration inhibitors for treatment of tumor metastasis: in vivo and mechanistic studies on the migrastatin core ether analog. Journal of the American Chemical Society. 132: 3224-8. PMID 20155906 DOI: 10.1021/Ja9101503  0.781
2010 Tsukano C, Siegel DR, Danishefsky SJ. Total syntheses of polycyclic polyp renylated acylphloroglucinols Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry. 68: 592-600. DOI: 10.5059/Yukigoseikyokaishi.68.592  0.664
2010 GRIFFITH DA, DANISHEFSKY SJ. ChemInform Abstract: Total Synthesis of Allosamidin: An Application of the Sulfonamidoglycosylation of Glycals. Cheminform. 22: no-no. DOI: 10.1002/chin.199144276  0.622
2010 Wilson R, Danishefsky S. Cover Picture: On the Reach of Chemical Synthesis: Creation of a Mini-Pipeline from an Academic Laboratory (Angew. Chem. Int. Ed. 35/2010) Angewandte Chemie International Edition. 49: 6003-6003. DOI: 10.1002/Anie.201004265  0.35
2010 Wilson R, Danishefsky S. Titelbild: Zum Wirkungsbereich der chemischen Synthese: Aufbau einer Minipipeline in einem akademischen Labor (Angew. Chem. 35/2010) Angewandte Chemie. 122: 6139-6139. DOI: 10.1002/Ange.201004265  0.308
2009 Zhu J, Wu X, Danishefsky SJ. On the Preparation of Enantiomerically Pure Isonitriles from Amino Acid Esters and Peptides. Tetrahedron Letters. 50: 577-579. PMID 21869850 DOI: 10.1016/J.Tetlet.2008.11.069  0.531
2009 Zhu J, Wan Q, Yang G, Ouerfelli O, Danishefsky SJ. Synthesis of Human Cancer Associated Globo-H (MBr1) Glycosylamino Acid: Some Mechanistic and Conformational Reinvestigations. Heterocycles. 79: 441-449. PMID 21423783 DOI: 10.3987/Com-08-S(D)82  0.637
2009 Lee JH, Kim WH, Danishefsky SJ. Syntheses of Isomerically Pure Reference Octalins and Hydrindanes. Tetrahedron Letters. 50: 5482-5484. PMID 20711484 DOI: 10.1016/J.Tetlet.2009.07.068  0.466
2009 Yuan Y, Chen J, Wan Q, Tan Z, Chen G, Kan C, Danishefsky SJ. Toward homogeneous erythropoietin: fine tuning of the C-terminal acyl donor in the chemical synthesis of the Cys29-Gly77 glycopeptide domain. Journal of the American Chemical Society. 131: 5432-7. PMID 20560636 DOI: 10.1021/Ja808705V  0.714
2009 Peng F, Yu M, Danishefsky SJ. Synthetic Studies towards Maoecrystal V. Tetrahedron Letters. 50: 6586. PMID 20174449 DOI: 10.1016/J.Tetlet.2009.09.050  0.5
2009 Yuan Y, Zhu J, Li X, Wu X, Danishefsky SJ. Preparation and reactions of N-thioformyl peptides from amino thioacids and isonitriles. Tetrahedron Letters. 50: 2329-2333. PMID 20161291 DOI: 10.1016/J.Tetlet.2009.02.205  0.446
2009 Wu X, Yuan Y, Li X, Danishefsky SJ. Thio-mediated synthesis of derivatized N-linked glycopeptides using isonitrile chemistry. Tetrahedron Letters. 50: 4666-4669. PMID 20161157 DOI: 10.1016/J.Tetlet.2009.06.005  0.353
2009 Stockdill JL, Wu X, Danishefsky SJ. Coupling reactions of hindered isonitriles and hindered alkyl thioacids: Mechanistic studies. Tetrahedron Letters. 50: 5152-5155. PMID 20160954 DOI: 10.1016/J.Tetlet.2009.06.129  0.732
2009 Kim WH, Angeles AR, Lee JH, Danishefsky SJ. Concise Synthesis of the Xenibellols Core. Tetrahedron Letters. 50: 6440-6441. PMID 20160940 DOI: 10.1016/J.Tetlet.2009.08.131  0.816
2009 Rao Y, Li X, Nagorny P, Hayashida J, Danishefsky SJ. A Simple Method for the Conversion of Carboxylic Acids into Thioacids with Lawesson's Reagent. Tetrahedron Letters. 50: 6684-6686. PMID 20160926 DOI: 10.1016/J.Tetlet.2009.09.080  0.589
2009 Zhu J, Wan Q, Danishefsky SJ. Synthesis of Biotinylated Tumor-Associated Carbohydrate Antigens for Immunological Studies. Tetrahedron Letters. 50: 712-714. PMID 20157341 DOI: 10.1016/J.Tetlet.2008.11.113  0.612
2009 Wang P, Zhu J, Yuan Y, Danishefsky SJ. Total synthesis of the 2,6-sialylated immunoglobulin G glycopeptide fragment in homogeneous form. Journal of the American Chemical Society. 131: 16669-71. PMID 19886622 DOI: 10.1021/Ja907136D  0.588
2009 Jeon I, Iyer K, Danishefsky SJ. A practical total synthesis of globo-H for use in anticancer vaccines. The Journal of Organic Chemistry. 74: 8452-5. PMID 19874068 DOI: 10.1021/Jo901682P  0.583
2009 Zhu J, Warren JD, Danishefsky SJ. Synthetic carbohydrate-based anticancer vaccines: the Memorial Sloan-Kettering experience. Expert Review of Vaccines. 8: 1399-413. PMID 19803761 DOI: 10.1586/Erv.09.95  0.561
2009 Jeon I, Lee D, Krauss IJ, Danishefsky SJ. A new model for the presentation of tumor-associated antigens and the quest for an anticancer vaccine: a solution to the synthesis challenge via ring-closing metathesis. Journal of the American Chemical Society. 131: 14337-44. PMID 19746915 DOI: 10.1021/Ja9052625  0.717
2009 Wang Z, Min SJ, Danishefsky SJ. Total synthesis and structural revision of (+/-)-tricholomalides A and B. Journal of the American Chemical Society. 131: 10848-9. PMID 19722666 DOI: 10.1021/Ja9049433  0.562
2009 Kim WH, Lee JH, Danishefsky SJ. Improved dienophilicity of nitrocycloalkenes: prospects for the development of a trans-Diels-Alder paradigm. Journal of the American Chemical Society. 131: 12576-8. PMID 19685875 DOI: 10.1021/Ja9058926  0.469
2009 Hayden AE, DeChancie J, George AH, Dai M, Yu M, Danishefsky SJ, Houk KN. Origins of the regioselectivities in the Diels-Alder reactions of vinylindenes with 1,4-quinone monoketal and acrolein dienophiles. The Journal of Organic Chemistry. 74: 6770-6. PMID 19663431 DOI: 10.1021/Jo901473H  0.538
2009 Nagorny P, Kim WH, Wan Q, Lee D, Danishefsky SJ. On the emerging role of chemistry in the fashioning of biologics: synthesis of a bidomainal fucosyl GM1-based vaccine for the treatment of small cell lung cancer. The Journal of Organic Chemistry. 74: 5157-62. PMID 19555091 DOI: 10.1021/Jo900918M  0.674
2009 Zhu J, Wan Q, Lee D, Yang G, Spassova MK, Ouerfelli O, Ragupathi G, Damani P, Livingston PO, Danishefsky SJ. From synthesis to biologics: preclinical data on a chemistry derived anticancer vaccine. Journal of the American Chemical Society. 131: 9298-303. PMID 19518111 DOI: 10.1021/Ja901415S  0.597
2009 Nagorny P, Fasching B, Li X, Chen G, Aussedat B, Danishefsky SJ. Toward fully synthetic homogeneous beta-human follicle-stimulating hormone (beta-hFSH) with a biantennary N-linked dodecasaccharide. synthesis of beta-hFSH with chitobiose units at the natural linkage sites. Journal of the American Chemical Society. 131: 5792-9. PMID 19341309 DOI: 10.1021/Ja809554X  0.716
2009 Tan Z, Shang S, Halkina T, Yuan Y, Danishefsky SJ. Toward homogeneous erythropoietin: non-NCL-based chemical synthesis of the Gln78-Arg166 glycopeptide domain. Journal of the American Chemical Society. 131: 5424-31. PMID 19334683 DOI: 10.1021/Ja808704M  0.49
2009 Kan C, Trzupek JD, Wu B, Wan Q, Chen G, Tan Z, Yuan Y, Danishefsky SJ. Toward homogeneous erythropoietin: chemical synthesis of the Ala1-Gly28 glycopeptide domain by "alanine" ligation. Journal of the American Chemical Society. 131: 5438-43. PMID 19334679 DOI: 10.1021/Ja808707W  0.722
2009 Lee LS, Stephenson KK, Fahey JW, Parsons TL, Lietman PS, Andrade AS, Lei X, Yun H, Soon GH, Shen P, Danishefsky S, Flexner C. Induction of chemoprotective phase 2 enzymes by ginseng and its components. Planta Medica. 75: 1129-33. PMID 19326326 DOI: 10.1055/S-0029-1185508  0.473
2009 Zhu J, Wan Q, Ragupathi G, George CM, Livingston PO, Danishefsky SJ. Biologics through chemistry: total synthesis of a proposed dual-acting vaccine targeting ovarian cancer by orchestration of oligosaccharide and polypeptide domains. Journal of the American Chemical Society. 131: 4151-8. PMID 19253940 DOI: 10.1021/Ja810147J  0.572
2009 Dai M, Danishefsky SJ. An oxidative dearomatization cyclization model for cortistatin A Heterocycles. 77: 157-161. DOI: 10.3987/Com-08-S(F)6  0.422
2008 Lei X, Danishefsky SJ. Efficient Synthesis of a Novel Resorcyclide as Anticancer Agent Based on Hsp90 Inhibition. Advanced Synthesis & Catalysis. 350: 1677-1681. PMID 21442009 DOI: 10.1002/Adsc.200800187  0.35
2008 Ng F, Yun H, Lei X, Danishefsky SJ, Fahey J, Stephenson K, Flexner C, Lee L. (3R, 9R, 10R)-Panaxytriol: A molecular-based nutraceutical with possible application to cancer prevention and treatment. Tetrahedron Letters. 49: 7178-7179. PMID 20011028 DOI: 10.1016/J.Tetlet.2008.09.169  0.485
2008 Dai M, Wang Z, Danishefsky SJ. A novel α,β-unsaturated nitrone-aryne [3+2] cycloaddition and its application in the synthesis of the cortistatin core. Tetrahedron Letters. 49: 6613-6616. PMID 19924220 DOI: 10.1016/J.Tetlet.2008.09.019  0.654
2008 Dai M, Danishefsky SJ. A concise synthesis of the cortistatin core. Tetrahedron Letters. 49: 6610-6612. PMID 19924219 DOI: 10.1016/J.Tetlet.2008.09.018  0.53
2008 Lei X, Dai M, Hua Z, Danishefsky SJ. Biomimetic total synthesis of tricycloillicinone and mechanistic studies toward the rearrangement of prenyl phenyl ethers. Tetrahedron Letters. 49: 6383-6385. PMID 19890380 DOI: 10.1016/J.Tetlet.2008.07.184  0.581
2008 Polara A, Cook SP, Danishefsky SJ. Multiple chirality transfers in the enantioselective synthesis of 11-O-debenzoyltashironin. Chiroptical analysis of the key cascade. Tetrahedron Letters. 49: 5906-5908. PMID 19812682 DOI: 10.1016/J.Tetlet.2008.07.139  0.702
2008 Wright BJ, Hartung J, Peng F, Van de Water R, Liu H, Tan QH, Chou TC, Danishefsky SJ. Synthesis of pluraflavin A "aglycone". Journal of the American Chemical Society. 130: 16786-90. PMID 19049469 DOI: 10.1021/Ja805936V  0.8
2008 Dai M, Krauss IJ, Danishefsky SJ. Total synthesis of spirotenuipesines A and B. The Journal of Organic Chemistry. 73: 9576-83. PMID 18973385 DOI: 10.1021/Jo8016814  0.764
2008 Wan Q, Chen J, Yuan Y, Danishefsky SJ. Oxo-ester mediated native chemical ligation: concept and applications. Journal of the American Chemical Society. 130: 15814-6. PMID 18855357 DOI: 10.1021/Ja804993Y  0.531
2008 Joyce JG, Krauss IJ, Song HC, Opalka DW, Grimm KM, Nahas DD, Esser MT, Hrin R, Feng M, Dudkin VY, Chastain M, Shiver JW, Danishefsky SJ. An oligosaccharide-based HIV-1 2G12 mimotope vaccine induces carbohydrate-specific antibodies that fail to neutralize HIV-1 virions. Proceedings of the National Academy of Sciences of the United States of America. 105: 15684-9. PMID 18838688 DOI: 10.1073/Pnas.0807837105  0.683
2008 Chen J, Wan Q, Yuan Y, Zhu J, Danishefsky SJ. Native chemical ligation at valine: a contribution to peptide and glycopeptide synthesis. Angewandte Chemie (International Ed. in English). 47: 8521-4. PMID 18833563 DOI: 10.1002/Anie.200803523  0.652
2008 Li X, Danishefsky SJ. Noncatalytic reaction of isonitriles and carboxylic acids en route to amide-type linkages. Nature Protocols. 3: 1666-70. PMID 18833204 DOI: 10.1038/Nprot.2008.153  0.317
2008 Angeles AR, Waters SP, Danishefsky SJ. Total syntheses of (+)- and (-)-peribysin E. Journal of the American Chemical Society. 130: 13765-70. PMID 18783227 DOI: 10.1021/Ja8048207  0.786
2008 Li X, Yuan Y, Kan C, Danishefsky SJ. Addressing mechanistic issues in the coupling of isonitriles and carboxylic acids: potential routes to peptidic constructs. Journal of the American Chemical Society. 130: 13225-7. PMID 18783225 DOI: 10.1021/Ja804709S  0.376
2008 Jones GO, Li X, Hayden AE, Houk KN, Danishefsky SJ. The coupling of isonitriles and carboxylic acids occurring by sequential concerted rearrangement mechanisms. Organic Letters. 10: 4093-6. PMID 18707109 DOI: 10.1021/Ol8016287  0.302
2008 Li X, Danishefsky SJ. New chemistry with old functional groups: on the reaction of isonitriles with carboxylic acids--a route to various amide types. Journal of the American Chemical Society. 130: 5446-8. PMID 18370392 DOI: 10.1021/Ja800612R  0.318
2008 Wright BJ, Chan C, Danishefsky SJ. Synthesis and cytotoxic evaluation of some cribrostatin-ecteinascidin analogues. Journal of Natural Products. 71: 409-14. PMID 18278868 DOI: 10.1021/Np800022X  0.617
2008 Yu M, Danishefsky SJ. A direct route to fluostatin C by a fascinating Diels-Alder reaction. Journal of the American Chemical Society. 130: 2783-5. PMID 18254631 DOI: 10.1021/Ja7113757  0.331
2008 Tsukano C, Siegel DR, Danishefsky SJ. Synthesis of Nemorosone and Clusianone Synfacts. 2008: 337-337. DOI: 10.1055/S-2008-1042888  0.691
2007 Wan Q, Danishefsky SJ. Free-radical-based, specific desulfurization of cysteine: a powerful advance in the synthesis of polypeptides and glycopolypeptides. Angewandte Chemie (International Ed. in English). 46: 9248-52. PMID 18046687 DOI: 10.1002/Anie.200704195  0.412
2007 Tsukano C, Siegel DR, Danishefsky SJ. Differentiation of nonconventional "carbanions"-the total synthesis of nemorosone and clusianone. Angewandte Chemie (International Ed. in English). 46: 8840-4. PMID 17935090 DOI: 10.1002/Anie.200703886  0.66
2007 Chen G, Wan Q, Tan Z, Kan C, Hua Z, Ranganathan K, Danishefsky SJ. Development of efficient methods for accomplishing cysteine-free peptide and glycopeptide coupling. Angewandte Chemie (International Ed. in English). 46: 7383-7. PMID 17828726 DOI: 10.1002/Anie.200702865  0.679
2007 Krauss IJ, Joyce JG, Finnefrock AC, Song HC, Dudkin VY, Geng X, Warren JD, Chastain M, Shiver JW, Danishefsky SJ. Fully synthetic carbohydrate HIV antigens designed on the logic of the 2G12 antibody. Journal of the American Chemical Society. 129: 11042-4. PMID 17711286 DOI: 10.1021/Ja074804R  0.748
2007 Velthuisen EJ, Danishefsky SJ. Total synthesis of (+)-suaveolindole: establishment of its absolute configuration. Journal of the American Chemical Society. 129: 10640-1. PMID 17696355 DOI: 10.1021/Ja075100K  0.82
2007 Krauss IJ, Mandal M, Danishefsky SJ. Total synthesis of (+)-isomigrastatin. Angewandte Chemie (International Ed. in English). 46: 5576-9. PMID 17583888 DOI: 10.1002/Anie.200701837  0.751
2007 Angeles AR, Dorn DC, Kou CA, Moore MA, Danishefsky SJ. Total synthesis of peribysin E necessitates revision of the assignment of its absolute configuration. Angewandte Chemie (International Ed. in English). 46: 1451-4. PMID 17387656 DOI: 10.1002/Anie.200604308  0.778
2007 Li C, Chan C, Heimann AC, Danishefsky SJ. Total synthesis of phalarine. Angewandte Chemie (International Ed. in English). 46: 1448-50. PMID 17387655 DOI: 10.1002/anie.200604072  0.711
2007 Li C, Chan C, Heimann AC, Danishefsky SJ. On the rearrangement of an azaspiroindolenine to a precursor to phalarine: mechanistic insights. Angewandte Chemie (International Ed. in English). 46: 1444-7. PMID 17387654 DOI: 10.1002/Anie.200604071  0.698
2007 Dai M, Danishefsky SJ. The total synthesis of spirotenuipesines A and B. Journal of the American Chemical Society. 129: 3498-9. PMID 17335213 DOI: 10.1021/ja069164r  0.47
2007 Min SJ, Danishefsky SJ. Total synthesis of paecilomycine A. Angewandte Chemie (International Ed. in English). 46: 2199-202. PMID 17300126 DOI: 10.1002/Anie.200605058  0.301
2007 Dai M, Sarlah D, Yu M, Danishefsky SJ, Jones GO, Houk KN. Highly selective Diels-Alder reactions of directly connected enyne dienophiles. Journal of the American Chemical Society. 129: 645-57. PMID 17227028 DOI: 10.1021/Ja065762U  0.697
2007 Wilson RM, Danishefsky SJ. Promising agents at the interface of biology and oncology derived through chemical synthesis Pure and Applied Chemistry. 79: 2189-2216. DOI: 10.1351/Pac200779122189  0.343
2007 Danishefsky S, Angeles A, Dorn D, Kou C, Moore M. Synthesis of ent-Peribysin E Synfacts. 2007: 0678-0678. DOI: 10.1055/S-2007-968601  0.784
2007 Maloney DJ, Danishefsky SJ. Studies toward the total synthesis of grandisine a: Synthesis of 9-epi-grandisine A Heterocycles. 72: 167-174.  0.313
2006 Chen J, Chen G, Wu B, Wan Q, Tan Z, Hua Z, Danishefsky SJ. Mature Homogeneous Erythropoietin-Level Building Blocks by Chemical Synthesis: The EPO 114-166 Glycopeptide Domain, Presenting the O-Linked Glycophorin. Tetrahedron Letters. 47: 8013-8016. PMID 17426819 DOI: 10.1016/J.Tetlet.2006.09.045  0.696
2006 Cook SP, Polara A, Danishefsky SJ. The total synthesis of (+/-)-11-O-debenzoyltashironin. Journal of the American Chemical Society. 128: 16440-1. PMID 17177359 DOI: 10.1021/Ja0670254  0.681
2006 Cook SP, Danishefsky SJ. An interesting issue of Diels-Alder selectivity discovered en route to 11-O-debenzoyltashironin. Organic Letters. 8: 5693-5. PMID 17134249 DOI: 10.1021/Ol062067I  0.569
2006 Yoshino T, Ng F, Danishefsky SJ. A total synthesis of xestodecalactone a and proof of its absolute stereochemistry: interesting observations on dienophilic control with 1,3-disubstituted nonequivalent allenes. Journal of the American Chemical Society. 128: 14185-91. PMID 17061903 DOI: 10.1021/Ja064270E  0.416
2006 Wan Q, Chen J, Chen G, Danishefsky SJ. A potentially valuable advance in the synthesis of carbohydrate-based anticancer vaccines through extended cycloaddition chemistry. The Journal of Organic Chemistry. 71: 8244-9. PMID 17025318 DOI: 10.1021/Jo061406I  0.627
2006 Chen G, Warren JD, Chen J, Wu B, Wan Q, Danishefsky SJ. Studies related to the relative thermodynamic stability of C-terminal peptidyl esters of O-hydroxy thiophenol: emergence of a doable strategy for non-cysteine ligation applicable to the chemical synthesis of glycopeptides. Journal of the American Chemical Society. 128: 7460-2. PMID 16756298 DOI: 10.1021/Ja061588Y  0.73
2006 Wu B, Chen J, Warren JD, Chen G, Hua Z, Danishefsky SJ. Building complex glycopeptides: Development of a cysteine-free native chemical ligation protocol. Angewandte Chemie (International Ed. in English). 45: 4116-25. PMID 16710874 DOI: 10.1002/anie.200600538  0.611
2006 Cheong PH, Yun H, Danishefsky SJ, Houk KN. Torsional steering controls the stereoselectivity of epoxidation in the guanacastepene a synthesis. Organic Letters. 8: 1513-6. PMID 16597098 DOI: 10.1021/Ol052862G  0.594
2006 Zheng S, Chan C, Furuuchi T, Wright BJ, Zhou B, Guo J, Danishefsky SJ. Stereospecific formal total synthesis of ecteinascidin 743. Angewandte Chemie (International Ed. in English). 45: 1754-9. PMID 16496274 DOI: 10.1002/Anie.200503983  0.819
2006 Chan C, Zheng S, Zhou B, Guo J, Heid RM, Wright BJ, Danishefsky SJ. The solution to a deep stereochemical conundrum: studies toward the tetrahydroisoquinoline alkaloids. Angewandte Chemie (International Ed. in English). 45: 1749-54. PMID 16496273 DOI: 10.1002/Anie.200503982  0.749
2006 Ragupathi G, Koide F, Livingston PO, Cho YS, Endo A, Wan Q, Spassova MK, Keding SJ, Allen J, Ouerfelli O, Wilson RM, Danishefsky SJ. Preparation and evaluation of unimolecular pentavalent and hexavalent antigenic constructs targeting prostate and breast cancer: a synthetic route to anticancer vaccine candidates. Journal of the American Chemical Society. 128: 2715-25. PMID 16492059 DOI: 10.1021/Ja057244+  0.501
2006 Liu H, Siegel DR, Danishefsky SJ. Studies directed toward the synthesis of terreulactone A: rapid construction of the A, B, C rings. Organic Letters. 8: 423-5. PMID 16435850 DOI: 10.1021/Ol052618P  0.643
2006 Siegel DR, Danishefsky SJ. Total synthesis of garsubellin A. Journal of the American Chemical Society. 128: 1048-9. PMID 16433500 DOI: 10.1021/Ja057418N  0.645
2006 Carcache DA, Cho YS, Hua Z, Tian Y, Li YM, Danishefsky SJ. Total synthesis of (+/-)-jiadifenin and studies directed to understanding its SAR: probing mechanistic and stereochemical issues in palladium-mediated allylation of enolate-like structures. Journal of the American Chemical Society. 128: 1016-22. PMID 16417394 DOI: 10.1021/Ja056980A  0.376
2006 Lambert TH, Danishefsky SJ. Total synthesis of UCS1025A. Journal of the American Chemical Society. 128: 426-7. PMID 16402826 DOI: 10.1021/Ja0574567  0.643
2006 Chan C, Danishefsky SJ. Synthetic studies toward cribrostatin IV: An intriguing epimerization Heterocycles. 70: 113-118. DOI: 10.3987/Com-06-S(W)35  0.326
2006 Danishefsky S, Zheng S, Chan C, Furuuchi T, Wright B, Zhou B, Guo J. Synthesis of Ecteinascidin 743 Synfacts. 2006: 0755-0755. DOI: 10.1055/S-2006-941932  0.793
2006 Danishefsky S, Lambert T. Synthesis of UCS1025A Synfacts. 2006: 0536-0536. DOI: 10.1055/S-2006-934495  0.686
2006 Wu B, Tan Z, Chen G, Chen J, Hua Z, Wan Q, Ranganathan K, Danishefsky SJ. Mature homogeneous erythropoietin building blocks by chemical synthesis: the EPO 22-37 glycopeptide domain presenting the full N-linked dodecasaccharide Tetrahedron Letters. 47: 8009-8011. DOI: 10.1016/J.Tetlet.2006.09.050  0.644
2006 Yun H, Gagnon A, Danishefsky SJ. Toward the synthesis of xestocyclamine A: investigation of double Michael reaction and direct aza Diels-Alder reaction Tetrahedron Letters. 47: 5311-5315. DOI: 10.1016/J.Tetlet.2006.05.126  0.709
2006 Wu B, Hua Z, Warren JD, Ranganathan K, Wan Q, Chen G, Tan Z, Chen J, Endo A, Danishefsky SJ. Synthesis of the fucosylated biantennary N-glycan of erythropoietin Tetrahedron Letters. 47: 5577-5579. DOI: 10.1016/J.Tetlet.2006.05.086  0.772
2006 Chan C, Li C, Zhang F, Danishefsky SJ. Studies toward the total synthesis of phalarine: a survey of some biomimetic possibilities Tetrahedron Letters. 47: 4839-4841. DOI: 10.1016/J.Tetlet.2006.05.041  0.514
2006 Wu B, Warren JD, Chen J, Chen G, Hua Z, Danishefsky SJ. Reiterative cysteine-based coupling leading to complex, homogeneous glycopeptides Tetrahedron Letters. 47: 5219-5223. DOI: 10.1016/J.Tetlet.2006.04.132  0.498
2006 Chen J, Warren JD, Wu B, Chen G, Wan Q, Danishefsky SJ. A route to cyclic peptides and glycopeptides by native chemical ligation using in situ derived thioesters Tetrahedron Letters. 47: 1969-1972. DOI: 10.1016/J.Tetlet.2006.01.077  0.734
2006 Wang ZG, Warren JD, Dudkin VY, Zhang X, Iserloh U, Visser M, Eckhardt M, Seeberger PH, Danishefsky SJ. A highly convergent synthesis of an N-linked glycopeptide presenting the H-type 2 human blood group determinant Tetrahedron. 62: 4954-4978. DOI: 10.1016/J.Tet.2006.02.080  0.678
2005 Mandal M, Yun H, Dudley GB, Lin S, Tan DS, Danishefsky SJ. Total synthesis of guanacastepene a: a route to enantiomeric control. The Journal of Organic Chemistry. 70: 10619-37. PMID 16355979 DOI: 10.1021/Jo051470K  0.81
2005 Yun H, Chou TC, Dong H, Tian Y, Li YM, Danishefsky SJ. Total synthesis as a resource in drug discovery: the first in vivo evaluation of panaxytriol and its derivatives. The Journal of Organic Chemistry. 70: 10375-80. PMID 16323847 DOI: 10.1021/Jo0515475  0.562
2005 Hua Z, Carcache DA, Tian Y, Li YM, Danishefsky SJ. The synthesis and preliminary biological evaluation of a novel steroid with neurotrophic activity: NGA0187. The Journal of Organic Chemistry. 70: 9849-56. PMID 16292815 DOI: 10.1021/Jo051556D  0.386
2005 Ouerfelli O, Warren JD, Wilson RM, Danishefsky SJ. Synthetic carbohydrate-based antitumor vaccines: challenges and opportunities. Expert Review of Vaccines. 4: 677-85. PMID 16221069 DOI: 10.1586/14760584.4.5.677  0.433
2005 Cho YS, Wan Q, Danishefsky SJ. Organic synthesis in pursuit of immunology: large-scale synthesis of peracetylated GM2 glycosylamino acid for preparation of a multiantigenic prostate cancer vaccine. Bioorganic & Medicinal Chemistry. 13: 5259-66. PMID 16006132 DOI: 10.1016/J.Bmc.2005.06.018  0.521
2005 Rivkin A, Chou TC, Danishefsky SJ. On the remarkable antitumor properties of fludelone: how we got there. Angewandte Chemie (International Ed. in English). 44: 2838-50. PMID 15880547 DOI: 10.1002/Anie.200461751  0.332
2005 Chou TC, Guan Y, Soenen DR, Danishefsky SJ, Boger DL. Potent reversal of multidrug resistance by ningalins and its use in drug combinations against human colon carcinoma xenograft in nude mice. Cancer Chemotherapy and Pharmacology. 56: 379-90. PMID 15875185 DOI: 10.1007/S00280-005-1019-Y  0.317
2005 Chan C, Heid R, Zheng S, Guo J, Zhou B, Furuuchi T, Danishefsky SJ. Total synthesis of cribrostatin IV: fine-tuning the character of an amide bond by remote control. Journal of the American Chemical Society. 127: 4596-8. PMID 15796524 DOI: 10.1021/Ja050203T  0.815
2005 Shan D, Chen L, Njardarson JT, Gaul C, Ma X, Danishefsky SJ, Huang XY. Synthetic analogues of migrastatin that inhibit mammary tumor metastasis in mice. Proceedings of the National Academy of Sciences of the United States of America. 102: 3772-6. PMID 15728385 DOI: 10.1073/Pnas.0500658102  0.558
2005 Meng Z, Danishefsky SJ. A synthetic pathway to either enantiomer of merrilactone A. Angewandte Chemie (International Ed. in English). 44: 1511-3. PMID 15690391 DOI: 10.1002/Anie.200462509  0.489
2005 Kagan E, Ragupathi G, Yi SS, Reis CA, Gildersleeve J, Kahne D, Clausen H, Danishefsky SJ, Livingston PO. Comparison of antigen constructs and carrier molecules for augmenting the immunogenicity of the monosaccharide epithelial cancer antigen Tn. Cancer Immunology, Immunotherapy : Cii. 54: 424-30. PMID 15625606 DOI: 10.1007/S00262-004-0584-Y  0.496
2005 Yun H, Meng Z, Danishefsky SJ. Enantiotopic synthesis of natural products: Merrilactone and guanacastepene Heterocycles. 66: 711-725. DOI: 10.3987/REV-05-SR(K)2  0.635
2005 Cho YS, Wu KD, Moore MAS, Chou TC, Danishefsky SJ. Second-generation epothilones: Discovery of fludelone and its extraordinary antitumor properties Drugs of the Future. 30: 737-745. DOI: 10.1358/Dof.2005.030.07.895806  0.334
2005 Wan Q, Young SC, Lambert TH, Danishefsky SJ. Olefin cross-metathesis: A powerful tool for constructing vaccines composed of multimeric antigens Journal of Carbohydrate Chemistry. 24: 425-440. DOI: 10.1081/Car-200066992  0.682
2005 Chan C, Heid R, Zheng S, Guo J, Zhou B, Furuuchi T, Danishefsky SJ. Total Synthesis of Cribrostatin IV:  Fine-Tuning the Character of an Amide Bond by Remote Control   [J. Am. Chem. Soc.2005,127, 4596−4598].  Journal of the American Chemical Society. 127: 7262-7262. DOI: 10.1021/Ja059909D  0.787
2005 Yun H, Danishefsky SJ. A protocol to accomplish 'homo-Robinson' annulation: Application to the guanacastepene problem Tetrahedron Letters. 46: 3879-3882. DOI: 10.1016/J.Tetlet.2005.03.191  0.553
2005 Cook SP, Christoph G, Danishefsky SJ. En route to the total synthesis of tashironin: On the exercise of stereochemical control by a methyl group in mediating remote cyclization reactions Tetrahedron Letters. 46: 843-847. DOI: 10.1016/J.Tetlet.2004.11.148  0.628
2005 Endo A, Danishefsky SJ. Total Synthesis of Salinosporamide A (I). Cheminform. 36. DOI: 10.1002/chin.200544233  0.301
2004 Gaul C, Njardarson JT, Shan D, Dorn DC, Wu KD, Tong WP, Huang XY, Moore MA, Danishefsky SJ. The migrastatin family: discovery of potent cell migration inhibitors by chemical synthesis. Journal of the American Chemical Society. 126: 11326-37. PMID 15355116 DOI: 10.1021/Ja048779Q  0.679
2004 Rivkin A, Yoshimura F, Gabarda AE, Cho YS, Chou TC, Dong H, Danishefsky SJ. Discovery of (E)-9,10-dehydroepothilones through chemical synthesis: on the emergence of 26-trifluoro-(E)-9,10-dehydro-12,13-desoxyepothilone B as a promising anticancer drug candidate. Journal of the American Chemical Society. 126: 10913-22. PMID 15339176 DOI: 10.1021/Ja046992G  0.341
2004 Warren JD, Miller JS, Keding SJ, Danishefsky SJ. Toward fully synthetic glycoproteins by ultimately convergent routes: a solution to a long-standing problem. Journal of the American Chemical Society. 126: 6576-8. PMID 15161285 DOI: 10.1021/ja0491836  0.511
2004 Njardarson JT, Gaul C, Shan D, Huang XY, Danishefsky SJ. Discovery of potent cell migration inhibitors through total synthesis: lessons from structure-activity studies of (+)-migrastatin. Journal of the American Chemical Society. 126: 1038-40. PMID 14746469 DOI: 10.1021/Ja039714A  0.641
2004 Dudkin VY, Miller JS, Danishefsky SJ. Chemical synthesis of normal and transformed PSA glycopeptides. Journal of the American Chemical Society. 126: 736-8. PMID 14733546 DOI: 10.1021/Ja037988S  0.303
2004 Geng X, Yang ZQ, Danishefsky SJ. Synthetic development of radicicol and cycloproparadicicol: Highly promising anticancer agents targeting Hsp90 Synlett. 1325-1333. DOI: 10.1055/S-2004-829052  0.327
2004 Mandal M, Danishefsky SJ. Probing the formation and chemistry of enoxyoxirane derivatives in the C-ring en route to guanacastepene Tetrahedron Letters. 45: 3831-3833. DOI: 10.1016/J.Tetlet.2004.02.162  0.31
2004 Mandal M, Danishefsky SJ. Probing competitive pathways in building a hydroazulene moiety by reductive cyclization Tetrahedron Letters. 45: 3827-3829. DOI: 10.1016/J.Tetlet.2004.02.161  0.31
2003 Slovin SF, Ragupathi G, Musselli C, Olkiewicz K, Verbel D, Kuduk SD, Schwarz JB, Sames D, Danishefsky S, Livingston PO, Scher HI. Fully synthetic carbohydrate-based vaccines in biochemically relapsed prostate cancer: clinical trial results with alpha-N-acetylgalactosamine-O-serine/threonine conjugate vaccine. Journal of Clinical Oncology : Official Journal of the American Society of Clinical Oncology. 21: 4292-8. PMID 14645418 DOI: 10.1200/JCO.2003.04.112  0.662
2003 Siu T, Cox CD, Danishefsky SJ. Total synthesis of lactonamycinone. Angewandte Chemie (International Ed. in English). 42: 5629-34. PMID 14639735 DOI: 10.1002/Anie.200352592  0.576
2003 Cox CD, Siu T, Danishefsky SJ. Studies directed toward the total synthesis of lactonamycin: control of the sense of cycloaddition of a quinone through directed intramolecular catalysis. Angewandte Chemie (International Ed. in English). 42: 5625-9. PMID 14639734 DOI: 10.1002/Anie.200352591  0.548
2003 Yamamoto K, Hentemann MF, Allen JG, Danishefsky SJ. On the total synthesis and determination of the absolute configuration of rishirilide B: exploitation of subtle effects to control the sense of cycloaddition of o-quinodimethides. Chemistry (Weinheim An Der Bergstrasse, Germany). 9: 3242-52. PMID 12866068 DOI: 10.1002/Chem.200304931  0.382
2003 Gaul C, Njardarson JT, Danishefsky SJ. The total synthesis of (+)-migrastatin. Journal of the American Chemical Society. 125: 6042-3. PMID 12785819 DOI: 10.1021/Ja0349103  0.654
2003 Yun H, Danishefsky SJ. Straightforward synthesis of panaxytriol: an active component of Red Ginseng. The Journal of Organic Chemistry. 68: 4519-22. PMID 12762760 DOI: 10.1021/Jo0341665  0.515
2003 Zhang X, Houk KN, Lin S, Danishefsky SJ. Mechanism of cis-enamide formation from N-(alpha-silyl)allyl amides: synthetic potential of stepwise dyotropic rearrangements. Journal of the American Chemical Society. 125: 5111-4. PMID 12708862 DOI: 10.1021/Ja029576+  0.317
2003 Coltart DM, Danishefsky SJ. Novel synthetic approach to the 8,10-dimethyl anti-syn-anti-perhydrophenanthrene skeleton. Organic Letters. 5: 1289-92. PMID 12688741 DOI: 10.1021/Ol034213F  0.639
2003 Yamamoto K, Garbaccio RM, Stachel SJ, Solit DB, Chiosis G, Rosen N, Danishefsky SJ. Total synthesis as a resource in the discovery of potentially valuable antitumor agents: cycloproparadicicol. Angewandte Chemie (International Ed. in English). 42: 1280-4. PMID 12645064 DOI: 10.1002/Anie.200390329  0.321
2003 Rivkin A, Yoshimura F, Gabarda AE, Chou TC, Dong H, Tong WP, Danishefsky SJ. Complex target-oriented total synthesis in the drug discovery process: the discovery of a highly promising family of second generation epothilones. Journal of the American Chemical Society. 125: 2899-901. PMID 12617656 DOI: 10.1021/Ja029695P  0.356
2003 Ng FW, Lin H, Chiu P, Danishefsky SJ. Explorations in Organic Chemistry Leading to the Total Synthesis of (±)-Gelsemine [J. Am. Chem. Soc. 2002, 124, 9812−9824]. Journal of the American Chemical Society. 125: 13303-13303. DOI: 10.1021/Ja0334558  0.5
2002 Zhang F, Danishefsky SJ. An efficient stereoselective total synthesis of DL-sesquicillin, a glucocorticoid antagonist. Angewandte Chemie (International Ed. in English). 41: 1434-7. PMID 19750790 DOI: 10.1002/1521-3773(20020415)41:8<1434::Aid-Anie1434>3.0.Co;2-A  0.441
2002 Gagnon A, Danishefsky SJ. Evaluation of Diene hierarchies for Diels--Alder reactions en route to xestocyclamine A: elaboration of an Ansa bridge by B-alkyl Suzuki macrocyclization. Angewandte Chemie (International Ed. in English). 41: 1581-4. PMID 19750672 DOI: 10.1002/1521-3773(20020503)41:9<1581::Aid-Anie1581>3.0.Co;2-F  0.582
2002 Lin S, Dudley GB, Tan DS, Danishefsky SJ. A stereoselective route to guanacastepene A through a surprising epoxidation. Angewandte Chemie (International Ed. in English). 41: 2188-91. PMID 19746640 DOI: 10.1002/1521-3773(20020617)41:12<2188::Aid-Anie2188>3.0.Co;2-J  0.779
2002 Tan DS, Dudley GB, Danishefsky SJ. Synthesis of the functionalized tricyclic skeleton of guanacastepene A: a tandem epoxide-opening beta-elimination/knoevenagel cyclization. Angewandte Chemie (International Ed. in English). 41: 2185-8. PMID 19746639 DOI: 10.1002/1521-3773(20020617)41:12<2185::Aid-Anie2185>3.0.Co;2-0  0.768
2002 Njardarson JT, Biswas K, Danishefsky SJ. Application of hitherto unexplored macrocyclization strategies in the epothilone series: novel epothilone analogs by total synthesis. Chemical Communications (Cambridge, England). 2759-61. PMID 12478733 DOI: 10.1039/B209941A  0.7
2002 Rivkin A, Biswas K, Chou TC, Danishefsky SJ. On the introduction of a trifluoromethyl substituent in the epothilone setting: chemical issues related to ring forming olefin metathesis and earliest biological findings. Organic Letters. 4: 4081-4. PMID 12423091 DOI: 10.1021/Ol0268283  0.377
2002 Rivkin A, Njardarson JT, Biswas K, Chou TC, Danishefsky SJ. Total syntheses of [17]- and [18]dehydrodesoxyepothilones B via a concise ring-closing metathesis-based strategy: correlation of ring size with biological activity in the epothilone series. The Journal of Organic Chemistry. 67: 7737-40. PMID 12398497 DOI: 10.1021/Jo0204294  0.63
2002 Chappell MD, Harris CR, Kuduk SD, Balog A, Wu Z, Zhang F, Lee CB, Stachel SJ, Danishefsky SJ, Chou TC, Guan Y. Probing the SAR of dEpoB via chemical synthesis: a total synthesis evaluation of C26-(1,3-dioxolanyl)-12,13-desoxyepothilone B. The Journal of Organic Chemistry. 67: 7730-6. PMID 12398496 DOI: 10.1021/Jo020180Q  0.507
2002 Ragupathi G, Coltart DM, Williams LJ, Koide F, Kagan E, Allen J, Harris C, Glunz PW, Livingston PO, Danishefsky SJ. On the power of chemical synthesis: immunological evaluation of models for multiantigenic carbohydrate-based cancer vaccines. Proceedings of the National Academy of Sciences of the United States of America. 99: 13699-704. PMID 12359877 DOI: 10.1073/Pnas.202427599  0.655
2002 Ujaque G, Lee PS, Houk KN, Hentemann MF, Danishefsky SJ. The origin of endo stereoselectivity in the hetero-Diels-Alder reactions of aldehydes with ortho-xylylenes: CH-pi, pi-pi, and steric effects on stereoselectivity. Chemistry (Weinheim An Der Bergstrasse, Germany). 8: 3423-30. PMID 12203322 DOI: 10.1002/1521-3765(20020802)8:15<3423::Aid-Chem3423>3.0.Co;2-X  0.305
2002 Coltart DM, Royyuru AK, Williams LJ, Glunz PW, Sames D, Kuduk SD, Schwarz JB, Chen XT, Danishefsky SJ, Live DH. Principles of mucin architecture: structural studies on synthetic glycopeptides bearing clustered mono-, di-, tri-, and hexasaccharide glycodomains. Journal of the American Chemical Society. 124: 9833-44. PMID 12175243 DOI: 10.1021/Ja020208F  0.787
2002 Biswas K, Lin H, Njardarson JT, Chappell MD, Chou TC, Guan Y, Tong WP, He L, Horwitz SB, Danishefsky SJ. Highly concise routes to epothilones: the total synthesis and evaluation of epothilone 490. Journal of the American Chemical Society. 124: 9825-32. PMID 12175242 DOI: 10.1021/Ja0262333  0.649
2002 Ng FW, Lin H, Chiu P, Danishefsky SJ. Explorations in organic chemistry leading to the total synthesis of (+/-)-gelsemine. Journal of the American Chemical Society. 124: 9812-24. PMID 12175241 DOI: 10.1021/ja0204675  0.498
2002 Ragupathi G, Deshpande PP, Coltart DM, Kim HM, Williams LJ, Danishefsky SJ, Livingston PO. Constructing an adenocarcinoma vaccine: immunization of mice with synthetic KH-1 nonasaccharide stimulates anti-KH-1 and anti-Le(y) antibodies. International Journal of Cancer. Journal International Du Cancer. 99: 207-12. PMID 11979435 DOI: 10.1002/Ijc.10305  0.657
2002 Birman VB, Danishefsky SJ. The total synthesis of (+/-)-merrilactone A. Journal of the American Chemical Society. 124: 2080-1. PMID 11878938 DOI: 10.1021/ja012495d  0.319
2002 Zhou B, Guo J, Danishefsky SJ. Studies directed to the total synthesis of ET 743 and analogues thereof: an expeditious route to the ABFGH subunit. Organic Letters. 4: 43-6. PMID 11772086 DOI: 10.1021/Ol016844K  0.561
2002 Garbaccio RM, Stachel SJ, Baeschlin DK, Danishefsky SJ. Concise asymmetric syntheses of radicicol and monocillin I. Journal of the American Chemical Society. 123: 10903-8. PMID 11686693 DOI: 10.1021/Ja011364+  0.371
2002 Danishefsky S, Schuda P, Kato K. Synthesis of vernolepin. Diels-Alder approach to the angularly functionalized AB system Cheminform. 7. PMID 1255288 DOI: 10.1021/Jo00869A001  0.352
2002 Gaul C, Danishefsky SJ. Synthesis of the macrolide core of migrastatin Tetrahedron Letters. 43: 9039-9042. DOI: 10.1016/S0040-4039(02)02281-5  0.412
2002 Dudley GB, Danishefsky SJ, Sukenick G. On the use of deuterium isotope effects in chemical synthesis Tetrahedron Letters. 43: 5605-5606. DOI: 10.1016/S0040-4039(02)01114-0  0.617
2002 Ng FW, Lin H, Tan Q, Danishefsky SJ. The synthesis of a key intermediate en route to gelsemine: a program based on intramolecular displacement of the carbonoxygen bond of a strategic oxetane Tetrahedron Letters. 43: 545-548. DOI: 10.1016/S0040-4039(01)02212-2  0.406
2002 Danishefsky S, Etheredge SJ, Dynak J, McCurry P. A Route To Furanoid Systems By Intramolecular Homoconjugate Addition Cheminform. 5. DOI: 10.1002/Chin.197450236  0.774
2002 Lin S, Dudley GB, Tan DS, Danishefsky SJ. A Stereoselective Route to Guanacastepene A through a Surprising Epoxidation This work was supported by the National Institutes of Health (CA-28824). S.L. is a US Army breast cancer research program postdoctoral fellow (DAMD-17-99-1-9373). G.B.D. is an NIH postdoctoral fellow (1 F32 NS11150-01). D.S.T. is a Damon Runyon Cancer Research Foundation postdoctoral fellow (DRG-1641). We thank Dr. George Sukenick and Sylvi Rusli (NMR Core Facility, CA-02848) for mass spectral analyses. Angewandte Chemie International Edition. 41: 2188. DOI: 10.1002/1521-3773(20020617)41:12<2188::AID-ANIE2188>3.0.CO;2-J  0.719
2002 Tan DS, Dudley GB, Danishefsky SJ. Synthesis of the Functionalized Tricyclic Skeleton of Guanacastepene A: A Tandem Epoxide-Opening β-Elimination/Knoevenagel Cyclization This work was supported by the National Institutes of Health (HL-25848 and CA-28824). D.S.T. is a Damon Runyon Cancer Research Foundation postdoctoral fellow (DRG-1641). G.B.D. is an NIH postdoctoral fellow (1 F32 NS11150-01). We thank Dr. George Sukenick and Sylvi Rusli (NMR Core Facility, CA-02848) for mass spectral analyses. Angewandte Chemie International Edition. 41: 2185. DOI: 10.1002/1521-3773(20020617)41:12<2185::AID-ANIE2185>3.0.CO;2-0  0.734
2002 Gagnon A, Danishefsky SJ. Evaluation of diene hierarchies for Diels-Alder reactions en route to xestocyclamine A: Elaboration of an ansa bridge by B-alkyl Suzuki macrocyclization Angewandte Chemie - International Edition. 41: 1581-1584. DOI: 10.1002/1521-3773(20020503)41:9<1581::AID-ANIE1581>3.0.CO;2-F  0.533
2002 Zhang F, Danishefsky SJ. An Efficient Stereoselective Total Synthesis of dl-Sesquicillin, a Glucocorticoid Antagonist This work was supported by the National Institutes of Health (Grant Number: HL25848). We thank Dr. Yashuiro Itagaki, Columbia University for high-resolution mass-spectral analysis. F.Z. would also like to thank Columbia University and Pharmacia & Upjohn for a graduate fellowship. Angewandte Chemie. 114: 1492. DOI: 10.1002/1521-3757(20020415)114:8<1492::Aid-Ange1492>3.0.Co;2-V  0.434
2001 Carson MW, Kim G, Hentemann MF, Trauner D, Danishefsky SJ. Concise Stereoselective Routes to Advanced Intermediates Related to Natural and Unnatural Pinnaic Acid This work was supported by the National Institutes of Health (Grant Numbers: CA28824). Postdoctoral Fellowship support is gratefully acknowledged by M.W.C. (U.S. Army BCRP, DAMD17-98-1-8154), M.F.H. (5T32 CA62948-05), and D.T. (Schering Research Foundation, Berlin). We thank Dr. George Sukenick of the MSKCC NMR Core Facility for NMR and mass spectral analyses. Angewandte Chemie (International Ed. in English). 40: 4450-4452. PMID 12404442 DOI: 10.1002/1521-3773(20011203)40:23<4450::AID-ANIE4450>3.0.CO;2-M  0.333
2001 Siu T, Qin D, Danishefsky SJ. The Total Synthesis of Heliquinomycinone This work was supported by the National Institutes of Health (Grant numbers: AI 16943 and HL25848). The authors thank Dr. Makoto Chino of Nippon Kayaku Co., Ltd. for kindly providing a sample of heliquinomycin, and Yashuiro Itagaki of Columbia University for high-resolution mass spectral analyses. Angewandte Chemie (International Ed. in English). 40: 4713-4716. PMID 12404392 DOI: 10.1002/1521-3773(20011217)40:24<4713::Aid-Anie4713>3.0.Co;2-N  0.519
2001 Qin D, Ren RX, Siu T, Zheng C, Danishefsky SJ. Studies in the Total Synthesis of Heliquinomycinone: Proof of Concept and Assembly of a Fully Mature Spirocyclization Precursor This work was supported by the National Institutes of Health (Grant numbers: AI 16943 and HL25848). A Postdoctoral Fellowship is gratefully acknowledged by R.X.R. (NIH, Grant Number IF32EY06750-0181). The authors thank Dr. Daniel Chen for important initial experiments, Dr. Brian Bridgewater and Prof. Ged Parkin of Columbia University for X-ray crystal structure analysis of 11 a, and Yashuiro Itagaki for high-resolution mass spectral analyses. Angewandte Chemie (International Ed. in English). 40: 4709-4713. PMID 12404391 DOI: 10.1002/1521-3773(20011217)40:24<4709::AID-ANIE4709>3.0.CO;2-Q  0.454
2001 Chemler SR, Trauner D, Danishefsky SJ. The B-Alkyl Suzuki-Miyaura Cross-Coupling Reaction: Development, Mechanistic Study, and Applications in Natural Product Synthesis A list of abbreviations can be found at the end of the article. Angewandte Chemie (International Ed. in English). 40: 4544-4568. PMID 12404358 DOI: 10.1002/1521-3773(20011217)40:24<4544::Aid-Anie4544>3.0.Co;2-N  0.684
2001 Chemler SR, Iserloh U, Danishefsky SJ. Enantioselective synthesis of the oxadecalin core of phomactin A via a highly stereoselective Diels-Alder reaction. Organic Letters. 3: 2949-51. PMID 11554815 DOI: 10.1021/Ol0161357  0.632
2001 Cox C, Danishefsky SJ. Concise synthesis of a lactonamycin model system by diastereoselective dihydroxylation of a highly functionalized naphthoquinone. Organic Letters. 3: 2899-902. PMID 11529785 DOI: 10.1021/Ol016361G  0.416
2001 Dudley GB, Danishefsky SJ. A four-step synthesis of the hydroazulene core of guanacastepene Organic Letters. 3: 2399-2402. PMID 11463326 DOI: 10.1021/Ol016222Z  0.631
2001 Allen JR, Harris CR, Danishefsky SJ. Pursuit of optimal carbohydrate-based anticancer vaccines: Preparation of a multiantigenic unimolecular glycopeptide containing the Tn, MBr1, and Lewisy antigens Journal of the American Chemical Society. 123: 1890-1897. PMID 11456809 DOI: 10.1021/Ja002779I  0.381
2001 Inoue M, Carson MW, Frontier AJ, Danishefsky SJ. Total synthesis and determination of the absolute configuration of frondosin B. Journal of the American Chemical Society. 123: 1878-89. PMID 11456808 DOI: 10.1021/Ja0021060  0.579
2001 Stachel SJ, Chul Bom Lee, Spassova M, Chappell MD, Bornmann WG, Danishefsky SJ, Chou TC, Guan Y. On the interactivity of complex synthesis and tumor pharmacology in the drug discovery process: Total synthesis and comparative in vivo evaluations of the 15-Aza epothilones Journal of Organic Chemistry. 66: 4369-4378. PMID 11397179 DOI: 10.1021/Jo010275C  0.348
2001 Qin D, Ren RX, Siu T, Zheng C, Danishefsky SJ. Studies in the Total Synthesis of Heliquinomycinone: Proof of Concept and Assembly of a Fully Mature Spirocyclization Precursor Angewandte Chemie. 113: 4845-4849. DOI: 10.1002/1521-3757(20011217)113:24<4845::Aid-Ange4845>3.0.Co;2-B  0.59
2001 Chemler SR, Trauner D, Danishefsky SJ. DieB-Alkyl-Suzuki-Miyaura-Kreuzkupplung: Entwicklung, Untersuchungen zum Mechanismus und Anwendungen in der Naturstoffsynthese Angewandte Chemie. 113: 4676-4701. DOI: 10.1002/1521-3757(20011217)113:24<4676::Aid-Ange4676>3.0.Co;2-B  0.666
2000 Wu Z, Zhang F, Danishefsky SJ. Subtle Variations in the Long-Range Transmission of Stereochemical Information: Matched and Mismatched Aldol Reactions This work was supported by the National Institutes of Health (Grant Nos. CA-28824 and HL-25848). Angewandte Chemie (International Ed. in English). 39: 4505-4508. PMID 11169651 DOI: 10.1002/1521-3773(20001215)39:24<4505::Aid-Anie4505>3.0.Co;2-2  0.401
2000 Danishefsky SJ, Inoue M, Trauner D. Synthesis of immunomodulatory marine natural products. Ernst Schering Research Foundation Workshop. 1-24. PMID 11077604 DOI: 10.1007/978-3-662-04042-3_1  0.424
2000 Garbaccio RM, Danishefsky SJ. Efficient asymmetric synthesis of radicicol dimethyl ether: a novel application of ring-forming olefin metathesis. Organic Letters. 2: 3127-9. PMID 11009362 DOI: 10.1021/Ol0063252  0.419
2000 Chemler SR, Danishefsky SJ. Transannular macrocyclization via intramolecular B-alkyl Suzuki reaction Organic Letters. 2: 2695-2698. PMID 10990430 DOI: 10.1021/Ol0062547  0.618
2000 Stachel SJ, Chappell MD, Lee CB, Danishefsky SJ, Chou TC, He L, Horwitz SB. On the total synthesis and preliminary biological evaluations of 15(R) and 15(S) aza-dEpoB: a Mitsunobu inversion at C15 in pre-epothilone fragments. Organic Letters. 2: 1637-9. PMID 10841498 DOI: 10.1021/Ol005932M  0.335
2000 Allen JR, Allen JG, Zhang XF, Williams LJ, Zatorski A, Ragupathi G, Livingston PO, Danishefsky SJ. A second generation synthesis of the MBr1 (globo-H) breast tumor antigen: new application of the n-pentenyl glycoside method for achieving complex carbohydrate protein linkages. Chemistry (Weinheim An Der Bergstrasse, Germany). 6: 1366-75. PMID 10840960 DOI: 10.1002/(Sici)1521-3765(20000417)6:8<1366::Aid-Chem1366>3.0.Co;2-K  0.332
2000 Martello LA, McDaid HM, Regl DL, Yang CP, Meng D, Pettus TR, Kaufman MD, Arimoto H, Danishefsky SJ, Smith AB, Horwitz SB. Taxol and discodermolide represent a synergistic drug combination in human carcinoma cell lines. Clinical Cancer Research : An Official Journal of the American Association For Cancer Research. 6: 1978-87. PMID 10815923  0.589
2000 Bhattacharya SK, Danishefsky SJ. A total synthesis of the methyl glycoside of ganglioside GM1 Journal of Organic Chemistry. 65: 144-151. PMID 10813908 DOI: 10.1021/Jo9912496  0.721
2000 Inoue M, Frontier AJ, Danishefsky SJ. The Total Synthesis of Frondosin B. Angewandte Chemie (International Ed. in English). 39: 761-764. PMID 10760861 DOI: 10.1002/(Sici)1521-3757(20000218)112:4<777::Aid-Ange777>3.0.Co;2-K  0.533
2000 Frontier AJ, Raghavan S, Danishefsky SJ. A highly stereoselective total synthesis of hispidospermidin: Derivation of a pharmacophore model Journal of the American Chemical Society. 122: 6151-6159. DOI: 10.1021/Ja9944960  0.609
2000 Allen JG, Hentemann aMF, Danishefsky SJ. A Powerful o-Quinone Dimethide Strategy for Intermolecular Diels−Alder Cycloadditions Journal of the American Chemical Society. 122: 571-575. DOI: 10.1021/Ja993627U  0.337
2000 Glunz PW, Hintermann S, Williams LJ, Schwarz JB, Kuduk SD, Kudryashov V, Lloyd KO, Danishefsky SJ. Design and Synthesis of Ley-Bearing Glycopeptides that Mimic Cell Surface LeyMucin Glycoprotein Architecture Journal of the American Chemical Society. 122: 7273-7279. DOI: 10.1021/Ja0011820  0.323
2000 Pettus TRR, Inoue M, Chen XT, Danishefsky SJ. A fully synthetic route the neurotrophic illicinones: Syntheses of tricycloillicinone and bicycloillicinone aldehyde Journal of the American Chemical Society. 122: 6160-6168. DOI: 10.1021/Ja000521M  0.381
2000 Zhou B, Guo J, Danishefsky SJ. A novel face specific Mannich closure providing access to the saframycin-ecteinascidin series of piperazine based alkaloids Tetrahedron Letters. 41: 2043-2046. DOI: 10.1016/S0040-4039(00)00106-4  0.468
2000 Zhou B, Edmondson S, Padron J, Danishefsky SJ. Synthetic explorations in the saframycin-ecteinascidin series: Construction of major chiral subunits through catalytic asymmetric induction Tetrahedron Letters. 41: 2039-2042. DOI: 10.1016/S0040-4039(00)00105-2  0.508
2000 Trauner D, Churchill D, Danishefsky S. On the Conformations of Halichlorine and the Pinnaic Acids: Nitrogen Inversion as a Possible Determinant of Biological Profile Helvetica Chimica Acta. 83: 2344-2351. DOI: 10.1002/1522-2675(20000906)83:9<2344::Aid-Hlca2344>3.0.Co;2-2  0.474
2000 Allen JR, Danishefsky SJ. Synthesis of Non-NaturalO-Glycosylamino Acids Derived fromn-Pentenyl Glycosides; Model Studies and Proof of Principle for Glycopeptide Synthesis Journal Fur Praktische Chemie-Chemiker-Zeitung. 342: 736-744. DOI: 10.1002/1521-3897(200010)342:8<736::Aid-Prac736>3.0.Co;2-#  0.408
1999 Ragupathi G, Slovin SF, Adluri S, Sames D, Kim IJ, Kim HM, Spassova M, Bornmann WG, Lloyd KO, Scher HI, Livingston PO, Danishefsky SJ. A Fully Synthetic Globo H Carbohydrate Vaccine Induces a Focused Humoral Response in Prostate Cancer Patients: A Proof of Principle. Angewandte Chemie (International Ed. in English). 38: 563-566. PMID 29711780 DOI: 10.1002/(Sici)1521-3773(19990215)38:4<563::Aid-Anie563>3.0.Co;2-3  0.674
1999 Meng D, Danishefsky SJ. Stereospecific Sulfur-Mediated Cleavage of a Spirocyclobutanone: Synthesis of a Fully Functional Precursor to the CP Compounds. Angewandte Chemie (International Ed. in English). 38: 1485-1488. PMID 29711567 DOI: 10.1002/(Sici)1521-3773(19990517)38:10<1485::Aid-Anie1485>3.0.Co;2-1  0.373
1999 Trauner D, Schwarz JB, Danishefsky SJ. Total Synthesis of (+)-Halichlorine: An Inhibitor of VCAM-1 Expression. Angewandte Chemie (International Ed. in English). 38: 3542-3545. PMID 10602236 DOI: 10.1002/(Sici)1521-3773(19991203)38:23<3542::Aid-Anie3542>3.0.Co;2-I  0.458
1999 Meng D, Tan Q, Danishefsky SJ. Discovery Through Total Synthesis-Epimerization at C7 in the CP Compounds: Is (7S)-CP-263,114 a Fermentation Product? Angewandte Chemie. 38: 3197-3201. PMID 10556901 DOI: 10.1002/(Sici)1521-3773(19991102)38:21<3197::Aid-Anie3197>3.0.Co;2-6  0.317
1999 McDaid HM, Bhattacharya SK, Chen XT, He L, Shen HJ, Gutteridge CE, Horwitz SB, Danishefsky SJ. Structure-activity profiles of eleutherobin analogs and their cross-resistance in Taxol-resistant cell lines. Cancer Chemotherapy and Pharmacology. 44: 131-7. PMID 10412947 DOI: 10.1007/S002800050957  0.663
1999 Live DH, Williams LJ, Kuduk SD, Schwarz JB, Glunz PW, Chen XT, Sames D, Kumar RA, Danishefsky SJ. Probing cell-surface architecture through synthesis: an NMR-determined structural motif for tumor-associated mucins. Proceedings of the National Academy of Sciences of the United States of America. 96: 3489-93. PMID 10097062 DOI: 10.1073/Pnas.96.7.3489  0.689
1999 Allen JR, Danishefsky SJ. New Applications of then-Pentenyl Glycoside Method in the Synthesis and Immunoconjugation of Fucosyl GM1:  A Highly Tumor-Specific Antigen Associated with Small Cell Lung Carcinoma Journal of the American Chemical Society. 121: 10875-10882. DOI: 10.1021/Ja992594F  0.377
1999 Schkeryantz JM, Woo JCG, Siliphaivanh P, Depew KM, Danishefsky SJ. Total synthesis of gypsetin, deoxybrevianamide E, brevianamide E, and tryprostatin B: Novel constructions of 2,3-disubstituted indoles Journal of the American Chemical Society. 121: 11964-11975. DOI: 10.1021/Ja9925249  0.424
1999 Glunz PW, Hintermann S, Schwarz JB, Kuduk SD, Chen XT, Williams LJ, Sames D, Danishefsky SJ, Kudryashov V, Lloyd KO. Probing cell surface 'glyco-architecture' through total synthesis. Immunological consequences of a human blood group determinant in a clustered mucin-like context [6] Journal of the American Chemical Society. 121: 10636-10637. DOI: 10.1021/Ja992309S  0.691
1999 Harris CR, Kuduk SD, Balog A, Savin K, Glunz PW, Danishefsky SJ. New Chemical Synthesis of the Promising Cancer Chemotherapeutic Agent 12,13-Desoxyepothilone B: Discovery of a Surprising Long-Range Effect on the Diastereoselectivity of an Aldol Condensation Journal of the American Chemical Society. 121: 7050-7062. DOI: 10.1021/Ja991189L  0.354
1999 Chen XT, Bhattacharya SK, Zhou B, Gutteridge CE, Pettus TRR, Danishefsky SJ. The total synthesis of eleutherobin Journal of the American Chemical Society. 121: 6563-6579. DOI: 10.1021/Ja990215C  0.769
1999 Schwarz JB, Kuduk SD, Chen XT, Sames D, Glunz PW, Danishefsky SJ. A broadly applicable method for the efficient synthesis of α-O-linked glycopeptides and clustered sialic acid residues Journal of the American Chemical Society. 121: 2662-2673. DOI: 10.1021/Ja9833265  0.687
1999 Trauner D, Danishefsky SJ. Studies towards the total synthesis of halichlorine: asymmetric synthesis of the spiroquinolizidine subunit Tetrahedron Letters. 40: 6513-6516. DOI: 10.1016/S0040-4039(99)01170-3  0.502
1999 Bhattacharya SK, Chen X, Gutteridge CE, Danishefsky SJ. A remarkable pyranose to furanose isomerization mediated by an “anomeric" silyloxy function Tetrahedron Letters. 40: 3313-3316. DOI: 10.1016/S0040-4039(99)00499-2  0.691
1999 Harris CR, Kuduk SD, Savin K, Balog A, Danishefsky SJ. Dianion equivalents corresponding to the polypropionate domain of epothilone B Tetrahedron Letters. 40: 2263-2266. DOI: 10.1016/S0040-4039(99)00221-X  0.345
1999 Trauner D, Schwarz J, Danishefsky S. Totalsynthese von (+)-Halichlorin, einem Inhibitor der Expression von VCAM-1 Angewandte Chemie. 111: 3756-3758. DOI: 10.1002/(Sici)1521-3757(19991203)111:23<3756::Aid-Ange3756>3.0.Co;2-9  0.379
1999 Meng D, Danishefsky SJ. Stereospezifische, schwefelunterstützte Spaltung eines Spirocylobutanons: Synthese einer vollständig funktionalisierten Vorstufe der CP-Verbindungen Angewandte Chemie. 111: 1582-1585. DOI: 10.1002/(Sici)1521-3757(19990517)111:10<1582::Aid-Ange1582>3.0.Co;2-S  0.317
1999 Ragupathi G, Slovin SF, Adluri S, Sames D, Kim IJ, Kim HM, Spassova M, Bornmann WG, Lloyd KO, Scher HI, Livingston PO, Danishefsky SJ. Ein totalsynthetischer Globo-H-Kohlenhydrat-Impfstoff verursacht eine gezielte humorale Immunantwort bei Prostatakrebs-Patienten: der Beweis des Prinzips Angewandte Chemie. 111: 590-594. DOI: 10.1002/(Sici)1521-3757(19990215)111:4<590::Aid-Ange590>3.0.Co;2-A  0.659
1998 Chen XT, Zhou B, Bhattacharya SK, Gutteridge CE, Pettus TRR, Danishefsky SJ. The Total Synthesis of Eleutherobin: A Surprise Ending. Angewandte Chemie (International Ed. in English). 37: 789-792. PMID 29711384 DOI: 10.1002/(Sici)1521-3773(19980403)37:6<789::Aid-Anie789>3.0.Co;2-3  0.75
1998 Zheng C, Seeberger PH, Danishefsky SJ. Amidoglycosylation of Polymer-Bound Glycals: A Complete Solid-Phase Synthesis of the Oligosaccharide Domain of the Lewis Blood Group Determinant. Angewandte Chemie (International Ed. in English). 37: 786-789. PMID 29711374 DOI: 10.1002/(Sici)1521-3773(19980403)37:6<786::Aid-Anie786>3.0.Co;2-F  0.571
1998 Zheng C, Seeberger PH, Danishefsky SJ. Solid Support Oligosaccharide Synthesis:  Construction of β-Linked Oligosaccharides by Coupling of Glycal Derived Thioethyl Glycosyl Donors The Journal of Organic Chemistry. 63: 1126-1130. DOI: 10.1021/Jo971606H  0.565
1998 Pettus TRR, Chen XT, Danishefsky SJ. A fully synthetic route to the neurotrophic illicinones by sequential aromatic Claisen rearrangements [10] Journal of the American Chemical Society. 120: 12684-12685. DOI: 10.1021/Ja982582E  0.374
1998 Kuduk SD, Schwarz JB, Chen X, Glunz PW, Sames D, Ragupathi G, Livingston PO, Danishefsky SJ. Synthetic and Immunological Studies on Clustered Modes of Mucin-Related Tn and TF O-Linked Antigens:  The Preparation of a Glycopeptide-Based Vaccine for Clinical Trials against Prostate Cancer† Journal of the American Chemical Society. 120: 12474-12485. DOI: 10.1021/Ja9825128  0.674
1998 Roberge JY, Beebe X, Danishefsky SJ. Convergent Synthesis ofN-Linked Glycopeptides on a Solid Support Journal of the American Chemical Society. 120: 3915-3927. DOI: 10.1021/Ja9740071  0.371
1998 Deshpande PP, Kim HM, Zatorski A, Park T, Ragupathi G, Livingston PO, Live D, Danishefsky SJ. Strategy in Oligosaccharide Synthesis:  An Application to a Concise Total Synthesis of the KH-1(adenocarcinoma) Antigen Journal of the American Chemical Society. 120: 1600-1614. DOI: 10.1021/Ja9725864  0.41
1998 Kwon O, Su D, Meng D, Deng W, D'Amico DC, Danishefsky SJ. A Stereospecific Geminal Alkylation Scheme En Route To CP‐225, 917 and CP‐263,114 Angewandte Chemie. 37: 1880-1882. DOI: 10.1002/(Sici)1521-3773(19980803)37:13/14<1880::Aid-Anie1880>3.0.Co;2-5  0.54
1998 Chen XT, Zhou B, Bhattacharya SK, Gutteridge CE, Pettus TRR, Danishefsky SJ. The total synthesis of eleutherobin: A surprise ending Angewandte Chemie - International Edition. 37: 789-792. DOI: 10.1002/(SICI)1521-3773(19980403)37:6<789::AID-ANIE789>3.0.CO;2-3  0.76
1998 Kwon O, Su D, Meng D, Deng W, D'Amico DC, Danishefsky SJ. Eine stereospezifische geminale Alkylierung auf dem Weg zu CP-225,917 und CP-263,114 Angewandte Chemie. 110: 1981-1983. DOI: 10.1002/(Sici)1521-3757(19980703)110:13/14<1981::Aid-Ange1981>3.0.Co;2-5  0.526
1998 Kwon O, Su D, Meng D, Deng W, D'Amico DC, Danishefsky SJ. Bildung einer Matrixstruktur für die Totalsynthese von CP-225,917 und CP-263,114 durch Aldol- und intramolekulare Heck-Reaktion Angewandte Chemie. 110: 1978-1981. DOI: 10.1002/(Sici)1521-3757(19980703)110:13/14<1978::Aid-Ange1978>3.0.Co;2-2  0.528
1998 Chen X, Zhou B, Bhattacharya S, Gutteridge C, Pettus T, Danishefsky S. Totalsynthese von Eleutherobin: zum Schluß eine Überraschung Angewandte Chemie. 110: 835-838. DOI: 10.1002/(Sici)1521-3757(19980316)110:6<835::Aid-Ange835>3.0.Co;2-0  0.752
1998 Zheng C, Seeberger P, Danishefsky S. Amidoglycosylierung von polymergebundenen Glycalen: eine komplette Festphasensynthese des Oligosaccharidteils der Blutgruppendeterminante Lewisb Angewandte Chemie. 110: 831-834. DOI: 10.1002/(Sici)1521-3757(19980316)110:6<831::Aid-Ange831>3.0.Co;2-G  0.506
1998 Chen X, Gutteridge C, Bhattacharya S, Zhou B, Pettus T, Hascall T, Danishefsky S. Eine konvergente Route zur Totalsynthese der Eleutheside Angewandte Chemie. 110: 195-197. DOI: 10.1002/(Sici)1521-3757(19980116)110:1/2<195::Aid-Ange195>3.0.Co;2-C  0.775
1997 Sames D, Chen XT, Danishefsky SJ. Convergent total synthesis of a tumour-associated mucin motif. Nature. 389: 587-91. PMID 9335496 DOI: 10.1038/39292  0.728
1997 Deshpande PP, Danishefsky SJ. Total synthesis of the potential anticancer vaccine KH-1 adenocarcinoma antigen. Nature. 387: 164-6. PMID 9144285 DOI: 10.1038/387164A0  0.327
1997 Zhong G, Hoffmann T, Lerner RA, Danishefsky S, Barbas CF. Antibody-catalyzed enantioselective Robinson annulation Journal of the American Chemical Society. 119: 8131-8132. DOI: 10.1021/Ja970944X  0.322
1997 Frontier AJ, Raghavan S, Danishefsky SJ. Stereocontrolled total synthesis of hispidospermidin Journal of the American Chemical Society. 119: 6686-6687. DOI: 10.1021/Ja970889S  0.636
1997 Meng D, Su DS, Balog A, Bertinato P, Sorensen EJ, Danishefsky SJ, Zheng YH, Chou TC, He L, Horwitz SB. Remote effects in macrolide formation through ring-forming olefin metathesis: An application to the synthesis of fully active epothilone congeners Journal of the American Chemical Society. 119: 2733-2734. DOI: 10.1021/Ja964275J  0.553
1997 Balog A, Bertinato P, Su DS, Meng D, Sorensen E, Danishefsky SJ, Zheng YH, Chou TC, He L, Horwitz SB. Stereoselective syntheses and evaluation of compounds in the 8-desmethylepothilone a series: Some surprising observations regarding their chemical and biological properties Tetrahedron Letters. 38: 4529-4532. DOI: 10.1016/S0040-4039(97)00931-3  0.485
1997 Su D, Meng D, Bertinato P, Balog A, Sorensen EJ, Danishefsky SJ, Zheng Y, Chou T, He L, Horwitz SB. Total Synthesis of(–)-Epothilone B: An Extension of the Suzuki Coupling Method and Insights into Structure–Activity Relationships of the Epothilones Angewandte Chemie International Edition in English. 36: 757-759. DOI: 10.1002/Anie.199707571  0.326
1997 Seeberger PH, Beebe X, Sukenick GD, Pochapsky S, Danishefsky SJ. Monitoring the Progress of Solid-Phase Oligosaccharide Synthesis by High-Resolution Magic Angle Spinning NMR: Observations of Enhanced Selectivity forβ-Glycoside Formation fromα-1,2-Anhydrosugar Donors in Solid-Phase Couplings Angewandte Chemie International Edition in English. 36: 491-493. DOI: 10.1002/Anie.199704911  0.541
1997 Su D, Meng D, Bertinato P, Balog A, Sorensen EJ, Danishefsky SJ, Chou T, He L, Horwitz SB. Totalsynthese von ( - )-Epothilon B: eine Erweiterung der Suzuki-Kupplung und Erkenntnisse über Struktur-Wirkungs-Beziehungen der Epothilone Angewandte Chemie. 109: 775-777. DOI: 10.1002/Ange.19971090719  0.499
1997 Seeberger PH, Beebe X, Danishefsky SJ, Sukenick GD, Pochapsky S. Verfolgung von Festphasen-Oligosaccharidsynthesen mit hochauflösender MAS-NMR-Spektroskopie: Selektivität der Festphasenkupplung von α-1,2-Didehydrozuckerdonoren zu β-Glycosiden Angewandte Chemie. 109: 507-510. DOI: 10.1002/Ange.19971090511  0.516
1996 Bertinato P, Sorensen EJ, Meng D, Danishefsky SJ. Studies toward a Synthesis of Epothilone A: Stereocontrolled Assembly of the Acyl Region and Models for Macrocyclization. The Journal of Organic Chemistry. 61: 8000-8001. PMID 11667778  0.523
1996 Meng D, Sorensen EJ, Bertinato P, Danishefsky SJ. Studies toward a Synthesis of Epothilone A: Use of Hydropyran Templates for the Management of Acyclic Stereochemical Relationships. The Journal of Organic Chemistry. 61: 7998-7999. PMID 11667777 DOI: 10.1021/Jo961673W  0.5
1996 Seeberger PH, Cirillo PF, Hu S, Beebe X, Bilodeau MT, Danishefsky SJ. Synthesis of the pentasaccharide core structure of asparagine-linked glycoprotein oligosaccharides by the glycal assembly method. Enantiomer. 1: 311-23. PMID 9676275  0.559
1996 Live DH, Kumar RA, Beebe X, Danishefsky SJ. Conformational influences of glycosylation of a peptide: a possible model for the effect of glycosylation on the rate of protein folding. Proceedings of the National Academy of Sciences of the United States of America. 93: 12759-61. PMID 8917491 DOI: 10.1073/Pnas.93.23.12759  0.323
1996 Bertinato P, Sorensen EJ, Meng D, Danishefsky SJ. Studies toward a synthesis of epothilone A: Stereocontrolled assembly of the acyl region and models for macrocyclization Journal of Organic Chemistry. 61: 8000-8001. DOI: 10.1021/jo961674o  0.523
1996 Meng D, Sorensen EJ, Bertinato P, Danishefsky SJ. Studies toward a synthesis of epothilone A: Use of hydropyran templates for the management of acyclic stereochemical relationships Journal of Organic Chemistry. 61: 7998-7999. DOI: 10.1021/jo961673w  0.5
1996 Danishefsky SJ, Shair MD. Observations in the Chemistry and Biology of Cyclic Enediyne Antibiotics: Total Syntheses of Calicheamicin γ1I and Dynemicin A Journal of Organic Chemistry. 61: 16-44. DOI: 10.1021/Jo951560X  0.658
1996 Park TK, Kim IJ, Hu S, Bilodeau MT, Randolph JT, Kwon O, Danishefsky SJ. Total Synthesis and Proof of Structure of a Human Breast Tumor (Globo-H) Antigen Journal of the American Chemical Society. 118: 11488-11500. DOI: 10.1021/Ja962048B  0.352
1996 Shair MD, Yoon TY, Mosny KK, Chou TC, Danishefsky SJ. The total synthesis of dynemicin A leading to development of a fully contained bioreductively activated enediyne prodrug Journal of the American Chemical Society. 118: 9509-9525. DOI: 10.1021/Ja960040W  0.666
1996 Link JT, Raghavan S, Gallant M, Danishefsky SJ, Chou TC, Ballas LM. Staurosporine andent-Staurosporine:  The First Total Syntheses, Prospects for a Regioselective Approach, and Activity Profiles1 Journal of the American Chemical Society. 118: 2825-2842. DOI: 10.1021/Ja952907G  0.346
1996 Liu KK‐, Danishefsky SJ. A Paradigm Case for the Merging of Glycal and Enzymatic Assembly Methods in Glycoconjugate Synthesis: A Highly Efficient Chemo‐Enzymatic Synthesis of GM3 Chemistry: a European Journal. 2: 1359-1362. DOI: 10.1002/Chem.19960021105  0.39
1996 Balog A, Meng D, Kamenecka T, Bertinato P, Su D, Sorensen EJ, Danishefsky SJ. Totalsynthese von (—)-Epothilon A Angewandte Chemie. 108: 2976-2978. DOI: 10.1002/Ange.19961082318  0.477
1995 Roberge JY, Beebe X, Danishefsky SJ. A strategy for a convergent synthesis of N-linked glycopeptides on a solid support. Science (New York, N.Y.). 269: 202-4. PMID 7618080 DOI: 10.1126/Science.7618080  0.792
1995 Hitchcock SA, Chu-Moyer MY, Boyer SH, Olson SH, Danishefsky SJ. A Remarkable Glycosidation Reaction: The Total Synthesis of Calicheamicin .gamma.1I Journal of the American Chemical Society. 117: 5750-5756. DOI: 10.1021/Ja00126A014  0.374
1995 Randolph JT, McClure KF, Danishefsky SJ. Major Simplifications in Oligosaccharide Syntheses Arising from a Solid-Phase Based Method: An Application to the Synthesis of the Lewis b Antigen Journal of the American Chemical Society. 117: 5712-5719. DOI: 10.1021/Ja00126A012  0.324
1995 Randolph JT, Danishefsky SJ. First Synthesis of a Digitalis Saponin. Demonstration of the Scope and Limitations of a Convergent Scheme for Branched Oligosaccharide Synthesis by the Logic of Glycal Assembly Journal of the American Chemical Society. 117: 5693-5700. DOI: 10.1021/Ja00126A010  0.365
1995 Schkeryantz JM, Danishefsky SJ. Total Synthesis of (.+-.)-FR-900482 Journal of the American Chemical Society. 117: 4722-4723. DOI: 10.1021/Ja00121A037  0.418
1995 Danishefsky SJ, Gervay J, Peterson JM, McDonald FE, Koseki K, Griffith DA, Oriyama T, Marsden SP. Application of Glycals to the Synthesis of Oligosaccharides: Convergent Total Syntheses of the Lewis X Trisaccharide Sialyl Lewis X Antigenic Determinant and Higher Congeners Journal of the American Chemical Society. 117: 1940-1953. DOI: 10.1021/Ja00112A007  0.706
1995 Shair MD, Yoon T, Danishefsky SJ. Total Synthesis of(±)-Dynemicin A Angewandte Chemie International Edition in English. 34: 1721-1723. DOI: 10.1002/Anie.199517211  0.605
1995 Shair MD, Danishefsky SJ, Yoon T, Chou T. Enediyne Quinone Imines: Truncated, Biologically Active Dynemicin Congeners Angewandte Chemie International Edition in English. 33: 2477-2479. DOI: 10.1002/Anie.199424771  0.619
1995 Shair MD, Yoon T, Danishefsky SJ. Totalsynthese von (±)-Dynemicin A Angewandte Chemie. 107: 1883-1885. DOI: 10.1002/Ange.19951071616  0.586
1994 Roche CJ, Berkowitz D, Sulikowski GA, Danishefsky SJ, Crothers DM. Binding affinity and site selectivity of daunomycin analogues. Biochemistry. 33: 936-42. PMID 8305441 DOI: 10.1021/Bi00170A012  0.747
1994 Ho SN, Boyer SH, Schreiber SL, Danishefsky SJ, Crabtree GR. Specific inhibition of formation of transcription complexes by a calicheamicin oligosaccharide: a paradigm for the development of transcriptional antagonists. Proceedings of the National Academy of Sciences of the United States of America. 91: 9203-7. PMID 7937742 DOI: 10.1073/Pnas.91.20.9203  0.408
1994 Snyder L, Shen W, Bornmann WG, Danishefsky SJ. Synthesis of 18-Noranhydrocamptothecin Analogs Which Retain Topoisomerase I Inhibitory Function Journal of Organic Chemistry. 59: 7033-7037. DOI: 10.1021/Jo00102A030  0.37
1994 Chu-Moyer MY, Danishefsky SJ, Schulte GK. Total Synthesis of (.+-.)-Myrocin C Journal of the American Chemical Society. 116: 11213-11228. DOI: 10.1021/Ja00104A002  0.345
1994 Yoon T, Shair MD, Danishefsky SJ. An advanced dynemicin A model: Stabilization of the 3,8-epoxide by anthraquinone functionality in the absence of the bridging enediyne Tetrahedron Letters. 35: 6259-6262. DOI: 10.1016/S0040-4039(00)73406-X  0.574
1994 Link J, Danishefsky SJ. Regioselective imide reduction : An issue in the total synthesis of staurosporine Tetrahedron Letters. 35: 9135-9138. DOI: 10.1016/0040-4039(94)88446-3  0.421
1994 Olson SH, Danishefsky SJ. Reductive desilanolation as a route to benzonitriles. An application to a concise synthesis of the aromatic sector of calicheamicin Tetrahedron Letters. 35: 7901-7904. DOI: 10.1016/0040-4039(94)80006-5  0.395
1994 Hitchcock SA, Boyer SH, Chu-Moyer MY, Olson SH, Danishefsky SJ. A Convergent Total Synthesis of Calicheamicinγ1I Angewandte Chemie. 33: 858-862. DOI: 10.1002/Anie.199408581  0.397
1994 Shair MD, Yoon T, Chou T, Danishefsky SJ. Endiin-Chinonimine: verkleinerte, biologisch aktive Dynemicinanaloga Angewandte Chemie. 106: 2578-2580. DOI: 10.1002/Ange.19941062337  0.632
1994 Randolph JT, Danishefsky SJ. Strategie für den Zusammenbau verzweigter Oligosaccharide mit der Festphasenmethode: kurze Synthese der Blutgruppendeterminante Lewisb in konjugatbildender Form Angewandte Chemie. 106: 1538-1541. DOI: 10.1002/Ange.19941061415  0.301
1994 Behar V, Danishefsky SJ. Hochkonvergente Synthese der Blutgruppen-determinante Lewisy in konjugatbildender Form Angewandte Chemie. 106: 1536-1538. DOI: 10.1002/Ange.19941061414  0.301
1993 Grandi MJD, Jung DK, Krol WJ, Danishefsky SJ. Synthesis of competent nucleophiles for delivering the A ring of taxol Journal of Organic Chemistry. 58: 4989-4992. DOI: 10.1021/Jo00070A040  0.389
1993 Isaacs RCA, Grandi MJD, Danishefsky SJ. Synthesis of an enantiomerically pure intermediate containing the CD substructure of taxol Journal of Organic Chemistry. 58: 3938-3941. DOI: 10.1021/Jo00067A028  0.359
1993 Queneau Y, Krol WJ, Bornmann WG, Danishefsky SJ. A ready synthesis of intermediates containing the A-ring substructure of taxol: a Diels-Alder route to the B-seco taxane series. [Erratum to document cited in CA117(3):26833h] The Journal of Organic Chemistry. 58: 798-798. DOI: 10.1021/Jo00055A048  0.332
1993 Shen W, Coburn CA, Bornmann WG, Danishefsky SJ. Concise total syntheses of dl-camptothecin and related anticancer drugs Journal of Organic Chemistry. 58: 611-617. DOI: 10.1021/Jo00055A012  0.331
1993 Gallant M, Link JT, Danishefsky SJ. A stereoselective synthesis of indole-.beta.-N-glycosides: an application to the synthesis of rebeccamycin The Journal of Organic Chemistry. 58: 343-349. DOI: 10.1021/Jo00054A015  0.378
1993 Liu KKC, Danishefsky SJ. A striking example of the interfacing of glycal chemistry with enzymatically mediated sialylation: a concise synthesis of ganglioside GM3 Journal of the American Chemical Society. 115: 4933-4934. DOI: 10.1021/Ja00064A082  0.38
1993 Link JT, Gallant M, Danishefsky SJ, Huber S. The first synthesis of a fully functionalized core structure of staurosporine : sequential indolyl glycosidation by endo and exo glycals Journal of the American Chemical Society. 115: 3782-3783. DOI: 10.1021/Ja00062A057  0.352
1993 Yohannes D, Myers CD, Danishefsky SJ. Degradation of rapamycin: Synthesis of a rapamycin derived fragment containing the tricarbonyl and triene sectors Tetrahedron Letters. 34: 2075-2078. DOI: 10.1016/S0040-4039(00)60349-0  0.632
1992 Queneau Y, Krol WJ, Bornmann WG, Danishefsky SJ. A ready synthesis of intermediates containing the A-ring substructure of taxol : a Diels-Alder route to the B-seco taxane series Journal of Organic Chemistry. 57: 4043-4047. DOI: 10.1021/Jo00040A064  0.384
1992 Magee TV, Bornmann WG, Isaacs RCA, Danishefsky SJ. A straightforward route to functionalized intermediates containing the CD substructure of taxol. Journal of Organic Chemistry. 57: 3274-3276. DOI: 10.1021/Jo00038A008  0.357
1992 Dushin RG, Danishefsky SJ. Stereospecific synthesis of aryl .beta.-glucosides: an application to the synthesis of a prototype corresponding to the aryloxy carbohydrate domain of vancomycin Journal of the American Chemical Society. 114: 3471-3475. DOI: 10.1021/Ja00035A047  0.327
1992 Yohannes D, Danishefsky SJ. Degradation of rapamycin: Retrieval of major intact subunits. Tetrahedron Letters. 33: 7469-7472. DOI: 10.1016/S0040-4039(00)60797-9  0.603
1991 Drak J, Iwasawa N, Danishefsky S, Crothers DM. The carbohydrate domain of calicheamicin gamma I1 determines its sequence specificity for DNA cleavage. Proceedings of the National Academy of Sciences of the United States of America. 88: 7464-8. PMID 1881884 DOI: 10.1073/Pnas.88.17.7464  0.518
1991 Chen SH, Horvath RF, Joglar J, Fisher MJ, Danishefsky SJ. Application of the Ibuka-Yamamoto reaction to a problem in stereochemical communication: a strategy for the stereospecific synthesis and stabilization of the triene substructure of rapamycin through sulfone substitution The Journal of Organic Chemistry. 56: 5834-5845. DOI: 10.1021/Jo00020A027  0.338
1991 Fisher MJ, Chow K, Villalobos A, Danishefsky SJ. On the remarkable propensity for carbon-carbon bond cleavage reactions in the C(8)-C(10) region of FK-506 Journal of Organic Chemistry. 56: 2900-2907. DOI: 10.1021/Jo00008A055  0.307
1991 McClure KF, Benbow JW, Danishefsky SJ, Schulte GK. A novel photochemical route to the mitomycin and FR-900482 series Journal of the American Chemical Society. 113: 8185-8186. DOI: 10.1021/Ja00021A064  0.326
1991 Haseltine JN, Paz Cabal M, Mantlo NB, Iwasawa N, Yamashita DS, Coleman RS, Danishefsky SJ, Schulte GK. Total synthesis of calicheamicinone: new arrangements for actuation of the reductive cycloaromatization of aglycon congeners Journal of the American Chemical Society. 113: 3850-3866. DOI: 10.1021/Ja00010A030  0.674
1991 Sulikowski GA, Turos E, Danishefsky SJ, Shulte GM. An entry to the ring B:ring C bishydroquinone leucodaunomycin series containing an intact carbohydrate Journal of the American Chemical Society. 113: 1373-1377. DOI: 10.1021/Ja00004A045  0.775
1991 Berkowitz DB, Danishefsky SJ. Enzymatic resolution of racemic glycals: an application of the wong acylation method Tetrahedron Letters. 32: 5497-5500. DOI: 10.1016/0040-4039(91)80067-G  0.558
1990 Chow K, Danishefsky S. Stereospecific Vorbrueggen-like reactions of 1,2-anhydro sugars. An alternative route to the synthesis of nucleosides The Journal of Organic Chemistry. 55: 4211-4214. DOI: 10.1021/Jo00300A049  0.338
1990 Jones AB, Villalobos A, Linde RG, Danishefsky SJ. A formal synthesis of FK-506. Exploration of some alternatives to macrolactamization The Journal of Organic Chemistry. 55: 2786-2797. DOI: 10.1021/Jo00296A042  0.347
1990 Villalobos A, Danishefsky SJ. Stereoselective routes to the C10−C19 fragment of FK-506 Journal of Organic Chemistry. 55: 2776-2786. DOI: 10.1021/Jo00296A041  0.323
1990 Linde RG, Egbertson M, Coleman RS, Jones AB, Danishefsky SJ. Efficient preparation of intermediates corresponding to C22-C27 and C28-C34 of FK-506 The Journal of Organic Chemistry. 55: 2771-2776. DOI: 10.1021/Jo00296A040  0.497
1990 Wittman MD, Halcomb RL, Danishefsky SJ. On the conversion of biologically interesting amines to hydroxylamines The Journal of Organic Chemistry. 55: 1981-1983. DOI: 10.1021/Jo00294A005  0.32
1990 Wittman MD, Halcomb RL, Danishefsky SJ, Golik J, Vyas D. A route to glycals in the allal and gulal series: synthesis of the thiosugar of esperamicin A1 Journal of Organic Chemistry. 55: 1979-1981. DOI: 10.1021/Jo00294A004  0.386
1990 Myles DC, Danishefsky SJ, Schulte G. Development of a fully synthetic stereoselective route to 6-deoxyerythronolide B by reiterative applications of the Lewis acid catalyzed diene aldehyde cyclocondensation reaction: a remarkable instance of diastereofacial selectivity Journal of Organic Chemistry. 55: 1636-1648. DOI: 10.1021/Jo00292A045  0.409
1990 Fang FG, Maier ME, Danishefsky SJ, Schulte G. New Routes To Functionalized Benzazepine Substructures : A Novel Transformation Of An Alpha -Diketone Thioamide Induced By Trimethyl Phosphite Journal of Organic Chemistry. 55: 831-838. DOI: 10.1021/Jo00290A011  0.582
1990 Griffith DA, Danishefsky SJ. Sulfonamidoglycosylation of glycals. A route to oligosaccharides with 2-aminohexose subunits Journal of the American Chemical Society. 112: 5811-5819. DOI: 10.1021/Ja00171A021  0.579
1990 Kim G, Chu-Moyer MY, Danishefsky SJ. The total synthesis of dl-indolizomycin Journal of the American Chemical Society. 112: 2003-2005. DOI: 10.1021/Ja00161A059  0.403
1989 Myles DC, Danishefsky SJ. The synthesis of polyoxygenated natural products via fully synthetic branched pyranose derivatives: Application to the erythronolide problem Pure and Applied Chemistry. 61: 1235-1242. DOI: 10.1351/Pac198961071235  0.367
1989 Chow K, Danishefsky S. Total synthesis of 13-oxygenated prostanoids derived from arachidonate: an instance of extraordinary variability in the stereochemical sense of a Mukaiyama aldol reaction The Journal of Organic Chemistry. 54: 6016-6018. DOI: 10.1021/Jo00287A009  0.353
1989 Chenault HK, Danishefsky SJ. Characterization of 2-siloxyoxiranes formed by epoxidation of silyl enol ethers with dimethyldioxirane Journal of Organic Chemistry. 54: 4249-4250. DOI: 10.1021/Jo00278A055  0.331
1989 Jones AB, Yamaguchi M, Patten A, Danishefsky SJ, Ragan JA, Smith DB, Schreiber SL. Studies relating to the synthesis of the immunosuppressive agent FK-506: coupling of fragments via a stereoselective trisubstituted olefin forming reaction sequence The Journal of Organic Chemistry. 54: 17-19. DOI: 10.1021/Jo00262A008  0.5
1989 Villalobos A, Danishefsky SJ. Stereoselective syntheses of FK-506 subunits by the rhodium(I)-catalyzed hdrogenation of dienes. The synthesis and coupling of a C10-C19 fragment Journal of Organic Chemistry. 54: 12-15. DOI: 10.1021/Jo00262A006  0.352
1989 Turos E, Audia JE, Danishefsky SJ. Total synthesis of the Fusarium toxin equisetin: proof of the stereochemical relationship of the tetramate and terpenoid sectors Journal of the American Chemical Society. 111: 8231-8236. DOI: 10.1021/ja00203a026  0.606
1989 Halcomb RL, Danishefsky SJ. On the direct epoxidation of glycals: application of a reiterative strategy for the synthesis of .beta.-linked oligosaccharides Journal of the American Chemical Society. 111: 6661-6666. DOI: 10.1021/Ja00199A028  0.313
1989 Danishefsky S, Lee JY. Total synthesis of (±)-pancratistatin Journal of the American Chemical Society. 111: 4829-4837. DOI: 10.1021/Ja00195A039  0.304
1989 Fang FG, Prato M, Kim G, Danishefsky SJ. The aza-robinson annulation: An application to the synthesis of iso-A58365A Tetrahedron Letters. 30: 3625-3628. DOI: 10.1016/S0040-4039(01)80465-2  0.465
1988 Danishefsky SJ, Simoneau B. Synthetic studies in the mevinoid field. The total synthesis of ML236A Pure and Applied Chemistry. 60: 1555-1562. DOI: 10.1351/Pac198860111555  0.387
1988 Feigelson GB, Danishefsky SJ. On the synthesis and extraordinary configurational stability of the C9a-hydroxylated mitomycins in the 10-decarbamoyloxy-9-dehydro series: fully synthetic routes to novel mitomycin congeners Journal of Organic Chemistry. 53: 3391-3393. DOI: 10.1021/Jo00249A061  0.329
1988 Patten AD, Huy NN, Danishefsky SJ. A concise total synthesis of defucogilvocarcin V by application of the meyers biaryl strategy: ortho- and para-selective functionalizations of the A ring Journal of Organic Chemistry. 53: 1003-1007. DOI: 10.1021/Jo00240A012  0.358
1988 Danishefsky SJ, Mantlo N. Total synthesis of (.+-.)-heptelidic acid Journal of the American Chemical Society. 110: 8129-8133. DOI: 10.1021/Ja00232A027  0.346
1988 Danishefsky SJ, Selnick HG, Zelle RE, DeNinno MP. Total synthesis of zincophorin Journal of the American Chemical Society. 110: 4368-4378. DOI: 10.1021/Ja00221A043  0.418
1987 Danishefsky SJ, Danishefsky S, Feigelson GB. Polonovski reactions of mitosane derivatives Heterocycles. 25: 301-304. DOI: 10.3987/S-1987-01-0301  0.306
1987 Askin D, Angst C, Danishefsky S. An approach to the synthesis of bactobolin and the total synthesis of N-acetylactinobolamine: some remarkably stable hemiacetals Journal of Organic Chemistry. 52: 622-635. DOI: 10.1021/Jo00380A025  0.386
1987 Danishefsky SJ, Selnick HG, DeNinno MP, Zelle RE. The total synthesis of zincophorin Journal of the American Chemical Society. 109: 1572-1574. DOI: 10.1021/Ja00239A049  0.418
1987 Danishefsky SJ, Panek JS. Total synthesis of (.+-.)-3-demethoxyerythratidinone: demonstration of a radical cyclization route to a site specific enol derivative Journal of the American Chemical Society. 109: 917-918. DOI: 10.1021/Ja00237A057  0.59
1987 Danishefsky SJ, Myles DC, Harvey DF. Expeditious synthesis of the polypropionate sector of rifamycin S by reiterative Diene-Aldehyde cyclocondensation reactions Journal of the American Chemical Society. 109: 862-867. DOI: 10.1021/Ja00237A037  0.37
1986 Zelle RE, DeNinno MP, Selnick HG, Danishefsky SJ. A systematic degradation of zincophorin: a stereoselective synthesis of the C17-C25 fragment Journal of Organic Chemistry. 51: 5032-5036. DOI: 10.1021/Jo00375A060  0.312
1986 Danishefsky SJ, Vogel C. A concise total synthesis of (±)-ipalbidine by application of the aldimine-diene cyclocondensation reaction Journal of Organic Chemistry. 51: 3915-3916. DOI: 10.1021/Jo00370A039  0.33
1986 Danishefsky SJ, DeNinno MP. The total synthesis of (.+-.)-N-acetylneuraminic acid (NANA). A remarkable hydroxylation of a (Z)-enoate The Journal of Organic Chemistry. 51: 2615-2617. DOI: 10.1021/Jo00363A047  0.331
1986 Bednarski M, Danishefsky S. Interactivity of chiral catalysts and chiral auxiliaries in the cycloaddition of activated dienes with aldehydes: a synthesis of L-glucose Journal of the American Chemical Society. 108: 7060-7067. DOI: 10.1021/Ja00282A035  0.6
1986 Danishefsky SJ, Egbertson M. On the characterization of intermediates in the mitomycin activation cascade: a practical synthesis of an aziridinomitosene Journal of the American Chemical Society. 108: 4648-4650. DOI: 10.1021/Ja00275A065  0.34
1986 Danishefsky SJ, Egbertson M. Characterization of Intermediates in the Mitomycin Activation Cascade: A Practical Synthesis of an Aziridinomitosene. Cheminform. 17. DOI: 10.1002/Chin.198648348  0.34
1986 Askin D, Angst C, Danishefsky S. A Total Synthesis of N-Acetylactinobolamine (I). Cheminform. 17. DOI: 10.1002/Chin.198621317  0.336
1986 Danishefsky S, Chao K-, Schulte G. Variations in the Stereochemistry of the Boron Trifluoride Mediated Cyclocondensation Reaction of Aldehydes with Siloxy Dienes. Cheminform. 17. DOI: 10.1002/Chin.198618104  0.318
1986 Danishefsky S, Maring C. A Fully Synthetic Route to Hikosamine. Cheminform. 17. DOI: 10.1002/Chin.198613322  0.354
1985 Askin D, Angst C, Danishefsky S. A total synthesis of N-acetylactinobolamine Journal of Organic Chemistry. 50: 5005-5007. DOI: 10.1021/Jo00224A082  0.336
1985 Danishefsky S, Maring C. A fully synthetic route to hikosamine Journal of the American Chemical Society. 107: 7762-7764. DOI: 10.1021/Ja00311A090  0.354
1985 Danishefsky S, Barbachyn M. A fully synthetic route to tunicaminyluracil Journal of the American Chemical Society. 107: 7761-7762. DOI: 10.1021/Ja00311A089  0.354
1985 Danishefsky S, Berman EM, Ciufolini M, Etheredge SJ, Segmuller BE. A stereospecific route to aziridinomitosanes: the synthesis of novel mitomycin congeners Journal of the American Chemical Society. 107: 3891-3898. DOI: 10.1021/Ja00299A022  0.817
1985 Danishefsky S, Chackalamannil S, Harrison P, Silvestri M. Synthetic studies toward aflavinine: a synthesis of 3-demethylaflavinine via a [2 + 2 + 2] annulation Journal of the American Chemical Society. 107: 2474-2484. DOI: 10.1021/Ja00294A046  0.607
1985 Danishefsky SJ, Harrison PJ, Webb RR, O'Neill BT. Total synthesis of quinocarcinol methyl ester Journal of the American Chemical Society. 107: 1421-1423. DOI: 10.1021/Ja00291A058  0.334
1985 Danishefsky S, Uang BJ, Quallich G. Total synthesis of vineomycinone B2 methyl ester Journal of the American Chemical Society. 107: 1285-1293. DOI: 10.1021/Ja00291A031  0.359
1985 Danishefsky SJ, Pearson WH, Segmuller BE. Total synthesis of (.+-.)-3-deoxy-D-manno-2-octulopyranosate Journal of the American Chemical Society. 107: 1280-1285. DOI: 10.1021/Ja00291A030  0.771
1985 Danishefsky SJ, Pearson WH, Harvey DF, Maring CJ, Springer JP. Chelation-controlled facially selective cyclocondensation reactions of chiral alkoxy aldehydes: syntheses of a mouse androgen and of a carbon-linked disaccharide Journal of the American Chemical Society. 107: 1256-1268. DOI: 10.1021/Ja00291A027  0.568
1985 Danishefsky S, Chackalamannil S, Harrison P, Silvestri M, Cole P. Synthetic Studies Toward Aflavinine: A Synthesis Of 3-Demethylaflavinine Via A (2 + 2 + 2) Annulation Cheminform. 16. DOI: 10.1002/Chin.198534342  0.696
1985 Danishefsky SJ, Uang BJ, Quallich G. Total Synthesis Of Vineomycinone B2 Methyl Ester Cheminform. 16. DOI: 10.1002/Chin.198529367  0.321
1985 Danishefsky S, Maring C. A new approach to the synthesis of hexoses: an entry to (.+-.)-fucose and (.+-.)-daunosamine Journal of the American Chemical Society. 107: 1269-1274. DOI: 10.1002/Chin.198529338  0.335
1984 Danishefsky S, Bednarski M, Izawa T, Maring C. A general route to 1-alkoxy-3-[(trimethylsilyl)oxy]-1,3-butadienes: vinylogous transesterification The Journal of Organic Chemistry. 49: 2290-2292. DOI: 10.1021/jo00186a044  0.56
1984 Danishefsky S, Webb RR. Lewis acid catalyzed cyclocondensations of formaldehyde with activated dienes: a direct route to pyranosidal pentoses Journal of Organic Chemistry. 49: 1955-1958. DOI: 10.1021/Jo00185A024  0.306
1984 Danishefsky S, Uang B, Quallich G. Additions and Corrections - Total Synthesis of Vinemycin B2Aglycon Journal of the American Chemical Society. 106: 5388-5388. DOI: 10.1021/Ja00330A602  0.399
1984 Danishefsky SJ, Pearson WH, Harvey D. On the relationship of topological and diastereofacial control in the Lewis acid catalyzed cyclocondensation reaction of alkoxyaldehydes with activated dienes: metal tunable asymmetric induction Journal of the American Chemical Society. 106: 2456-2458. DOI: 10.1021/Ja00320A051  0.571
1984 Danishefsky SJ, Pearson WH, Harvey DF. Diastereofacial control in the Lewis acid catalyzed cyclocondensation reaction of aldehydes with activated dienes: a synthesis of the Mus musculus pheromone Journal of the American Chemical Society. 106: 2455-2456. DOI: 10.1021/Ja00320A050  0.608
1984 Danishefsky S, Webb RRI. Lewis Acid Catalyzed Cyclocondensations Of Formaldehyde With Activated Dienes. A Direct Route To Pyranosidal Pentoses Cheminform. 15. DOI: 10.1002/Chin.198452208  0.306
1984 Danishefsky SJ, Pearson WH, Harvey DF. Diastereofacial Control In The Lewis Acid Catalyzed Cyclocondensation Reaction Of Aldehydes With Activated Dienes: A Synthesis Of The Mus Musculus Pheromone Cheminform. 15. DOI: 10.1002/Chin.198430344  0.605
1984 Danishefsky SJ, Uang BJ, Quallich G. Total Synthesis Of Vineomycin B2 Aglycon Cheminform. 15. DOI: 10.1002/Chin.198430338  0.333
1984 Danishefsky SJ, Pearson WH, Harvey DF. On The Relationship Of Topological And Diastereofacial Control In The Lewis Acid Catalyzed Cyclocondensation Reaction Of Alkoxyaldehydes With Activated Dienes: Metal Tunable Asymmetric Induction Cheminform. 15. DOI: 10.1002/Chin.198430102  0.562
1984 Danishefsky S, Chackalamannil S, Silvestri M, Springer J. Stereospecific 2 + 2 + 2 Annulation Cheminform. 15. DOI: 10.1002/Chin.198414176  0.661
1984 Bednarski M, Danishefsky S. On The Interactivity Of Chiral Auxiliaries With Chiral Catalysts In The Hetero Diels-Alder Reaction: A New Route To L-Glycolipids Cheminform. 15. DOI: 10.1002/Chin.198409318  0.6
1984 Larson ER, Danishefsky S. A Totally Synthetic Route To Lincosamine Cheminform. 15. DOI: 10.1002/Chin.198406320  0.347
1983 Danishefsky SJ, Pearson WH. A new strategy for the synthesis of spiro ketals Journal of Organic Chemistry. 15: 3865-3866. DOI: 10.1021/Jo00169A070  0.365
1983 Danishefsky S, Chackalamannil S, Silvestri M, Springer J. A stereospecific 2+2+2 annulation Journal of Organic Chemistry. 48: 3615-3616. DOI: 10.1021/Jo00168A067  0.583
1983 Bednarski M, Danishefsky S. On the interactivity of chiral auxiliaries with chiral catalysts in the hetero Diels-Alder reaction: a new route to L-glycolipids Journal of the American Chemical Society. 105: 6968-6969. DOI: 10.1021/Ja00361A042  0.6
1983 Larson ER, Danishefsky S. A totally synthetic route to lincosamine Journal of the American Chemical Society. 105: 6715-6716. DOI: 10.1021/Ja00360A030  0.347
1982 Danishefsky S, Etheredge SJ. Annulative route to enediones Journal of Organic Chemistry. 14: 4791-4793. DOI: 10.1021/Jo00145A042  0.304
1982 Danishefsky S, Kato N, Askin D, Kerwin JF. Stereochemical consequences of the Lewis acid catalyzed cyclocondensation of oxygenated dienes with aldehydes. A rapid and stereoselective entry to various natural products derived from propionate Journal of the American Chemical Society. 104: 360-362. DOI: 10.1021/Ja00365A096  0.31
1981 Danishefsky S, Regan J, Doehner R. Approaches to the synthesis of the mitomycins. A route to the mitosanes involving activated cyclopropanes The Journal of Organic Chemistry. 46: 5255-5261. DOI: 10.1021/Jo00339A001  0.362
1981 Danishefsky S, Vaughan K, Gadwood R, Tsuzuki K. Total synthesis of dl-quadrone Journal of the American Chemical Society. 103: 4136-4141. DOI: 10.1021/Ja00404A026  0.712
1981 Danishefsky S, Morris J, Clizbe LA. Total synthesis of pretyrosine (arogenate) Journal of the American Chemical Society. 103: 1602-1604. DOI: 10.1021/Ja00396A070  0.418
1980 Danishefsky S, Tsuzuki K. Control of remote relative chiralities: a stereospecific total synthesis of dl-widdrol Journal of the American Chemical Society. 102: 6891-6893. DOI: 10.1021/Ja00542A059  0.357
1980 Danishefsky S, Funk RL, Kerwin JF. Claisen rearrangements of lactonic (silyl) enolates: a new route to functionalized cycloalkenes Journal of the American Chemical Society. 102: 6889-6891. DOI: 10.1021/Ja00542A058  0.62
1980 Danishefsky S, Etheredge SJ. Simple Synthetic Route To Lasiodiplodin Cheminform. 11. DOI: 10.1002/Chin.198014290  0.351
1980 DANISHEFSKY S, YAN C, SINGH RK, GAMMILL RB, MCCURRY PMJ, FRITSCH N, CLARDY J. ChemInform Abstract: DERIVATIVES OF 1-METHOXY-3-TRIMETHYLSILYLOXY-1,3-BUTADIENE FOR DIELS-ALDER REACTIONS Chemischer Informationsdienst. 11. DOI: 10.1002/Chin.198007114  0.301
1979 Danishefsky S, Etheredge SJ. Simple synthetic route to lasiodiplodin Journal of Organic Chemistry. 44: 4716-4717. DOI: 10.1021/Jo00393A058  0.351
1979 Danishefsky S, Yan C, Singh RK, Gammill RB, McCurry PM, Fritsch N, Clardy J. Derivatives of 1-methoxy-3-trimethylsilyloxy-1,3-butadiene for Diels-Alder reactions Journal of the American Chemical Society. 101: 7001-7008. DOI: 10.1021/Ja00517A037  0.788
1979 Danishefsky S, Berman E, Clizbe LA, Hirama M. A simple synthesis of L-.gamma.-carboxyglutamate and derivatives thereof Journal of the American Chemical Society. 101: 4385-4386. DOI: 10.1021/Ja00509A062  0.313
1978 Danishefsky S, Hirama M, Gombatz K, Harayama T, Berman E, Schuda P. Stereospecific total synthesis of dl-pentalenolactone Journal of the American Chemical Society. 100: 6536-6538. DOI: 10.1021/Ja00488A063  0.408
1978 Danishefsky S, Hirama M. Total Synthesis Of Disodium Prephenate Cheminform. 9. DOI: 10.1002/Chin.197808327  0.418
1977 Danishefsky S, Hirama M. Total synthesis of disodium prephenate. Journal of the American Chemical Society. 99: 7740-7741. PMID 915167 DOI: 10.1021/Ja00465A072  0.418
1977 Danishefsky S, Yan CF, McCurry PM. A Diels-Alder route to functionalized cyclohexadienones Journal of Organic Chemistry. 42: 1819-1821. DOI: 10.1021/Jo00430A040  0.78
1977 Danishefsky S, Tsai M, Kitahara T. Specific directing effects in the opening of vicinal hydroxy epoxides The Journal of Organic Chemistry. 42: 394-396. DOI: 10.1021/Jo00422A066  0.487
1977 Danishefsky S, McKee R, Singh RK. Stereospecific total synthesis of dl-hastanecine and dl-dihydroxyheliotridane Journal of the American Chemical Society. 99: 7711-7713. DOI: 10.1021/Ja00465A054  0.381
1977 Danishefsky S, Schuda PF, Kitahara T, Etheredge SJ. The total synthesis of dl-vernolepin and dl-vernomenin Journal of the American Chemical Society. 99: 6066-6075. DOI: 10.1021/Ja00460A038  0.555
1977 DANISHEFSKY S, YAN CF, MCCURRY PMJ. ChemInform Abstract: A DIELS-ALDER ROUTE TO FUNCTIONALIZED CYCLOHEXADIENONES Chemischer Informationsdienst. 8: no-no. DOI: 10.1002/Chin.197743131  0.305
1977 Danishefsky S, Tsai M-, Kitahara T. Specific Directing Effects In The Opening Of Vicinal Hydroxy Epoxides Cheminform. 8. DOI: 10.1002/Chin.197722204  0.487
1977 Danishefsky S, Schuda PF, Mazza S, Kato K. Diels-Alder Reactions Of O-Benzoquinones. A Route To Derivatives Of Δ2-1-Octalone Cheminform. 8. DOI: 10.1002/Chin.197706171  0.304
1976 Danishefsky S, Zimmer A. The direction of base-catalyzed aldol cyclization of 1,5 diketones Journal of Organic Chemistry. 41: 4059-4064. DOI: 10.1021/Jo00888A002  0.355
1976 Danishefsky S, Schuda PF, Mazza S, Kato K. Diels-Alder reactions of o-benzoquinones. A route to derivatives of .DELTA.2-1-octalone Journal of Organic Chemistry. 41: 3468-3473. DOI: 10.1021/Jo00883A033  0.304
1976 Danishefsky S, Kitahara T, Tsai M, Dynak J. Functionalized alanes for the conversion of epoxides to trans-fused .gamma.-lactones The Journal of Organic Chemistry. 41: 1669-1671. DOI: 10.1021/Jo00871A052  0.478
1976 Danishefsky S, Kitahara T, McKee R, Schuda PF. Reactions of silyl enol ethers and lactone enolates with dimethyl(methylene)ammonium iodide. The bis-.alpha.-methylenation of pre-vernolepin and pre-vernomenin Journal of the American Chemical Society. 98: 6715-6717. DOI: 10.1021/Ja00437A058  0.503
1975 Danishefsky S, Cain P, Nagel A. Bis annelations via 6-methyl-2-vinylpyridine. Efficient synthesis of dl-D-homoestrone Journal of the American Chemical Society. 97: 380-387. PMID 1133355 DOI: 10.1021/Ja00835A028  0.319
1975 Danishefsky S, Cain P, Nagel A. Bis Annelations Via 6-Methyl-2-Vinylpyridine, An Efficient Synthesis Of Dl-D-Homoestrone Cheminform. 6. DOI: 10.1002/Chin.197514388  0.319
1975 Danishefsky S, Etheredge SJ. Synthesis And Biological Evaluation Of De-Ab-Camptothecin Cheminform. 6. DOI: 10.1002/Chin.197511473  0.361
1974 Danishefsky S, Etheredge SJ. Synthesis and biological evaluation of DE-AB-camptothecin. Journal of Organic Chemistry. 39: 3430-3432. PMID 4427189 DOI: 10.1021/Jo00937A034  0.361
1974 Danishefsky S, Etheredge SJ, Dynak J, McCurry P. Route to furanoid system by intramolecular homoconjugate addition Journal of Organic Chemistry. 39: 2658-2659. DOI: 10.1021/Jo00931A058  0.8
1971 Volkmann R, Danishefsky S, Eggler J, Solomon DM. Total synthesis of (+-)-camptothecine Journal of the American Chemical Society. 93: 5576-5577. DOI: 10.1021/ja00750a045  0.302
1971 Danishefsky S, Crawley LS, Solomon DM, Heggs P. Novel construction of steroid skeleton. Utility of di-tert-butyl acetonedicarboxylate Journal of the American Chemical Society. 93: 2356-2357. DOI: 10.1021/Ja00738A063  0.302
1967 Stork G, Danishefsky S, Ohashi M. Isoxazole annelation reaction. Method for the construction of cyclohexenone rings in polycyclic systems Journal of the American Chemical Society. 89: 5459-5460. DOI: 10.1021/Ja00997A031  0.513
1965 Danishefsky S, Cunningham R. The Reaction of Enamines with Activated Butadienes. A One-Step Synthesis of Benzenes1 Journal of Organic Chemistry. 30: 3676-3679. DOI: 10.1021/Jo01022A020  0.389
1962 Yates P, Danishefsky S. A Novel Type of Alkyl Shift Journal of the American Chemical Society. 84: 879-880. DOI: 10.1021/Ja00864A051  0.443
1961 Morrison H, Danishefsky S, Yates P. Communications- Preparation of α-Diazo Ketones The Journal of Organic Chemistry. 26: 2617-2618. DOI: 10.1021/Jo01351A658  0.57
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