| Year |
Citation |
Score |
| 2005 |
Frick JA, Klassen JB, Rapoport H. Diastereo- and enantioselective synthesis of 2-substituted 1-aminocyclopropane-1-carboxylic acids. Application to the synthesis of protected 2,3-methano analogs of ornithine and glutamic acid Synthesis. 1751-1756. DOI: 10.1055/S-2005-870007 |
0.393 |
|
| 2003 |
Rapoport H, Chen Y, Mohareb RM, Ahn JH, Sim TB, Ho JZ. An efficient procedure for the preparation of (1S,3R)- and (1S,3S)-1-amino-3-(hydroxymethyl)cyclopentanes. Chemical & Pharmaceutical Bulletin. 51: 1153-6. PMID 14519920 DOI: 10.1002/CHIN.200412213 |
0.321 |
|
| 2003 |
Hart BP, Verma SK, Rapoport H. Asymmetric synthesis of the carbapenam core from serine. The Journal of Organic Chemistry. 68: 187-90. PMID 12515481 DOI: 10.1021/Jo026499S |
0.384 |
|
| 2003 |
Paleo MR, Aurrecoechea N, Jung KY, Rapoport H. Formal enantiospecific synthesis of (+)-FR900482. The Journal of Organic Chemistry. 68: 130-8. PMID 12515471 DOI: 10.1021/Jo0206521 |
0.383 |
|
| 2003 |
Ho JZ, Mohareb RM, Ahn JH, Sim TB, Rapoport H. Enantiospecific synthesis of carbapentostatins. The Journal of Organic Chemistry. 68: 109-14. PMID 12515468 DOI: 10.1021/Jo020612X |
0.418 |
|
| 2003 |
McLaughlin M, Mohareb RM, Rapoport H. An efficient procedure for the preparation of 4-substituted 5-aminoimidazoles. The Journal of Organic Chemistry. 68: 50-4. PMID 12515460 DOI: 10.1021/Jo026257S |
0.386 |
|
| 2003 |
Jamison TF, Lubell WD, Dener JM, Krisché MJ, Rapoport H. 9‐Bromo‐9‐Phenylfluorene Organic Syntheses. 220-220. DOI: 10.1002/0471264180.Os071.28 |
0.618 |
|
| 2002 |
Holden KG, Mattson MN, Cha KH, Rapoport H. Synthesis of chiral pilocarpine analogues via a C-8 ketone intermediate. The Journal of Organic Chemistry. 67: 5913-8. PMID 12182622 DOI: 10.1021/Jo0111210 |
0.403 |
|
| 2002 |
Verma SK, Atanes MN, Busto JH, Thai DL, Rapoport H. Hydroxylated pyrrolidines. Enantiospecific synthesis of all-cis 2,3,4,5-substituted pyrrolidine derivatives from serine. The Journal of Organic Chemistry. 67: 1314-8. PMID 11846680 DOI: 10.1021/Jo011008+ |
0.385 |
|
| 2001 |
Lennox JR, Turner SC, Rapoport H. Enantiospecific synthesis of annulated nicotine analogues from D-glutamic acid. 7-Azabicyclo[2.2.1]heptano[2.3-c]pyridines. The Journal of Organic Chemistry. 66: 7078-83. PMID 11597233 DOI: 10.1021/Jo010534Y |
0.354 |
|
| 2000 |
Pickersgill IF, Rapoport H. Preparation of functionalized, conformationally constrained DTPA analogues from L- or D-serine and trans-4-hydroxy-L-proline. Hydroxymethyl substituents on the central acetic acid and on the backbone. The Journal of Organic Chemistry. 65: 4048-57. PMID 10866623 DOI: 10.1021/Jo000071G |
0.363 |
|
| 2000 |
Turner SC, Zhai H, Rapoport H. Enantiospecific synthesis of annulated nicotine analogues from D- and L- glutamic acid. Pyridotropanes Journal of Organic Chemistry. 65: 861-870. DOI: 10.1021/Jo991609P |
0.375 |
|
| 1999 |
Hart BP, Rapoport H. Conformationally Constrained 7-Azabicyclo[2.2.1]heptane Amino Acids. Synthesis of a Glutamic Acid Analogue. The Journal of Organic Chemistry. 64: 2050-2056. PMID 11674299 DOI: 10.1021/Jo982327C |
0.376 |
|
| 1999 |
Hurt CR, Lin R, Rapoport H. Enantiospecific Synthesis of (R)-4-Amino-5-oxo-1,3,4,5-tetrahydrobenz[cd]indole, an Advanced Intermediate Containing the Tricyclic Core of the Ergots. The Journal of Organic Chemistry. 64: 225-233. PMID 11674107 DOI: 10.1021/Jo981723S |
0.376 |
|
| 1999 |
Xu YZ, Choi J, Isabel Calaza M, Turner S, Rapoport H. Conformationally constrained nicotines. 1-Pyridinyl-7- azabicyclo[2.2.1]heptane and 1-pyridinyl-8-azabicyclo[3.2.1] octane analogues Journal of Organic Chemistry. 64: 4069-4078. DOI: 10.1021/Jo990130U |
0.346 |
|
| 1998 |
Folmer JJ, Acero C, Thai DL, Rapoport H. Synthesis of carbacephems from serine Journal of Organic Chemistry. 63: 8170-8182. DOI: 10.1021/Jo980592S |
0.391 |
|
| 1998 |
Lin R, Castells J, Rapoport H. Enantiospecific synthesis of natural (-)-cocaine and unnatural (+)- cocaine from D- and L- glutamic acid Journal of Organic Chemistry. 63: 4069-4078. DOI: 10.1021/Jo980153T |
0.304 |
|
| 1996 |
FRYDMAN B, DESPUY ME, RAPOPORT H. PYRROLES FROM AZAINDOLES. A SYNTHESIS OF PORPHOBILINOGEN. Journal of the American Chemical Society. 87: 3530-1. PMID 14322546 DOI: 10.1021/Ja01093A061 |
0.416 |
|
| 1996 |
Campbell JA, Rapoport H. Chirospecific Syntheses of Conformationally Constrained 7-Azabicycloheptane Amino Acids by Transannular Alkylation. The Journal of Organic Chemistry. 61: 6313-6325. PMID 11667473 DOI: 10.1021/Jo960759M |
0.594 |
|
| 1996 |
Berrée F, Chang K, Cobas A, Rapoport H. Synthesis of Anisolylated Aspartyl and Glutamyl Tripeptides. The Journal of Organic Chemistry. 61: 715-721. PMID 11666995 DOI: 10.1021/Jo951754C |
0.34 |
|
| 1996 |
Mattson MN, Rapoport H. A new method for expeditious ketone synthesis from acids via acyl hemiacetals Journal of Organic Chemistry. 61: 6071-6074. DOI: 10.1021/Jo9607471 |
0.369 |
|
| 1996 |
Hernández AS, Thaler A, Castells J, Rapoport H. Enantiospecific synthesis of (+)- and (-)-ferruginine from L-glutamic acid. Synthesis of tropanes via intramolecular iminium ion cyclization Journal of Organic Chemistry. 61: 314-323. DOI: 10.1021/Jo9515081 |
0.396 |
|
| 1995 |
Grote CW, Kim DJ, Rapoport H. Stereocontrolled synthesis of DTPA analogues branched in the ethylene unit Journal of Organic Chemistry. 60: 6987-6997. DOI: 10.1021/Jo00126A059 |
0.374 |
|
| 1995 |
Campbell JA, Lee WK, Rapoport H. Chirospecific syntheses of precursors of cyclopentane and cyclopentene carbocyclic nucleosides by [3 + 3]-coupling and transannular alkylation Journal of Organic Chemistry. 60: 4602-4616. DOI: 10.1021/Jo00119A044 |
0.582 |
|
| 1995 |
Hernández A, Marcos M, Rapoport H. Synthesis of (+)- and (-)-N-BOC-7-azabicyclo[2.2.1]heptan-2-ones, versatile intermediates for the enantiospecific synthesis of (+)-and (-)-epibatidine and analogues Journal of Organic Chemistry. 60: 2683-2691. DOI: 10.1021/Jo00114A015 |
0.403 |
|
| 1995 |
Nam KC, Rapoport H. Synthesis of deuterium labeled plant ethylene precursor Journal of Labelled Compounds and Radiopharmaceuticals. 36: 431-437. DOI: 10.1002/Jlcr.2580360505 |
0.348 |
|
| 1994 |
Chang HS, Bergmeier SC, Frick JA, Bathe A, Rapoport H. Synthesis of (1R,3R,5S)-1-Amino-3-(hydroxymethyl)bicyclo[3.1.0]hexane as a Precursor for the Synthesis of Carbocyclic Nucleosides The Journal of Organic Chemistry. 59: 5336-5342. DOI: 10.1021/Jo00097A040 |
0.34 |
|
| 1994 |
Peterli-Roth P, Maguire MP, León E, Rapoport H. Syntheses of 6-deaminosinefungin and (S)-6-methyl-6-deaminosinefungin Journal of Organic Chemistry. 59: 4186-4193. DOI: 10.1021/Jo00094A033 |
0.357 |
|
| 1994 |
Civitello ER, Rapoport H. Synthesis of the enantiomeric furobenzofurans, late precursors for the synthesis of (+)- and (-)-aflatoxins B1, B2, G1, and G2 Journal of Organic Chemistry. 59: 3775-3782. DOI: 10.1021/Jo00093A008 |
0.315 |
|
| 1994 |
Williams MA, Rapoport H. Synthesis of conformationally constrained DTPA analogues. Incorporation of the ethylenediamine units as aminopyrrolidines Journal of Organic Chemistry. 59: 3616-3625. DOI: 10.1021/Jo00092A022 |
0.37 |
|
| 1994 |
Hernandez A, Rapoport H. Conformationally constrained analogues of anatoxin. Chirospecific synthesis of s-Trans carbonyl ring-fused analogues Journal of Organic Chemistry. 59: 1058-1066. DOI: 10.1021/Jo00084A023 |
0.317 |
|
| 1994 |
Park KH, Rapoport H. Enantioselective synthesis of (1R,4S)-1-amino-4-(hydroxymethyl)-2-cyclopentene, a precursor for carbocyclic nucleoside synthesis Journal of Organic Chemistry. 59: 394-399. DOI: 10.1021/Jo00081A019 |
0.393 |
|
| 1993 |
Truong TV, Rapoport H. Chirospecific synthesis of the tetrahydroimidazodiazepinol aglycon of pentostatin and its analogs Journal of Organic Chemistry. 58: 6090-6096. DOI: 10.1021/Jo00074A041 |
0.383 |
|
| 1993 |
Bergmeier SC, Lee WK, Rapoport H. Chirospecific synthesis of (1S,3R)-1-amino-3-(hydroxymethyl)cyclopentane, a precursor for carbocyclic nucleoside synthesis. Intramolecular aziridine cyclizations The Journal of Organic Chemistry. 58: 5019-5022. DOI: 10.1021/Jo00070A050 |
0.394 |
|
| 1993 |
Bergmeier SC, Cobas AA, Rapoport H. Chirospecific synthesis of (1S,3R)-1-amino-3-(hydroxymethyl)cyclopentane, precursor for carbocyclic nucleoside synthesis. Dieckmann cyclization with an .alpha.-amino acid The Journal of Organic Chemistry. 58: 2369-2376. DOI: 10.1021/Jo00061A006 |
0.388 |
|
| 1993 |
Dener JM, Zhang LH, Rapoport H. An effective chirospecific synthesis of (+)-pilocarpine from L-aspartic acid Journal of Organic Chemistry. 58: 1159-1166. DOI: 10.1021/Jo00057A031 |
0.405 |
|
| 1993 |
Williams MA, Rapoport H. Synthesis of enantiomerically pure diethylenetriaminepentaacetic acid analogs. L-Phenylalanine as the educt for substitution at the central acetic acid Journal of Organic Chemistry. 58: 1151-1158. DOI: 10.1021/Jo00057A030 |
0.338 |
|
| 1992 |
Frick JA, Klassen JB, Bathe A, Abramson JM, Rapoport H. An Efficient Synthesis of Enantiomerically Pure (R)-(2-Benzyloxyethyl)oxirane from (S)-Aspartic Acid Synthesis. 1992: 621-623. DOI: 10.1055/S-1992-26176 |
0.395 |
|
| 1992 |
Bierer DE, O'Connell JF, Parquette JR, Thompson CM, Rapoport H. Regiospecific synthesis of the aminoimidazoquinoxaline (IQx) mutagens from cooked foods Journal of Organic Chemistry. 57: 1390-1405. DOI: 10.1021/Jo00031A017 |
0.584 |
|
| 1992 |
Civitello ER, Rapoport H. The regioselective cleavage of aryl tosylates by electrochemical reduction Journal of Organic Chemistry. 57: 834-840. DOI: 10.1021/Jo00029A010 |
0.315 |
|
| 1992 |
Park KK, Rapoport H. Synthesis of substituted 1H‐pyrrolo[3,2‐c]quinolines Journal of Heterocyclic Chemistry. 29: 1031-1032. DOI: 10.1002/Jhet.5570290464 |
0.312 |
|
| 1991 |
Gerspacher M, Rapoport H. 2-Amino-2-deoxyhexoses as chiral educts for hydroxylated indolizidines. Synthesis of (+)-castanospermine and (+)-6-epicastanospermine Journal of Organic Chemistry. 56: 3700-3706. DOI: 10.1021/Jo00011A047 |
0.351 |
|
| 1991 |
Bishop JE, Nagy JO, O'Connell JF, Rapoport H. Diastereoselective synthesis of phycocyanobilin-cysteine adducts Journal of the American Chemical Society. 113: 8024-8035. DOI: 10.1021/Ja00021A032 |
0.425 |
|
| 1990 |
Sardina FJ, Howard MH, Morningstar M, Rapoport H. Enantiodivergent synthesis of (+)- and (-)-anatoxin from L-glutamic acid Journal of Organic Chemistry. 55: 5025-5033. DOI: 10.1021/Jo00304A012 |
0.362 |
|
| 1990 |
Dunn PJ, Haener R, Rapoport H. Stereoselective synthesis of 2,3-diamino acids. 2,3-Diamino-4-phenylbutanoic acid Journal of Organic Chemistry. 55: 5017-5025. DOI: 10.1021/Jo00304A011 |
0.344 |
|
| 1990 |
Lubell WD, Jamison TF, Rapoport H. N-(9-phenylfluoren-9-yl)-α-amino ketones and N-(9-phenylfluoren-9-yl)-α-amino aldehydes as chiral educts for the synthesis of optically pure 4-alkyl-3-hydroxy-2-amino acids. Synthesis of the C-9 amino acid MeBmt present in cyclosporin Journal of Organic Chemistry. 55: 3511-3522. DOI: 10.1021/Jo00298A025 |
0.683 |
|
| 1990 |
Gmeiner P, Feldman PL, Chu-Moyer MY, Rapoport H. An efficient and practical total synthesis of (+)-vincamine from L-aspartic acid Journal of Organic Chemistry. 55: 3068-3074. DOI: 10.1021/Jo00297A023 |
0.375 |
|
| 1990 |
Howard MH, Sardina FJ, Rapoport H. Chirospecific syntheses of nitrogen and side-chain-modified anatoxin analogs. Synthesis of (1R)-anatoxinal and (1R)-anatoxinic acid derivatives Journal of Organic Chemistry. 55: 2829-2838. DOI: 10.1021/Jo00296A050 |
0.329 |
|
| 1990 |
Jones RJ, Rapoport H. Enantiospecific synthesis of an aziridinobenzazocinone, an advanced intermediate containing the core nucleus of FR900482 and FK973 Journal of Organic Chemistry. 55: 1144-1146. DOI: 10.1021/Jo00291A010 |
0.37 |
|
| 1990 |
VanSickle AP, Rapoport H. Azapsoralens. Synthesis of 8-azapsoralens Journal of Organic Chemistry. 55: 895-901. DOI: 10.1021/Jo00290A019 |
0.364 |
|
| 1989 |
Saljoughian M, Morimoto H, Rapoport H. Synthesis Of Monotritiomethyl Iodide From Thioethers: Hydrogenolysis In The Presence Of Thioethers Journal of Organic Chemistry. 54: 4689-4691. DOI: 10.1021/Jo00280A044 |
0.371 |
|
| 1989 |
Sardina FJ, Howard MH, Koskinen AMP, Rapoport H. Chirospecific synthesis of nitrogen and side chain modified analogs of (+)-anatoxin Journal of Organic Chemistry. 54: 4654-4660. DOI: 10.1021/Jo00280A037 |
0.38 |
|
| 1989 |
Lubell W, Rapoport H. Surrogates for chiral aminomalondialdehyde. Synthesis of N-(9-phenylfluoren-9-yl)serinal and N-(9-phenylfluoren-9-yl)vinylglycinal The Journal of Organic Chemistry. 54: 3824-3831. DOI: 10.1021/Jo00277A016 |
0.543 |
|
| 1989 |
Wolf JP, Rapoport H. Conformationally constrained peptides. Chirospecific synthesis of 4-alkyl-substituted .gamma.-lactam-bridged dipeptides from L-aspartic acid Journal of Organic Chemistry. 54: 3164-3173. DOI: 10.1021/Jo00274A037 |
0.318 |
|
| 1989 |
Bishop JE, Dagam SA, Rapoport H. Synthesis and characterization of monothiosuccinimides Journal of Organic Chemistry. 54: 1876-1883. DOI: 10.1021/Jo00269A024 |
0.408 |
|
| 1989 |
Roemmele RC, Rapoport H. Chirospecific synthesis of .beta.-hydroxy .alpha.-amino acids Journal of Organic Chemistry. 54: 1866-1875. DOI: 10.1021/Jo00269A023 |
0.316 |
|
| 1989 |
Koskinen AMP, Rapoport H. Synthesis of 4-substituted prolines as conformationally constrained amino acid analogs Journal of Organic Chemistry. 54: 1859-1866. DOI: 10.1021/Jo00269A022 |
0.388 |
|
| 1989 |
Saljoughian M, Morimoto H, Dorsky AM, Rapoport H, Andres H. A new and efficient synthesis of monotritiomethyl iodide Journal of Labelled Compounds and Radiopharmaceuticals. 27: 767-776. DOI: 10.1002/Jlcr.2580270705 |
0.387 |
|
| 1988 |
Lagarias JC, Klotz AV, Dallas JL, Glazer AN, Bishop JE, O'Connell JF, Rapoport H. Exclusive A-ring linkage for singly attached phycocyanobilins and phycoerythrobilins in phycobiliproteins. Absence of singly D-ring-linked bilins. The Journal of Biological Chemistry. 263: 12977-85. PMID 3417648 |
0.482 |
|
| 1988 |
O'Connell JF, Parquette J, Yelle WE, Wang W, Rapoport H. Convenient synthesis of methyl 1-methyl-2,4-dibromo-5-imidazolecarboxylate Synthesis. 1988: 767-771. DOI: 10.1055/S-1988-27702 |
0.31 |
|
| 1988 |
Lubell WD, Rapoport H. .alpha.-Amino acids as chiral educts for asymmetric products. Alkylation of N-phenylfluorenyl .alpha.-amino ketones. Synthesis of optically pure .alpha.-alkyl carboxylic acids Journal of the American Chemical Society. 110: 7447-7455. DOI: 10.1021/Ja00230A027 |
0.556 |
|
| 1988 |
Saljoughian M, Morimoto H, Rapoport H. A new route to the synthesis of multi-tritiated methyl iodide International Journal of Radiation Applications and Instrumentation. Part a. Applied Radiation and Isotopes. 39: 607. DOI: 10.1016/0883-2889(88)90382-6 |
0.354 |
|
| 1987 |
Maurer PJ, Rapoport H. Nitrogen-bridged conformationally constrained etorphine analogues. Synthesis and biological evaluation. Journal of Medicinal Chemistry. 30: 2016-26. PMID 3669010 DOI: 10.1021/Jm00394A016 |
0.336 |
|
| 1987 |
Feldman PL, Rapoport H. Synthesis of (-)-vindoline Journal of the American Chemical Society. 109: 1603-1604. DOI: 10.1021/Ja00239A069 |
0.406 |
|
| 1987 |
Bishop JE, Rapoport H, Klotz AV, Chan CF, Glazer AN, Fueglistaller P, Zuber H. Chromopeptides from phycoerythrocyanin. Structure and linkage of the three bilin groups Journal of the American Chemical Society. 109: 875-881. DOI: 10.1021/Ja00237A039 |
0.317 |
|
| 1987 |
Lubell WD, Rapoport H. Configurational stability of N-protected .alpha.-amino aldehydes Journal of the American Chemical Society. 109: 236-239. DOI: 10.1021/Ja00235A035 |
0.551 |
|
| 1986 |
Rapoport H, Waterhouse AL, Thompson CM, O'Connell JF. Synthesis and radiolabeling of heterocyclic food mutagens. Environmental Health Perspectives. 67: 41-5. PMID 3757958 DOI: 10.1289/Ehp.866741 |
0.639 |
|
| 1986 |
Bishop JE, Lagarias JC, Nagy JO, Schoenleber RW, Rapoport H, Klotz AV, Glazer AN. Phycobiliprotein-bilin linkage diversity. I. Structural studies on A- and D-ring-linked phycocyanobilins. The Journal of Biological Chemistry. 261: 6790-6. PMID 3084489 |
0.467 |
|
| 1986 |
Feldman PL, Rapoport H. Convenient Synthesis of 6-Methoxyindole and 6-Methoxytryptophyl Bromide Synthesis. 1986: 735-737. DOI: 10.1055/S-1986-31759 |
0.421 |
|
| 1986 |
Boutin RH, Rapoport H. .alpha.-Amino acid derivatives as chiral educts for asymmetric products. Synthesis of sphingosine from .alpha.'-amino-.alpha.,.beta.-ynones Journal of Organic Chemistry. 51: 5320-5327. DOI: 10.1021/Jo00376A050 |
0.301 |
|
| 1986 |
Feldman PL, Rapoport H. Synthesis of optically pure .DELTA.4-tetrahydroquinolinic acids and hexahydroindolo[2,3-a]quinolizines from L-aspartic acid. Racemization on the route to vindoline Journal of Organic Chemistry. 51: 3882-3890. DOI: 10.1021/Jo00370A025 |
0.329 |
|
| 1986 |
Moyer MP, Feldman PL, Rapoport H. Intramolecular N-H, O-H and S-H Insertion Reactions. Synthesis of Heterocycles from α-Diazo β-Keto Esters. Cheminform. 17. DOI: 10.1002/Chin.198623110 |
0.303 |
|
| 1986 |
Shaw KJ, Luly JR, Rapoport H. Routes to Mitomycins. Chirospecific Synthesis of Aziridinomitosenes. Cheminform. 17. DOI: 10.1002/Chin.198618364 |
0.389 |
|
| 1986 |
Cupps TL, Boutin RH, Rapoport H. α-Amino Acids as Chiral Educts for Asymmetric Products. The Synthesis of α′-Amino-α,β-ynones. Cheminform. 17. DOI: 10.1002/Chin.198609130 |
0.315 |
|
| 1985 |
Koskinen AM, Rapoport H. Synthetic and conformational studies on anatoxin-a: a potent acetylcholine agonist. Journal of Medicinal Chemistry. 28: 1301-9. PMID 4032432 DOI: 10.1002/Chin.198552240 |
0.609 |
|
| 1985 |
Knipmeyer LL, Rapoport H. Analgesics of the 6,14-ethenomorphinan type. 6-deoxy-7 alpha-orvinols and 6-deoxy-8 alpha-orvinols. Journal of Medicinal Chemistry. 28: 461-6. PMID 3981537 DOI: 10.1021/Jm00382A013 |
0.324 |
|
| 1985 |
Shaw KJ, Luly JR, Rapoport H. Routes to mitomycins. Chirospecific synthesis of aziridinomitosenes Journal of Organic Chemistry. 50: 4515-4523. DOI: 10.1021/Jo00223A019 |
0.389 |
|
| 1985 |
Cupps TL, Boutin RH, Rapoport H. .alpha.-Amino acids as chiral educts for asymmetric products. The synthesis of .alpha.'-amino-.alpha.,.beta.-ynones Journal of Organic Chemistry. 50: 3972-3979. DOI: 10.1021/Jo00221A004 |
0.312 |
|
| 1985 |
Christie BD, Rapoport H. Synthesis of optically pure pipecolates from L-asparagine. Application to the total synthesis of (+)-apovincamine through amino acid decarbonylation and iminium ion cyclization Journal of Organic Chemistry. 50: 1239-1246. DOI: 10.1021/Jo00208A017 |
0.356 |
|
| 1985 |
Shiosaki K, Rapoport H. .alpha.-Amino acids as chiral educts for asymmetric products. Chirospecific syntheses of the 5-butyl-2-heptylpyrrolidines from glutamic acid Journal of Organic Chemistry. 50: 1229-1239. DOI: 10.1021/Jo00208A016 |
0.321 |
|
| 1985 |
Maurer PJ, Knudsen CG, Palkowitz AD, Rapoport H. .alpha.-Amino acids as chiral educts for asymmetric products. Chirospecific syntheses of methyl L-sibirosaminide and its C-3 epimer from L-allothreonine Journal of Organic Chemistry. 50: 325-332. DOI: 10.1021/Jo00203A008 |
0.323 |
|
| 1985 |
Waddell TG, Rapoport H. Synthesis of [3-14C]-2′-methylreticuline and its incorporation into alkaloid fractions of Papaver somniferum Phytochemistry. 24: 469-472. DOI: 10.1016/S0031-9422(00)80749-9 |
0.345 |
|
| 1985 |
Waterhouse AL, Rapoport H. Synthesis and tritium labeling of the food mutagens IQ and methyl‐IQ Journal of Labelled Compounds and Radiopharmaceuticals. 22: 201-216. DOI: 10.1002/Jlcr.2580220302 |
0.577 |
|
| 1985 |
Bauman JG, Hawley RC, Rapoport H. An Efficient Synthesis Of Aklavinone And Related 11-Deoxyanthracyclinones Cheminform. 16. DOI: 10.1002/Chin.198537331 |
0.343 |
|
| 1985 |
Christie BD, Rapoport H. Synthesis Of Optically Pure Pipecolates From L-Asparagine. Application To The Total Synthesis Of (+)-Apovincamine Through Amino Acid Decarbonylation And Iminium Ion Cyclization Cheminform. 16. DOI: 10.1002/Chin.198535327 |
0.356 |
|
| 1985 |
Duclos RIJ, Tung JS, Rapoport H. A High-Yield Modification Of The Pschorr Phenanthrene Synthesis Cheminform. 16. DOI: 10.1002/Chin.198528147 |
0.377 |
|
| 1985 |
Maurer PJ, Knudsen CG, Palkowitz AD, Rapoport H. α-AMINO ACIDS AS CHIRAL EDUCTS FOR ASYMMETRIC PRODUCTS. CHIROSPECIFIC SYNTHESES OF METHYL L-SIBIROSAMINIDE AND ITS C-3 EPIMER FROM L-ALLOTHREONINE Cheminform. 16. DOI: 10.1002/Chin.198525359 |
0.324 |
|
| 1985 |
Bauman JG, Hawley RC, Rapoport H. Synthesis Of A Cyclohexadiene Monoepoxide By Intramolecular Darzens Condensation. Efficient Synthesis Of An A Ring Anthracyclinone Precursor Cheminform. 16. DOI: 10.1002/Chin.198511186 |
0.412 |
|
| 1985 |
Petersen JS, Toeteberg-Kaulen S, Rapoport H. Synthesis Of (.+-.)-Ω-Aza(X.Y.1)Bicycloalkanes By An Intramolecular Mannich Reaction Cheminform. 16. DOI: 10.1002/Chin.198503253 |
0.668 |
|
| 1984 |
Kanne D, Rapoport H, Hearst JE. 8-Methoxypsoralen-nucleic acid photoreaction. Effect of methyl substitution on pyrone vs. furan photoaddition. Journal of Medicinal Chemistry. 27: 531-4. PMID 6708053 DOI: 10.1021/Jm00370A017 |
0.55 |
|
| 1984 |
Hutchins CW, Rapoport H. Analgesics of the orvinol type. 19-Deoxy and 6,20-epoxy derivatives. Journal of Medicinal Chemistry. 27: 521-7. PMID 6708052 DOI: 10.1002/Chin.198438334 |
0.314 |
|
| 1984 |
Hearst JE, Isaacs ST, Kanne D, Rapoport H, Straub K. The reaction of the psoralens with deoxyribonucleic acid. Quarterly Reviews of Biophysics. 17: 1-44. PMID 6385057 DOI: 10.1017/S0033583500005242 |
0.524 |
|
| 1984 |
Duclos RI, Tung JS, Rapoport H. A high-yield modification of the Pschorr phenanthrene synthesis Journal of Organic Chemistry. 49: 5243-5246. DOI: 10.1021/Jo00200A046 |
0.367 |
|
| 1984 |
Castellino AJ, Rapoport H. Synthesis of benzofurans from oxygenated phenoxyamines Journal of Organic Chemistry. 49: 4399-4404. DOI: 10.1021/Jo00197A014 |
0.356 |
|
| 1984 |
Bauman JG, Hawley RC, Rapoport H. Synthesis of a cyclohexadiene monoepoxide by intramolecular darzens condensation efficient synthesis of an a ring anthracyclinone precursor Journal of Organic Chemistry. 49: 3791-3796. DOI: 10.1021/Jo00194A023 |
0.36 |
|
| 1984 |
Petersen JS, Toeteberg-Kaulen S, Rapoport H. Synthesis of (.+-.)-.omega.-aza[x.y.1]bicycloalkanes by an intramolecular Mannich reaction Journal of Organic Chemistry. 49: 2948-2953. DOI: 10.1021/Jo00190A020 |
0.671 |
|
| 1984 |
Luly JR, Rapoport H. Routes to mitomycins. An improved synthesis of 7-methoxymitosene using palladium catalysis Journal of Organic Chemistry. 49: 1671-1672. DOI: 10.1021/Jo00183A042 |
0.375 |
|
| 1984 |
Castellino AJ, Rapoport H. Synthesis of phenoxyamines Journal of Organic Chemistry. 49: 1348-1352. DOI: 10.1021/Jo00182A007 |
0.342 |
|
| 1984 |
Rosenberg SH, Rapoport H. Convergent and efficient synthesis of spiro[benzofuran-3(2H),4'-piperidines] Journal of Organic Chemistry. 49: 56-62. DOI: 10.1021/Jo00175A011 |
0.338 |
|
| 1984 |
Petersen JS, Fels G, Rapoport H. Chirospecific syntheses of (+)- and (-)-anatoxin a Journal of the American Chemical Society. 106: 4539-4547. DOI: 10.1021/Ja00328A040 |
0.69 |
|
| 1984 |
Schoenleber RW, Kim Y, Rapoport H. Relative stereochemistry of the A ring of plant bile pigments Journal of the American Chemical Society. 106: 2645-2651. DOI: 10.1021/Ja00321A026 |
0.344 |
|
| 1984 |
Maurer PJ, Takahata H, Rapoport H. .alpha.-Amino acids as chiral educts for asymmetric products. A general synthesis of D-.alpha.-amino acids from L-serine Journal of the American Chemical Society. 106: 1095-1098. DOI: 10.1021/Ja00316A047 |
0.324 |
|
| 1984 |
Petersen JS, Fels G, Rapoport H. Chirospecific Syntheses Of (+)- And (-)-Anatoxin A Cheminform. 15. DOI: 10.1002/Chin.198447346 |
0.69 |
|
| 1984 |
Luly JR, Rapoport H. Routes To Mitomycins. An Improved Synthesis Of 7-Methoxymitosene Using Palladium Catalysis Cheminform. 15. DOI: 10.1002/Chin.198440160 |
0.375 |
|
| 1984 |
Maurer PJ, Takahata H, Rapoport H. α-Amino Acids as Chiral Educts for Asymmetric Products. A General Synthesis of D-α-Amino Acids from L-Serine. Cheminform. 15. DOI: 10.1002/Chin.198421322 |
0.332 |
|
| 1984 |
Buckley TFI, Rapoport H. α-Amino Acids as Chiral Educts for Asymmetric Products. Chirally Specific Syntheses of Tylophorine and Cryptopleurine. Cheminform. 15. DOI: 10.1002/Chin.198418340 |
0.335 |
|
| 1984 |
Bender DR, Kanne D, Frazier JD, Rapoport H. Synthesis and Derivatization of 8-Acetylpsoralens. Acetyl Migrations During Claisen Rearrangement. Cheminform. 15. DOI: 10.1002/Chin.198401213 |
0.395 |
|
| 1983 |
Kim SH, Peckler S, Graves B, Kanne D, Rapoport H, Hearst JE. Sharp kink of DNA at psoralen-cross-link site deduced from crystal structure of psoralen-thymine monoadduct. Cold Spring Harbor Symposia On Quantitative Biology. 47: 361-5. PMID 6574850 DOI: 10.1101/Sqb.1983.047.01.042 |
0.461 |
|
| 1983 |
Bender DR, Kanne D, Frazier JD, Rapoport H. Synthesis and derivatization of 8-acetylpsoralens. Acetyl migrations during Claisen rearrangement Journal of Organic Chemistry. 48: 2709-2719. DOI: 10.1021/Jo00164A015 |
0.395 |
|
| 1983 |
Knudsen CG, Rapoport H. .alpha.-Amino acids as chiral educts for asymmetric products. Aminoacylation of metallo alkyls and alkenyls Journal of Organic Chemistry. 48: 2260-2266. DOI: 10.1021/Jo00161A023 |
0.325 |
|
| 1983 |
Moos WH, Gless RD, Rapoport H. Codeine analogs. Synthesis of 4a-aryldecahydroisoquinolines containing nitrogen ring functionality and of octahydro-1H-indeno[1,2,3-ef]isoquinolines. A total synthesis of codeine Journal of Organic Chemistry. 48: 227-238. DOI: 10.1021/Jo00150A017 |
0.658 |
|
| 1983 |
Luly JR, Rapoport H. Routes to mitomycins. New syntheses of the 2,3,5,8-tetrahydro-5,8-dioxo-1H-pyrrolo[1,2-a]indole ring system. An efficient synthesis of 7-methoxymitosene Journal of the American Chemical Society. 105: 2859-2866. DOI: 10.1021/Ja00347A055 |
0.386 |
|
| 1983 |
Lagarias JC, Yokoyama WH, Bordner J, Shih WC, Klein MP, Rapoport H. Cyclopeptide alkaloids. Conformational analysis of the dihydro-p-phencyclopeptine nucleus Journal of the American Chemical Society. 105: 1031-1040. DOI: 10.1021/Ja00342A064 |
0.522 |
|
| 1983 |
Knudsen CG, Rapoport H. .alpha.-Amino acids as chiral educts for asymmetric products. Aminoacylation of metallo alkyls and alkenyls Cheminform. 14. DOI: 10.1002/Chin.198348138 |
0.325 |
|
| 1983 |
Moos WH, Gless RD, Rapoport H. Codeine Analogs. Synthesis Of 4A‐Aryldecahydroisoquinolines Containing Nitrogen Ring Functionality And Of Octahydro‐1H‐Indeno(1,2,3‐Ef)Isoquinolines. A Total Synthesis Of Codeine Cheminform. 14. DOI: 10.1002/Chin.198323256 |
0.676 |
|
| 1982 |
Peckler S, Graves B, Kanne D, Rapoport H, Hearst JE, Kim SH. Structure of a psoralen-thymine monoadduct formed in photoreaction with DNA. Journal of Molecular Biology. 162: 157-72. PMID 7154093 DOI: 10.1016/0022-2836(82)90166-8 |
0.498 |
|
| 1982 |
Kanne D, Straub K, Rapoport H, Hearst JE. Psoralen-deoxyribonucleic acid photoreaction. Characterization of the monoaddition products from 8-methoxypsoralen and 4,5'8-trimethylpsoralen. Biochemistry. 21: 861-71. PMID 7074056 DOI: 10.1021/Bi00534A008 |
0.519 |
|
| 1982 |
Moos WH, Gless RD, Rapoport H. Codeine analogs. Synthesis of 4a-(2,3-dimethoxyphenyl)decahydroisoquinolines and octahydro-1H-[1]benzopyrano[4,3,2-e,f]isoquinolines Journal of Organic Chemistry. 47: 1831-1837. DOI: 10.1021/Jo00349A006 |
0.607 |
|
| 1982 |
Watkins BE, Rapoport H. Synthesis of benzyl and benzyloxycarbonyl base-blocked 2'-deoxyribonucleosides Journal of Organic Chemistry. 14: 4471-4477. DOI: 10.1021/Jo00144A014 |
0.383 |
|
| 1982 |
Kashdan DS, Schwartz JA, Rapoport H. Synthesis of 1,2,3,4-Tetrahydroisoquinolines Journal of Organic Chemistry. 13: 2638-2643. DOI: 10.1021/Jo00134A025 |
0.409 |
|
| 1982 |
Panetta JA, Rapoport H. Synthesis of thiocoumarins from acrylic and propiolic ortho esters and benzenethiols Journal of Organic Chemistry. 13: 2626-2628. DOI: 10.1021/Jo00134A022 |
0.436 |
|
| 1982 |
Luly JR, Rapoport H. Routes to mitomycins. Application of iminium salts to the synthesis of 7-methoxymitosene Journal of Organic Chemistry. 13: 2404-2413. DOI: 10.1021/Jo00133A034 |
0.363 |
|
| 1982 |
Kanne D, Straub K, Hearst JE, Rapoport H. Isolation and characterization of pyrimidine-psoralen-pyrimidine photodiadducts from DNA Journal of the American Chemical Society. 104: 6754-6764. DOI: 10.1021/Ja00388A046 |
0.478 |
|
| 1982 |
Watkins BE, Kiely JS, Rapoport H. Synthesis of oligodeoxyribonucleotides using N-benzyloxycarbonyl-blocked nucleosides Journal of the American Chemical Society. 104: 5702-5708. DOI: 10.1021/Ja00385A026 |
0.324 |
|
| 1982 |
Buckley TF, Rapoport H. Mild and simple biomimetic conversion of amines to carbonyl compounds Journal of the American Chemical Society. 104: 4446-4450. DOI: 10.1021/Ja00380A019 |
0.307 |
|
| 1982 |
Isaacs ST, Rapoport H, Hearst JE. Synthesis of deuterium and tritium labeled psoralens Journal of Labelled Compounds and Radiopharmaceuticals. 19: 345-356. DOI: 10.1002/Jlcr.2580190306 |
0.554 |
|
| 1982 |
Moos WH, Gless RD, Rapoport H. Codeine analogs. Synthesis of 4a-(2,3-dimethoxyphenyl)decahydroisoquinolines and octahydro-1H-[1]benzopyrano[4,3,2-e,f]isoquinolines Cheminform. 13. DOI: 10.1002/Chin.198243245 |
0.616 |
|
| 1982 |
Moos WH, Gless RD, Rapoport H. Codeine Analogs. Synthesis Of Spiro(Benzofuran‐3(2H)4′‐Piperidines) And Octahydro‐1H‐Benzofuro(3,2‐E)Isoquinolines Cheminform. 13. DOI: 10.1002/Chin.198222242 |
0.605 |
|
| 1982 |
Johansen JE, Christie BD, Rapoport H. Iminium salts from .alpha.-amino acid decarbonylation. Application to the synthesis of octahydroindolo[2,3-a]quinolizines Cheminform. 13. DOI: 10.1002/Chin.198216329 |
0.336 |
|
| 1981 |
Hutchins CW, Cooper GK, Pürro S, Rapoport H. 6-Demethoxythebaine and its conversion to analgesics of the 6,14-ethenomorphinan type. Journal of Medicinal Chemistry. 24: 773-7. PMID 7277381 DOI: 10.1002/Chin.198147294 |
0.311 |
|
| 1981 |
Gendler PL, Rapoport H. Permethyl analogue of the pyrrolic antibiotic distamycin A. Journal of Medicinal Chemistry. 24: 33-8. PMID 7009865 DOI: 10.1021/Jm00133A008 |
0.4 |
|
| 1981 |
Moos WH, Gless RD, Rapoport H. Codeine analogs. Synthesis of spiro[benzofuran-3(2H)4'-piperidines] and octahydro-1H-benzofuro[3,2-e]isoquinolines Journal of Organic Chemistry. 46: 5064-5074. DOI: 10.1021/Jo00338A003 |
0.61 |
|
| 1981 |
Johansen JE, Christie BD, Rapoport H. Iminium salts from .alpha.-amino acid decarbonylation. Application to the synthesis of octahydroindolo[2,3-a]quinolizines Journal of Organic Chemistry. 46: 4914-4920. DOI: 10.1021/Jo00337A018 |
0.336 |
|
| 1981 |
Luly JR, Rapoport H. Amine addition to unsymmetrical benzoquinones Journal of Organic Chemistry. 12: 2745-2752. DOI: 10.1021/Jo00326A029 |
0.373 |
|
| 1981 |
Ghera E, David YB, Rapoport H. Synthesis of functionalized quinoline derivatives by annulation of pyridines Journal of Organic Chemistry. 12: 2059-2065. DOI: 10.1021/Jo00323A016 |
0.381 |
|
| 1981 |
Buckley TF, Rapoport H. .alpha.-Amino acids as chiral educts for asymmetric products. Amino acylation with N-acylamino acids Journal of the American Chemical Society. 103: 6157-6163. DOI: 10.1021/Ja00410A030 |
0.318 |
|
| 1981 |
Straub K, Kanne D, Hearst JE, Rapoport H. Isolation and characterization of pyrimidine-psoralen photoadducts from DNA Journal of the American Chemical Society. 103: 2347-2355. DOI: 10.1021/Ja00399A035 |
0.497 |
|
| 1980 |
Goff D, Lagarias JC, Shih WC, Klein MP, Rapoport H. Cyclopeptide alkaloids. Synthetic, spectroscopic and conformational studies of phencyclopeptine model compounds The Journal of Organic Chemistry. 45: 4813-4817. DOI: 10.1021/Jo01312A001 |
0.575 |
|
| 1980 |
Falling SN, Rapoport H. Routes to mitomycins. Application of iminium salts to the synthesis of naphthoquinone mitosene analogs Journal of Organic Chemistry. 45: 1260-1270. DOI: 10.1021/Jo01295A020 |
0.376 |
|
| 1980 |
Lagarias JC, Rapoport H. Chromopeptides from phytochrome. The structure and linkage of the PR form of the phytochrome chromophore Journal of the American Chemical Society. 102: 4821-4828. DOI: 10.1021/Ja00534A042 |
0.502 |
|
| 1980 |
Buckley TF, Rapoport H. Dependence of aryl ether acylation upon Lewis acid stoichiometry Journal of the American Chemical Society. 102: 3056-3062. DOI: 10.1021/Ja00529A031 |
0.33 |
|
| 1980 |
Falling SN, Rapoport H. Routes To Mitomycins. Application Of Iminium Salts To The Synthesis Of Naphthoquinone Mitosene Analogs Cheminform. 11. DOI: 10.1002/Chin.198030345 |
0.376 |
|
| 1980 |
Padgett HC, Csendes IG, Rapoport H. The Alkoxycarbonyl Moiety As Blocking Group. A Generally Useful Variation Of The Malonic Ester Synthesis Cheminform. 11. DOI: 10.1002/Chin.198006176 |
0.34 |
|
| 1979 |
Lagarias JC, Goff D, Klein FK, Rapoport H. Cyclopeptide Alkaloids. Phencyclopeptines From the Polymorphic Species Ceanothus integerrimus. Journal of Natural Products. 42: 220-227. PMID 27802386 DOI: 10.1021/Np50002A013 |
0.439 |
|
| 1979 |
Csendes IG, Lee YY, Padgett HC, Rapoport H. Iminium salts from .alpha.-amino acid decarbonylation. Application to the synthesis of some 1-azabicyclo[x.y.0]systems Journal of Organic Chemistry. 11: 4173-4178. DOI: 10.1021/Jo01337A034 |
0.313 |
|
| 1979 |
Padgett HC, Csendes IG, Rapoport H. The alkoxycarbonyl moiety as blocking group. A generally useful variation of the malonic ester synthesis Journal of Organic Chemistry. 44: 3492-3496. DOI: 10.1021/Jo01334A009 |
0.34 |
|
| 1979 |
Hauske JR, Rapoport H. A New And Convenient Synthesis Of 2-Deoxy-D-Ribose From 2 ,4-O-Ethylidene-D-Erythrose Journal of Organic Chemistry. 44: 2472-2476. DOI: 10.1021/Jo01328A029 |
0.31 |
|
| 1979 |
Bender DR, Hearst JE, Rapoport H. Psoralen synthesis. Improvements in furano ring formation. Application to the synthesis of 4,5′,8-trimethylpsoralen Journal of Organic Chemistry. 44: 2176-2180. DOI: 10.1021/Jo01327A030 |
0.595 |
|
| 1979 |
Hannan RL, Barber RB, Rapoport H. Synthesis of bromonaphthoquinones from 1,5-dimethoxynaphthalene Journal of Organic Chemistry. 10: 2153-2158. DOI: 10.1021/Jo01327A025 |
0.407 |
|
| 1979 |
Houghten RA, Simpson RA, Hanson RN, Rapoport H. Bicyclic guanidino ketones Journal of Organic Chemistry. 11: 4536-4543. DOI: 10.1021/Jo00393A017 |
0.369 |
|
| 1979 |
Lagarias JC, Glazer AN, Rapoport H. Chromopeptides from C-phycocyanin. Structure and linkage of a phycocyanobilin bound to the .beta. subunit Journal of the American Chemical Society. 101: 5030-5037. DOI: 10.1021/Ja00511A038 |
0.508 |
|
| 1979 |
Bates HA, Rapoport H. Synthesis of anatoxin a via intramolecular cyclization of iminium salts Journal of the American Chemical Society. 101: 1259-1265. DOI: 10.1021/Ja00499A035 |
0.397 |
|
| 1979 |
Dean RT, Rapoport H. STEREOSPECIFIC CYCLIZATIONS OF IMINIUM SALTS FROM α‐AMINO ACID DECARBONYLATION. SYNTHESIS OF 8‐ AND 13‐METHYLBERBINES Cheminform. 10. DOI: 10.1002/Chin.197913381 |
0.395 |
|
| 1978 |
Barker P, Gendler P, Rapoport H. 2-(Trichloroacetyl)pyrroles as intermediates in the preparation of 2,4-disubstituted pyrroles Journal of Organic Chemistry. 10: 4849-4853. DOI: 10.1021/Jo00419A029 |
0.377 |
|
| 1978 |
Dean RT, Rapoport H. Stereospecific cyclizations of iminium salts from .alpha.-amino acid decarbonylation. Synthesis of 8- and 13-methylberbines Journal of Organic Chemistry. 43: 4183-4189. DOI: 10.1021/Jo00415A043 |
0.353 |
|
| 1978 |
Dean RT, Rapoport H. Iminium salts from .alpha.-amino acid decarbonylation. Application to the synthesis of berbines Journal of Organic Chemistry. 43: 2115-2122. DOI: 10.1021/Jo00405A006 |
0.335 |
|
| 1978 |
Lagarias JC, Houghten RA, Rapoport H. Cyclopeptide alkaloids. Synthesis of the ring system and its ion affinity Journal of the American Chemical Society. 100: 8202-8209. DOI: 10.1021/Ja00494A030 |
0.551 |
|
| 1978 |
Musich JA, Rapoport H. Synthesis of anthopleurine, the alarm pheromone from Anthopleura elegantissima Journal of the American Chemical Society. 100: 4865-4872. DOI: 10.1021/Ja00483A037 |
0.402 |
|
| 1978 |
Schmidtchen FP, Rapoport H. Polyprenylpyridinols. Synthesis Of Piericidin Analogs Cheminform. 9. DOI: 10.1002/Chin.197803371 |
0.412 |
|
| 1977 |
Isaacs ST, Shen CK, Hearst JE, Rapoport H. Synthesis and characterization of new psoralen derivatives with superior photoreactivity with DNA and RNA. Biochemistry. 16: 1058-64. PMID 849407 DOI: 10.1021/Bi00625A005 |
0.517 |
|
| 1977 |
Musich JA, Rapoport H. Reaction of O-methyl-N,N'-diisopropylisourea with amino acids and amines. The Journal of Organic Chemistry. 42: 139-41. PMID 830852 DOI: 10.1002/Chin.197720240 |
0.3 |
|
| 1977 |
Schmidtchen FP, Rapoport H. Polyprenylpyridinols. Synthesis of piericidin analogues. Journal of the American Chemical Society. 99: 7014-9. PMID 561812 DOI: 10.1021/Ja00463A041 |
0.421 |
|
| 1977 |
Miller MJ, Rapoport H. Porphyrin-protein bond of cytochrome c558 from Euglena gracilis. Journal of the American Chemical Society. 99: 3479-85. PMID 192772 DOI: 10.1002/Chin.197733339 |
0.409 |
|
| 1977 |
Slama JT, Willson CG, Grimshaw CE, Rapoport H. Stereochemistry of the porphyrin-protein bond of cytochrome c. Stereochemical comparison of Rhodospirillum rubrum, yeast, and horse heart porphyrins c. Biochemistry. 16: 1750-4. PMID 192273 DOI: 10.1021/Bi00627A036 |
0.486 |
|
| 1977 |
Weller DD, Gless RD, Rapoport H. Synthesis of 4a-aryldecahydroisoquinolines. Functionality in the carbocyclic ring Journal of Organic Chemistry. 42: 1485-1495. DOI: 10.1021/Jo00429A001 |
0.321 |
|
| 1977 |
Dean RT, Padgett HC, Rapoport H. A High Yield Regiospecific Preparation Of Iminium Salts Cheminform. 8. DOI: 10.1002/Chin.197706135 |
0.304 |
|
| 1976 |
Barber RB, Rapoport H. Conversion of Thebaine to Codeine. Journal of Medicinal Chemistry. 19: 1175-80. PMID 994146 DOI: 10.1002/Chin.197705347 |
0.351 |
|
| 1976 |
Weller DD, Rapoport H. A practical synthesis of codeine from dihydrothebainone. Journal of Medicinal Chemistry. 19: 1171-5. PMID 994145 DOI: 10.1021/Jm00232A001 |
0.357 |
|
| 1976 |
Dean RT, Padgett HC, Rapoport H. A high yield regiospecific preparation of iminium salts Journal of the American Chemical Society. 98: 7448-7449. DOI: 10.1021/Ja00439A069 |
0.304 |
|
| 1975 |
Lee DL, Rapoport H. Synthesis of tabtoxinine-delta-lactam. The Journal of Organic Chemistry. 40: 3491-5. PMID 1185324 DOI: 10.1021/Jo00912A005 |
0.405 |
|
| 1975 |
Barber RB, Rapoport H. Synthesis of thebaine and oripavine from codeine and morphine. Journal of Medicinal Chemistry. 18: 1074-7. PMID 1177252 DOI: 10.1002/Chin.197608340 |
0.32 |
|
| 1975 |
Tang CS, Morrow CJ, Rapoport H. A total syntheses of dl-camptothecin. Journal of the American Chemical Society. 97: 159-67. PMID 1133329 DOI: 10.1021/Ja00834A028 |
0.324 |
|
| 1975 |
Slama JT, Smith HW, Willson CG, Rapoport H. Porphyrin-protein bond of cytochrome C. Structure of porphyrin C. Journal of the American Chemical Society. 97: 6556-62. PMID 171295 DOI: 10.1002/Chin.197602358 |
0.48 |
|
| 1974 |
Jacobson SJ, Willson CG, Rapoport H. Mechanism of cystine racemization in strong acid. The Journal of Organic Chemistry. 39: 1074-7. PMID 4847772 DOI: 10.1002/Chin.197436414 |
0.506 |
|
| 1974 |
Plattner JJ, Gless RD, Cooper GK, Rapoport H. Synthesis of some DE and CDE ring analogs of camptothecin. The Journal of Organic Chemistry. 39: 303-11. PMID 4820107 DOI: 10.1002/Chin.197420342 |
0.383 |
|
| 1974 |
Snyder CD, Rapoport H. Synthesis of menaquinones. Journal of the American Chemical Society. 96: 8046-54. PMID 4464316 DOI: 10.1002/Chin.197511481 |
0.407 |
|
| 1974 |
Snyder CD, Rapoport H. Stereochemistry Of Quinate-Shikimate Conversions, Synthesis Of (-)-4-Epi-Shikimic Acid Cheminform. 5. DOI: 10.1002/Chin.197404175 |
0.392 |
|
| 1973 |
Bosin TR, Hanson RN, Rodricks JV, Simpson RA, Rapoport H. Routes to functionalized guanidines. The synthesis of guanidino diesters. The Journal of Organic Chemistry. 38: 1591-600. PMID 4708892 DOI: 10.1021/Jo00948A031 |
0.353 |
|
| 1973 |
Baldwin RM, Snyder CD, Rapoport H. Biosynthesis of menaquinones. Dissymmetry in the naphthalenic intermediate. Journal of the American Chemical Society. 95: 276-8. PMID 4682897 DOI: 10.1021/Ja00782A067 |
0.315 |
|
| 1973 |
Moore RE, Rapoport H. Geissovelline, a new alkaloid from Geissospermum vellossi The Journal of Organic Chemistry. 38: 215-230. DOI: 10.1021/Jo00942A007 |
0.408 |
|
| 1973 |
Snyder CD, Rapoport H. Stereochemistry of quinate-shikimate conversions. Synthesis of (-)-4-epi-shikimic acid Journal of the American Chemical Society. 95: 7821-7828. DOI: 10.1021/Ja00804A044 |
0.392 |
|
| 1973 |
BOSIN TR, HANSON RN, RODRICKS JV, SIMPSON RA, RAPOPORT H. ChemInform Abstract: WEGE ZU GUANIDINEN MIT FUNKTIONELLEN GRUPPEN, SYNTHESE VON GUANIDINODIESTERN Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/Chin.197332208 |
0.33 |
|
| 1972 |
Tang C, Rapoport H. A total synthesis of dl-camptothecin. Journal of the American Chemical Society. 94: 8615-6. PMID 4638996 DOI: 10.1021/JA00779A073 |
0.382 |
|
| 1972 |
Plattner JJ, Gless RD, Rapoport H. Synthesis of some DE and CDE ring analogs of camptothecin. Journal of the American Chemical Society. 94: 8613-5. PMID 4638995 DOI: 10.1021/Ja00779A072 |
0.383 |
|
| 1972 |
McDowell BL, Rapoport H. Acidic aromatic hydrocarbons. Analogs of fluoradene Journal of Organic Chemistry. 37: 3261-3265. DOI: 10.1021/Jo00986A015 |
0.307 |
|
| 1971 |
Frydman B, Los M, Rapoport H. Synthesis of substituted 1,5- and 1,7-naphthyridines and related lactams. The Journal of Organic Chemistry. 36: 450-454. PMID 27807974 DOI: 10.1021/Jo00802A018 |
0.4 |
|
| 1971 |
Rapoport H, Rodricks JV. Synthesis of cyclic guanidines Journal of Organic Chemistry. 36: 46-48. DOI: 10.1021/Jo00800A012 |
0.41 |
|
| 1971 |
Rapoport H, Frydman B, Reil S, Valasinas A, Frydman RB. Synthesis of 2-aminomethyldipyrrolylmethanes of biosynthetic interest Journal of the American Chemical Society. 93: 2738-2745. DOI: 10.1021/Ja00740A026 |
0.409 |
|
| 1971 |
Rapoport H, Plattner JJ. Synthesis of d- and 1-sirenin and their absolute configurations Journal of the American Chemical Society. 93: 1758-1761. DOI: 10.1021/Ja00736A030 |
0.313 |
|
| 1970 |
Nutting WH, Jewell RA, Rapoport H. 4-(4-Nitrophenylazo)benzoic acid. Improved synthesis of its acid chloride and spectroscopic properties of its esters Journal of Organic Chemistry. 35: 505-508. DOI: 10.1021/Jo00827A050 |
0.349 |
|
| 1970 |
Bhalerao UT, Plattner JJ, Rapoport H. Synthesis of dl-sirenin and dl-isosirenin Journal of the American Chemical Society. 92: 3429-3433. DOI: 10.1021/Ja00714A034 |
0.365 |
|
| 1970 |
Frydman B, Reil S, Despuy ME, Rapoport H. Additions and Corrections - Pyrroles from Azaindoles. A Synthesis of Porphobilinogen and Related Pyrroles. Journal of the American Chemical Society. 92: 1810-1810. DOI: 10.1021/Ja00709A603 |
0.365 |
|
| 1969 |
Frydman B, Reil S, Despuy ME, Rapoport H. Pyrroles from azaindoles. A synthesis of porphobilinogen and related pyrroles. Journal of the American Chemical Society. 91: 2338-42. PMID 5784185 DOI: 10.1021/Ja01037A025 |
0.375 |
|
| 1969 |
Martin PK, Rapoport H, Smith HW, Wong JL. Synthesis of cyclopenin and isocyclopenin Journal of Organic Chemistry. 34: 1359-1363. DOI: 10.1021/Jo01257A035 |
0.406 |
|
| 1969 |
Rapoport H, Snyder CD, Bondinell WE. Synthesis of chlorobiumquinone Journal of the American Chemical Society. 36: 3951-3960. DOI: 10.1021/Jo00824A023 |
0.406 |
|
| 1969 |
Plattner JJ, Bhalerao UT, Rapoport H. Synthesis of dl-sirenin Journal of the American Chemical Society. 91: 4933-4934. DOI: 10.1021/Ja01045A066 |
0.393 |
|
| 1968 |
Bondinell WE, DiMari SJ, Frydman B, Matsumoto K, Rapoport H. Synthesis of 2-methyl-3-vinyl-1,4-naphthoquinones Journal of Organic Chemistry. 33: 4351-4362. DOI: 10.1021/Jo01276A010 |
0.356 |
|
| 1968 |
Frydman B, Reil SJ, Boned J, Rapoport H. Synthesis of substituted 4- and 6-azaindoles Journal of Organic Chemistry. 33: 3762-3766. DOI: 10.1021/Jo01274A017 |
0.428 |
|
| 1968 |
Martin PK, Matthews HR, Rapoport H, Thyagarajan G. Synthesis of 1,4-substituted imidazoles Journal of Organic Chemistry. 33: 3758-3761. DOI: 10.1021/Jo01274A016 |
0.432 |
|
| 1968 |
Chan KC, Jewell RA, Nutting WH, Rapoport H. Synthesis and stereochemical assignment of trans-2-methyl-2-pentenoic acid and the corresponding esters, aldehydes, and alcohols Journal of Organic Chemistry. 33: 3382-3385. DOI: 10.1021/Jo01273A004 |
0.344 |
|
| 1968 |
Flaugh ME, Rapoport H. Synthesis of porphyrins. Deoxophylloerythroetioporphyrin Journal of the American Chemical Society. 90: 6877-6879. DOI: 10.1021/Ja01026A076 |
0.41 |
|
| 1968 |
Smith H, Wegfahrt P, Rapoport H. The synthesis of cyclopenin Journal of the American Chemical Society. 90: 1668-1669. DOI: 10.1021/Ja01008A059 |
0.406 |
|
| 1967 |
Blaschke G, Parker HI, Rapoport H. Codeinone as the intermediate in the biosynthetic conversion of thebaine to codeine. Journal of the American Chemical Society. 89: 1540-1. PMID 6041360 DOI: 10.1021/Ja00982A056 |
0.304 |
|
| 1967 |
Rapoport H, Lovell CH, Reist HR, Warren ME. The synthesis of thebaine and northebaine from codeinone dimethyl ketal. Journal of the American Chemical Society. 89: 1942-7. PMID 6040525 DOI: 10.1021/Ja00984A032 |
0.423 |
|
| 1967 |
Moore RE, Rapoport H. Synthesis of some ethyl-6,7-dimethoxycarbazoles and interpretation of their nuclear magnetic resonance spectra The Journal of Organic Chemistry. 32: 3335-3339. DOI: 10.1021/Jo01286A013 |
0.428 |
|
| 1965 |
Alworth WL, Rapoport H. Biosynthesis of the nicotine alkaloids in Nicotiana glutinosa. Interrelationships among nicotine, nornicotine, anabasine, and anatabine. Archives of Biochemistry and Biophysics. 112: 45-53. PMID 5865121 DOI: 10.1016/0003-9861(65)90008-1 |
0.507 |
|
| 1965 |
Bordner J, Rapoport H. Synthesis of 2,2'-Bipyrroles from 2-Pyrrolinones1a Journal of Organic Chemistry. 30: 3824-3828. DOI: 10.1021/Jo01022A053 |
0.406 |
|
| 1965 |
Wong JL, Brown MS, Rapoport H. The Synthesis of Pyrrolo[1,2-c]pyrimidine (6-Azapyrrocoline)1 Journal of Organic Chemistry. 30: 2398-2402. DOI: 10.1021/Jo01018A070 |
0.341 |
|
| 1964 |
Rapoport H, Bordner J. Synthesis of Substituted 2,2'-Bipyrroles1a Journal of Organic Chemistry. 29: 2727-2731. DOI: 10.1021/Jo01032A062 |
0.428 |
|
| 1964 |
Rapoport H, Castagnoli N, Holden KG. 2,2':5',2″-Terpyrrole1a The Journal of Organic Chemistry. 29: 883-885. DOI: 10.1021/Jo01027A029 |
0.492 |
|
| 1964 |
Blake J, Willson CD, Rapoport H. 3-Pyrrolidinones by Intramolecular Condensation Journal of the American Chemical Society. 86: 5293-5299. DOI: 10.1021/Ja01077A049 |
0.35 |
|
| 1964 |
Alworth WL, De Selms RC, Rapoport H. The Biosynthesis of Nicotine inNicotiana glutinosafrom Carbon-14 Dioxide Journal of the American Chemical Society. 86: 1608-1616. DOI: 10.1021/Ja01062A034 |
0.491 |
|
| 1963 |
Rapoport H, Batcho AD. 1,5-Naphthyridine and Some of Its Alkyl Derivatives Journal of Organic Chemistry. 28: 1753-1759. DOI: 10.1021/Jo01042A005 |
0.35 |
|
| 1962 |
Rapoport H, Moore RE. Alkaloids of Geissospermum vellosii. Isolation and Structure Determinations of Vellosimine, Vellosiminol, and Geissolosimine The Journal of Organic Chemistry. 27: 2981-2985. DOI: 10.1021/Jo01056A004 |
0.408 |
|
| 1962 |
Rapoport H, Castagnoli N. 2,2″-Bipyrrole Journal of the American Chemical Society. 84: 2178-2181. DOI: 10.1021/Ja00870A032 |
0.492 |
|
| 1961 |
Rapoport H, Willson CD. Synthesis of Pyrrole-3-carboxylic Acids Journal of Organic Chemistry. 26: 1102-1104. DOI: 10.1021/Jo01063A030 |
0.386 |
|
| 1960 |
Rapoport H, Iwamoto R, Tretter JR. The Synthesis of 2,2'-Biquinolyls and Related Compounds by Catalytic Dehydrogenation Journal of Organic Chemistry. 25: 372-373. DOI: 10.1021/Jo01073A015 |
0.344 |
|
| 1960 |
Rapoport H, Holden KG. The Synthesis of Prodigiosin Journal of the American Chemical Society. 82: 5510-5511. DOI: 10.1021/Ja00863A026 |
0.406 |
|
| 1957 |
Rapoport H, Chadha MS, Lovell CH. Preparation and Cleavage of Some Codeine Glycols1 Journal of the American Chemical Society. 79: 4694-4697. DOI: 10.1021/Ja01574A031 |
0.318 |
|
| 1956 |
Rapoport H, Reist HN, Lovell CH. Codeinone Dimethyl Ketal And Its Conversion To Thebaine Journal of the American Chemical Society. 78: 5128-5128. DOI: 10.1021/Ja01600A086 |
0.302 |
|
| 1956 |
Rapoport H, Volcheck EJ. The Synthesis of Desoxycarpyrinic and Carpyrinic Acids Journal of the American Chemical Society. 78: 2451-2455. DOI: 10.1021/Ja01592A029 |
0.376 |
|
| 1955 |
Rapoport H, Masamune S. The Stereochemistry of 10-Hydroxycodeine Derivatives1,2 Journal of the American Chemical Society. 77: 4330-4335. DOI: 10.1021/Ja01621A045 |
0.377 |
|
| 1955 |
Rapoport H, Allen RH, Cisney ME. The Synthesis of Isocolchinol Methyl Ether Journal of the American Chemical Society. 77: 670-675. DOI: 10.1021/Ja01608A039 |
0.357 |
|
| 1955 |
Rapoport H, Lavigne JB. The Preparation of Colchicide1(Demethoxycolchicine) Journal of the American Chemical Society. 77: 667-670. DOI: 10.1021/Ja01608A038 |
0.302 |
|
| 1954 |
Rapoport H, Christian CG, Spencer G. The Synthesis Of Some Compounds Related To Cuscohygrine Journal of Organic Chemistry. 19: 840-844. DOI: 10.1021/Jo01370A024 |
0.333 |
|
| 1953 |
Rapoport H, Look M. A Synthesis of 3,2'-Nornicotyrine1 Journal of the American Chemical Society. 75: 4605-4607. DOI: 10.1021/Ja01114A526 |
0.406 |
|
| 1951 |
Rapoport H, King TP, Lavigne JB. The Preparation of Some Acenaphthoxyacetic Acids Journal of the American Chemical Society. 73: 2718-2721. DOI: 10.1021/Ja01150A082 |
0.307 |
|
| 1951 |
Rapoport H, Campion JE. The Synthesis of 2,3,4-Trimethoxybenzcyclohepten-6-one1 Journal of the American Chemical Society. 73: 2239-2241. DOI: 10.1021/Ja01149A091 |
0.407 |
|
| 1950 |
Rapoport H, Bonner RM. The Preparation of Some Tetrasubstituted Amidrazones Journal of the American Chemical Society. 72: 2783-2784. DOI: 10.1021/Ja01162A523 |
0.317 |
|
| 1950 |
Rapoport H, Williams AR, Cisney ME. The Synthesis of DL-Colchinol Methyl Ether1,2 Journal of the American Chemical Society. 72: 1414-1421. DOI: 10.1021/Ja01148A005 |
0.355 |
|
| 1949 |
RAPOPORT H, JORGENSEN E. THE SYNTHESIS OF CUSCOHYGRINE The Journal of Organic Chemistry. 14: 664-669. DOI: 10.1021/Jo01156A021 |
0.406 |
|
| 1949 |
Rapoport H, Williams AR. A Synthesis of Dibenzocycloheptadiene Journal of the American Chemical Society. 71: 1774-1778. DOI: 10.1021/Ja01173A069 |
0.406 |
|
| 1947 |
Small L, Rapoport H. Nuclear substituted morphine derivatives Journal of Organic Chemistry. 12: 284-292. PMID 20291137 DOI: 10.1021/Jo01166A012 |
0.352 |
|
| 1947 |
Rapoport H, Small L. The Mannich reaction with dihydrocodeinone Journal of Organic Chemistry. 12: 834-838. PMID 18919736 DOI: 10.1021/Jo01170A016 |
0.311 |
|
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