Clayton H. Heathcock, Ph.D. - Publications

Affiliations: 
1964-2005 Chemistry University of California, Berkeley, Berkeley, CA 
 2005- QB3 Lawrence Berkeley National Laboratory, Berkeley, CA, USA 
Area:
natural products chemistry
Website:
http://heathcock.org/chhgrp/

261 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2010 Takai K, Heathcock CH. Generation of novel nucleophilic organometallic species and their applications to organic synthesis Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry. 68: 3-18. DOI: 10.5059/Yukigoseikyokaishi.68.3  0.4
2010 HEATHCOCK CH, BROWN RCD, NORMAN TC. ChemInform Abstract: Synthesis of Petrosins C (I) and D (II). Cheminform. 29: no-no. DOI: 10.1002/chin.199849271  0.654
2010 WALKER MA, HEATHCOCK CH. ChemInform Abstract: Acyclic Stereoselection. Part 54. Extending the Scope of the Evans Asymmetric Aldol Reaction: Preparation of anti- and “Non-Evans” syn- Aldols. Cheminform. 23: no-no. DOI: 10.1002/chin.199208067  0.328
2010 OARE DA, HEATHCOCK CH. ChemInform Abstract: Acyclic Stereocontrol in Michael Addition Reactions of Enamines and Enol Ethers Cheminform. 22: no-no. DOI: 10.1002/chin.199132288  0.785
2007 Oare DA, Heathcock CH. Acyclic stereocontrol in Michael addition reactions of enamines and enol ethers Topics in Stereochemistry. 20: 87-170. DOI: 10.1002/9780470147290.Ch2  0.793
2007 Oare DA, Heathcock CH. Stereochemistry of the Base‐Promoted Michael Addition Reaction Topics in Stereochemistry. 19: 227-407. DOI: 10.1002/9780470147283.Ch5  0.779
2004 Christie HS, Heathcock CH. Total synthesis of (+/-)-halichlorine, (+/-)-pinnaic acid, and (+/-)-tauropinnaic acid. Proceedings of the National Academy of Sciences of the United States of America. 101: 12079-84. PMID 15299146 DOI: 10.1073/Pnas.0403887101  0.449
2004 Brito-Arias M, Pereda-Miranda R, Heathcock CH. Synthesis of tricolorin F. The Journal of Organic Chemistry. 69: 4567-70. PMID 15230576 DOI: 10.1021/Jo030244C  0.382
2003 Heathcock CH, McLaughlin M, Medina J, Hubbs JL, Wallace GA, Scott R, Claffey MM, Hayes CJ, Ott GR. Multigram synthesis of the C29-C51 subunit and completion of the total synthesis of altohyrtin C (spongistatin 2). Journal of the American Chemical Society. 125: 12844-9. PMID 14558833 DOI: 10.1021/Ja030317+  0.791
2003 Hubbs JL, Heathcock CH. A second-generation synthesis of the C1-C28 portion of the altohyrtins (spongistatins). Journal of the American Chemical Society. 125: 12836-43. PMID 14558832 DOI: 10.1021/Ja030316H  0.719
2003 Young SD, Buse CT, Heathcock CH. 2‐Methyl‐2‐(Trimethylsiloxy)Pentan‐3‐one Organic Syntheses. 79-79. DOI: 10.1002/0471264180.Os063.09  0.38
2003 Heathcock CH, Hassner A. Methyl (trans‐2‐Iodo‐1‐Tetralin)Carbamate Organic Syntheses. 112-112. DOI: 10.1002/0471264180.Os051.28  0.333
2003 Heathcock CH, Hassner A. Aziridines from β-Iodocarbamates: 1,2,3,4-Tetrahydronaphthalene(1,2)imine Organic Syntheses. 53-53. DOI: 10.1002/0471264180.Os051.12  0.309
2002 Skyler D, Heathcock CH. The pyridoacridine family tree: a useful scheme for designing synthesis and predicting undiscovered natural products. Journal of Natural Products. 65: 1573-81. PMID 12444679 DOI: 10.1021/Np020016Y  0.76
2002 Fell JD, Heathcock CH. Oxidative fragmentation of pregna-14,16-dien-20-ones to 14 beta-hydroxyandrost-15-en-17-ones. The Journal of Organic Chemistry. 67: 4742-6. PMID 12098283 DOI: 10.1021/Jo011175+  0.805
2002 Blazey CM, Heathcock CH. Regiochemistry in 1,3-dipolar cycloadditions of the azomethine ylide formed from diethyl aminomalonate and paraformaldehyde. The Journal of Organic Chemistry. 67: 298-300. PMID 11777476 DOI: 10.1021/Jo010645X  0.804
2002 Kedrowski BL, Heathcock CH. Thiazoline ring formation from 2-methylcysteines and 2-halomethylalanines Heterocycles. 58: 601-634. DOI: 10.3987/Com-02-S(M)60  0.789
2001 Skyler D, Heathcock CH. A simple biomimetic synthesis of styelsamine B. Organic Letters. 3: 4323-4. PMID 11784208 DOI: 10.1021/Ol010262L  0.803
2001 Hinman MM, Heathcock CH. A synthetic approach to the Stemona alkaloids. The Journal of Organic Chemistry. 66: 7751-6. PMID 11701032 DOI: 10.1021/Jo0106391  0.356
2001 Wallace GA, Heathcock CH. Further studies of the Daphniphyllum alkaloid polycyclization cascade. The Journal of Organic Chemistry. 66: 450-4. PMID 11429813 DOI: 10.1021/Jo001145R  0.731
2000 Yamamoto K, Heathcock CH. alpha,beta-epoxy vinyl triflates in Pd-catalyzed reactions. Organic Letters. 2: 1709-12. PMID 10880207 DOI: 10.1021/Ol000064E  0.572
2000 Wallace GA, Scott RW, Heathcock CH. Synthesis of the C29-C44 portion of spongistatin 1 (altohyrtin A). The Journal of Organic Chemistry. 65: 4145-52. PMID 10866633 DOI: 10.1021/jo0002801  0.672
2000 Toczko MA, Heathcock CH. Total synthesis of (+/-)-aspidospermidine. The Journal of Organic Chemistry. 65: 2642-5. PMID 10808435 DOI: 10.1021/Jo991599S  0.826
1999 Claffey MM, Hayes CJ, Heathcock CH. Synthesis of the C1-C28 Portion of Spongistatin 1 (Altohyrtin A). The Journal of Organic Chemistry. 64: 8267-8274. PMID 11674747 DOI: 10.1021/Jo9910987  0.38
1999 Liu JF, Heathcock CH. Total Synthesis of (+/-)-Cylindricines A and B. The Journal of Organic Chemistry. 64: 8263-8266. PMID 11674746 DOI: 10.1021/Jo991020Q  0.401
1999 Mapp AK, Heathcock CH. Total Synthesis of Myxalamide A. The Journal of Organic Chemistry. 64: 23-27. PMID 11674080 DOI: 10.1021/Jo9813742  0.698
1999 Aubart KM, Heathcock CH. A Biomimetic Approach to the Discorhabdin Alkaloids: Total Syntheses of Discorhabdins C and E and Dethiadiscorhabdin D. The Journal of Organic Chemistry. 64: 16-22. PMID 11674079 DOI: 10.1021/Jo9815397  0.365
1999 Hubbs JL, Heathcock CH. Total synthesis of (+/-)-isoschizogamine. Organic Letters. 1: 1315-7. PMID 10825981 DOI: 10.1021/Ol9902632  0.743
1999 Chi S, Heathcock CH. Total syntheses of (+/-)-preussomerins G and I. Organic Letters. 1: 3-5. PMID 10822527 DOI: 10.1021/Ol990020+  0.387
1998 Denhart DJ, Griffith DA, Heathcock CH. Synthesis of the tricyclic core of sarain A. Use of formaldehyde in an intramolecular Grigg azomethine ylide cyclization Journal of Organic Chemistry. 63: 9616-9617. DOI: 10.1021/Jo981801B  0.669
1998 Scott RW, Epperson J, Heathcock CH. Total Synthesis of Petrosin, Petrosin A, and Petrosin B Journal of Organic Chemistry. 63: 5001-5012. DOI: 10.1021/Jo9801768  0.411
1997 Larson DP, Heathcock CH. Total Synthesis of Tricolorin A. The Journal of Organic Chemistry. 62: 8406-8418. PMID 11671979 DOI: 10.1021/jo971413u  0.321
1997 Szczepankiewicz BG, Heathcock CH. A novel method for suppression of the abnormal Fischer indole synthesis Tetrahedron. 53: 8853-8870. DOI: 10.1016/S0040-4020(97)90396-3  0.379
1996 McDermott TS, Mortlock AA, Heathcock CH. Total Syntheses of (-)-Papuamine and (-)-Haliclonadiamine. The Journal of Organic Chemistry. 61: 700-709. PMID 11666993 DOI: 10.1021/Jo951647I  0.406
1996 Heathcock CH. Nature knows best: an amazing reaction cascade is uncovered by design and discovery. Proceedings of the National Academy of Sciences of the United States of America. 93: 14323-7. PMID 8962049 DOI: 10.1073/Pnas.93.25.14323  0.371
1996 Scott RW, Heathcock CH. An efficient synthesis of 3,4,6-tri-O-benzyl-2-C-methyl-D-glucal. Carbohydrate Research. 291: 205-8. PMID 8864231 DOI: 10.1016/S0008-6215(96)00162-0  0.342
1996 Parsons RL, Heathcock CH. Total Synthesis of (-)-Tantazole B Synlett. 1996: 1168-1170. DOI: 10.1055/S-1996-5716  0.328
1996 Marshall KA, Mapp AK, Heathcock CH. Synthesis of a 2,7-dioxatricyclo[4.2.1.03,8]nonane: A model study for possible application in a synthesis of dictyoxetane Journal of Organic Chemistry. 61: 9135-9145. DOI: 10.1021/Jo961680K  0.676
1996 Caron S, Stoermer D, Mapp AK, Heathcock CH. Total synthesis of zaragozic acid A (squalestatin S1). Synthesis of the relay compound Journal of Organic Chemistry. 61: 9126-9134. DOI: 10.1021/Jo961534E  0.688
1996 Stoermer D, Caron S, Heathcock CH. Total synthesis of zaragozic acid A (squalestatin S1). Degradation to a relay compound and reassembly of the natural product Journal of Organic Chemistry. 61: 9115-9125. DOI: 10.1021/Jo961533M  0.395
1996 Larson DP, Heathcock CH. Synthesis of the macrolactone disaccharide subunit of tricolorin A Journal of Organic Chemistry. 61: 5208-5209. DOI: 10.1021/Jo960655B  0.376
1996 Brimble MA, Heathcock CH, Nobin GN. Synthesis and ene reactions of di-(-)-methyl diazenedicarboxylate Tetrahedron Asymmetry. 7: 2007-2016. DOI: 10.1016/0957-4166(96)00242-X  0.487
1996 Caron S, McDonald AI, Heathcock CH. An improved synthesis of 1,6-anhydro-2,3-di-O-benzyl-β-D-xylo-hexopyranos-4-ulose Carbohydrate Research. 281: 179-182. DOI: 10.1016/0008-6215(95)00335-5  0.303
1995 Heathcock CH, Clasby M, Griffith DA, Henke BR, Sharp MJ. Progress toward the Synthesis of Sarain A Synlett. 1995: 467-474. DOI: 10.1055/S-1995-5298  0.659
1995 Raimundo BC, Heathcock CH. Further Studies on the Anti-Selective Aldol Reaction of Chiral Imides Synlett. 1995: 1213-1214. DOI: 10.1055/S-1995-5246  0.366
1995 Caron S, McDonald AI, Heathcock CH. Synthesis of 1-substituted and 1,4-disubstituted 2,3-di-O-benzyl-1,6-anhydrogalactofuranoses Journal of Organic Chemistry. 60: 2780-2785. DOI: 10.1021/Jo00114A028  0.356
1995 Heathcock CH, Kath JC, Ruggeri RB. Daphniphyllum alkaloids. 16. Total synthesis of (+)-codaphniphylline Journal of Organic Chemistry. 60: 1120-1130. DOI: 10.1021/Jo00110A013  0.424
1995 Griffith DA, Heathcock CH. Progress toward the synthesis of sarain A: An unanticipated rearrangement Tetrahedron Letters. 36: 2381-2384. DOI: 10.1016/0040-4039(95)00283-I  0.67
1994 Heathcock CH, Smith SC. Synthesis and biological activity of unsymmetrical bis-steroidal pyrazines related to the cytotoxic marine natural product cephalostatin 1 Journal of Organic Chemistry. 59: 6828-6839. DOI: 10.1021/Jo00101A052  0.338
1994 Szczepankiewicz BG, Heathcock CH. Total synthesis of diplamine, a cytotoxic pyridoacridine alkaloid from a Pacific tunicate Journal of Organic Chemistry. 59: 3512-3513. DOI: 10.1021/Jo00092A002  0.395
1994 Scott RW, Epperson JR, Heathcock CH. Total Synthesis of Petrosin Journal of the American Chemical Society. 116: 8853-8854. DOI: 10.1021/Ja00098A073  0.417
1994 Parsons RL, Heathcock CH. Total synthesis of mirabazole B Tetrahedron Letters. 35: 1383-1384. DOI: 10.1016/S0040-4039(00)76224-1  0.328
1994 Parsons RL, Heathcock CH. Revision of the stereostructure of mirabazole C Tetrahedron Letters. 35: 1379-1382. DOI: 10.1016/S0040-4039(00)76223-X  0.316
1994 Sharp MJ, Heathcock CH. An unusual isomerization under Lawesson thiation conditions Tetrahedron Letters. 35: 3651-3652. DOI: 10.1016/S0040-4039(00)73062-0  0.321
1993 Ganesan A, Heathcock CH. Synthesis of unsymmetrical pyrazines by reaction of an oxadiazinone with enamines Journal of Organic Chemistry. 58: 6155-6157. DOI: 10.1021/Jo00074A058  0.601
1993 Clark DL, Heathcock CH. Studies on the alkylation of chiral enolates: Application toward the total synthesis of discodermolide Journal of Organic Chemistry. 58: 5878-5879. DOI: 10.1021/Jo00074A005  0.385
1993 Brimble MA, Heathcock CH. Allylic amination by the Lewis-acid-mediated ene reaction of diethyl azodicarboxylate with alkenes Journal of Organic Chemistry. 58: 5261-5263. DOI: 10.1021/Jo00071A042  0.43
1993 Stoermer D, Heathcock CH. Total synthesis of (-)-alloaristoteline, (-)-serratoline, and (+)-aristotelone Journal of Organic Chemistry. 58: 564-568. DOI: 10.1021/Jo00055A007  0.399
1993 Ihle NC, Heathcock CH. Palladium-catalyzed intramolecular alkyne-carbon monoxide-alkene insertion cascade for synthesis of .alpha.-methylenecyclopentenones Journal of Organic Chemistry. 58: 560-563. DOI: 10.1021/Jo00055A006  0.41
1993 Theisen PD, Heathcock CH. Prochiral recognition in the reaction of 3-substituted glutaric anhydrides with chiral secondary alcohols Journal of Organic Chemistry. 58: 142-146. DOI: 10.1021/Jo00053A027  0.361
1993 Ganosan A, Heathcock CH. A Stereochemical test of the mechanism of electrophilic substitution in 3-substituted indoles Tetrahedron Letters. 34: 439-440. DOI: 10.1016/0040-4039(93)85096-F  0.437
1992 Henke BR, Kouklis AJ, Heathcock CH. Intramolecular 1,3-dipolar cycloaddition of stabilized azomethine ylides to unactivated dipolarophiles Journal of Organic Chemistry. 57: 7056-7066. DOI: 10.1021/Jo00052A015  0.316
1992 Smith SC, Heathcock CH. A convenient procedure for the synthesis of bis-steroidal pyrazines: Models for the cephalostatins Journal of Organic Chemistry. 57: 6379-6380. DOI: 10.1021/Jo00050A002  0.375
1992 Thompson SK, Heathcock CH. Total synthesis of some marasmane and lactarane sesquiterpenes Journal of Organic Chemistry. 57: 5979-5989. DOI: 10.1021/Jo00048A036  0.363
1992 Van Draanen NA, Arseniyadis S, Crimmins MT, Heathcock CH. Protocols for the preparation of each of the four possible stereoisomeric .alpha.-alkyl-.beta.-hydroxy carboxylic acids from a single chiral aldol reagent. [Erratum to document cited in CA114(17):163485y] The Journal of Organic Chemistry. 57: 5802-5802. DOI: 10.1021/Jo00047A053  0.342
1992 Walker MA, Heathcock CH. Total synthesis of (−)-mirabazole C Journal of Organic Chemistry. 57: 5566-5568. DOI: 10.1021/Jo00047A005  0.357
1992 Kerwin SM, Heathcock CH. Remote oxidation of perhydrophenanthrenes by template-directed hydrogen atom abstraction Journal of Organic Chemistry. 57: 4005-4013. DOI: 10.1021/Jo00040A050  0.683
1992 Heathcock CH, Ruggeri RB, McClure KF. Daphniphyllum alkaloids. 15. Total syntheses of (.+-.)-methyl homodaphniphyllate and (.+-.)-daphnilactone A The Journal of Organic Chemistry. 57: 2585-2594. DOI: 10.1021/Jo00035A012  0.301
1992 Heathcock CH, Stafford JA, Clark DL. Daphniphyllum alkaloids. 14. Total synthesis of (.+-.)-bukittinggine Journal of Organic Chemistry. 57: 2575-2585. DOI: 10.1021/Jo00035A011  0.374
1992 Heathcock CH, Piettre S, Ruggeri RB, Ragan JA, Kath JC. Daphniphyllum alkaloids. 12. A proposed biosynthesis of the pentacyclic skeleton. Proto-daphniphylline Journal of Organic Chemistry. 57: 2554-2566. DOI: 10.1021/Jo00035A009  0.35
1992 Heathcock CH, Hansen MM, Ruggeri RB, Kath JC. Daphniphyllum alkaloids. 11. Biomimetic total synthesis of methyl homosecodaphniphyllate. Development of the tetracyclization reaction Journal of Organic Chemistry. 57: 2544-2553. DOI: 10.1021/Jo00035A008  0.467
1992 Heathcock CH, Davidsen SK, Mills SG, Sanner MA. Daphniphyllum alkaloids. 10. Classical total synthesis of methyl homodaphniphyllate Journal of Organic Chemistry. 57: 2531-2544. DOI: 10.1021/Jo00035A007  0.442
1992 Munchhof MJ, Heathcock CH. The stereochemistry of enolate formation in THF-hexane mixtures Tetrahedron Letters. 33: 8005-8006. DOI: 10.1016/S0040-4039(00)74701-0  0.327
1992 Lopes RSC, Lopes CC, Heathcock CH. Synthesis of pancratistatin models Tetrahedron Letters. 33: 6775-6778. DOI: 10.1016/S0040-4039(00)61773-2  0.352
1992 Heathcock CH. The enchanting alkaloids of Yuzuriha Angewandte Chemie (International Edition in English). 31: 665-681. DOI: 10.1002/Anie.199206653  0.37
1992 Heathcock CH, Stafford JA. Daphniphyllum alkaloids. 13. Asymmetric total synthesis of (-)-secodaphniphylline Journal of Organic Chemistry. 57: 2566-2574.  0.328
1991 Walker MA, Heathcock CH. Acyclic stereoselection. 54. Extending the scope of the Evans asymmetric aldol reaction: preparation of anti and "non-Evans" syn aldols Journal of Organic Chemistry. 56: 5747-5750. DOI: 10.1021/Jo00020A006  0.417
1991 Van Draanen NA, Arseniyadis S, Crimmins MT, Heathcock CH. Protocols for the preparation of each of the four possible stereoisomeric α-alkyl-β-hydroxy carboxylic acids from a single chiral aldol reagent Journal of Organic Chemistry. 56: 2499-2506. DOI: 10.1021/Jo00007A043  0.454
1990 Piettre S, Heathcock CH. Biomimetic total synthesis of proto-daphniphylline. Science (New York, N.Y.). 248: 1532-4. PMID 17818314 DOI: 10.1126/Science.248.4962.1532  0.358
1990 Montgomery SH, Pirrung MC, Heathcock CH. De novo synthesis of carbohydrates by stereoselective aldol reaction: L-cladinose. Carbohydrate Research. 202: 13-32. PMID 2224887 DOI: 10.1016/0008-6215(90)84068-6  0.715
1990 Heathcock CH, Piettre S, Kath J. Mechanistic investigations of a biomimetic polycyclization process that leads to the Daphniphyllum alkaloids Pure and Applied Chemistry. 62: 1911-1920. DOI: 10.1351/Pac199062101911  0.385
1990 Danda H, Hansen MM, Heathcock CH. Acyclic stereoselection. 48. Reversal of stereochemistry in the aldol reactions of a chiral boron enolate [Erratum to document cited in CA112(5):35733z] The Journal of Organic Chemistry. 55: 6231-6231. DOI: 10.1021/Jo00312A039  0.373
1990 Mori I, Ishihara K, Flippin LA, Nozaki K, Yamamoto H, Bartlett PA, Heathcock CH. Acyclic stereoselection. 52. On the mechanism of Lewis acid mediated nucleophilic substitution reactions of acetals The Journal of Organic Chemistry. 55: 6107-6115. DOI: 10.1021/Jo00312A015  0.553
1990 Mori I, Bartlett PA, Heathcock CH. Stereoselective additions of nucleophilic alkenes to chiral thionium ions Journal of Organic Chemistry. 55: 5966-5977. DOI: 10.1021/Jo00311A013  0.338
1990 Stafford JA, Heathcock CH. Daphniphyllum alkaloids. Part 8. Asymmetric total synthesis of (-)-secodaphniphylline The Journal of Organic Chemistry. 55: 5433-5434. DOI: 10.1021/Jo00307A006  0.495
1990 Ruggeri RB, Heathcock CH. Daphniphyllum alkaloids. Part 7. Biomimetic total synthesis of (.+-.)-methyl homodaphniphyllate The Journal of Organic Chemistry. 55: 3714-3715. DOI: 10.1021/Jo00299A006  0.366
1990 Thompson SK, Heathcock CH. Effect of cation, temperature, and solvent on the stereoselectivity of the Horner-Emmons reaction of trimethyl phosphonoacetate with aldehydes Journal of Organic Chemistry. 55: 3386-3388. DOI: 10.1021/Jo00297A076  0.363
1990 Thompson SK, Heathcock CH. Total synthesis of (.+-.)-isovelleral, a mutagenic sesquiterpene dialdehyde from Lactarius vellereus Journal of Organic Chemistry. 55: 3004-3005. DOI: 10.1021/Jo00297A009  0.422
1990 Mori I, Ishihara K, Heathcock CH. Acyclic stereoselection. 50. New stereoselective propanal/propanoic acid synthons for aldol reactions The Journal of Organic Chemistry. 55: 1114-1117. DOI: 10.1021/Jo00290A060  0.375
1990 Danda H, Hansen MM, Heathcock CH. Reversal of stereochemistry in the aldol reactions of a chiral boron enolate Journal of Organic Chemistry. 55: 173-181. DOI: 10.1021/Jo00288A029  0.304
1990 Oare DA, Heathcock CH. Acyclic stereoselection. 47. Stereochemistry of the Michael addition of ester and ketone enolates to .alpha.,.beta.-unsaturated ketones The Journal of Organic Chemistry. 55: 157-172. DOI: 10.1021/Jo00288A028  0.766
1990 Oare DA, Henderson MA, Sanner MA, Heathcock CH. Acyclic stereoselection. 46. Stereochemistry of the Michael addition of N,N-disubstituted amide and thioamide enolates to .alpha.,.beta.-unsaturated ketones The Journal of Organic Chemistry. 55: 132-157. DOI: 10.1021/Jo00288A027  0.746
1990 OARE DA, HEATHCOCK CH. ChemInform Abstract: Acyclic Stereoselection. Part 47. Stereochemistry of the Michael Addition of Ester and Ketone Enolates to α,β-Unsaturated Ketones. Cheminform. 21. DOI: 10.1002/chin.199027098  0.758
1990 Stafford JA, Heathcock CH. Asymmetric total synthesis of (-)-secodaphniphylline Journal of Organic Chemistry. 55: 5433-5434.  0.322
1989 Heathcock CH, Davis BR, Hadley CR. Synthesis and biological evaluation of a monocyclic, fully functional analogue of compactin. Journal of Medicinal Chemistry. 32: 197-202. PMID 2909732 DOI: 10.1021/Jm00121A036  0.335
1989 Ruggeri RB, Heathcock CH. A proposal for biosynthesis of the Daphniphyllum alkaloids Pure and Applied Chemistry. 61: 289-292. DOI: 10.1351/Pac198961030289  0.355
1989 Heathcock CH, Blumenkopf TA, Smith KM. Total synthesis of (.+-.)-fawcettimine The Journal of Organic Chemistry. 54: 1548-1562. DOI: 10.1021/Jo00268A015  0.417
1989 Ruggeri RB, McClure KF, Heathcock CH. Daphniphyllum alkaloids. Part 5. Total synthesis of (.+-.)-daphnilactone A: a novel fragmentation reaction Journal of the American Chemical Society. 111: 1530-1531. DOI: 10.1021/Ja00186A075  0.459
1989 Dickman DA, Heathcock CH. Total synthesis of (.+-.)-vallesamidine Journal of the American Chemical Society. 111: 1528-1530. DOI: 10.1021/Ja00186A074  0.417
1989 Slough GA, Bergman RG, Heathcock CH. Synthesis of .eta.1 oxygen-bound rhodium enolates. Applications to catalytic aldol chemistry Journal of the American Chemical Society. 111: 938-949. DOI: 10.1021/Ja00185A025  0.348
1989 Ishihara K, Yamamoto H, Heathcock CH. Diastereoselective aldol synthesis using acetal templates Tetrahedron Letters. 30: 1825-1828. DOI: 10.1016/S0040-4039(00)99590-X  0.445
1989 OARE DA, HEATHCOCK CH. ChemInform Abstract: Synthesis of the Cyclic Hexapeptide Echinocandin D. New Approaches to the Asymmetric Synthesis of β-Hydroxy-α-amino Acids Cheminform. 20. DOI: 10.1002/chin.198916362  0.767
1988 Burkhardt ER, Doney JJ, Slough GA, Stack JM, Heathcock CH, Bergman RG. Carbon-Carbon bond forming reactions of organotransition metal enolate complexes Pure and Applied Chemistry. 60: 1-6. DOI: 10.1351/Pac198860010001  0.318
1988 Henderson MA, Heathcock CH. Acyclic stereoselection. 44. Diastereoselectivity in the ortho ester Claisen rearrangement of chiral propargylic alcohols. Use of β-allenic esters as chiral methylmalonaldehyde synthons Journal of Organic Chemistry. 53: 4736-4745. DOI: 10.1021/Jo00255A014  0.35
1988 Hoagland S, Morita Y, Bai DL, Märki HP, Kees K, Brown L, Heathcock CH. Acyclic stereoselection. 43. Stereoselective synthesis of the C-8 to C-15 moiety of erythronolide A Journal of Organic Chemistry. 53: 4730-4735. DOI: 10.1021/Jo00255A013  0.35
1988 Norman MH, Heathcock CH. Improved synthesis of N-benzyl-5-ethyl-1,2,3,4-tetrahydropyridine Journal of Organic Chemistry. 53: 3370-3371. DOI: 10.1021/Jo00249A050  0.339
1988 Heathcock CH, Finkelstein BL, Jarvi ET, Radel PA, Hadley CR. Acyclic stereoselection. Part 42. 1,4- and 1,5-Stereoselection by sequential aldol addition to a .alpha.,.beta.-unsaturated aldehydes followed by Claisen rearrangement. Application to total synthesis of the vitamin E side chain and the archaebacterial C40 diol The Journal of Organic Chemistry. 53: 1922-1942. DOI: 10.1021/Jo00244A017  0.38
1988 Ruggeri RB, Hansen MM, Heathcock CH. Total synthesis of (.+-.)-methyl homosecodaphniphyllate. A remarkable new tetracyclization reaction Journal of the American Chemical Society. 110: 8734-8736. DOI: 10.1021/Ja00234A046  0.451
1987 Heathcock CH, Hadley CR, Rosen T, Theisen PD, Hecker SJ. Total synthesis and biological evaluation of structural analogues of compactin and dihydromevinolin. Journal of Medicinal Chemistry. 30: 1858-73. PMID 3656359 DOI: 10.1021/Jm00393A030  0.396
1987 Heathcock CH, Geldern TWv. Total synthesis of (+)-norsecurinine Heterocycles. 25: 75-78. DOI: 10.3987/S-1987-01-0075  0.417
1987 Hansen MM, Bartlett PA, Heathcock CH. Preparation and reactions of an alkylzinc enolate Organometallics. 6: 2069-2074. DOI: 10.1021/Om00153A006  0.406
1987 Kerwin SM, Paul AG, Heathcock CH. Quassinoid synthesis. 2. Preparation of a tetracyclic intermediate having the bruceantin tetrahydrofuran ring Journal of Organic Chemistry. 52: 1686-1695. DOI: 10.1021/Jo00385A008  0.651
1987 Ruggeri RB, Heathcock CH. Synthesis of polycyclic lactam and lactone ethers by intramolecular reformatsky reactions. A model for construction of the daphnilactone a ring system Journal of Organic Chemistry. 52: 5745-5746. DOI: 10.1021/Jo00235A020  0.384
1987 Hecker S, Heathcock C. Correction. Total Synthesis of (+)-Dihydromevinolin Journal of the American Chemical Society. 109: 7583-7583. DOI: 10.1021/Ja00258A600  0.386
1987 Lodge EP, Heathcock CH. Acyclic stereoselection. 40. Steric effects, as well as .sigma.*-orbital energies, are important in diastereoface differentiation in additions to chiral aldehydes Journal of the American Chemical Society. 109: 3353-3361. DOI: 10.1021/Ja00245A027  0.349
1987 Lodge EP, Heathcock CH. Acyclic stereoselection. 39. The origin of diastereofacial selectivity in additions to chiral aldehydes and ketones: trajectory analysis Journal of the American Chemical Society. 109: 2819-2820. DOI: 10.1021/Ja00243A042  0.368
1987 Burkhardt ER, Doney JJ, Bergman RG, Heathcock CH. Tungsten and molybdenum 2-oxaallyl [.eta.1-(C)-enolate] complexes: functional group transformations, photochemical aldol reactions, and alkyne/carbon monoxide migratory insertion reactions Journal of the American Chemical Society. 109: 2022-2039. DOI: 10.1021/Ja00241A020  0.367
1987 Oare DA, Heathcock CH. Influence of enolate geometry on the stereochemistry of Michael additions of ketone enolates to α,β-unsaturated ketones Tetrahedron Letters. 28: 1354. DOI: 10.1016/S0040-4039(00)85424-6  0.775
1987 OARE DA, HEATHCOCK CH. ChemInform Abstract: Acyclic Stereoselection. Part 38. Influence of Enolate Geometry on the Stereochemistry of Michael Additions of Ketone Enolates to α,β-Unsaturated Ketones. Cheminform. 18. DOI: 10.1002/chin.198725063  0.754
1987 HEATHCOCK CH, RADEL PA. ChemInform Abstract: Acyclic Stereoselection. Part 37. Total Synthesis of a Slightly Unnatural Product. Confirmation of the Stereostructure of the Archaebacterial C40 Diol by Synthesis of a Stereoisomer. Cheminform. 18. DOI: 10.1002/chin.198717320  0.323
1986 Heathcock CH, Radel PA. Total synthesis of a slightly unnatural product. Confirmation of the stereostructure of the archaebacterial C40 diol by synthesis of a stereoisomer Journal of Organic Chemistry. 51: 4322-4323. DOI: 10.1021/Jo00372A051  0.37
1986 Heathcock CH, Davidsen SK, Hug KT, Flippin LA. Acyclic stereoselection. XXXVI: Simple diastereoselection in the Lewis acid mediated reactions of enol silanes with aldehydes Journal of Organic Chemistry. 51: 3027-3037. DOI: 10.1021/Jo00365A033  0.447
1986 Heathcock CH, Uehling DE. Acyclic stereoselection. Part 34. Stereoselection in the Michael addition reaction. 4. Diastereofacial preferences in Lewis acid-mediated additions of enolsilanes to chiral enones The Journal of Organic Chemistry. 51: 279-280. DOI: 10.1021/Jo00352A040  0.446
1986 Heathcock CH, Davidsen SK, Mills S, Sanner MA. Total synthesis of (.+-.)-methyl homodaphniphyllate Journal of the American Chemical Society. 108: 5650-5651. DOI: 10.1021/Ja00278A061  0.384
1986 Heathcock CH, Smith KM, Blumenkopf TA. Total synthesis of (±)-fawcettimine (Burnell's base A) Journal of the American Chemical Society. 108: 5022-5024. DOI: 10.1021/Ja00276A062  0.343
1986 Heathcock CH, Davidsen SK, Hug KT, Flippin LA. Acyclic stereoselection. 36. Simple diastereoselection in the Lewis acid mediated reactions of enol silanes with aldehydes Journal of Organic Chemistry. 51: 3027-3037. DOI: 10.1016/S0040-4039(01)81736-6  0.438
1986 Rosen T, Heathcock CH. The synthesis of mevinic acids Tetrahedron. 42: 4909-4951. DOI: 10.1016/S0040-4020(01)88045-5  0.304
1986 Hecker SJ, Heathcock CH. Total synthesis of (+)-dihydromevinolin Journal of the American Chemical Society. 108: 4586-4594. DOI: 10.1002/Chin.198648343  0.417
1986 HEATHCOCK CH, UEHLING DE. ChemInform Abstract: Acyclic Stereoselection. Part 34. Stereoselection in the Michael Addition Reactions. Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198627088  0.342
1986 Takai K, Heathcock CH. Acyclic Stereoselection. Part 32. Synthesis and Characterization of the Diastereomeric (4S)‐Pentane‐1,2,3,4‐tetrols. Cheminform. 17. DOI: 10.1002/Chin.198601076  0.4
1986 Heathcock CH, Uehling DE. Stereoselection in the Michael addition reaction. 4. Diastereofacial preferences in Lewis acid mediated additions of enolsilanes to chiral enones Journal of Organic Chemistry. 51: 279-280.  0.331
1985 Hecker SJ, Heathcock CH. An approach to the synthesis of mevinolin based on intramolecular Diels-Alder cycloaddition Journal of Organic Chemistry. 50: 5159-5166. DOI: 10.1021/Jo00225A037  0.398
1985 Takai K, Heathcock CH. Acyclic stereoselection. 32. Synthesis and characterization of the diastereomeric (4S)-pentane-1,2,3,4-tetrols Journal of Organic Chemistry. 50: 3247-3251. DOI: 10.1021/Jo00218A001  0.395
1985 Heathcock CH, Oare DA. Acyclic stereoselection. 31. Stereoselection in the Michael addition reaction. 3. Relationship between ester enolate geometry and adduct stereochemistry in the kinetic Michael reaction of lithium enolates with enones Journal of Organic Chemistry. 50: 3022-3024. DOI: 10.1021/Jo00216A051  0.779
1985 Heathcock CH, Henderson MA, Oare DA, Sanner MA. Acyclic stereoselection. 30. Stereoselection in the Michael addition reaction. 2. Stereochemistry of the kinetic Michael reaction of amide enolates with enones The Journal of Organic Chemistry. 50: 3019-3022. DOI: 10.1021/Jo00216A050  0.768
1985 Rosen T, Heathcock CH. Synthetic and biological studies of compactin and related compounds. 4. Total synthesis of (+)-compactin Journal of the American Chemical Society. 107: 3731-3733. DOI: 10.1021/Ja00298A062  0.369
1985 Doney JJ, Bergman RG, Heathcock CH. Synthesis, structure, and carbon-carbon bond-forming reactions of carbon-bound molybdenum, tungsten, and rhenium enolates. Detection of an .eta.3-oxaallyl intermediate Journal of the American Chemical Society. 107: 3724-3726. DOI: 10.1021/Ja00298A057  0.327
1985 Heathcock CH, Norman MH, Uehling DE. Acyclic stereoselection. 29. Stereoselection in the Michael addition reaction. 1. The Mukaiyama-Michael reaction Journal of the American Chemical Society. 107: 2797-2799. DOI: 10.1021/Ja00295A037  0.412
1985 Heathcock CH, Montgomery SH. Acyclic stereoselection. 28. Use of stereoselective aldol methodology in the total synthesis of cladinose. Tetrahedron Letters. 26: 1001-1004. DOI: 10.1016/S0040-4039(00)98496-X  0.453
1985 Heathcock CH, Arseniyadis S. Acyclic stereoselection. 35. Effect of cation on diastereofacial selectivity in aldol reactions of a chiral α-silyloxy ketone Tetrahedron Letters. 26: 6009-6012. DOI: 10.1016/S0040-4039(00)95111-6  0.442
1985 Heathcock CH, Doney JJ, Bergman RG. Synthesis and carbon-carbon bond-forming reactions of tungsten, molybdenum, and rhenium enolates Pure and Applied Chemistry. 57: 1789-1798. DOI: 10.1002/Chin.198614380  0.336
1985 Connolly PJ, Heathcock CH. An approach to the total synthesis of dendrobine Journal of Organic Chemistry. 50: 4135-4144. DOI: 10.1002/Chin.198610368  0.344
1985 Heathcock CH, Oare DA. Acyclic Stereoselection. 31. Stereoselection In The Michael Addition Reaction. 3. Relationship Between Ester Enolate Geometry And Adduct Stereochemistry In The Kinetic Michael Reaction Of Lithium Enolates With Enones Cheminform. 16. DOI: 10.1002/Chin.198551087  0.796
1985 Heathcock CH, Young SD, Hagen JP, Pilli R, Badertscher U. Acyclic stereoselection. 25. Stereoselective synthesis of the C-1 to C-7 moiety of erythronolide A Journal of Organic Chemistry. 50: 2095-2105. DOI: 10.1002/Chin.198547330  0.595
1985 HEATHCOCK CH, NORMAN MH, UEHLING DE. ChemInform Abstract: ACYCLIC STEREOSELECTION. 29. STEREOSELECTION IN THE MICHAEL ADDITION REACTION. 1. THE MUKAIYAMA-MICHAEL REACTION Chemischer Informationsdienst. 16. DOI: 10.1002/chin.198536086  0.307
1985 Heathcock CH, Von Geldern TW, Lebrilla CB, Maier WF. Nucleophilic substitution with inversion of configuration at the nucleophile Journal of Organic Chemistry. 50: 968-972. DOI: 10.1002/Chin.198535174  0.426
1985 Rosen T, Taschner MJ, Thomas JA, Heathcock CH. Synthetic and biological studies of compactin and related compounds. 3. Synthesis of the hexalin portion of compactin Journal of Organic Chemistry. 50: 1190-1201. DOI: 10.1002/Chin.198535148  0.337
1985 Rosen T, Heathcock CH. Total synthesis of (+)-compactin Journal of the American Chemical Society. 107: 3731-3733.  0.302
1985 Heathcock CH, Oare DA. Stereoselection in the Michael addition reaction. 3. Relationship between ester enolate geometry and adduct stereochemistry in the kinetic Michael reaction of lithium enolates with enones Journal of Organic Chemistry. 50: 3022-3024.  0.781
1984 Heathcock CH, Pirrung MC, Young SD, Hagen JP, Jarvi ET, Badertscher U, Märki HP, Montgomery SH. Acyclic stereoselection. 23. Lactaldehyde enolate equivalents Journal of the American Chemical Society. 106: 8161-8174. DOI: 10.1021/Ja00338A027  0.655
1984 Heathcock CH, Hug KT, Flippin LA. Acyclic stereoselection. 27. Simple diastereoselection in the lewis acid mediated reactions of enolsilanes with aldehydes Tetrahedron Letters. 25: 5973-5976. DOI: 10.1016/S0040-4039(01)81736-6  0.326
1984 Kiyooka Si, Sasaoka H, Fujiyama R, Heathcock CH. Diastereofacial selectivity in the Lewis acid mediated reactions of allylsilane with chiral β-alkoxy acetal Tetrahedron Letters. 25: 5331-5334. DOI: 10.1016/S0040-4039(01)81596-3  0.39
1984 Heathcock CH, Jarvi ET, Rosen T. Acyclic stereoselection. 21. Synthesis of an ionophore synthon having four asymmetric carbons by sequential aldol addition, claisen rearrangement and hydroboration Tetrahedron Letters. 25: 243-246. DOI: 10.1016/S0040-4039(00)99851-4  0.399
1984 Heathcock CH, Kiyooka SI, Blumenkopf TA. Acyclic stereoselection. 22. Diastereofacial selectivity in the Lewis acid mediated reactions of allylsilanes with chiral aldehydes and enones Journal of Organic Chemistry. 49: 4214-4223. DOI: 10.1002/Chin.198519094  0.431
1984 Rosen T, Taschner MJ, Heathcock CH. Synthetic and biological studies of compactin and related compounds. 2. Synthesis of the lactone moiety of compactin Journal of Organic Chemistry. 49: 3994-4003. DOI: 10.1002/Chin.198515272  0.354
1984 HEATHCOCK CH. ChemInform Abstract: Stereoselective Aldol Condensations Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198449357  0.301
1984 HEATHCOCK CH, MONTGOMERY SH. ChemInform Abstract: ACYCLIC STEREOSELECTION. 19. TOTAL SYNTHESIS OF (.+-.)-RISTOSAMINE AND (.+-.)-MEGALOSAMINE Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198407309  0.347
1983 Heathcock CH, Jennings RA, Von Geldern TW. Studies directed toward the total synthesis of securinega alkaloids Journal of Organic Chemistry. 48: 3428-3431. DOI: 10.1021/Jo00168A011  0.345
1983 Blumenkopf TA, Heathcock CH. Stereochemistry of the Sakurai reaction. Additions to cyclohexenones and cycloheptenones Journal of the American Chemical Society. 105: 2354-2358. DOI: 10.1021/Ja00346A041  0.393
1983 Heathcock CH, Flippin LA. Acyclic stereoselection. 16. High diastereofacial selectivity in Lewis acid mediated additions of enolsilanes to chiral aldehydes Journal of the American Chemical Society. 105: 1667-1668. DOI: 10.1021/Ja00344A050  0.371
1983 Kiyooka Si, Heathcock CH. Acyclic stereoselection. 20. High diastereofacial selectivity in the stannic chloride mediated reactions of allylsilanes with chiral α- and β-alkoxy aldehydes Tetrahedron Letters. 24: 4765-4768. DOI: 10.1016/S0040-4039(00)94002-4  0.366
1983 Heathcock CH, Montgomery SH. Acyclic stereoselection. 19. Total synthesis of (±)-ristosamine and (±)-megalosamine. Tetrahedron Letters. 24: 4637-4640. DOI: 10.1016/S0040-4039(00)86214-0  0.322
1983 Heathcock CH, Lampe J. Acyclic stereoselection. 17. Simple diastereoselection in the addition of medium- and long-chain n-alkyl ketone lithium enolates to aldehydes Journal of Organic Chemistry. 48: 4330-4337. DOI: 10.1002/Chin.198418091  0.361
1982 Heathcock CH, Tice CM, Germroth TC. Synthesis of sesquiterpene antitumor lactones. 10. Total synthesis of (.+-.)-parthenin Journal of the American Chemical Society. 104: 6081-6091. DOI: 10.1021/Ja00386A040  0.438
1982 Heathcock CH, DelMar EG, Graham SL. Synthesis of sesqui terpene anti tumor lactones 9. the hydro naphthalene route to pseudo guaianes total synthesis of racemic confertin Journal of the American Chemical Society. 104: 1907-1917. DOI: 10.1021/Ja00371A020  0.364
1982 Heathcock CH, Kleinman EF, Binkley ES. Total synthesis of lycopodium alkaloids: (.+-.)-lycopodine, (.+-.)-lycodine, and (.+-.)-lycodoline Journal of the American Chemical Society. 104: 1054-1068. DOI: 10.1021/Ja00368A024  0.424
1982 Heathcock CH, Jarvi ET. Acyclic stereoselection. 15. Sequential aldol-claisen as a method for 1,5-stereoselection. Total synthesis of the vitamin-E side chain Tetrahedron Letters. 23: 2825-2828. DOI: 10.1016/S0040-4039(00)88423-3  0.398
1982 Heathcock CH, Taschner MJ, Rosen T, A. Thomas J, Hadley CR, Popják G. Synthesis and biological activity of the hexalin moiety of compactin (ML-236B) Tetrahedron Letters. 23: 4747-4750. DOI: 10.1016/S0040-4039(00)85703-2  0.306
1982 Heathcock CH, DelMar EG, Graham SL. Synthesis of sesquiterpene antitumor lactones. 9. The hydronaphthalene route to pseudoguaianes. Total synthesis of (±)-confertin Journal of the American Chemical Society. 104: 1907-1917. DOI: 10.1002/Chin.198231297  0.358
1981 Heathcock CH. Acyclic stereocontrol through the aldol condensation. Science (New York, N.Y.). 214: 395-400. PMID 17730226 DOI: 10.1002/Chin.198209364  0.372
1981 Heathcock CH, Pirrung MC, Lampe J, Buse CT, Young SD. Acyclic stereoselection. 12. Double stereodifferentiation with mutual kinetic resolution. A superior class of reagents for control of Cram's rule stereoselection in synthesis of erythro-.alpha.-alkyl-.beta.-hydroxy carboxylic acids from chiral aldehydes Journal of Organic Chemistry. 46: 2290-2300. DOI: 10.1021/Jo00324A017  0.717
1981 Heathcock CH, White CT, Morrison JJ, VanDerveer D. Acyclic stereoselection. 11. Double stereodifferentiation as a method for achieving superior Cram's rule selectivity in aldol condensations with chiral aldehydes Journal of Organic Chemistry. 46: 1296-1309. DOI: 10.1021/Jo00320A014  0.336
1981 White CT, Heathcock CH. Acyclic stereoselection. 10. A general synthesis of erythro-.alpha.-alkyl-.beta.-hydroxy ketones The Journal of Organic Chemistry. 46: 191-192. DOI: 10.1021/Jo00314A047  0.371
1981 Tice CM, Heathcock CH. Synthesis of sesquiterpene antitumor lactones. 8. An approach to the synthesis of pseudoguianolides based on oxy-Cope rearrangement Journal of Organic Chemistry. 46: 9-13. DOI: 10.1021/Jo00314A003  0.409
1981 Heathcock CH, Hagen JP, Jarvi ET, Pirrung MC, Young SD. Acyclic stereoselection. 14. O-alkyllactic acid esters: reagents for the stereoselective construction of erythro- and threo-.alpha.-methyl-.alpha.,.beta.-dihydroxy carbonyl compounds Journal of the American Chemical Society. 103: 4972-4974. DOI: 10.1021/Ja00406A064  0.679
1981 Heathcock CH, Kleinman EF. Total synthesis of (.+-.)-lycodoline Journal of the American Chemical Society. 103: 222-223. DOI: 10.1021/Ja00391A055  0.417
1981 Schinzer D, Heathcock CH. Fluoride-catalyzed conversion of acylsilanes to aldehydes and ketones Tetrahedron Letters. 22: 1881-1884. DOI: 10.1016/S0040-4039(01)90467-8  0.347
1981 Heathcock CH, Pirrung MC, Montgomery SH, Lampe J. Acyclic stereoselection-13. Aryl esters: reagents for threo-aldolization Tetrahedron. 37: 4087-4095. DOI: 10.1016/S0040-4020(01)93284-3  0.736
1981 Heathcock CH, Pirrung MC, Lampe J, Buse CT, Young SD. Acyclic stereoselection. 12. Double stereodifferentiation with mutual kinetic resolution. A superior class of reagents for control of Cram's rule stereoselection in synthesis of erythro-.alpha.-alkyl-.beta.-hydroxy carboxylic acids from chiral aldehydes Cheminform. 12. DOI: 10.1002/Chin.198142079  0.717
1981 Heathcock CH, Hagen JP, Jarvi ET, Pirrung MC, Young SD. Acyclic stereoselection. 14. O-alkyllactic acid esters: Reagents for the stereoselective construction of erythro- and threo-α-methyl-α,β-dihydroxy carbonyl compounds Journal of the American Chemical Society. 103: 4972-4974.  0.663
1981 Heathcock CH, Pirrung MC, Lampe J, Buse CT, Young SD. Acyclic stereoselection. 12. Double stereodifferentiation with mutual kinetic resolution. A superior class of reagents for control of cram's rule stereoselection in synthesis of erythro-α-alkyl-β-hydroxy carboxylic acids from chiral aldehydes Journal of Organic Chemistry. 46: 2290-2300.  0.696
1980 Dugger RW, Heathcock CH. An Efficient Preparation oftrans, trans-β-Ionylideneacetaldehyde Synthetic Communications. 10: 509-515. DOI: 10.1080/00397918008069326  0.413
1980 Heathcock CH, Young SD, Hagen JP, Pirrung MC, White CT, VanDerveer D. Acyclic stereoselection. 9. Stereochemistry of the addition of lithium enolates to .alpha.-alkoxy aldehydes Journal of Organic Chemistry. 12: 3846-3856. DOI: 10.1021/Jo01307A023  0.679
1980 Pirrung MC, Heathcock CH. Acyclic stereoselection. 8. A new class of reagents for the highly stereoselective preparation of threo-2-alkyl-3-hydroxycarboxylic acids by the aldol condensation Journal of Organic Chemistry. 45: 1727-1728. DOI: 10.1021/Jo01297A057  0.719
1980 Dugger RW, Heathcock CH. A general synthesis of 5,6-dihydro-.alpha.-pyrones The Journal of Organic Chemistry. 45: 1181-1185. DOI: 10.1021/Jo01295A002  0.318
1980 Heathcock CH, Buse CT, Kleschick WA, Pirrung MC, Sohn JE, Lampe J. Acyclic stereoselection. 7. Stereoselective synthesis of 2-alkyl-3-hydroxy carbonyl compounds by aldol condensation Journal of Organic Chemistry. 45: 1066-1081. DOI: 10.1021/Jo01294A030  0.732
1980 Heathcock CH, Buse CT, Kleschick WA, Pirrung MC, Sohn JE, Lampe J. Correction. Acyclic Stereoselection. 7. Stereoselective Synthesis of 2-Alkyl-3-hydroxy Carbonyl Compounds by Aldol Condensation Journal of Organic Chemistry. 45: 1066-1081. DOI: 10.1021/Jo00339A601  0.73
1980 Thomas JA, Heathcock CH. A reagent for cyclohexene annelation Tetrahedron Letters. 21: 3235-3236. DOI: 10.1016/S0040-4039(00)78654-0  0.421
1980 Graham SL, Heathcock CH. Stereoselectivity in the alkylation of sulfonium salts Tetrahedron Letters. 21: 3865-3868. DOI: 10.1016/0040-4039(80)80201-2  0.385
1980 Heathcock CH, Pirrung MC, Buse CT, Hagen JP, Young SD, Sohn JE. Acyclic stereoselection. 6. A reagent for achieving high 1,2-diastereoselection in the aldol conversion of chiral aldehydes into 3-hydroxy-2-methylcarboxylic acids Cheminform. 11. DOI: 10.1002/Chin.198007106  0.702
1980 Heathcock CH, Young SD, Hagen JP, Pirrung MC, White CT, VanDerveer D. Acyclic stereoselection. 9. Stereochemistry of the addition of lithium enolates to α-alkoxy aldehydes Journal of Organic Chemistry. 45: 3846-3856.  0.674
1979 Davalian D, Heathcock CH. Synthesis of 7,8-epoxy-7,8-dihydroretinoids The Journal of Organic Chemistry. 44: 4458-4461. DOI: 10.1021/Jo01338A049  0.434
1979 Heathcock CH, Pirrung MC, Sohn JE. Acyclic stereoselection. 4. Assignment of stereostructure to .beta.-hydroxycarbonyl compounds by carbon-13 nuclear magnetic resonance The Journal of Organic Chemistry. 44: 4294-4299. DOI: 10.1021/Jo01338A015  0.633
1979 Heathcock CH, Germroth TC, Graham SL. Stereochemistry of cuprate addition to 4-, 5-, and 6-alkylcycloheptenones The Journal of Organic Chemistry. 44: 4481-4487. DOI: 10.1021/Jo00393A004  0.398
1979 Heathcock CH, Pirrung MC, Buse CT, Hagen JP, Young SD, Sohn JE. Acyclic stereoselection. 6. A reagent for achieving high 1,2-diastereoselection in the aldol conversion of chiral aldehydes into 3-hydroxy-2-methylcarboxylic acids Journal of the American Chemical Society. 101: 7077-7079. DOI: 10.1021/Ja00517A056  0.719
1979 Heathcock CH, White CT. Acyclic stereoselection. 5. Use of double stereodifferentiation to enhance 1,2 diastereoselection in aldol condensations of chiral aldehydes Journal of the American Chemical Society. 101: 7076-7077. DOI: 10.1021/Ja00517A055  0.395
1979 Plavac F, Heathcock CH. Synthesis of sesquiterpene antitumor lactones. 7. Studies directed toward the total synthesis of pentalenolactone. Intramolecular ene reaction. Tetrahedron Letters. 20: 2115-2118. DOI: 10.1016/S0040-4039(01)86277-8  0.492
1978 Kleschick WA, Heathcock CH. Synthesis and chemistry of ethyl 2-diethylphosphonoacrylate The Journal of Organic Chemistry. 43: 1256-1259. DOI: 10.1021/Jo00400A056  0.45
1978 Heathcock CH, Kleinman E, Binkley ES. A highly efficient total synthesis of (.+-.)-lycopodine Journal of the American Chemical Society. 100: 8036-8037. DOI: 10.1021/Ja00493A057  0.381
1978 Buse CT, Heathcock CH. Acyclic stereoselection. III. Synthesis of threo-3-hydroxy-2-methylcarboxylic acids Tetrahedron Letters. 19: 1685-1688. DOI: 10.1016/S0040-4039(01)94640-4  0.421
1977 Kozar LG, Clark RD, Heathcock CH. Synthesis of bicyclo[2.2.2]octenes and bicyclo[3.2.2]nonenes by .pi.-cyclization The Journal of Organic Chemistry. 42: 1386-1389. DOI: 10.1021/Jo00428A026  0.654
1977 Buse CT, Heathcock CH. Acyclic stereoselection. 2. Synthesis of 3-hydroxy-2-methyl- and 3-hydroxy-2,4-dimethylcarboxylic acids Journal of the American Chemical Society. 99: 8109-8110. DOI: 10.1021/Ja00466A085  0.428
1977 Kleschick WA, Buse CT, Heathcock CH. Stereoselection in the aldol condensation Journal of the American Chemical Society. 99: 247-248. DOI: 10.1021/Ja00443A046  0.451
1976 Clark RD, Heathcock CH. Synthesis of a cytotoxic vernolepin prototype. Ozonization of silyloxyalkenes. The Journal of Organic Chemistry. 41: 1396-403. PMID 1263006 DOI: 10.1002/Chin.197634228  0.617
1976 Wege PM, Clark RD, Heathcock CH. Synthesis of sesquiterpene antitumor lactones. 6. cis-8a-Vinyloctahydro-3H-2-benzopyran-3,7-dione, a precursor to vernolepin. The Journal of Organic Chemistry. 41: 3144-8. PMID 966107 DOI: 10.1002/Chin.197652369  0.546
1976 Chavdarian CG, Heathcock CH. Synthesis of Sesquiterpene Anti-Tumor Lactones. IV1. A Stereoselective Synthesis oftrans-2,3-Epoxycyclohexanol Synthetic Communications. 6: 277-280. DOI: 10.1080/00397917608063522  0.358
1976 Ellis JE, Dutcher JS, Heathcock CH. Pentacyclic triterpene synthesis. 6. Synthesis of a bicyclic intermediate corresponding to rings D and E of .beta.-amyrin The Journal of Organic Chemistry. 41: 2670-2676. DOI: 10.1021/Jo00878A002  0.402
1976 Dutcher JS, Macmillan JG, Heathcock CH. Pentacyclic triterpene synthesis. 5. Synthesis of optically pure ring AB precursors The Journal of Organic Chemistry. 41: 2663-2669. DOI: 10.1021/Jo00878A001  0.395
1976 Clark RD, Heathcock CH. Preparation and reactions of .beta.-chloro-.alpha.,.beta.-unsaturated ketones The Journal of Organic Chemistry. 41: 636-643. DOI: 10.1021/Jo00866A012  0.557
1976 Chavdarian CG, Woo SL, Clark RD, Heathcock CH. Synthesis of sesquiterpene antitumor lactones. V. a model for rings B and C of vernolepin Tetrahedron Letters. 17: 1769-1772. DOI: 10.1016/S0040-4039(00)93778-X  0.569
1976 ELLIS JE, DUTCHER JS, HEATHCOCK CH. ChemInform Abstract: PENTACYCLIC TRITERPENE SYNTHESIS. 6. SYNTHESIS OF A BICYCLIC INTERMEDIATE CORRESPONDING TO RINGS D AND E OF β-AMYRIN Chemischer Informationsdienst. 7: no-no. DOI: 10.1002/Chin.197645370  0.42
1975 Chavdarian CG, Heathcock CH. Synthesis of delta-lactones from cyclohexenones. Preparation of a vernolepin analog. The Journal of Organic Chemistry. 40: 2970-1. PMID 1177076 DOI: 10.1021/Jo00908A031  0.446
1975 Clark RD, Kozar LG, Heathcock CH. Cyclopentenones from β, ε-Diketo Phosphonates. Synthesis of cis-Jasmone Synthetic Communications. 5: 1-5. DOI: 10.1080/00397917508063507  0.611
1975 CLARK RD, KOZAR LG, HEATHCOCK CH. Alkylation of Diethyl 2-Oxoalkanephosphonates Synthesis. 1975: 635-636. DOI: 10.1055/S-1975-23860  0.632
1975 Clark RD, Heathcock CH. Synthesis of spiro lactones and ketones via conjugate addition to cyclopropyl malonates and β-keto esters Tetrahedron Letters. 16: 529-532. DOI: 10.1016/S0040-4039(00)71912-5  0.611
1975 CLARK RD, KOZAR LG, HEATHCOCK CH. ChemInform Abstract: CYCLOPENTENONES FROM BETA,EPSILON-DIKETO PHOSPHONATES. SYNTHESIS OF CIS-JASMONE Chemischer Informationsdienst. 6: no-no. DOI: 10.1002/Chin.197529407  0.316
1974 Ellis JE, Dutcher JS, Heathcock CH. Pentacyclic Triterpene Synthesis. IV a New Method for Accomplishing Robinson-Nazarov Annelations Synthetic Communications. 4: 71-77. DOI: 10.1080/00397917408062058  0.378
1974 CLARK RD, HEATHCOCK CH. A New Procedure for the Preparation of β-Chloro-α,β-unsaturated Ketones Synthesis. 1974: 47-48. DOI: 10.1055/S-1974-23238  0.54
1974 Clark RD, Heathcock CH. Ozonization of silyloxyalkenes Tetrahedron Letters. 15: 2027-2030. DOI: 10.1016/S0040-4039(01)82622-8  0.471
1974 Clark RD, Heathcock CH. A new synthesis of the vernolepin a-ring Tetrahedron Letters. 15: 1713-1715. DOI: 10.1016/S0040-4039(01)82561-2  0.604
1974 Dutcher JS, Heathcock CH. Pentacyclic triterpene synthesis. III. Preparation of an optically active synthon for rings A and B Tetrahedron Letters. 15: 933-936. DOI: 10.1016/S0040-4039(01)82372-8  0.335
1974 Dutcher JS, Macmillan JG, Heathcock CH. Pentacyclic triterpene synthesis. II. Preparation of an AB synthon Tetrahedron Letters. 15: 929-932. DOI: 10.1016/S0040-4039(01)82371-6  0.359
1973 Brattesani DN, Heathcock CH. A Convenient Procedure for the Alkylation of Acetylenes Synthetic Communications. 3: 245-248. DOI: 10.1080/00397917308065910  0.375
1973 Clark RD, Ellis JE, Heathcock CH. Methylation of Dimedone Synthetic Communications. 3: 347-354. DOI: 10.1080/00397917308063488  0.565
1973 Clark RD, Heathcock CH. Reduction of .beta.-halo-.alpha.,.beta.-unsaturated ketones The Journal of Organic Chemistry. 38: 3658-3658. DOI: 10.1021/Jo00960A060  0.519
1972 Amano Y, Heathcock CH. (+)-Occidentalol: Absolute Stereostructure and Total Synthesis Canadian Journal of Chemistry. 50: 340-345. DOI: 10.1139/V72-051  0.409
1972 Ratcliffe BE, Heathcock CH. Synthesis and Characterization of S-Methylspiro[4.5]-dec-7-en-6-one and 6-methylspiro[4.5]dec-6-en-8-one Synthetic Communications. 2: 157-163. DOI: 10.1080/00397917208081758  0.79
1972 Heathcock CH, Ratcliffe R, Van J. Synthesis of hydroazulenes by solvolytic rearrangement of 9-methyl-1-declyl tosylates The Journal of Organic Chemistry. 37: 1796-1807. DOI: 10.1021/Jo00976A029  0.398
1972 Heathcock CH, Ratcliffe BE. Acid-catalyzed rearrangement of 6-methyltricyclo[4.4.0.02,7]decan-3-one The Journal of Organic Chemistry. 37: 1298-1304. DOI: 10.1021/Jo00974A003  0.787
1972 Ratcliffe BE, Heathcock CH. Acid-catalyzed rearrangement of tricyclo[4.4.0.2,7]decan-3-ols The Journal of Organic Chemistry. 37: 531-537. DOI: 10.1021/Jo00969A001  0.79
1972 Heathcock CH, Badger RA. Photochemistry of 1,6-cyclodecadienes. II. Synthesis and photochemistry of 6-methyl-1,6-cyclodecadien-3-one The Journal of Organic Chemistry. 37: 234-238. DOI: 10.1021/Jo00967A013  0.788
1972 Heathcock CH, Badger RA, Starkey RA. Photochemistry of 1,6-cyclodecadienes. I. 1-Methyl-(E,E)-1,6-cyclodecadiene The Journal of Organic Chemistry. 37: 231-234. DOI: 10.1021/Jo00967A012  0.758
1972 Heathcock CH, Badger RA, Starkey RH. Correction. Photochemistry of 1,6-Cyclodecadienes. I. 1-Methyl-(E,E)-1,6-cyclodecadiene The Journal of Organic Chemistry. 37: 3754-3754. DOI: 10.1021/Jo00796A619  0.758
1972 HEATHCOCK CH, ELLIS JE, MCMURRY JE, COPPOLINO A. ChemInform Abstract: SAEURE-KATALYSIERTE ROBINSON-ANNELLIERUNGSRK. Chemischer Informationsdienst. 3: no-no. DOI: 10.1002/Chin.197214260  0.594
1971 Heathcock CH, Ellis JE. Pentacyclic triterpene synthesis. Preparation of a useful intermediate Journal of the Chemical Society D: Chemical Communications. 1474-1475. DOI: 10.1039/C29710001474  0.342
1971 Heathcock CH, Ratcliffe R. Stereoselective total synthesis of the guaiazulenic sesquiterpenoids .alpha.-bulnesene and bulnesol Journal of the American Chemical Society. 93: 1746-1757. DOI: 10.1021/Ja00736A029  0.338
1971 Heathcock CH, Ellis JE, McMurry JE, Coppolino A. Acid-catalyzed Robinson Annelations Tetrahedron Letters. 12: 4995-4996. DOI: 10.1016/S0040-4039(01)97609-9  0.627
1970 Hassner A, Hoblitt RP, Heathcock C, Kropp JE, Lorber M. Stereochemistry. XLV. Electronic vs. steric effects in the addition of iodine isocyanate to olefins Journal of the American Chemical Society. 92: 1326-1331. DOI: 10.1021/Ja00708A036  0.454
1970 HASSNER A, HOBLITT RP, HEATHCOCK C, KROPP JE, LORBER M. ChemInform Abstract: ELEKTRONISCHE UND STERISCHE EINFLUESSE BEI DER ADDITION VON JODISOCYANAT AN OLEFINE Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/Chin.197023122  0.519
1969 Heathcock CH, Poulter SR. Catalytic hydrogenation of cyclopropyl alkenes. III. On the mechanism of homogeneous hydrogenation in the presence of tris(triphenylphosphine)chlororhodium(I). Tetrahedron Letters. 10: 2755-2758. DOI: 10.1016/S0040-4039(01)88261-7  0.751
1969 Heathcock CH, Gulick LC, Dehlinger T. Reaction of furyllithium with carboxylic acids Journal of Heterocyclic Chemistry. 6: 141-142. DOI: 10.1002/Jhet.5570060130  0.381
1969 Heathcock CH, Ellis JE, Badger RA. Reaction of alkyllithium reagents with 2,2-dialkyi-l,3-dioxolanes Journal of Heterocyclic Chemistry. 6: 139-140. DOI: 10.1002/Jhet.5570060129  0.779
1969 Heathcock CH. A New Synthesis of Alkyl Azides Angewandte Chemie International Edition in English. 8: 134-135. DOI: 10.1002/Anie.196901341  0.421
1969 Heathcock CH. Neue Synthese für Alkylazide Angewandte Chemie. 81: 148-149. DOI: 10.1002/Ange.19690810405  0.348
1968 Heathcock CH, Kelly TR. Total synthesis of nor-ketoagarofuran Chemical Communications (London). DOI: 10.1039/C1968000267a  0.55
1968 Heathcock CH, Badger RA. Synthesis and photocyclization of a cyclodecadienone Chemical Communications (London). 1510-1511. DOI: 10.1039/C19680001510  0.812
1968 Heathcock CH, Ratcliffe BE. Unusual cyclobutane pyrolysis The Journal of Organic Chemistry. 33: 3650-3651. DOI: 10.1021/Jo01273A071  0.767
1968 Heathcock CH, Poulter SR. The effect of cyclopropyl substitution on the .pi.->.pi.* transition of simple olefins Journal of the American Chemical Society. 90: 3766-3769. DOI: 10.1021/Ja01016A028  0.764
1968 Poulter SR, Heathcock CH. Catalytic hydrogenation of cyclopropyl alkenes. II. Nature of the intermediates in the heterogeneous hydrogenolysis reaction Tetrahedron Letters. 9: 5343-5347. DOI: 10.1016/S0040-4039(00)75380-9  0.784
1968 Poulter SR, Heathcock CH. Catalytic hydrogenation of cyclopropyl alkenes. I. Effect of alkyl substitution on the heterogeneous hydrogenolysis reaction Tetrahedron Letters. 9: 5339-5342. DOI: 10.1016/S0040-4039(00)75379-2  0.799
1968 Heathcock C, Kelly T. Sesquiterpenoids—IV Tetrahedron. 24: 3753-3765. DOI: 10.1016/S0040-4020(01)92007-1  0.434
1967 Hassner A, Lorber ME, Heathcock C. Addition of iodine isocyanate to olefins. Scope and synthetic utility. The Journal of Organic Chemistry. 32: 540-9. PMID 6042109 DOI: 10.1021/Jo01278A006  0.571
1967 Heathcock CH, Badger RA, Patterson JW. Total synthesis of (.+-.)-copaene and (.+-.)-ylangene. General method for the synthesis of tricyclo [4.4.0.02,7]decanes Journal of the American Chemical Society. 89: 4133-4145. DOI: 10.1021/Ja00992A032  0.804
1966 Heathcock CH. The synthesis of 1-methyltricyclo[4.4.0.02,7]decanes Tetrahedron Letters. 7: 2043-2047. DOI: 10.1016/S0040-4039(00)76293-9  0.431
1965 Hassner A, Heathcock C. Additions and Corrections-On the Mechanism of the Conversion of β-Iodo Carbamates to Aziridines The Journal of Organic Chemistry. 30: 4395-4395. DOI: 10.1021/Jo01023A611  0.458
1965 Hassner A, Heathcock C. Synthesis and Ring Opening of Fused Steroidal Aziridines*,1 The Journal of Organic Chemistry. 30: 1748-1752. DOI: 10.1021/Jo01017A010  0.561
1965 Jorgenson MJ, Heathcock CH. Photochemistry of Cyclopropylacrylic Esters Journal of the American Chemical Society. 87: 5264-5266. DOI: 10.1021/Ja00950A060  0.399
1964 Hassner A, Heathcock C. On the Mechanism of the Conversion of β-Iodo Carbamates to Aziridines1 The Journal of Organic Chemistry. 29: 3640-3645. DOI: 10.1021/Jo01035A052  0.445
1964 Hassner A, Heathcock C. Reaction of Nitrosyl Chloride with Steroid 5-Enes.1Nuclear Magnetic Resonance as a Stereochemical Tool in Steroids The Journal of Organic Chemistry. 29: 1350-1355. DOI: 10.1021/Jo01029A019  0.473
1964 Hassner A, Heathcock C. Synthesis of fused ethyleneimines from cyclic olefins Tetrahedron. 20: 1037-1042. DOI: 10.1016/S0040-4020(01)98439-X  0.349
1963 Hassner A, Heathcock C. The stereochemistry of ethyleneimines fused to six-membered rings Tetrahedron Letters. 4: 393-395. DOI: 10.1016/S0040-4039(01)90644-6  0.425
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