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Paul Knochel - Publications

Affiliations: 
1987-1992 University of Michigan, Ann Arbor, Ann Arbor, MI 
 1992-1999 Philipps-Universität Marburg, Marburg, Hessen, Germany 
 1999- Chemistry Ludwig-Maximilians-Universität München, München, Bayern, Germany 
Area:
organic synthesis, asymmetric catalysis and natural product synthesis
Website:
http://www.knochel.cup.uni-muenchen.de/index.php?prof-dr-paul-knochel-1

316 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Leroux M, Huang WY, Lemke Y, Koller T, Karaghiosoff K, Knochel P. Pyrrole Protected β-Aminoalkylzinc Reagents for the Enantioselective Synthesis of Amino-Derivatives. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 32196786 DOI: 10.1002/chem.202000870  0.32
2020 Lutter FH, Grokenberger L, Spieß P, Hammann JM, Karaghiosoff K, Knochel P. Cobalt-Catalyzed Cross-Coupling of Functionalized Alkylzinc Reagents with (Hetero)Aryl Halides. Angewandte Chemie (International Ed. in English). PMID 31909546 DOI: 10.1002/anie.201914490  0.6
2019 Li J, Ren Q, Cheng X, Karaghiosoff K, Knochel P. Chromium(II)-Catalyzed Diastereoselective and Chemoselective Csp2‒Csp3 Cross-Couplings Using Organomagnesium Reagents. Journal of the American Chemical Society. PMID 31634428 DOI: 10.1021/jacs.9b08586  0.32
2019 Balkenhohl M, Jangra H, Lenz T, Ebeling M, Zipse H, Karaghiosoff K, Knochel P. Lewis Acid Directed Regioselective Metalations of Pyridazine. Angewandte Chemie (International Ed. in English). PMID 31034125 DOI: 10.1002/anie.201903839  0.36
2019 Leroux M, Vorherr T, Lewis I, Schaefer M, Koch G, Karaghiosoff K, Knochel P. Late-stage Functionalization of Peptides and Cyclopeptides using Organozinc reagents. Angewandte Chemie (International Ed. in English). PMID 30946517 DOI: 10.1002/anie.201902454  0.32
2019 Lemaire S, Diène C, Gavryushin A, Du Jourdin XM, Paolini L, Jusseau X, Knochel P, Farina V. Preparation of 2'-Deoxy-2'-spirocyclopropylcytidine via an Alternative Cyclopropanation Reaction. The Journal of Organic Chemistry. PMID 30721067 DOI: 10.1021/acs.joc.8b02784  0.52
2019 Anthore-Dalion L, Benischke AD, Wei B, Berionni G, Knochel P. The Halogen-Samarium Exchange Reaction. Synthetic Applications and Kinetics. Angewandte Chemie (International Ed. in English). PMID 30664831 DOI: 10.1002/anie.201814373  0.72
2018 Hofmayer MS, Lutter FH, Grokenberger L, Hammann JM, Knochel P. Practical Ni-Catalyzed Cross-Coupling of Unsaturated Zinc Pivalates with Unsaturated Nonaflates and Triflates. Organic Letters. PMID 30561216 DOI: 10.1021/acs.orglett.8b03417  0.6
2018 Simon M, Karaghiosoff K, Knochel P. Diastereoselective Intramolecular Carbolithiations of Stereodefined Secondary Alkyllithiums Bearing a Remote Alkynylsilane. Organic Letters. PMID 29874088 DOI: 10.1021/acs.orglett.8b01290  0.36
2018 Balkenhohl M, Salgues B, Hirai T, Karaghiosoff K, Knochel P. Regioselective Metalation and Functionalization of the Pyrazolo[1,5- a]pyridine Scaffold Using Mg- and Zn-TMP Bases. Organic Letters. 20: 3114-3118. PMID 29738248 DOI: 10.1021/acs.orglett.8b01204  0.32
2018 Benischke AD, Anthore-Dalion L, Kohl F, Knochel P. Synthesis of Polyfunctionalized Triaryllanthanum Reagents Using Ph3La and Related Species as Exchange Reagents. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29733471 DOI: 10.1002/chem.201801527  0.72
2018 Ziegler DS, Karaghiosoff K, Knochel P. Aryl and Heteroaryl Magnesium Reagents in Toluene via a Br/Mg- or a Cl/Mg-Exchange. Angewandte Chemie (International Ed. in English). PMID 29656503 DOI: 10.1002/anie.201802123  0.32
2018 Thomas L, Lutter FH, Hofmayer MS, Karaghiosoff K, Knochel P. Cobalt-Catalyzed Diastereoselective Cross-Couplings between Alkynylzinc Pivalates and Functionalized Cyclic Iodides or Bromides. Organic Letters. PMID 29624060 DOI: 10.1021/acs.orglett.8b00784  0.32
2018 Morozova V, Skotnitzki J, Moriya K, Karaghiosoff K, Knochel P. Preparation of Optically Enriched Secondary Alkyllithium and Alkylcopper Reagents. Synthesis of (-)-Lardolure and Siphonarienal. Angewandte Chemie (International Ed. in English). PMID 29512307 DOI: 10.1002/anie.201800792  0.36
2017 Benischke AD, Anthore-Dalion L, Berionni G, Knochel P. Preparation of Functionalized Diaryl- and Diheteroaryl- Lanthanum Reagents via a Fast Halogen-Lanthanum Exchange. Angewandte Chemie (International Ed. in English). PMID 29052932 DOI: 10.1002/anie.201709553  0.72
2017 Ziegler DS, Greiner R, Lumpe H, Kqiku L, Karaghiosoff K, Knochel P. Directed Zincation or Magnesiation of the 2-Pyridone and 2,7-Naphthyridone Scaffold Using TMP Bases. Organic Letters. PMID 29039957 DOI: 10.1021/acs.orglett.7b02690  0.32
2017 Makarov IS, Brocklehurst CE, Karaghiosoff K, Koch G, Knochel P. Convenient Preparation of Bicyclo[1.1.1]pentane Bioisosteres of Internal Alkynes and para-Disubstituted Benzenes using [1.1.1]Propellane. Angewandte Chemie (International Ed. in English). PMID 28786520 DOI: 10.1002/anie.201706799  0.32
2017 Balkenhohl M, Greiner R, Makarov IS, Heinz B, Karaghiosoff K, Zipse H, Knochel P. Zn-, Mg-, and Li-TMP Bases for the Successive Regioselective Metalations of the 1,5-Naphthyridine Scaffold. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28777497 DOI: 10.1002/chem.201703638  0.36
2017 Hammann JM, Thomas L, Chen YH, Haas D, Knochel P. Cobalt-Catalyzed Cross-Couplings of Bench-Stable Alkynylzinc Pivalates with (Hetero)Aryl and Alkenyl Halides. Organic Letters. PMID 28696711 DOI: 10.1021/acs.orglett.7b01722  0.6
2017 Ganiek MA, Becker MR, Berionni G, Zipse H, Knochel P. Barbier Continuous Flow Preparation and Reactions of Carbamoyllithiums for Nucleophilic Amidation. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28590518 DOI: 10.1002/chem.201702593  0.36
2017 Ketels M, Konrad DB, Karaghiosoff K, Trauner D, Knochel P. Selective Lithiation, Magnesiation, and Zincation of Unsymmetrical Azobenzenes Using Continuous Flow. Organic Letters. PMID 28296419 DOI: 10.1021/acs.orglett.7b00460  0.32
2017 Balkenhohl M, François C, Sustac Roman D, Quinio P, Knochel P. Transition-Metal-Free Amination of Pyridine-2-sulfonyl Chloride and Related N-Heterocycles Using Magnesium Amides. Organic Letters. PMID 28093909 DOI: 10.1021/acs.orglett.6b03703  0.72
2016 Castelló-Micó A, Nafe J, Higashida K, Karaghiosoff K, Gingras M, Knochel P. Selective Metalations of 1,4-Dithiins and Condensed Analogues Using TMP-Magnesium and -Zinc Bases. Organic Letters. PMID 28035825 DOI: 10.1021/acs.orglett.6b03539  0.32
2016 Auras F, Ascherl L, Hakimioun AH, Margraf JT, Hanusch FC, Reuter S, Bessinger D, Döblinger M, Hettstedt C, Karaghiosoff K, Herbert S, Knochel P, Clark T, Bein T. Synchronized Offset Stacking: A Concept for Growing Large-Domain and Highly Crystalline 2D Covalent Organic Frameworks. Journal of the American Chemical Society. PMID 27992179 DOI: 10.1021/jacs.6b09787  0.32
2016 Hammann JM, Lutter FH, Haas D, Knochel P. A Robust and Broadly Applicable Cobalt-Catalyzed Cross-Coupling of Functionalized Bench-Stable Organozinc Pivalates with Unsaturated Halides. Angewandte Chemie (International Ed. in English). PMID 27981715 DOI: 10.1002/anie.201610324  0.6
2016 Hofmayer MS, Hammann JM, Haas D, Knochel P. Cobalt-Catalyzed C(sp(2))-C(sp(3)) Cross-Coupling Reactions of Diarylmanganese Reagents with Secondary Alkyl Iodides. Organic Letters. 18: 6456-6459. PMID 27978689 DOI: 10.1021/acs.orglett.6b03349  0.6
2016 Haas D, Sustac-Roman D, Schwarz S, Knochel P. Directed Zincation with TMPZnCl·LiCl and Further Functionalization of the Tropolone Scaffold. Organic Letters. 18: 6380-6383. PMID 27978661 DOI: 10.1021/acs.orglett.6b03270  0.44
2016 Benischke AD, Le Corre G, Knochel P. Preparation of Polyfunctional Organozinc Halides by an InX₃- and LiCl-Catalyzed Zinc Insertion to Aryl and Heteroaryl Iodides and Bromides. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27862462 DOI: 10.1002/chem.201605139  0.72
2016 Cai Y, Benischke A, Knochel P, Gosmini C. Cobalt-Catalyzed Reductive Cross-Coupling Between Styryl and Benzyl Halides. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27762460 DOI: 10.1002/chem.201603832  0.44
2016 Greshock TJ, Moore KP, McClain RT, Bellomo A, Chung CK, Dreher SD, Kutchukian PS, Peng Z, Davies IW, Vachal P, Ellwart M, Manolikakes SM, Knochel P, Nantermet PG. Synthesis of Complex Druglike Molecules by the Use of Highly Functionalized Bench-Stable Organozinc Reagents. Angewandte Chemie (International Ed. in English). PMID 27690172 DOI: 10.1002/anie.201604652  0.56
2016 Hammann JM, Haas D, Tüllmann CP, Karaghiosoff K, Knochel P. Diastereoselective Cobalt-Mediated Cross-Couplings of Cycloalkyl Iodides with Alkynyl or (Hetero)Aryl Grignard Reagents. Organic Letters. PMID 27649388 DOI: 10.1021/acs.orglett.6b02119  0.6
2016 Nickel J, Fernández M, Klier L, Knochel P. Synthesis of Pyrrolo[2,3-d]pyrimidines by Copper-Mediated Carbomagnesiations of N-Sulfonyl Ynamides and Application to the Preparation of Rigidin A and a 7-Azaserotonin Derivative. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27529336 DOI: 10.1002/chem.201602519  0.32
2016 Benischke AD, Leroux M, Knoll I, Knochel P. Iron-Catalyzed Acylation of Polyfunctionalized Aryl- and Benzylzinc Halides with Acid Chlorides. Organic Letters. PMID 27457108 DOI: 10.1021/acs.orglett.6b01677  0.72
2016 Fernandez S, Ganiek MA, Karpacheva M, Hanusch FC, Reuter S, Bein T, Auras F, Knochel P. Synthesis and Reactivity of Triazaphenanthrenes. Organic Letters. PMID 27321707 DOI: 10.1021/acs.orglett.6b01373  1
2016 Morozova V, Moriya K, Mayer P, Knochel P. Stereoselective Synthesis and Retentive Trapping of α-Chiral Secondary Alkyllithiums Leading to Stereodefined α,β-Dimethyl Carboxylic Esters. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27140953 DOI: 10.1002/chem.201601911  0.4
2016 Shen ZL, Dhayalan V, Benischke AD, Greiner R, Karaghiosoff K, Mayer P, Knochel P. Polyfunctional Lithium, Magnesium, and Zinc Alkenyl Reagents as Building Blocks for the Synthesis of Complex Heterocycles. Angewandte Chemie (International Ed. in English). PMID 26991941 DOI: 10.1002/anie.201600961  1
2016 Barroso S, Lemaire S, Farina V, Steib AK, Blanc R, Knochel P. Cine Substitution with Arylzinc Reagents: Scope and Mechanistic Studies. The Journal of Organic Chemistry. PMID 26914598 DOI: 10.1021/acs.joc.6b00074  1
2016 Klier L, Aranzamendi E, Ziegler D, Nickel J, Karaghiosoff K, Carell T, Knochel P. Lewis Acid Triggered Regioselective Magnesiation and Zincation of Uracils, Uridines, and Cytidines. Organic Letters. PMID 26883782 DOI: 10.1021/acs.orglett.6b00190  1
2016 Haas D, Hammann JM, Lutter FH, Knochel P. Mild Cobalt-Catalyzed Negishi Cross-Couplings of (Hetero)arylzinc Reagents with (Hetero)aryl Halides. Angewandte Chemie (International Ed. in English). PMID 26879151 DOI: 10.1002/anie.201510665  1
2016 Ganiek MA, Becker MR, Ketels M, Knochel P. Continuous Flow Magnesiation or Zincation of Acrylonitriles, Acrylates, and Nitroolefins. Application to the Synthesis of Butenolides. Organic Letters. PMID 26863289 DOI: 10.1021/acs.orglett.6b00086  1
2016 Benischke AD, Knoll I, Rérat A, Gosmini C, Knochel P. A practical cobalt-catalyzed cross-coupling of benzylic zinc reagents with aryl and heteroaryl bromides or chlorides. Chemical Communications (Cambridge, England). PMID 26806016 DOI: 10.1039/c5cc10272c  1
2016 Benischke AD, Breuillac AJA, Moyeux A, Cahiez G, Knochel P. Iron-Catalyzed Cross-Coupling of Benzylic Manganese Chlorides with Aryl and Heteroaryl Halides Synlett. 27: 471-476. DOI: 10.1055/s-0035-1560812  1
2016 Nafe J, Knochel P. Selective Metalation of 1,3-Dithiole-2-thiones: An Effective Preparation of New Symmetrically and Nonsymmetrically Tetraarylated Tetrathiafulvalenes Synthesis (Germany). 48: 103-114. DOI: 10.1055/s-0035-1560728  1
2016 Greiner R, Blanc R, Petermayer C, Karaghiosoff K, Knochel P. Preparation of functionalized 2,7-naphthyridines by directed lithiation with (2,2,6,6-tetramethylpiperidyl)lithium and their regioselective iron-catalyzed cross couplings Synlett. 27: 231-236. DOI: 10.1055/s-0035-1560703  1
2016 Haas D, Hammann JM, Greiner R, Knochel P. Recent Developments in Negishi Cross-Coupling Reactions Acs Catalysis. 6: 1540-1552. DOI: 10.1021/acscatal.5b02718  1
2015 Castelló-Micó A, Herbert SA, León T, Bein T, Knochel P. Functionalizations of Mixtures of Regioisomeric Aryllithium Compounds by Selective Trapping with Dichlorozirconocene. Angewandte Chemie (International Ed. in English). PMID 26586204 DOI: 10.1002/anie.201508719  1
2015 Druzhinin SI, Galievsky VA, Demeter A, Kovalenko SA, Senyushkina TA, Dubbaka SR, Knochel P, Mayer P, Grosse C, Stalke D, Zachariasse KA. Two-State Intramolecular Charge Transfer (ICT) with 3,5-Dimethyl-4-(Dimethylamino)benzonitrile (MMD) and Its Meta-Isomer mMMD. Ground State Amino Twist Not Essential for ICT. The Journal of Physical Chemistry. A. PMID 26559045 DOI: 10.1021/acs.jpca.5b09368  1
2015 Nafe J, Auras F, Karaghiosoff K, Bein T, Knochel P. Selective Functionalization of Tetrathiafulvalene Using Mg- and Zn-TMP-Bases: Preparation of Mono-, Di-, Tri-, and Tetrasubstituted Derivatives. Organic Letters. 17: 5356-9. PMID 26469280 DOI: 10.1021/acs.orglett.5b02715  1
2015 Moriya K, Simon M, Mose R, Karaghiosoff K, Knochel P. Corrigendum: Stereoselective Retentive Domino Transmetalations of Secondary Alkyllithium Compounds to Functionalized Secondary Alkylcopper Reagents. Angewandte Chemie (International Ed. in English). 54: 12537. PMID 26465646 DOI: 10.1002/anie.201508286  0.36
2015 Quinio P, Roman DS, León T, William S, Karaghiosoff K, Knochel P. Transition-Metal-Free Cross-Coupling of Aryl and N-Heteroaryl Cyanides with Benzylic Zinc Reagents. Organic Letters. 17: 4396-9. PMID 26313453 DOI: 10.1021/acs.orglett.5b02380  1
2015 Moriya K, Simon M, Mose R, Karaghiosoff K, Knochel P. Stereoselective Retentive Domino Transmetalations of Secondary Alkyllithium Compounds to Functionalized Secondary Alkylcopper Reagents. Angewandte Chemie (International Ed. in English). 54: 10963-7. PMID 26277584 DOI: 10.1002/anie.201505740  1
2015 Ellwart M, Knochel P. Preparation of Solid, Substituted Allylic Zinc Reagents and Their Reactions with Electrophiles. Angewandte Chemie (International Ed. in English). PMID 26189654 DOI: 10.1002/anie.201504354  1
2015 Becker MR, Knochel P. Practical Continuous-Flow Trapping Metalations of Functionalized Arenes and Heteroarenes Using TMPLi in the Presence of Mg, Zn, Cu, or La Halides. Angewandte Chemie (International Ed. in English). PMID 25973885 DOI: 10.1002/anie.201502393  1
2015 Corral-Bautista F, Klier L, Knochel P, Mayr H. From Carbanions to Organometallic Compounds: Quantification of Metal Ion Effects on Nucleophilic Reactivities. Angewandte Chemie (International Ed. in English). PMID 25951612 DOI: 10.1002/anie.201501385  1
2015 Kuzmina OM, Steib AK, Fernandez S, Boudot W, Markiewicz JT, Knochel P. Practical Iron- and Cobalt-Catalyzed Cross-Coupling Reactions between N-Heterocyclic Halides and Aryl or Heteroaryl Magnesium Reagents. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 8242-9. PMID 25899175 DOI: 10.1002/chem.201500747  1
2015 Klatt T, Werner V, Maximova MG, Didier D, Apeloig Y, Knochel P. Preparation and Regioselective Magnesiation or Lithiation of Bis(trimethylsilyl)methyl-Substituted Heteroaryls for the Generation of Highly Functionalized Heterocycles. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 7830-4. PMID 25864885 DOI: 10.1002/chem.201500627  1
2015 Werner V, Ellwart M, Wagner AJ, Knochel P. Preparation of tertiary amines by the reaction of iminium ions derived from unsymmetrical aminals with zinc and magnesium organometallics. Organic Letters. 17: 2026-9. PMID 25849577 DOI: 10.1021/acs.orglett.5b00801  1
2015 Shen ZL, Knochel P. Stereoselective Preparation of Polyfunctional Alkenylindium(III) Halides and Their Cross-Coupling with Unsaturated Halides. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 7061-5. PMID 25820234 DOI: 10.1002/chem.201500943  1
2015 Haas D, Hofmayer MS, Bresser T, Knochel P. Zincation of 4,4-dimethyloxazoline using TMPZnCl·LiCl. A new preparation of 2-aryloxazolines. Chemical Communications (Cambridge, England). 51: 6415-7. PMID 25766645 DOI: 10.1039/c5cc01144b  1
2015 Hammann JM, Haas D, Knochel P. Cobalt-catalyzed negishi cross-coupling reactions of (hetero)arylzinc reagents with primary and secondary alkyl bromides and iodides. Angewandte Chemie (International Ed. in English). 54: 4478-81. PMID 25694155 DOI: 10.1002/anie.201411960  1
2015 Quinio P, François C, Escribano Cuesta A, Steib AK, Achrainer F, Zipse H, Karaghiosoff K, Knochel P. Preparation of tri- and tetrasubstituted allenes via regioselective lateral metalation of benzylic (trimethylsilyl)alkynes using TMPZnCl·LiCl. Organic Letters. 17: 1010-3. PMID 25662448 DOI: 10.1021/acs.orglett.5b00114  1
2015 Moriya K, Didier D, Simon M, Hammann JM, Berionni G, Karaghiosoff K, Zipse H, Mayr H, Knochel P. Stereoselective synthesis and reactions of secondary alkyllithium reagents functionalized at the 3-position. Angewandte Chemie (International Ed. in English). 54: 2754-7. PMID 25640227 DOI: 10.1002/anie.201409165  0.36
2015 Dhayalan V, Sämann C, Knochel P. Synthesis of polyfunctional secondary amines by the addition of functionalized zinc reagents to nitrosoarenes. Chemical Communications (Cambridge, England). 51: 3239-42. PMID 25610922 DOI: 10.1039/c4cc08846h  1
2015 Medina DD, Rotter JM, Hu Y, Dogru M, Werner V, Auras F, Markiewicz JT, Knochel P, Bein T. Room temperature synthesis of covalent-organic framework films through vapor-assisted conversion. Journal of the American Chemical Society. 137: 1016-9. PMID 25539131 DOI: 10.1021/ja510895m  1
2015 Steib AK, Kuzmina OM, Fernandez S, Malhotra S, Knochel P. Chemoselective chromium(II)-catalyzed cross-coupling reactions of dichlorinated heteroaromatics with functionalized aryl grignard reagents. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 1961-5. PMID 25470669 DOI: 10.1002/chem.201405275  1
2015 Nafe J, Herbert S, Auras F, Karaghiosoff K, Bein T, Knochel P. Functionalization of quinoxalines by using TMP bases: preparation of tetracyclic heterocycles with high photoluminescene quantum yields. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 1102-7. PMID 25404387 DOI: 10.1002/chem.201405240  1
2015 Benischke AD, Ellwart M, Becker MR, Knochel P. Polyfunctional Zinc and Magnesium Organometallics for Organic Synthesis: Some Perspectives Synthesis (Germany). DOI: 10.1055/s-0035-1561198  1
2015 Snieckus V, Knochel P. Cluster Preface: Resurgence of Synthetic Aromatic Chemistry Synlett. 26: 2782-2783. DOI: 10.1055/s-0035-1560959  1
2015 Dhayalan V, Alcañiz FR, Werner V, Karaghiosoff K, Knochel P. Preparation of a New Spirobi[thieno[2,3- c ]pyran] and Its Selective Mono- and Dimetalation: Application for the Preparation of Soluble Conjugated Oligothiophenes and Pyrene Derivatives Synthesis (Germany). 47: 3972-3982. DOI: 10.1055/s-0035-1560187  1
2015 Shen ZL, Sommer K, Knochel P. Expedient Preparation of Aryllithium and Arylzinc Reagents from Aryl Chlorides Using Lithium 4,4′-Di-tert-Butylbiphenylide and Zinc(II) Chloride Synthesis (Germany). DOI: 10.1055/s-0034-1380697  1
2015 Haas D, Hammann JM, Moyeux A, Cahiez G, Knochel P. Oxidative Homocoupling of Diheteroaryl- or Diarylmanganese Reagents Generated via Directed Manganation Using TMP2Mn Synlett. 26: 1515-1519. DOI: 10.1055/s-0034-1380424  1
2015 Hammann JM, Haas D, Steib AK, Knochel P. Highly Diastereoselective Cobalt-Mediated C(sp3)–C(sp2) Cross-Coupling Reactions of Cyclic Halohydrins with (Hetero)Aryl Grignard Reagents Synthesis (Germany). DOI: 10.1055/s-0034-1380407  1
2015 Kuzmina OM, Steib AK, Moyeux A, Cahiez G, Knochel P. Recent advances in iron-catalyzed Csp2-Csp2 cross-couplings Synthesis (Germany). 47: 1696-1705. DOI: 10.1055/s-0034-1380195  1
2015 Steib AK, Fernandez S, Kuzmina OM, Corpet M, Gosmini C, Knochel P. Chromium(II)-Catalyzed Amination of N-Heterocyclic Chlorides with Magnesium Amides Synlett. DOI: 10.1055/s-0034-1380178  1
2015 Quinio P, Benischke AD, Moyeux A, Cahiez G, Knochel P. New preparation of benzylic manganese chlorides by the direct insertion of magnesium into benzylic chlorides in the presence of MnCl2·2LiCl Synlett. 26. DOI: 10.1055/s-0034-1379944  1
2015 Barl NM, Malakhov V, Mathes C, Lustenberger P, Knochel P. Palladium-catalyzed cross-coupling between 7-azaindoles and reformatsky reagents Synthesis (Germany). 47: 692-700. DOI: 10.1055/s-0034-1379459  1
2015 Dhayalan V, Knochel P. Synthesis of Polyfunctional Secondary Amines by the Reaction of Functionalized Organomagnesium Reagents with Tertiary Nitroalkanes Synthesis (Germany). 47: 3246-3256. DOI: 10.1055/s-0034-1378871  1
2015 Becker MR, Ganiek MA, Knochel P. Practical and economic lithiations of functionalized arenes and heteroarenes using Cy2NLi in the presence of Mg, Zn or La halides in a continuous flow Chemical Science. 6: 6649-6653. DOI: 10.1039/c5sc02558c  1
2015 Shen ZL, Knochel P. C60-catalyzed preparation of aryl and heteroaryl magnesium and zinc reagents using Mg/LiCl Acs Catalysis. 5: 2324-2328. DOI: 10.1021/acscatal.5b00273  1
2015 Moegling J, Benischke AD, Hammann JM, Vepřek NA, Zoller F, Rendenbach B, Hoffmann A, Sievers H, Schuster M, Knochel P, Herres-Pawlis S. Bis(pyrazolyl)methane Copper Complexes as Robust and Efficient Catalysts for Sonogashira Couplings European Journal of Organic Chemistry. 2015: 7475-7483. DOI: 10.1002/ejoc.201501117  1
2015 Schlücker T, Dhayalan V, Langhals H, Sämann C, Knochel P. Soluble Adamantyl-Substituted Oligothiophenes with Short Fluorescence Decay: An Approach for Ultrafast Optical Signal Processing Asian Journal of Organic Chemistry. DOI: 10.1002/ajoc.201500150  1
2014 Hammann JM, Steib AK, Knochel P. Cobalt-mediated diastereoselective cross-coupling reactions between cyclic halohydrins and arylmagnesium reagents. Organic Letters. 16: 6500-3. PMID 25470419 DOI: 10.1021/ol503361m  1
2014 Kuzmina OM, Knochel P. Room-temperature chromium(II)-catalyzed direct arylation of pyridines, aryl oxazolines, and imines using arylmagnesium reagents. Organic Letters. 16: 5208-11. PMID 25230000 DOI: 10.1021/ol502623v  1
2014 Klier L, Diène CR, Schickinger M, Metzger A, Wagner AJ, Karaghiosoff K, Marek I, Knochel P. Isoxazole-embedded allylic zinc reagent for the diastereoselective preparation of highly functionalized aldol-type derivatives bearing a stereocontrolled quaternary center. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 14096-101. PMID 25204300 DOI: 10.1002/chem.201402733  1
2014 Manolikakes SM, Ellwart M, Stathakis CI, Knochel P. Air-stable solid aryl and heteroaryl organozinc pivalates: syntheses and applications in organic synthesis. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 12289-97. PMID 25116852 DOI: 10.1002/chem.201403015  1
2014 Petersen TP, Becker MR, Knochel P. Continuous flow magnesiation of functionalized heterocycles and acrylates with TMPMgCl⋅LiCl. Angewandte Chemie (International Ed. in English). 53: 7933-7. PMID 24962240 DOI: 10.1002/anie.201404221  1
2014 Frischmuth A, Fernández M, Barl NM, Achrainer F, Zipse H, Berionni G, Mayr H, Karaghiosoff K, Knochel P. New in situ trapping metalations of functionalized arenes and heteroarenes with TMPLi in the presence of ZnCl2 and other metal salts. Angewandte Chemie (International Ed. in English). 53: 7928-32. PMID 24923789 DOI: 10.1002/anie.201403688  1
2014 Werner V, Klatt T, Fujii M, Markiewicz J, Apeloig Y, Knochel P. Preparation and regioselective metalation of bis(trimethylsilyl)methyl-substituted aryl derivatives. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 8338-42. PMID 24890675 DOI: 10.1002/chem.201402531  1
2014 Chen Q, León T, Knochel P. Transition-metal-free BF₃-mediated oxidative and non-oxidative cross-coupling of pyridines. Angewandte Chemie (International Ed. in English). 53: 8746-50. PMID 24757070 DOI: 10.1002/anie.201400750  1
2014 Sämann C, Dhayalan V, Schreiner PR, Knochel P. Synthesis of substituted adamantylzinc reagents using a Mg-insertion in the presence of ZnCl₂ and further functionalizations. Organic Letters. 16: 2418-21. PMID 24735164 DOI: 10.1021/ol500781j  1
2014 Barl NM, Sansiaume-Dagousset E, Monzón G, Wagner AJ, Knochel P. Preparation and reactions of heteroarylmethylzinc reagents. Organic Letters. 16: 2422-5. PMID 24725243 DOI: 10.1021/ol500790p  1
2014 Klatt T, Markiewicz JT, Sämann C, Knochel P. Strategies to prepare and use functionalized organometallic reagents. The Journal of Organic Chemistry. 79: 4253-69. PMID 24697240 DOI: 10.1021/jo500297r  1
2014 Medina DD, Werner V, Auras F, Tautz R, Dogru M, Schuster J, Linke S, Döblinger M, Feldmann J, Knochel P, Bein T. Oriented thin films of a benzodithiophene covalent organic framework. Acs Nano. 8: 4042-52. PMID 24559375 DOI: 10.1021/nn5000223  1
2014 Klatt T, Roman DS, León T, Knochel P. TMP-magnesium and TMP-zinc bases for the regioselective metalation of the cinnoline scaffold. Organic Letters. 16: 1232-5. PMID 24512618 DOI: 10.1021/ol5001999  1
2014 Hernán-Gómez A, Herd E, Hevia E, Kennedy AR, Knochel P, Koszinowski K, Manolikakes SM, Mulvey RE, Schnegelsberg C. Organozinc pivalate reagents: segregation, solubility, stabilization, and structural insights. Angewandte Chemie (International Ed. in English). 53: 2706-10. PMID 24482294 DOI: 10.1002/anie.201309841  1
2014 Shen ZL, Peng Z, Yang CM, Helberg J, Mayer P, Marek I, Knochel P. Highly diastereoselective preparation of aldol products using new functionalized allylic aluminum reagents. Organic Letters. 16: 956-9. PMID 24479467 DOI: 10.1021/ol403692k  1
2014 Dagousset G, Moriya K, Mose R, Berionni G, Karaghiosoff K, Knochel P. Diastereoselective synthesis of open-chain secondary alkyllithium compounds and trapping reactions with electrophiles. Angewandte Chemie (International Ed. in English). 53: 1425-9. PMID 24459059 DOI: 10.1002/anie.201308679  1
2014 Moriya K, Knochel P. Diastereoconvergent Negishi cross-coupling using functionalized cyclohexylzinc reagents. Organic Letters. 16: 924-7. PMID 24428361 DOI: 10.1021/ol403673e  1
2014 Sämann C, Coya E, Knochel P. Full functionalization of the imidazole scaffold by selective metalation and sulfoxide/magnesium exchange. Angewandte Chemie (International Ed. in English). 53: 1430-4. PMID 24353035 DOI: 10.1002/anie.201309217  1
2014 Didier D, Delaye PO, Simaan M, Island B, Eppe G, Eijsberg H, Kleiner A, Knochel P, Marek I. Modulable and highly diastereoselective carbometalations of cyclopropenes. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 1038-48. PMID 24338953 DOI: 10.1002/chem.201303569  1
2014 Barl NM, Werner V, Sämann C, Knochel P. The halogen/magnesium-exchange using iPrMgCl•LiCl and related exchange reagents Heterocycles. 88: 827-844. DOI: 10.3987/REV-13-SR(S)4  1
2014 Dagousset G, François C, Len T, Blanc R, Sansiaume-Dagousset E, Knochel P. Preparation of functionalized lithium, magnesium, aluminum, zinc, manganese, and indium organometallics from functionalized organic halides Synthesis (Germany). 46: 3133-3171. DOI: 10.1055/s-0034-1378672  1
2014 León T, Quinio P, Chen Q, Knochel P. BF3-mediated oxidative cross-coupling of pyridines with alkynyllithium reagents and further reductive functionalizations of the pyridine scaffold Synthesis (Germany). 46: 1374-1379. DOI: 10.1055/s-0033-1341235  1
2014 Blanc R, Groll K, Bernhardt S, Stockmann PN, Knochel P. Efficient cross-coupling reactions of (pivaloyloxymethyl)zinc chloride Synthesis (Germany). 46: 1052-1058. DOI: 10.1055/s-0033-1340819  1
2014 Klatt T, Blümke TD, Ganiek MA, Knochel P. Synthesis of 1,2-dimetallic compounds via direct insertion of zinc powder in the presence of InCl3: Synthesis of ortho-bis-functionalized aromatics Synthesis (Germany). 46: 290-294. DOI: 10.1055/s-0033-1340106  1
2014 Enders D, Knochel P. Editorial Synthesis (Germany). 46: I-III. DOI: 10.1055/s-0033-1338582  1
2014 Knochel P. Introduction to Volume 7: Oxidation Comprehensive Organic Synthesis: Second Edition. 7: xiii-xiv. DOI: 10.1016/B978-0-08-097742-3.09037-6  1
2014 Knochel P, Molander GA. Preface Comprehensive Organic Synthesis: Second Edition. 1: xxiii. DOI: 10.1016/B978-0-08-097742-3.09005-4  1
2014 Knochel P, Molander GA. Comprehensive Organic Synthesis: Second Edition Comprehensive Organic Synthesis: Second Edition. 1: 1-9389.  1
2013 Haas D, Mosrin M, Knochel P. Regioselective functionalization of the oxazole scaffold using TMP-bases of Mg and Zn. Organic Letters. 15: 6162-5. PMID 24245558 DOI: 10.1021/ol403019c  1
2013 Colombe JR, Bernhardt S, Stathakis C, Buchwald SL, Knochel P. Synthesis of solid 2-pyridylzinc reagents and their application in Negishi reactions. Organic Letters. 15: 5754-7. PMID 24156393 DOI: 10.1021/ol402798z  0.64
2013 Steib AK, Kuzmina OM, Fernandez S, Flubacher D, Knochel P. Efficient chromium(II)-catalyzed cross-coupling reactions between Csp2 centers. Journal of the American Chemical Society. 135: 15346-9. PMID 24053764 DOI: 10.1021/ja409076z  1
2013 Unsinn A, Wunderlich SH, Jana A, Karaghiosoff K, Knochel P. A convenient alumination of functionalized aromatics by using the frustrated Lewis pair Et3 Al and TMPMgCl⋅LiCl. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 14687-96. PMID 24027191 DOI: 10.1002/chem.201301869  1
2013 Frischmuth A, Knochel P. Preparation of functionalized indoles and azaindoles by the intramolecular copper-mediated carbomagnesiation of ynamides. Angewandte Chemie (International Ed. in English). 52: 10084-8. PMID 23934952 DOI: 10.1002/anie.201304380  1
2013 Barl NM, Sansiaume-Dagousset E, Karaghiosoff K, Knochel P. Full functionalization of the 7-azaindole scaffold by selective metalation and sulfoxide/magnesium exchange. Angewandte Chemie (International Ed. in English). 52: 10093-6. PMID 23897626 DOI: 10.1002/anie.201303490  1
2013 Klatt T, Groll K, Knochel P. Generation of functionalized aryl and heteroaryl aluminum reagents by halogen-lithium exchange. Chemical Communications (Cambridge, England). 49: 6953-5. PMID 23802222 DOI: 10.1039/c3cc43356k  1
2013 Groll K, Manolikakes SM, du Jourdin XM, Jaric M, Bredihhin A, Karaghiosoff K, Carell T, Knochel P. Regioselective metalations of pyrimidines and pyrazines by using frustrated Lewis pairs of BF3·OEt2 and hindered magnesium- and zinc-amide bases. Angewandte Chemie (International Ed. in English). 52: 6776-80. PMID 23703866 DOI: 10.1002/anie.201301694  1
2013 Sämann C, Schade MA, Yamada S, Knochel P. Functionalized alkenylzinc reagents bearing carbonyl groups: preparation by direct metal insertion and reaction with electrophiles. Angewandte Chemie (International Ed. in English). 52: 9495-9. PMID 23666638 DOI: 10.1002/anie.201302058  1
2013 Berionni G, Morozova V, Heininger M, Mayer P, Knochel P, Mayr H. Electrophilic aromatic substitutions of aryltrifluoroborates with retention of the BF3- group: quantification of the activating and directing effects of the trifluoroborate group. Journal of the American Chemical Society. 135: 6317-24. PMID 23534556 DOI: 10.1021/ja4017655  1
2013 Kuzmina OM, Steib AK, Markiewicz JT, Flubacher D, Knochel P. Ligand-accelerated iron- and cobalt-catalyzed cross-coupling reactions between N-heteroaryl halides and aryl magnesium reagents. Angewandte Chemie (International Ed. in English). 52: 4945-9. PMID 23526682 DOI: 10.1002/anie.201210235  1
2013 Chen Q, du Jourdin XM, Knochel P. Transition-metal-free BF3-mediated regioselective direct alkylation and arylation of functionalized pyridines using Grignard or organozinc reagents. Journal of the American Chemical Society. 135: 4958-61. PMID 23506449 DOI: 10.1021/ja401146v  1
2013 Stathakis CI, Manolikakes SM, Knochel P. TMPZnOPiv•LiCl: a new base for the preparation of air-stable solid zinc pivalates of sensitive aromatics and heteroaromatics. Organic Letters. 15: 1302-5. PMID 23461805 DOI: 10.1021/ol400242r  1
2013 Unsinn A, Ford MJ, Knochel P. New preparation of TMPZnCl·LiCl by Zn insertion into TMPCl. Application to the functionalization of dibromodiazines. Organic Letters. 15: 1128-31. PMID 23421375 DOI: 10.1021/ol400248e  1
2013 Seel S, Dagousset G, Thaler T, Frischmuth A, Karaghiosoff K, Zipse H, Knochel P. Preparation of stereodefined secondary alkyllithium compounds. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 4614-22. PMID 23401284 DOI: 10.1002/chem.201204076  1
2013 Manolikakes SM, Jaric M, Karaghiosoff K, Knochel P. Metalated N-heterocyclic reagents prepared by the frustrated Lewis pair TMPMgCl·BF3 and their addition to aromatic aldehydes and activated ketones. Chemical Communications (Cambridge, England). 49: 2124-6. PMID 23389398 DOI: 10.1039/c3cc39040c  1
2013 Dogru M, Handloser M, Auras F, Kunz T, Medina D, Hartschuh A, Knochel P, Bein T. A photoconductive thienothiophene-based covalent organic framework showing charge transfer towards included fullerene. Angewandte Chemie (International Ed. in English). 52: 2920-4. PMID 23382014 DOI: 10.1002/anie.201208514  1
2013 Knochel P, Karaghiosoff K, Manolikakes S. Selective C-H activations using frustrated Lewis pairs. Applications in organic synthesis. Topics in Current Chemistry. 334: 171-90. PMID 23306865 DOI: 10.1007/128_2012_394  1
2013 Bernhardt S, Shen ZL, Knochel P. Preparation of functionalized organoindium reagents by means of magnesium insertion into organic halides in the presence of InCl3 at room temperature. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 828-33. PMID 23255158 DOI: 10.1002/chem.201203795  1
2013 Manolikakes SM, Barl NM, Sämann C, Knochel P. Regioselective functionalization of pyridines using a directed metalation or a halogen/metal exchange Zeitschrift Fur Naturforschung - Section B Journal of Chemical Sciences. 68: 411-422. DOI: 10.5560/ZNB.2013-3061  1
2013 Benhaim C, Lemaire S, Gaekens T, Govaerts T, Houpis IN, Reniers P, Van Looy A, Vermeulen WAA, Bernhardt S, Diène C, Knochel P, Farina V. Synthesis of (4′ R)-Azido-(2′ R)-2′-Deoxy-2′- C -Methyluridine and Its Esters by Direct Iodide Displacement Synlett. 24: 1697-1701. DOI: 10.1055/s-0033-1339293  1
2013 Crestey F, Zimdars S, Knochel P. Regioselective functionalization of purine derivatives at positions 8 and 6 using hindered TMP-amide bases of Zn and Mg Synthesis (Germany). 45: 3029-3037. DOI: 10.1055/s-0033-1338524  1
2013 Ila H, Markiewicz JT, Malakhov V, Knochel P. Metalated indoles, indazoles, benzimidazoles, and azaindoles and their synthetic applications Synthesis (Germany). 45: 2343-2371. DOI: 10.1055/s-0033-1338501  1
2013 Sämann C, Knochel P. A convenient synthesis of α-substituted β,γ-unsaturated ketones and esters via the direct addition of substituted allylic zinc reagents prepared by direct insertion Synthesis (Germany). 45: 1870-1876. DOI: 10.1055/s-0033-1338415  1
2013 Dogru M, Sonnauer A, Zimdars S, Döblinger M, Knochel P, Bein T. Facile synthesis of a mesoporous benzothiadiazole-COF based on a transesterification process Crystengcomm. 15: 1500-1502. DOI: 10.1039/c2ce26343b  1
2013 Knochel P, Blümke T, Groll K, Chen YH. Preparation of organoalanes for organic synthesis Topics in Organometallic Chemistry. 41: 173-186. DOI: 10.1007/3418-2012-36  1
2013 Unsinn A, Rohbogner CJ, Knochel P. Directed magnesiation of polyhaloaromatics using the tetramethylpiperidylmagnesium reagents TMP2Mg×2 LiCl and TMPMgCl×LiCl Advanced Synthesis and Catalysis. 355: 1553-1560. DOI: 10.1002/adsc.201300185  1
2013 Unsinn A, Wunderlich SH, Knochel P. Accelerated zincations for an efficient and mild functionalization of aromatics and heterocycles Advanced Synthesis and Catalysis. 355: 989-995. DOI: 10.1002/adsc.201300049  1
2012 Unsinn A, Dunst C, Knochel P. Stereoselective synthesis of tetrasubstituted alkenes via a sequential carbocupration and a new sulfur-lithium exchange. Beilstein Journal of Organic Chemistry. 8: 2202-6. PMID 23365630 DOI: 10.3762/bjoc.8.248  1
2012 Sämann C, Haag B, Knochel P. Highly regioselective preparation of heteroaryl-magnesium reagents by using a Br/Mg exchange. Chemistry (Weinheim An Der Bergstrasse, Germany). 18: 16145-52. PMID 23070798 DOI: 10.1002/chem.201202230  1
2012 Groll K, Blümke TD, Unsinn A, Haas D, Knochel P. Direct Pd-catalyzed cross-coupling of functionalized organoaluminum reagents. Angewandte Chemie (International Ed. in English). 51: 11157-61. PMID 23037856 DOI: 10.1002/anie.201205987  1
2012 Monzón G, Tirotta I, Nishii Y, Knochel P. The ortho and meta magnesiation of functionalized anilines and amino-substituted pyridines and pyrazines at room temperature. Angewandte Chemie (International Ed. in English). 51: 10624-7. PMID 22997059 DOI: 10.1002/anie.201205465  1
2012 Kuzmina OM, Steib AK, Flubacher D, Knochel P. Iron-catalyzed cross-coupling of N-heterocyclic chlorides and bromides with arylmagnesium reagents. Organic Letters. 14: 4818-21. PMID 22966964 DOI: 10.1021/ol302136c  1
2012 Blümke TD, Klatt T, Koszinowski K, Knochel P. InCl3-catalyzed synthesis of 1,2-dimetallic compounds by direct insertion of aluminum or zinc powder. Angewandte Chemie (International Ed. in English). 51: 9926-30. PMID 22951987 DOI: 10.1002/anie.201205169  1
2012 Stathakis CI, Bernhardt S, Quint V, Knochel P. Improved air-stable solid aromatic and heterocyclic zinc reagents by highly selective metalations for Negishi cross-couplings. Angewandte Chemie (International Ed. in English). 51: 9428-32. PMID 22907878 DOI: 10.1002/anie.201204526  1
2012 Mycka RJ, Duez S, Bernhardt S, Heppekausen J, Knochel P, Fleming FF. Cyclohexylcarbonitriles: diastereoselective arylations with TMPZnCl·LiCl. The Journal of Organic Chemistry. 77: 7671-6. PMID 22897673 DOI: 10.1021/jo301127n  1
2012 Klier L, Bresser T, Nigst TA, Karaghiosoff K, Knochel P. Lewis acid-triggered selective zincation of chromones, quinolones, and thiochromones: application to the preparation of natural flavones and isoflavones. Journal of the American Chemical Society. 134: 13584-7. PMID 22860983 DOI: 10.1021/ja306178q  1
2012 Dienstmaier JF, Medina DD, Dogru M, Knochel P, Bein T, Heckl WM, Lackinger M. Isoreticular two-dimensional covalent organic frameworks synthesized by on-surface condensation of diboronic acids. Acs Nano. 6: 7234-42. PMID 22775491 DOI: 10.1021/nn302363d  1
2012 Malysheva YB, Combes S, Allegro D, Peyrot V, Knochel P, Gavryushin AE, Fedorov AY. Synthesis and biological evaluation of novel anticancer bivalent colchicine-tubulizine hybrids. Bioorganic & Medicinal Chemistry. 20: 4271-8. PMID 22739088 DOI: 10.1016/j.bmc.2012.05.072  1
2012 Frischmuth A, Unsinn A, Groll K, Stadtmüller H, Knochel P. Preparations and reactions of SF5-substituted aryl and heteroaryl derivatives via Mg and Zn organometallics. Chemistry (Weinheim An Der Bergstrasse, Germany). 18: 10234-8. PMID 22714685 DOI: 10.1002/chem.201201485  1
2012 Shi L, Chu Y, Knochel P, Mayr H. Leaving group dependence of the rates of halogen-magnesium exchange reactions. Organic Letters. 14: 2602-5. PMID 22571332 DOI: 10.1021/ol300906a  1
2012 Duez S, Steib AK, Knochel P. Benzylic arylation of 2-methyl-5-membered heterocycles using TMP-bases. Organic Letters. 14: 1951-3. PMID 22489961 DOI: 10.1021/ol300517q  1
2012 Lemaire S, Houpis IN, Xiao T, Li J, Digard E, Gozlan C, Liu R, Gavryushin A, Diène C, Wang Y, Farina V, Knochel P. Stereoselective C-glycosylation reactions with arylzinc reagents. Organic Letters. 14: 1480-3. PMID 22385274 DOI: 10.1021/ol300220p  1
2012 Unsinn A, Knochel P. Regioselective zincation of indazoles using TMP2Zn and Negishi cross-coupling with aryl and heteroaryl iodides. Chemical Communications (Cambridge, England). 48: 2680-2. PMID 22307020 DOI: 10.1039/c2cc17804d  1
2012 Kunz T, Knochel P. Synthesis of functionalized benzo[b]thiophenes by the intramolecular copper-catalyzed carbomagnesiation of alkynyl(aryl)thioethers. Angewandte Chemie (International Ed. in English). 51: 1958-61. PMID 22253072 DOI: 10.1002/anie.201106734  1
2012 Langhals H, Knochel P, Walter A, Zimdars S. Benzothiadiazoloperylenes and benzoxadiazoloperylenes: Amorphous functional materials Synthesis (Germany). 44: 3465-3477. DOI: 10.1055/s-0032-1316785  1
2012 Malysheva YB, Combes S, Fedorov AY, Knochel P, Gavryushin AE. New method of synthesis and biological evaluation of some combretastatin A-4 analogues Synlett. 23: 1205-1208. DOI: 10.1055/s-0031-1290899  1
2012 Berionni G, Maji B, Knochel P, Mayr H. Nucleophilicity parameters for designing transition metal-free C-C bond forming reactions of organoboron compounds Chemical Science. 3: 878-882. DOI: 10.1039/c2sc00883a  1
2012 Brodmann T, Koos P, Metzger A, Knochel P, Ley SV. Continuous preparation of arylmagnesium reagents in flow with inline IR monitoring Organic Process Research and Development. 16: 1102-1113. DOI: 10.1021/op200275d  1
2011 Blümke TD, Groll K, Karaghiosoff K, Knochel P. New preparation of benzylic aluminum and zinc organometallics by direct insertion of aluminum powder. Organic Letters. 13: 6440-3. PMID 22098566 DOI: 10.1021/ol202733v  1
2011 Dienstmaier JF, Gigler AM, Goetz AJ, Knochel P, Bein T, Lyapin A, Reichlmaier S, Heckl WM, Lackinger M. Synthesis of well-ordered COF monolayers: surface growth of nanocrystalline precursors versus direct on-surface polycondensation. Acs Nano. 5: 9737-45. PMID 22040355 DOI: 10.1021/nn2032616  1
2011 Knochel P, Schade MA, Bernhardt S, Manolikakes G, Metzger A, Piller FM, Rohbogner CJ, Mosrin M. Functionalization of heterocyclic compounds using polyfunctional magnesium and zinc reagents. Beilstein Journal of Organic Chemistry. 7: 1261-77. PMID 21977211 DOI: 10.3762/bjoc.7.147  1
2011 Haag B, Mosrin M, Ila H, Malakhov V, Knochel P. Regio- and chemoselective metalation of arenes and heteroarenes using hindered metal amide bases. Angewandte Chemie (International Ed. in English). 50: 9794-824. PMID 21953742 DOI: 10.1002/anie.201101960  1
2011 Melzig L, Dennenwaldt T, Gavryushin A, Knochel P. Direct aminoalkylation of arenes, heteroarenes, and alkenes via Ni-catalyzed Negishi cross-coupling reactions. The Journal of Organic Chemistry. 76: 8891-906. PMID 21923124 DOI: 10.1021/jo201630e  1
2011 Bernhardt S, Manolikakes G, Kunz T, Knochel P. Preparation of solid salt-stabilized functionalized organozinc compounds and their application to cross-coupling and carbonyl addition reactions. Angewandte Chemie (International Ed. in English). 50: 9205-9. PMID 21919158 DOI: 10.1002/anie.201104291  1
2011 Dunst C, Knochel P. Regioselective functionalization of the thiazole scaffold using TMPMgCl·LiCl and TMP2Zn·2MgCl2·2LiCl. The Journal of Organic Chemistry. 76: 6972-8. PMID 21736384 DOI: 10.1021/jo201250n  1
2011 Duez S, Steib AK, Manolikakes SM, Knochel P. Lewis acid promoted benzylic cross-couplings of pyridines with aryl bromides. Angewandte Chemie (International Ed. in English). 50: 7686-90. PMID 21721092 DOI: 10.1002/anie.201103074  1
2011 Haag BA, Sämann C, Jana A, Knochel P. Practical one-pot preparation of magnesium di(hetero)aryl- and magnesium dialkenylboronates for Suzuki-Miyaura cross-coupling reactions. Angewandte Chemie (International Ed. in English). 50: 7290-4. PMID 21710516 DOI: 10.1002/anie.201103022  1
2011 Melzig L, Diène CR, Rohbogner CJ, Knochel P. Preparation of polyfunctional zinc organometallics using an Fe- or Co-catalyzed Cl/Zn-exchange. Organic Letters. 13: 3174-7. PMID 21595435 DOI: 10.1021/ol201100p  1
2011 Thaler T, Guo LN, Steib AK, Raducan M, Karaghiosoff K, Mayer P, Knochel P. Sulfoxide-alkene hybrids: a new class of chiral ligands for the Hayashi-Miyaura reaction. Organic Letters. 13: 3182-5. PMID 21591613 DOI: 10.1021/ol200841x  1
2011 Peng Z, Knochel P. Preparation of functionalized organomanganese(II) reagents by direct insertion of manganese to aromatic and benzylic halides. Organic Letters. 13: 3198-201. PMID 21574615 DOI: 10.1021/ol201109g  1
2011 Jaric M, Haag BA, Manolikakes SM, Knochel P. Selective and multiple functionalization of pyridines and alkaloids via Mg- and Zn-organometallic intermediates. Organic Letters. 13: 2306-9. PMID 21462960 DOI: 10.1021/ol200563j  1
2011 Melzig L, Rauhut CB, Naredi-Rainer N, Knochel P. Difunctionalisation of arenes and heteroarenes by directed metallation and sulfoxide-magnesium exchange. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 5362-72. PMID 21462274 DOI: 10.1002/chem.201003657  1
2011 Steib AK, Thaler T, Komeyama K, Mayer P, Knochel P. Highly diastereoselective iron-mediated C(sp2)-C(sp3) cross-coupling reactions between aryl Grignard reagents and cyclic iodohydrine derivatives. Angewandte Chemie (International Ed. in English). 50: 3303-7. PMID 21432956 DOI: 10.1002/anie.201007187  1
2011 Seel S, Thaler T, Takatsu K, Zhang C, Zipse H, Straub BF, Mayer P, Knochel P. Highly diastereoselective arylations of substituted piperidines. Journal of the American Chemical Society. 133: 4774-7. PMID 21388211 DOI: 10.1021/ja201008e  1
2011 Schade MA, Yamada S, Knochel P. Synthesis of polyfunctional allenes by successive copper-mediated substitutions. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 4232-7. PMID 21384450 DOI: 10.1002/chem.201003273  1
2011 Duez S, Bernhardt S, Heppekausen J, Fleming FF, Knochel P. Pd-catalyzed α-arylation of nitriles and esters and γ-arylation of unsaturated nitriles with TMPZnCl·LiCl. Organic Letters. 13: 1690-3. PMID 21366325 DOI: 10.1021/ol200194y  1
2011 Thaler T, Guo LN, Mayer P, Knochel P. Highly diastereoselective C(sp3)-C(sp) cross-coupling reactions between 1,3- and 1,4-substituted cyclohexylzinc reagents and bromoalkynes through remote stereocontrol. Angewandte Chemie (International Ed. in English). 50: 2174-7. PMID 21344579 DOI: 10.1002/anie.201006879  1
2011 Bresser T, Knochel P. Selective magnesiation or zincation of highly functionalized alkenes and cycloalkenes using 2,2,6,6-tetramethylpiperidyl bases. Angewandte Chemie (International Ed. in English). 50: 1914-7. PMID 21328669 DOI: 10.1002/anie.201006641  1
2011 Melzig L, Metzger A, Knochel P. Pd- and Ni-catalyzed cross-coupling reactions of functionalized organozinc reagents with unsaturated thioethers. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 2948-56. PMID 21280109 DOI: 10.1002/chem.201002850  1
2011 Zimdars S, Mollat du Jourdin X, Crestey F, Carell T, Knochel P. Trifunctionalization of the purine scaffold using Mg and Zn organometallic intermediates. Organic Letters. 13: 792-5. PMID 21247193 DOI: 10.1021/ol103057k  1
2011 Kunz T, Knochel P. Selective multiple magnesiations of the thieno[3,2-b]thiophene scaffold. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 866-72. PMID 21226101 DOI: 10.1002/chem.201002506  1
2011 Dogru M, Sonnauer A, Gavryushin A, Knochel P, Bein T. A Covalent Organic Framework with 4 nm open pores. Chemical Communications (Cambridge, England). 47: 1707-9. PMID 21206941 DOI: 10.1039/c0cc03792c  1
2011 Kienle M, Wagner AJ, Dunst C, Knochel P. Preparation of heterocyclic amines by an oxidative amination of zinc organometallics mediated by Cu(I): a new oxidative cycloamination for the preparation of annulated indole derivatives. Chemistry, An Asian Journal. 6: 517-23. PMID 20677325 DOI: 10.1002/asia.201000367  1
2011 Dunst C, Knochel P. Selective Mg insertion into substituted mono- and dichloro arenes in the presence of LiCl: A new preparation of boscalid Synlett. 2064-2068. DOI: 10.1055/s-0030-1261168  1
2011 Dunst C, Metzger A, Zaburdaeva EA, Knochel P. Stereoselective synthesis of polyfunctional tetrasubstituted alkenyl sulfides via a carbocupration of alkynyl sulfides with aryl and benzylic diorganozincs Synthesis. 3453-3462. DOI: 10.1055/s-0030-1260210  1
2011 Piller FM, Knochel P. Regio- and chemoselective synthesis of fully substituted furans Synthesis. 1751-1758. DOI: 10.1055/s-0030-1260035  1
2011 Zimdars S, Langhals H, Knochel P. Functionalization of the benzo[c][1,2,5]thiadiazole scaffold via Mg-, Zn- and Mn-intermediates Synthesis. 1302-1308. DOI: 10.1055/s-0030-1259966  1
2011 Zhang ZG, Haag BA, Li JS, Knochel P. Efficient preparation of polyfunctional indoles via a zinc organometallic variation of the Fischer indole synthesis Synthesis. 23-29. DOI: 10.1055/s-0030-1258348  1
2011 Li Y, Keilbach A, Kienle M, Goto Y, Inagaki S, Knochel P, Bein T. Hierarchically structured biphenylene-bridged periodic mesoporous organosilica Journal of Materials Chemistry. 21: 17338-17344. DOI: 10.1039/c1jm12023a  1
2011 Knochel P, Diène C. Preparation of functionalized Zn and Mg-organometallics. Application to the performance of diastereoselective cross-couplings Comptes Rendus Chimie. 14: 842-850. DOI: 10.1016/j.crci.2011.07.002  1
2010 Blümke T, Chen YH, Peng Z, Knochel P. Preparation of functionalized organoaluminiums by direct insertion of aluminium to unsaturated halides. Nature Chemistry. 2: 313-8. PMID 21124514 DOI: 10.1038/nchem.590  1
2010 Thaler T, Haag B, Gavryushin A, Schober K, Hartmann E, Gschwind RM, Zipse H, Mayer P, Knochel P. Highly diastereoselective Csp₃-Csp₂ Negishi cross-coupling with 1,2-, 1,3- and 1,4-substituted cycloalkylzinc compounds. Nature Chemistry. 2: 125-30. PMID 21124403 DOI: 10.1038/nchem.505  1
2010 Peng Z, Haag BA, Knochel P. Preparation of 2-magnesiated 1,3,5-triazines via an iodine-magnesium exchange. Organic Letters. 12: 5398-401. PMID 21043499 DOI: 10.1021/ol102173z  1
2010 Haag BA, Zhang ZG, Li JS, Knochel P. Fischer indole synthesis with organozinc reagents. Angewandte Chemie (International Ed. in English). 49: 9513-6. PMID 20979062 DOI: 10.1002/anie.201005319  1
2010 Jeganmohan M, Knochel P. tmp(4)Zr: an atom-economical base for the metalation of functionalized arenes and heteroarenes. Angewandte Chemie (International Ed. in English). 49: 8520-4. PMID 20839204 DOI: 10.1002/anie.201003558  1
2010 Schade MA, Fleckenstein JE, Knochel P, Koszinowski K. Charged tags as probes for analyzing organometallic intermediates and monitoring cross-coupling reactions by electrospray-ionization mass spectrometry. The Journal of Organic Chemistry. 75: 6848-57. PMID 20836538 DOI: 10.1021/jo101337a  1
2010 Peng Z, Blümke TD, Mayer P, Knochel P. Diastereoselective synthesis of homoallylic alcohols with adjacent tertiary and quaternary centers by using functionalized allylic aluminum reagents. Angewandte Chemie (International Ed. in English). 49: 8516-9. PMID 20821786 DOI: 10.1002/anie.201003813  1
2010 Jaric M, Haag BA, Unsinn A, Karaghiosoff K, Knochel P. Highly selective metalations of pyridines and related heterocycles using new frustrated Lewis pairs or tmp-zinc and tmp-magnesium bases with BF3.OEt2. Angewandte Chemie (International Ed. in English). 49: 5451-5. PMID 20818766 DOI: 10.1002/anie.201002031  1
2010 Schade MA, Manolikakes G, Knochel P. Preparation of primary amides from functionalized organozinc halides. Organic Letters. 12: 3648-50. PMID 20704410 DOI: 10.1021/ol101469f  1
2010 Guo LN, Gao H, Mayer P, Knochel P. Preparation of organoaluminum reagents from propargylic bromides and aluminum activated by PbCl2 and their regio- and diastereoselective addition to carbonyl derivatives. Chemistry (Weinheim An Der Bergstrasse, Germany). 16: 9829-34. PMID 20572180 DOI: 10.1002/chem.201000523  1
2010 Bresser T, Mosrin M, Monzon G, Knochel P. Regio- and chemoselective zincation of sensitive and moderately activated aromatics and heteroaromatics using TMPZnCl.LiCl. The Journal of Organic Chemistry. 75: 4686-95. PMID 20553051 DOI: 10.1021/jo100884u  1
2010 Piller FM, Bresser T, Fischer MK, Knochel P. Preparation of functionalized cyclic enol phosphates by halogen-magnesium exchange and directed deprotonation reactions. The Journal of Organic Chemistry. 75: 4365-75. PMID 20527975 DOI: 10.1021/jo100763f  1
2010 Kienle M, Unsinn A, Knochel P. Synthesis of dibenzothiophenes and related classes of heterocycles by using functionalized dithiocarbamates. Angewandte Chemie (International Ed. in English). 49: 4751-4. PMID 20514654 DOI: 10.1002/anie.201001025  1
2010 Kienle M, Knochel P. i-PrI acceleration of Negishi cross-coupling reactions. Organic Letters. 12: 2702-5. PMID 20481437 DOI: 10.1021/ol1007026  1
2010 Metzger A, Bernhardt S, Manolikakes G, Knochel P. MgCl2-accelerated addition of functionalized organozinc reagents to aldehydes, ketones, and carbon dioxide. Angewandte Chemie (International Ed. in English). 49: 4665-8. PMID 20480475 DOI: 10.1002/anie.201000634  1
2010 Rohbogner CJ, Wirth S, Knochel P. Phosphorodiamidate-directed metalation of N-heterocycles using Mg- and Zn-TMP bases. Organic Letters. 12: 1984-7. PMID 20356104 DOI: 10.1021/ol100453x  1
2010 Melzig L, Metzger A, Knochel P. Room temperature cross-coupling of highly functionalized organozinc reagents with thiomethylated N-heterocycles by nickel catalysis. The Journal of Organic Chemistry. 75: 2131-3. PMID 20192173 DOI: 10.1021/jo1001615  1
2010 Yamada S, Gavryushin A, Knochel P. Convenient electrophilic fluorination of functionalized aryl and heteroaryl magnesium reagents Angewandte Chemie - International Edition. 49: 2215-2218. PMID 20162637 DOI: 10.1002/anie.200905052  1
2010 Rohbogner CJ, Diène CR, Korn TJ, Knochel P. A cobalt-catalyzed sulfonate/copper exchange for the preparation of highly functionalized electron-deficient aryl copper reagents. Angewandte Chemie (International Ed. in English). 49: 1874-7. PMID 20140923 DOI: 10.1002/anie.200905379  1
2010 Bernhardt S, Metzger A, Knochel P. Direct addition of functionalized organozinc reagents to carbon dioxide, ketones, and aldehydes in the presence of MgCl2 Synthesis. 3802-3810. DOI: 10.1055/s-0030-1258314  1
2010 Metzger A, Melzig L, Knochel P. Scaled-up transition-metal-catalyzed cross-coupling reactions of thioether-substituted N-heterocycles with organozinc reagents Synthesis. 2853-2858. DOI: 10.1055/s-0030-1258145  1
2010 Dunst C, Kienle M, Knochel P. Preparation of heterocyclic amines via a copper(i)-mediated oxidative cross-coupling of organozinc reagents with lithium amides Synthesis. 2313-2318. DOI: 10.1055/s-0029-1220008  1
2010 Crestey F, Knochel P. Regioselective Functionalization of Chlorophthalazine Derivatives Synthesis. 1097-1106. DOI: 10.1055/s-0029-1219231  1
2010 Monzon G, Knochel P. Directed ortho-and meta-magnesiation or zincation of polyfunctional aryl nonaflates Synlett. 304-308. DOI: 10.1055/s-0029-1219165  1
2010 Wunderlich SH, Bresser T, Dunst C, Monzon G, Knochel P. Efficient preparation of polyfunctional organometallics via directed ortho -metalation Synthesis. 2670-2678. DOI: 10.1055/s-0029-1218845  1
2010 Yamada S, Knochel P. Large-scale preparation of aromatic fluorides via electrophilic fluorination with functionalized aryl- or heteroarylmagnesium reagents Synthesis. 2490-2494. DOI: 10.1055/s-0029-1218816  1
2010 Melzig L, Stemper J, Knochel P. A novel palladium-catalyzed cross-coupling of thiomethylated alkynes with functionalized organozinc reagents Synthesis. 2085-2091. DOI: 10.1055/s-0029-1218734  1
2010 Metzger A, Argyo C, Knochel P. Large-scale preparation of polyfunctional benzylic zinc reagents by direct insertion of zinc dust into benzylic chlorides in the presence of lithium chloride Synthesis. 882-891. DOI: 10.1055/S-0029-1217134  1
2010 Blümke TD, Piller FM, Knochel P. Preparation of highly functionalized alkylzinc halides from alkyl bromides using Mg, ZnCl2 and LiCl Chemical Communications. 46: 4082-4084. DOI: 10.1039/c001845g  1
2010 Knochel P, Wunderlich SH, Rohbogner CJ, Unsinn A. Scaleable preparation of functionalized organometallics via directed ortho metalation using Mg- and Zn-amide bases Organic Process Research and Development. 14: 339-345. DOI: 10.1021/op9002888  1
2010 Bresser T, Monzon G, Mosrin M, Knochel P. Scaleable preparation of sensitive functionalized aromatics and heteroaromatics via directed metalation using tmpZnCl.LiCl Organic Process Research and Development. 14: 1299-1303. DOI: 10.1021/op1001935  1
2010 Lotz M, Schuecker R, Mereiter K, Knochel P. Synthesis of exclusively centrostereogenic 1,3-bidentate ferrocenyldiphosphane ligands and their use in enantioselective hydrogenations Organometallics. 29: 6503-6508. DOI: 10.1021/om100830m  1
2010 Knochel P, Thaler T, Diene C. Pd-, Ni-, Fe-, and co-catalyzed cross-couplings using functionalized Zn-, Mg-, Fe-, and in-organometallics Israel Journal of Chemistry. 50: 547-557. DOI: 10.1002/ijch.201000033  1
2010 Brückl T, Thoma I, Wagner AJ, Knochel P, Carell T. Efficient synthesis of deazaguanosine-derived tRNA nucleosides PreQ 0, PreQ1, and archaeosine using the Turbo-Grignard method European Journal of Organic Chemistry. 6517-6519. DOI: 10.1002/ejoc.201000987  1
2010 Wunderlich S, Knochel P. Atom-economical preparation of aryl- And heteroaryl-lanthanum reagents by directed ortho metalation by using tmp3[La] Chemistry - a European Journal. 16: 3304-3307. DOI: 10.1002/chem.200903157  1
2009 Metzger A, Melzig L, Despotopoulou C, Knochel P. Pd-catalyzed cross-coupling of functionalized organozinc reagents with thiomethyl-substituted heterocycles. Organic Letters. 11: 4228-31. PMID 19691353 DOI: 10.1021/ol9017003  0.32
2009 Piller FM, Metzger A, Schade MA, Haag BA, Gavryushin A, Knochel P. Preparation of polyfunctional arylmagnesium, arylzinc, and benzylic zinc reagents by using magnesium in the presence of LiCl. Chemistry (Weinheim An Der Bergstrasse, Germany). 15: 7192-202. PMID 19544505 DOI: 10.1002/chem.200900575  1
2009 Dong Z, Clososki GC, Wunderlich SH, Unsinn A, Li J, Knochel P. Direct zincation of functionalized aromatics and heterocycles by using a magnesium base in the presence of ZnCl2 Chemistry - a European Journal. 15: 457-468. PMID 19035380 DOI: 10.1002/chem.200801558  1
2009 Thaler T, Ren H, Gommermann N, Clososki GC, Rohbogner CJ, Wunderlich SH, Knochel P. New Catalytic Cu-, Pd- and Stoichiometric Mg-, Zn-Mediated Bond Activations Activating Unreactive Substrates: the Role of Secondary Interactions. 359-377. DOI: 10.1002/9783527625468.ch20  1
2008 Metzger A, Piller FM, Knochel P. Polyfunctional benzylic zinc chlorides by the direct insertion of magnesium into benzylic chlorides in the presence of LiCl and ZnCl2. Chemical Communications (Cambridge, England). 5824-6. PMID 19009094 DOI: 10.1039/b812396a  0.32
2008 Manolikakes G, Muñoz Hernandez C, Schade MA, Metzger A, Knochel P. Palladium- and nickel-catalyzed cross-couplings of unsaturated halides bearing relatively acidic protons with organozinc reagents. The Journal of Organic Chemistry. 73: 8422-36. PMID 18834176 DOI: 10.1021/jo8015852  1
2008 Sase S, Jaric M, Metzger A, Malakhov V, Knochel P. One-pot Negishi cross-coupling reactions of in situ generated zinc reagents with aryl chlorides, bromides, and triflates. The Journal of Organic Chemistry. 73: 7380-2. PMID 18693766 DOI: 10.1021/jo801063c  0.32
2008 Schade MA, Metzger A, Hug S, Knochel P. Nickel-catalyzed cross-coupling reactions of benzylic zinc reagents with aromatic bromides, chlorides and tosylates. Chemical Communications (Cambridge, England). 3046-8. PMID 18688343 DOI: 10.1039/b803072c  1
2008 Metzger A, Schade MA, Manolikakes G, Knochel P. A general preparation of polyfunctional benzylic zinc organometallic compounds. Chemistry, An Asian Journal. 3: 1678-91. PMID 18604829 DOI: 10.1002/asia.200800161  1
2008 Manolikakes G, Schade MA, Hernandez CM, Mayr H, Knochel P. Negishi cross-couplings of unsaturated halides bearing relatively acidic hydrogen atoms with organozinc reagents. Organic Letters. 10: 2765-8. PMID 18529011 DOI: 10.1021/ol8009013  1
2008 Metzger A, Schade MA, Knochel P. LiCl-mediated preparation of highly functionalized benzylic zinc chlorides. Organic Letters. 10: 1107-10. PMID 18288850 DOI: 10.1021/ol7030697  1
2008 Rauhut CB, Vu VA, Fleming FF, Knochel P. Preparation of functionalized alkylmagnesium derivatives using an I/Mg-exchange. Organic Letters. 10: 1187-9. PMID 18275211 DOI: 10.1021/ol8000987  1
2008 Despotopoulou C, Bauer RC, Krasovskiy A, Mayer P, Stryker JM, Knochel P. Selective mono- and 1,2-difunctionalisation of cyclopentene derivatives via Mg and Cu intermediates. Chemistry (Weinheim An Der Bergstrasse, Germany). 14: 2499-506. PMID 18232043 DOI: 10.1002/chem.200701431  1
2008 Dunet G, Mayer P, Knochel P. Highly diastereoselective addition of cinnamylzinc derivatives to alpha-chiral carbonyl compounds. Organic Letters. 10: 117-20. PMID 18067308 DOI: 10.1021/ol702607t  0.4
2007 Kolodney G, Sklute G, Perrone S, Knochel P, Marek I. Diastereodivergent synthesis of enantiomerically pure homoallylic amine derivatives containing quaternary carbon stereocenters. Angewandte Chemie (International Ed. in English). 46: 9291-4. PMID 17893895 DOI: 10.1002/anie.200702981  1
2007 Ren H, Dunet G, Mayer P, Knochel P. Highly diastereoselective synthesis of homoallylic alcohols bearing adjacent quaternary centers using substituted allylic zinc reagents. Journal of the American Chemical Society. 129: 5376-7. PMID 17408274 DOI: 10.1021/ja071380s  0.4
2006 Korn TJ, Schade MA, Wirth S, Knochel P. Cobalt(II)-catalyzed cross-coupling between polyfunctional arylcopper reagents and aryl fluorides or tosylates. Organic Letters. 8: 725-8. PMID 16468752 DOI: 10.1021/ol0529142  1
2006 Ila H, Baron O, Wagner AJ, Knochel P. Functionalized magnesium organometallics as versatile intermediates for the synthesis of polyfunctional heterocycles. Chemical Communications (Cambridge, England). 583-93. PMID 16446819 DOI: 10.1039/b510866g  1
2006 Ila H, Baron O, Wagner AJ, Knochel P. Preparation and reactions of heteroaryl organomagnesium compounds Chemistry Letters. 35: 2-7. DOI: 10.1246/cl.2006.2  1
2005 Kopp F, Sklute G, Polborn K, Marek I, Knochel P. Stereoselective functionalization of cyclopropane derivatives using bromine/magnesium and sulfoxide/magnesium exchange reactions. Organic Letters. 7: 3789-91. PMID 16092876 DOI: 10.1021/ol051452p  1
2005 Leuser H, Perrone S, Liron F, Kneisel FF, Knochel P. Highly enantioselective preparation of tertiary alcohols and amines by copper-mediated diastereoselective allylic S(N)2' substitutions. Angewandte Chemie (International Ed. in English). 44: 4627-31. PMID 16003795 DOI: 10.1002/anie.200500672  0.76
2005 Lin W, Sapountzis I, Knochel P. Preparation of functionalized aryl magnesium reagents by the addition of magnesium aryl thiolates and amides to arynes. Angewandte Chemie (International Ed. in English). 44: 4258-61. PMID 15940729 DOI: 10.1002/anie.200500443  0.68
2005 Sapountzis I, Lin W, Kofink CC, Despotopoulou C, Knochel P. Iron-catalyzed aryl-aryl cross-couplings with magnesium-derived copper reagents. Angewandte Chemie (International Ed. in English). 44: 1654-8. PMID 15625666 DOI: 10.1002/anie.200462013  0.68
2004 Sapountzis I, Lin W, Fischer M, Knochel P. Preparation of polyfunctional arynes via 2-magnesiated diaryl sulfonates. Angewandte Chemie (International Ed. in English). 43: 4364-6. PMID 15368394 DOI: 10.1002/anie.200460417  0.68
2004 Varela JA, Peña D, Goldfuss B, Denisenko D, Kulhanek J, Polborn K, Knochel P. Diastereoselective remote C-H activation by hydroboration. Chemistry (Weinheim An Der Bergstrasse, Germany). 10: 4252-64. PMID 15352108 DOI: 10.1002/chem.200400023  1
2004 Duplais C, Bures F, Sapountzis I, Korn TJ, Cahiez G, Knochel P. An efficient synthesis of diaryl ketones by iron-catalyzed arylation of aroyl cyanides. Angewandte Chemie (International Ed. in English). 43: 2968-70. PMID 15170318 DOI: 10.1002/anie.200453696  1
2004 Heller B, Sundermann B, Fischer C, You J, Chen W, Drexler H, Knochel P, Bonrath W, Gutnov A. Facile and Racemization-Free Conversion of Chiral Nitriles into Pyridine Derivatives. Cheminform. 35. DOI: 10.1002/chin.200414155  0.32
2003 Gommermann N, Koradin C, Polborn K, Knochel P. Enantioselective, copper(I)-catalyzed three-component reaction for the preparation of propargylamines. Angewandte Chemie (International Ed. in English). 42: 5763-6. PMID 14661218 DOI: 10.1002/anie.200352578  1
2003 Dohle W, Staubitz A, Knochel P. Mild synthesis of polyfunctional benzimidazoles and indoles by the reduction of functionalized nitroarenes with phenylmagnesium chloride. Chemistry (Weinheim An Der Bergstrasse, Germany). 9: 5323-31. PMID 14613142 DOI: 10.1002/chem.200305090  1
2003 Knochel P, Dohle W, Gommermann N, Kneisel FF, Kopp F, Korn T, Sapountzis I, Vu VA. Highly functionalized organomagnesium reagents prepared through halogen-metal exchange. Angewandte Chemie (International Ed. in English). 42: 4302-20. PMID 14502700 DOI: 10.1002/anie.200300579  1
2003 Koradin C, Gommermann N, Polborn K, Knochel P. Synthesis of enantiomerically enriched propargylamines by copper-catalyzed addition of alkynes to enamines. Chemistry (Weinheim An Der Bergstrasse, Germany). 9: 2797-2811. PMID 12866545 DOI: 10.1002/chem.200204691  1
2003 Hupe E, Calaza MI, Knochel P. Substrate-controlled highly diastereoselective synthesis of primary and secondary diorganozinc reagents by hydroboration/boron-zinc exchange sequence. Chemistry (Weinheim An Der Bergstrasse, Germany). 9: 2789-96. PMID 12866543 DOI: 10.1002/chem.200204662  1
2003 Harrington-Frost N, Leuser H, Calaza MI, Kneisel FF, Knochel P. Highly stereoselective anti SN2' substitutions of (Z)-allylic pentafluorobenzoates with polyfunctionalized zinc-copper reagents. Organic Letters. 5: 2111-4. PMID 12790541 DOI: 10.1021/ol034525i  1
2003 Yang X, Rotter T, Piazza C, Knochel P. Successive iodine-magnesium or -copper exchange reactions for the selective functionalization of polyhalogenated aromatics. Organic Letters. 5: 1229-31. PMID 12688726 DOI: 10.1021/ol0341492  0.96
2003 Calaza MI, Hupe E, Knochel P. Highly anti-selective SN2' substitutions of chiral cyclic 2-iodo-allylic alcohol derivatives with mixed zinc-copper reagents. Organic Letters. 5: 1059-61. PMID 12659573 DOI: 10.1021/ol0340742  1
2003 Varchi G, Kofink C, Lindsay DM, Ricci A, Knochel P. Direct preparation of polyfunctional amino-substituted arylmagnesium reagents via an iodine-magnesium exchange reaction. Chemical Communications (Cambridge, England). 396-7. PMID 12613630  1
2003 Kloetzing RJ, Lotz M, Knochel P. New P,N-ferrocenyl ligands for rhodium-catalyzed hydroboration and palladium-catalyzed allylic alkylation Tetrahedron Asymmetry. 14: 255-264. DOI: 10.1016/S0957-4166(02)00827-3  1
2003 Koradin C, Dohle W, Rodriguez AL, Schmid B, Knochel P. Synthesis of polyfunctional indoles and related heterocycles mediated by cesium and potassium bases Tetrahedron. 59: 1571-1587. DOI: 10.1016/S0040-4020(03)00073-5  1
2003 Hupe E, Calaza MI, Knochel P. Synthesis and reaction of secondary and primary diorganozinc reagents using a boron-zinc exchange reaction. A useful method for the stereo- and regioselective formation of new carbon-carbon bonds Journal of Organometallic Chemistry. 680: 136-142. DOI: 10.1016/S0022-328X(03)00237-7  1
2003 Hupe E, Denisenko D, Knochel P. Stereoselective migration of sterically hindered organoboranes in cyclic and acyclic systems. A stereoselective allylic C-H activation reaction Tetrahedron. 59: 9187-9198. DOI: 10.1016/j.tet.2003.09.043  1
2002 Vu VA, Marek I, Polborn K, Knochel P. Preparation of new functionalized cyclopropylmagnesium reagents. Angewandte Chemie (International Ed. in English). 41: 351-2. PMID 12491430 DOI: 10.1002/1521-3773(20020118)41:2<351::AID-ANIE351>3.0.CO;2-5  1
2002 Lotz M, Polborn K, Knochel P. New ferrocenyl ligands with broad applications in asymmetric catalysis. Angewandte Chemie (International Ed. in English). 41: 4708-11. PMID 12481334 DOI: 10.1002/anie.200290024  1
2002 Piazza C, Knochel P. Sterically hindered lithium dialkylcuprates for the generation of highly functionalized mixed cuprates through a halogen-copper exchange. Angewandte Chemie (International Ed. in English). 41: 3263-5. PMID 12207410 DOI: 10.1002/1521-3773(20020902)41:17<3263::AID-ANIE3263>3.0.CO;2-8  0.96
2002 Koradin C, Polborn K, Knochel P. Enantioselective synthesis of propargylamines by copper-catalyzed addition of alkynes to enamines. Angewandte Chemie (International Ed. in English). 41: 2535-8. PMID 12203525 DOI: 10.1002/1521-3773(20020715)41:14<2535::AID-ANIE2535>3.0.CO;2-M  1
2002 Hupe E, Marek I, Knochel P. Diastereoselective reduction of alkenylboronic esters as a new method for controlling the stereochemistry of up to three adjacent centers in cyclic and acyclic molecules. Organic Letters. 4: 2861-3. PMID 12182574 DOI: 10.1021/ol0262486  1
2002 Lindsay DM, Dohle W, Jensen AE, Kopp F, Knochel P. Preparation of polyfunctional heterocycles using highly functionalized aminated arylmagnesium reagents as versatile scaffolds. Organic Letters. 4: 1819-22. PMID 12027622 DOI: 10.1021/ol025597x  1
2002 Jensen AE, Knochel P. Nickel-catalyzed cross-coupling between functionalized primary or secondary alkylzinc halides and primary alkyl halides. The Journal of Organic Chemistry. 67: 79-85. PMID 11777442 DOI: 10.1021/jo0105787  1
2002 Lotz M, Kramer G, Knochel P. Facile axial chirality control by using a precursor with central chirality. Application to the preparation of new axially chiral diphosphine complexes for asymmetric catalysis Chemical Communications. 8: 2546-2547. DOI: 10.1039/b207399d  1
2002 Hupe E, Knochel P, Szabó KJ. Mechanism of the stereoselective alkyl group exchange between alkylboranes and alkylzinc compounds. Quest for novel types of boron-metal exchange reactions Organometallics. 21: 2203-2207. DOI: 10.1021/om020083n  1
2002 Patti A, Lotz M, Knochel P. Synthesis of α,β-disubstituted ferrocenes via a ferrocenylepoxide intermediate. Preparation and catalytic activity of a new chiral ferrocenyloxazoline Tetrahedron Asymmetry. 12: 3375-3380. DOI: 10.1016/S0957-4166(02)00036-8  1
2002 Kneisel FF, Monguchi Y, Knapp KM, Zipse H, Knochel P. Stereoselective cyclizations mediated by functionalized organomagnesium reagents and catalyzed by cobalt or copper salts Tetrahedron Letters. 43: 4875-4879. DOI: 10.1016/S0040-4039(02)00839-0  1
2002 Thibonnet J, Vu VA, Bérillon L, Knochel P. Preparation of α-functionalized alkenylmagnesium reagents via a halide-magnesium exchange Tetrahedron. 58: 4787-4799. DOI: 10.1016/S0040-4020(02)00439-8  1
2002 Ragagnin G, Betzemeier B, Quici S, Knochel P. Copper-catalysed aerobic oxidation of alcohols using fluorous biphasic catalysis Tetrahedron. 58: 3985-3991. DOI: 10.1016/S0040-4020(02)00250-8  1
2002 Jensen AE, Knochel P. Preparation of 2-arylated-1,4-phenylenediamines by palladium-catalyzed cross-coupling reactions Journal of Organometallic Chemistry. 653: 122-128. DOI: 10.1016/S0022-328X(02)01156-7  1
2001 Sapountzis I, Dohle W, Knochel P. Stereoselective preparation of highly functionalized (Z)-3-magnesiated enoates by an iodine-magnesium exchange reaction. Chemical Communications (Cambridge, England). 2068-9. PMID 12240167  1
2001 Hupe E, Knochel P. Formal enantioselective Michael addition with umpolung of reactivity. Angewandte Chemie (International Ed. in English). 40: 3022-5. PMID 12203636 DOI: 10.1002/1521-3773(20010817)40:16<3022::AID-ANIE3022>3.0.CO;2-W  1
2001 Dohle W, Lindsay DM, Knochel P. Copper-mediated cross-coupling of functionalized arylmagnesium reagents with functionalized alkyl and benzylic halides. Organic Letters. 3: 2871-3. PMID 11529778 DOI: 10.1021/ol0163272  1
2001 Hupe E, Knochel P. Stereoselective synthesis of secondary organozinc reagents and their reaction with heteroatomic electrophiles. Organic Letters. 3: 127-30. PMID 11429854 DOI: 10.1021/ol0068400  1
2001 Demay S, Volant F, Knochel P. New C(2)-Symmetrical 1,2-Diphosphanes for the Efficient Rhodium-Catalyzed Asymmetric Hydroboration of Styrene Derivatives We thank the Deutsche Forschungsgemeinschaft (Leibniz program), The Institut de Recherches Servier (Suresnes, France), and PPG-SIPSY for financial support. We thank also BASF AG (Ludwigshafen), Chemetall GmbH (Frankfurt), and Degussa-Hüls AG (Hanau) for the generous gift of chemicals. Angewandte Chemie (International Ed. in English). 40: 1235-1238. PMID 11301435 DOI: 10.1002/1521-3773(20010401)40:7<1235::AID-ANIE1235>3.0.CO;2-Y  1
2001 Demay S, Lotz M, Polborn K, Knochel P. Preparation of a rigid bicyclic diphosphine by radical cyclisation Tetrahedron Asymmetry. 12: 909-914. DOI: 10.1016/S0957-4166(01)00123-9  1
2001 Hupe E, Calaza MI, Knochel P. Diastereoselective synthesis and reactions of diorganozinc reagents obtained after hydroborations with 9-BBN-H, thexylborane and catecholborane Tetrahedron Letters. 42: 8829-8831. DOI: 10.1016/S0040-4039(01)01916-5  1
2001 Boucley C, Cahiez G, Carini S, Cerè V, Comes-Franchini M, Knochel P, Pollicino S, Ricci A. Stereoselective addition of organomanganese reagents to chiral acylsilanes and aldehydes Journal of Organometallic Chemistry. 624: 223-228. DOI: 10.1016/S0022-328X(00)00902-5  1
2001 Piazza C, Millot N, Knochel P. New preparation of benzylic zinc reagents via a fragmentation reaction Journal of Organometallic Chemistry. 624: 88-95. DOI: 10.1016/S0022-328X(00)00840-8  1
2000 Boudier A, Bromm LO, Lotz M, Knochel P. New Applications of Polyfunctional Organometallic Compounds in Organic Synthesis Frequently used abbreviations are defined at the end of the article. Angewandte Chemie (International Ed. in English). 39: 4414-4435. PMID 11169635 DOI: 10.1002/1521-3773(20001215)39:24<4414::AID-ANIE4414>3.0.CO;2-C  1
2000 Goldfuss B, Knochel P, Bromm LO, Knapp K. C-H Activation by Direct Borane-Hydrocarbon Dehydrogenation: Kinetic and Thermodynamic Aspects This work was supported by the Fonds der Chemische Industrie (Sachbeihilfe and Liebig-Stipendium for B.G.), the Deutsche Forschungsgemeinschaft (GO 930/1-1 and Habilitationsstipendium for B.G.), the Research Pool Foundation of the University Heidelberg, Degussa-Hüls AG, and BASF AG. B.G. is grateful to Prof. P. Hofmann for support at Heidelberg and thanks Prof. A. Berndt (Marburg), Prof. G. Frenking (Marburg), and Prof. H. Mayr (München) for fruitful suggestions. Angewandte Chemie (International Ed. in English). 39: 4136-4139. PMID 11093231 DOI: 10.1002/1521-3773(20001117)39:22<4136::AID-ANIE4136>3.0.CO;2-F  0.84
2000 Rodriguez AL, Bunlaksananusorn T, Knochel P. Potassium tert-butoxide catalyzed addition of carbonyl derivatives to styrenes Organic Letters. 2: 3285-7. PMID 11029191  0.88
2000 Boudier A, Darcel C, Flachsmann F, Micouin L, Oestreich M, Knochel P. Stereoselective preparation and reactions of configurationally defined dialkylzinc compounds Chemistry (Weinheim An Der Bergstrasse, Germany). 6: 2748-61. PMID 10985723 DOI: 10.1002/1521-3765(20000804)6:15<2748::AID-CHEM2748>3.0.CO;2-Q  1
2000 Abarbri M, Thibonnet J, Berillon L, Dehmel F, Rottlander M, Knochel P. Preparation of new polyfunctional magnesiated heterocycles using a chlorine-, bromine-, or iodine-magnesium exchange The Journal of Organic Chemistry. 65: 4618-34. PMID 10959867 DOI: 10.1021/jo000235t  1
2000 Rodriguez AL, Koradin C, Dohle W, Knochel P. Versatile Indole Synthesis by a 5-endo-dig Cyclization Mediated by Potassium or Cesium Bases We thank the DFG (Leibniz-Programm) and the Fonds der Chemischen Industrie for generous financial support. A.L.R. and C. K. thank the Humboldt-Foundation and the BASF AG, respectively, for fellowships. W.D. was supported by the BMBF program (03 D 0056 2). We thank Dr. J. Henkelmann (BASF AG) for helpful discussions and the BASF AG for the generous gift of chemicals. Angewandte Chemie (International Ed. in English). 39: 2488-2490. PMID 10941112 DOI: 10.1002/1521-3773(20000717)39:14<2488::AID-ANIE2488>3.0.CO;2-E  1
2000 Boudier A, Hupe E, Knochel P. Highly Diastereoselective Synthesis of Monocyclic and Bicyclic Secondary Diorganozinc Reagents with Defined Configuration We thank the DFG (SFB 260, Leibniz-Program) and the Fonds der Chemischen Industrie for generous support (Kekulé-scholarship for E. H.). We thank BASF, Degussa-Hüls AG, and Chemetall GmbH AG for the generous gift of chemicals. Angewandte Chemie (International Ed. in English). 39: 2294-2297. PMID 10941068 DOI: 10.1002/1521-3773(20000703)39:13<2294::AID-ANIE2294>3.0.CO;2-J  1
2000 Lotz M, Ireland T, Tappe K, Knochel P. Preparation of new chiral borane-protected P,N-ferrocenyl ligands via a methoxy directed ortho-lithiation. Chirality. 12: 389-95. PMID 10824158 DOI: 10.1002/(SICI)1520-636X(2000)12:5/6<389::AID-CHIR16>3.0.CO;2-S  1
2000 Varchi G, Ricci A, Cahiez G, Knochel P. Copper catalyzed conjugate addition of highly functionalized arylmagnesium compounds to enones Tetrahedron. 56: 2727-2731. DOI: 10.1016/S0040-4020(00)00127-7  1
1999 Dübner F, Knochel P. Copper(I)-Catalyzed Enantioselective Substitution of Allyl Chlorides with Diorganozinc Compounds. Angewandte Chemie (International Ed. in English). 38: 379-381. PMID 29711661 DOI: 10.1002/(SICI)1521-3773(19990201)38:3<379::AID-ANIE379>3.0.CO;2-Y  1
1999 Tzalis D, Knochel P. Cesium Hydroxide: A Superior Base for the Catalytic Alkynylation of Aldehydes and Ketones and Catalytic Alkenylation of Nitriles. Angewandte Chemie (International Ed. in English). 38: 1463-1465. PMID 29711565 DOI: 10.1002/(SICI)1521-3773(19990517)38:10<1463::AID-ANIE1463>3.0.CO;2-H  0.6
1999 Millot N, Knochel P. Preparation and stereoselective additions of highly substituted cyclic allylzinc reagents: A zinc-ene cyclization Tetrahedron Letters. 40: 7779-7782. DOI: 10.1016/S0040-4039(99)01689-5  1
1999 Tzalis D, Koradin C, Knochel P. Cesium hydroxide catalyzed addition of alcohols and amine derivatives to alkynes and styrene Tetrahedron Letters. 40: 6193-6195. DOI: 10.1016/S0040-4039(99)01133-8  1
1999 Demay S, Harms K, Knochel P. Stereoselective preparation of phosphine oxides via a 2,3-sigmatropic shift of allylic diphenylphosphinites Tetrahedron Letters. 40: 4981-4984. DOI: 10.1016/S0040-4039(99)00952-1  1
1999 Boudier A, Knochel P. Palladium catalyzed stereoselective cross-couplings and acylations of chiral secondary diorganozincs Tetrahedron Letters. 40: 687-690. DOI: 10.1016/S0040-4039(98)02581-7  1
1998 Boymond L, Rottländer M, Cahiez G, Knochel P. Preparation of Highly Functionalized Grignard Reagents by an Iodine-Magnesium Exchange Reaction and its Application in Solid-Phase Synthesis. Angewandte Chemie (International Ed. in English). 37: 1701-1703. PMID 29711506 DOI: 10.1002/(SICI)1521-3773(19980703)37:12<1701::AID-ANIE1701>3.0.CO;2-U  1
1998 Lutz C, Lutz V, Knochel P. Enantioselective synthesis of 1,2-, 1,3- and 1,4- aminoalcohols by the addition of dialkylzincs to 1,2-, 1,3- and 1,4- aminoaldehydes Tetrahedron. 54: 6385-6402. DOI: 10.1016/S0040-4020(98)00297-X  1
1997 Prasad ASB, Stevenson TM, Citineni JR, Nyzam V, Knochel P. Preparation and reactions of new zincated nitrogen-containing heterocycles Tetrahedron. 53: 7237-7254. DOI: 10.1016/S0040-4020(97)00427-4  1
1996 Stevenson TM, Prasad ASB, Citineni JR, Knochel P. Preparation of zinc organometallics derived from nucleosides and nucleic acid bases and Pd(0) catalyzed coupling with aryl iodides Tetrahedron Letters. 37: 8375-8378. DOI: 10.1016/0040-4039(96)01934-X  1
1996 Klement I, Rottländer M, Tucker CE, Majid TN, Knochel P, Venegas P, Cahiez G. Preparation of polyfunctional aryl and alkenyl zinc halides from functionalized unsaturated organolithiums and their reactivity in cross-coupling and conjugated addition reactions Tetrahedron. 52: 7201-7220. DOI: 10.1016/0040-4020(96)00246-3  1
1996 Stadtmüller H, Vaupel A, Tucker CE, Stüdemann T, Knochel P. Stereoselective preparation of polyfunctional cyclopentane derivatives by radical nickel- or palladium-catalyzed carbozincations Chemistry - a European Journal. 2: 1204-1220. DOI: 10.1002/chem.19960021006  1
1994 Fürstner A, Singer R, Knochel P. A convenient preparation of functionalized arylzinc compounds by the reaction of zinc/silver-graphite with aryl iodides Tetrahedron Letters. 35: 1047-1050. DOI: 10.1016/S0040-4039(00)79962-X  1
1993 Stadtmüller H, Tucker CE, Vaupel A, Knochel P. Stereoselective synthesis of polyfunctional di- and trisubstituted cyclopentane derivatives using a new palladium catalyzed cyclization Tetrahedron Letters. 34: 7911-7914. DOI: 10.1016/S0040-4039(00)61508-3  1
1993 Semmelhack MF, Knochel P, Singleton T. A new approach to indole alkaloids via indole chromium complexes Tetrahedron Letters. 34: 5051-5054. DOI: 10.1016/S0040-4039(00)60673-1  1
1993 Klement I, Lennick K, Tucker CE, Knochel P. Preparation of polyfunctional nitriles by the cyanation of functionalized organozinc halides with p-toluenesulfonyl cyanide Tetrahedron Letters. 34: 4623-4626. DOI: 10.1016/S0040-4039(00)60640-8  1
1992 Cahiez G, Venegas P, Tucker CE, Majid TN, Knochel P. Addition of polyfunctional and pure (E or Z) alkenylcopper and arylcopper compounds to alkylidenemalonates Journal of the Chemical Society, Chemical Communications. 1406-1408. DOI: 10.1039/C39920001406  1
1991 Rozema MJ, Knochel P. Selective multiple methylene insertion reactions mediated by iodomethylzine iodide: Mechanistic considerations and synthetic applications Tetrahedron Letters. 32: 1855-1858. DOI: 10.1016/S0040-4039(00)85980-8  1
1988 Auvray P, Knochel P, Normant JF. 3-bromq-2-t-butylsulfonyl-1-propene. A versatile multi-coupling reagent part II Tetrahedron. 44: 4509-4519. DOI: 10.1016/S0040-4020(01)86152-4  1
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