Year |
Citation |
Score |
2020 |
Donkor IO, Xu J, Liu J, Cameron K. Synthesis and antiproliferative activity of sulfonamide-based peptidomimetic calpain inhibitors. Bioorganic & Medicinal Chemistry. 115433. PMID 32199690 DOI: 10.1016/j.bmc.2020.115433 |
0.461 |
|
2010 |
Saab NH, Donkor IO, Rodriguez L, Kador PF, Miller DD. ChemInform Abstract: Phenylsulfonylnitromethanes as Potent Irreversible Inhibitors of Aldose Reductase. Cheminform. 31: no-no. DOI: 10.1002/chin.200006244 |
0.422 |
|
2010 |
Donkor IO, Abdel-Ghany YS, Kador PF, Mizoguchi T, Bartoszko-Malik A, Miller DD. ChemInform Abstract: Synthesis and Biological Activity of Aldose Reductase Inhibitors with Michael Acceptor Substituents. Cheminform. 30: no-no. DOI: 10.1002/chin.199934174 |
0.383 |
|
2010 |
DONKOR IO, ABDEL-GHANY YS, KADOR PF, MIZOGUCHI T, BARTOSZKO-MALIK A, MILLER DD. ChemInform Abstract: Synthesis and Biological Activities of Aldose Reductase Inhibitors Bearing Acyl Benzenesulfonamides as Carboxylic Acid Surrogates. Cheminform. 29: no-no. DOI: 10.1002/chin.199828119 |
0.357 |
|
2008 |
Donkor IO, Korukonda R. Synthesis and calpain inhibitory activity of peptidomimetic compounds with constrained amino acids at the P2 position. Bioorganic & Medicinal Chemistry Letters. 18: 4806-8. PMID 18694642 DOI: 10.1016/J.Bmcl.2008.07.094 |
0.723 |
|
2008 |
Donkor IO, Assefa H, Liu J. Structural basis for the potent calpain inhibitory activity of peptidyl alpha-ketoacids. Journal of Medicinal Chemistry. 51: 4346-50. PMID 18636690 DOI: 10.1021/jm800182c |
0.379 |
|
2006 |
Korukonda R, Guan N, Dalton JT, Liu J, Donkor IO. Synthesis, calpain inhibitory activity, and cytotoxicity of P2-substituted proline and thiaproline peptidyl aldehydes and peptidyl alpha-ketoamides. Journal of Medicinal Chemistry. 49: 5282-90. PMID 16913717 DOI: 10.1021/Jm050849W |
0.725 |
|
2006 |
Huang TL, Vanden Eynde JJ, Mayence A, Donkor IO, Khan SI, Tekwani BL. Anti-plasmodial and anti-leishmanial activity of conformationally restricted pentamidine congeners. The Journal of Pharmacy and Pharmacology. 58: 1033-42. PMID 16872549 DOI: 10.1211/jpp.58.8.0003 |
0.301 |
|
2006 |
Guan N, Korukonda R, Hurh E, Schmittgen TD, Donkor IO, Dalton JT. Apoptosis induced by novel aldehyde calpain inhibitors in human tumor cell lines. International Journal of Oncology. 29: 655-63. PMID 16865282 DOI: 10.3892/Ijo.29.3.655 |
0.701 |
|
2006 |
Sanders ML, Donkor IO. A novel series of urea-based peptidomimetic calpain inhibitors. Bioorganic & Medicinal Chemistry Letters. 16: 1965-8. PMID 16412635 DOI: 10.1016/j.bmcl.2005.12.068 |
0.716 |
|
2005 |
Vanden Eynde JJ, Mayence A, Johnson MT, Huang TL, Collins MS, Rebholz S, Walzer PD, Cushion MT, Donkor IO. Antitumor and anti-Pneumocystis carinii activities of novel bisbenzamidines Medicinal Chemistry Research. 14: 143-157. DOI: 10.1007/S00044-005-0130-2 |
0.347 |
|
2004 |
Donkor IO, Han J, Zheng X. Design, synthesis, molecular modeling studies, and calpain inhibitory activity of novel alpha-ketoamides incorporating polar residues at the P1'-position. Journal of Medicinal Chemistry. 47: 72-9. PMID 14695821 DOI: 10.1021/jm0301336 |
0.307 |
|
2003 |
Donkor IO, Li H, Queener SF. Synthesis and DHFR inhibitory activity of a series of 6-substituted-2,4-diaminothieno[2,3-d]pyrimidines. European Journal of Medicinal Chemistry. 38: 605-11. PMID 12832132 DOI: 10.1016/S0223-5234(03)00101-6 |
0.32 |
|
2003 |
Donkor IO, Korukonda R, Huang TL, LeCour L. Peptidyl aldehyde inhibitors of calpain incorporating P2-proline mimetics. Bioorganic & Medicinal Chemistry Letters. 13: 783-4. PMID 12617890 DOI: 10.1016/S0960-894X(03)00021-0 |
0.734 |
|
2002 |
Sanders ML, Donkor IO. THE SYNTHESIS OF A SERIES OF 3,5-DISUBSTITUTED TETRAHYDRO- 1H-IMIDAZOLE-2,4-DIONES UTILIZING LITHIUM ALUMINUM HYDRIDE Synthetic Communications. 32: 1015-1021. DOI: 10.1081/Scc-120003149 |
0.332 |
|
2001 |
Donkor IO, Sanders ML. Synthesis of a reported calpain inhibitor isolated from Streptomyces griseus. Bioorganic & Medicinal Chemistry Letters. 11: 2647-9. PMID 11551769 DOI: 10.1016/S0960-894X(01)00524-8 |
0.685 |
|
2000 |
Donkor IO, Zheng X, Miller DD. Synthesis and calpain inhibitory activity of alpha-ketoamides with 2,3-methanoleucine stereoisomers at the P2 position. Bioorganic & Medicinal Chemistry Letters. 10: 2497-500. PMID 11086714 DOI: 10.1016/S0960-894X(00)00518-7 |
0.491 |
|
2000 |
Donkor IO. A survey of calpain inhibitors. Current Medicinal Chemistry. 7: 1171-88. PMID 11032966 DOI: 10.2174/0929867003374129 |
0.498 |
|
2000 |
Donkor IO, Zheng X, Han J, Miller DD. Asymmetric synthesis of 2,3-methanoleucine stereoisomers from common intermediates. Chirality. 12: 551-7. PMID 10861954 DOI: 10.1002/1520-636X(2000)12:7<551::Aid-Chir1>3.0.Co;2-C |
0.334 |
|
1999 |
Tao B, Huang TL, Zhang Q, Jackson L, Queener SF, Donkor IO. Synthesis and anti-Pneumocystis carinii activity of conformationally restricted analogues of pentamidine European Journal of Medicinal Chemistry. 34: 531-538. DOI: 10.1016/S0223-5234(99)80102-0 |
0.344 |
|
1999 |
Donkor IO, Abdel-Ghany YS, Kador PF, Mizoguchi T, Bartoszko-Malik A, Miller DD. Synthesis and biological activity of aldose reductase inhibitors with Michael acceptor substituents European Journal of Medicinal Chemistry. 34: 235-243. DOI: 10.1016/S0223-5234(99)80056-7 |
0.392 |
|
1998 |
Donkor IO, Zhou X, Schmidt J, Agrawal KC, Kishore V. Synthesis and radioprotective effects of adamantyl substituted 1,4-dihydropyridine derivatives. Bioorganic & Medicinal Chemistry. 6: 563-8. PMID 9629469 DOI: 10.1016/S0968-0896(98)00017-0 |
0.326 |
|
1998 |
Donkor IO, Abdel-Ghany YS, Kador PF, Mizoguchi T, Bartoszko-Malik A, Miller DD. Synthesis and biological activities of aldose reductase inhibitors bearing acyl benzenesulfonamides as carboxylic acid surrogates European Journal of Medicinal Chemistry. 33: 15-22. DOI: 10.1016/S0223-5234(99)80071-3 |
0.361 |
|
1996 |
Donkor IO, Devraj R, Queener SF, Barrows LR, Gangjee A. Synthesis of a Series of Diaminobenzo[f]- And Diaminobenzo[h]pyrimido[4,5-b]quinolines as 5-Deaza Tetracyclic Nonclassical Antifolates Journal of Heterocyclic Chemistry. 33: 1653-1660. DOI: 10.1002/Jhet.5570330618 |
0.361 |
|
1994 |
Donkor IO, Tidwell RR, Jones SK. Pentamidine congeners. 2. 2-butene-bridged aromatic diamidines and diimidazolines as potential anti-pneumocystis carinii pneumonia agents Journal of Medicinal Chemistry®. 37: 4554-4557. PMID 7799405 DOI: 10.1021/Jm00052A014 |
0.304 |
|
1991 |
Gangjee A, Donkor IO, Kisliuk RL, Gaumont Y, Thorndike J. Synthesis and biological activity of 5,11-methylenetetrahydro-5-deazahomofolic acid Journal of Medicinal Chemistry. 34: 611-616. PMID 1995884 DOI: 10.1021/Jm00106A022 |
0.521 |
|
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