Neil Vasdev, Ph.D. - Publications

Affiliations: 
2003 McMaster University, Hamilton, ON, Canada 
Area:
Radiation Chemistry

163 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2021 Knight AC, Varlow C, Tong J, Vasdev N. In Vitro and In Vivo Evaluation of GSK-3 Radioligands in Alzheimer's Disease: Preliminary Evidence of Sex Differences. Acs Pharmacology & Translational Science. 4: 1287-1294. PMID 34423266 DOI: 10.1021/acsptsci.1c00132  1
2021 Boyle AJ, Gaudet VC, Black SE, Vasdev N, Rosa-Neto P, Zukotynski KA. Artificial intelligence for molecular neuroimaging. Annals of Translational Medicine. 9: 822. PMID 34268435 DOI: 10.21037/atm-20-6220  0.01
2021 Murrell E, Tong J, Smil D, Kiyota T, Aman AM, Isaac MB, Watson IDG, Vasdev N. Leveraging Open Science Drug Development for PET: Preliminary Neuroimaging of C-Labeled ALK2 Inhibitors. Acs Medicinal Chemistry Letters. 12: 846-850. PMID 34055235 DOI: 10.1021/acsmedchemlett.1c00127  1
2021 Attwells S, Setiawan E, Rusjan PM, Xu C, Kish SJ, Vasdev N, Houle S, Santhirakumar A, Meyer JH. A double-blind placebo-controlled trial of minocycline on translocator protein distribution volume in treatment-resistant major depressive disorder. Translational Psychiatry. 11: 334. PMID 34052828 DOI: 10.1038/s41398-021-01450-3  1
2021 Pees A, Vosjan MJWD, Vasdev N, Windhorst AD, Vugts DJ. Fluorine-18 labelled Ruppert-Prakash reagent ([F]MeSiCF) for the synthesis of F-trifluoromethylated compounds. Chemical Communications (Cambridge, England). 57: 5286-5289. PMID 33942818 DOI: 10.1039/d1cc01789f  0.01
2021 Zukotynski K, Black SE, Kuo PH, Bhan A, Adamo S, Scott CJM, Lam B, Masellis M, Kumar S, Fischer CE, Tartaglia MC, Lang AE, Tang-Wai DF, Freedman M, Vasdev N, et al. Exploratory Assessment of K-means Clustering to Classify 18F-Flutemetamol Brain PET as Positive or Negative. Clinical Nuclear Medicine. PMID 33883495 DOI: 10.1097/RLU.0000000000003668  0.01
2021 Ding Y, Gao H, Zhang Y, Li Y, Vasdev N, Gao Y, Chen Y, Zhang Q. Correction to: Alantolactone selectively ablates acute myeloid leukemia stem and progenitor cells. Journal of Hematology & Oncology. 14: 61. PMID 33858468 DOI: 10.1186/s13045-021-01069-3  0.01
2021 Varlow C, Mossine AV, Bernard-Gauthier V, Scott PJH, Vasdev N. Radiofluorination of oxazole-carboxamides for preclinical PET neuroimaging of GSK-3. Journal of Fluorine Chemistry. 245. PMID 33840834 DOI: 10.1016/j.jfluchem.2021.109760  0.01
2021 Knight AC, Varlow C, Zi T, Liang SH, Josephson L, Schmidt K, Patel S, Vasdev N. Evaluation of [H]CPPC as a Tool Radioligand for CSF-1R. Acs Chemical Neuroscience. PMID 33667059 DOI: 10.1021/acschemneuro.0c00802  1
2021 Narayanaswami V, Tong J, Schifani C, Bloomfield PM, Dahl K, Vasdev N. Preclinical Evaluation of TSPO and MAO-B PET Radiotracers in an LPS Model of Neuroinflammation. Pet Clinics. 16: 233-247. PMID 33648665 DOI: 10.1016/j.cpet.2020.12.003  1
2021 Zhang L, Hu K, Shao T, Hou L, Zhang S, Ye W, Josephson L, Meyer JH, Zhang MR, Vasdev N, Wang J, Xu H, Wang L, Liang SH. Recent developments on PET radiotracers for TSPO and their applications in neuroimaging. Acta Pharmaceutica Sinica. B. 11: 373-393. PMID 33643818 DOI: 10.1016/J.Apsb.2020.08.006  1
2021 Lindberg A, Knight AC, Sohn D, Rakos L, Tong J, Radelet A, Mason NS, Stehouwer JS, Lopresti BJ, Klunk WE, Sandell J, Sandberg A, Hammarström P, Svensson S, Mathis CA, ... Vasdev N, et al. Radiosynthesis, and Evaluation of [F]CBD-2115 as a First-in-Class Radiotracer for Imaging 4R-Tauopathies. Acs Chemical Neuroscience. PMID 33497190 DOI: 10.1021/acschemneuro.0c00801  1
2021 Daniels RD, Clouston SAP, Hall CB, Anderson KR, Bennett DA, Bromet EJ, Calvert GM, Carreón T, DeKosky ST, Diminich ED, Finch CE, Gandy S, Kreisl WC, Kritikos M, Kubale TL, ... ... Vasdev N, et al. A Workshop on Cognitive Aging and Impairment in the 9/11-Exposed Population. International Journal of Environmental Research and Public Health. 18. PMID 33466931 DOI: 10.3390/ijerph18020681  0.01
2020 Hou L, Rong J, Haider A, Ogasawara D, Varlow C, Schafroth MA, Mu L, Gan J, Xu H, Fowler CJ, Zhang MR, Vasdev N, Ametamey S, Cravatt BF, Wang L, et al. Positron Emission Tomography Imaging of the Endocannabinoid System: Opportunities and Challenges in Radiotracer Development. Journal of Medicinal Chemistry. PMID 33379862 DOI: 10.1021/acs.jmedchem.0c01459  1
2020 Herth MM, Ametamey S, Antuganov D, Bauman A, Berndt M, Brooks AF, Bormans G, Choe YS, Gillings N, Häfeli UO, James ML, Kopka K, Kramer V, Krasikova R, Madsen J, ... ... Vasdev N, et al. On the consensus nomenclature rules for radiopharmaceutical chemistry - Reconsideration of radiochemical conversion. Nuclear Medicine and Biology. 93: 19-21. PMID 33232876 DOI: 10.1016/j.nucmedbio.2020.11.003  0.01
2020 Boyle AJ, Tong J, Zoghbi S, Pike VW, Innis R, Vasdev N. Repurposing [C]PS13 for PET imaging of cyclooxygenase-1 (COX-1) in ovarian cancer xenograft mouse models. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 32978284 DOI: 10.2967/jnumed.120.249367  1
2020 Gee AD, Herth MM, James ML, Korde A, Scott PJH, Vasdev N. Radionuclide Imaging for Neuroscience: Current Opinion and Future Directions. Molecular Imaging. 19: 1536012120936397. PMID 32907484 DOI: 10.1177/1536012120936397  1
2020 Dahl K, Turner T, Vasdev N. Radiosynthesis of a Bruton's Tyrosine Kinase Inhibitor, [ C]Tolebrutinib, via Palladium-NiXantphos-Mediated Carbonylation. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 32726870 DOI: 10.1002/Jlcr.3872  0.01
2020 Gee AD, Andersson J, Bhalla R, Choe YS, Dick DW, Herth MM, Hostetler ED, Jáuregui-Haza UJ, Huang YY, James ML, Jeong JM, Korde A, Kuge Y, Kung HF, Lapi SE, ... ... Vasdev N, et al. Training the next generation of radiopharmaceutical scientists. Nuclear Medicine and Biology. 88: 10-13. PMID 32650289 DOI: 10.1016/J.Nucmedbio.2020.06.004  1
2020 Murrell E, Pham JM, Sowa AR, Brooks AF, Kilbourn MR, Scott PJH, Vasdev N. Classics in Neuroimaging: Development of Positron Emission Tomography Tracers for Imaging the GABAergic Pathway. Acs Chemical Neuroscience. PMID 32578977 DOI: 10.1021/Acschemneuro.0C00343  0.01
2020 Varlow C, Boileau I, Wey HY, Liang SH, Vasdev N. Classics in Neuroimaging: Imaging the Endocannabinoid Pathway with PET. Acs Chemical Neuroscience. PMID 32559067 DOI: 10.1021/Acschemneuro.0C00305  1
2020 Narayanaswami V, Tong J, Fiorino F, Severino B, Sparaco R, Magli E, Giordano F, Bloomfield PM, Prabhakaran J, Mann JJ, Vasdev N, Dahl K, Kumar JSD. Synthesis, in vitro and in vivo evaluation of C-O-methylated arylpiperazines as potential serotonin 1A (5-HT) receptor antagonist radiotracers. Ejnmmi Radiopharmacy and Chemistry. 5: 13. PMID 32430632 DOI: 10.1186/S41181-020-00096-8  1
2020 Attwells S, Setiawan E, Rusjan PM, Xu C, Hutton C, Rafiei D, Varughese B, Kahn A, Kish SJ, Vasdev N, Houle S, Meyer JH. Translocator Protein Distribution Volume Predicts Reduction of Symptoms During Open-Label Trial of Celecoxib in Major Depressive Disorder. Biological Psychiatry. PMID 32402468 DOI: 10.1016/J.Biopsych.2020.03.007  1
2020 Duffy IR, Vasdev N, Dahl K. Copper(I)-Mediated C-Carboxylation of (Hetero)arylstannanes. Acs Omega. 5: 8242-8250. PMID 32309734 DOI: 10.1021/acsomega.0c00524  0.01
2020 Varlow C, Murrell E, Holland JP, Kassenbrock A, Shannon W, Liang SH, Vasdev N, Stephenson NA. Revisiting the Radiosynthesis of [F]FPEB and Preliminary PET Imaging in a Mouse Model of Alzheimer's Disease. Molecules (Basel, Switzerland). 25. PMID 32098347 DOI: 10.3390/Molecules25040982  1
2019 Attwells S, Setiawan E, Wilson AA, Rusjan PM, Miler L, Xu C, Hutton C, Husain MI, Kish S, Vasdev N, Houle S, Meyer JH. Replicating predictive serum correlates of greater translocator protein distribution volume in brain. Neuropsychopharmacology : Official Publication of the American College of Neuropsychopharmacology. PMID 31683271 DOI: 10.1038/S41386-019-0561-Y  1
2019 Bernard-Gauthier V, Mossine AV, Knight A, Patnaik D, Zhao W, Cheng C, Krishnan HS, Xuan LL, Chindavong PS, Reis SA, Chen JM, Shao X, Stauff J, Arteaga J, Sherman PS, ... ... Vasdev N, et al. Structural Basis for Achieving GSK-3 Inhibition with High Potency, Selectivity and Brain Exposure for PET Imaging and Drug Discovery. Journal of Medicinal Chemistry. PMID 31535859 DOI: 10.1021/Acs.Jmedchem.9B01030  1
2019 Duffy IR, Boyle AJ, Vasdev N. Improving PET Imaging Acquisition and Analysis With Machine Learning: A Narrative Review With Focus on Alzheimer's Disease and Oncology. Molecular Imaging. 18: 1536012119869070. PMID 31429375 DOI: 10.1177/1536012119869070  0.01
2019 Osovizky A, Laster B, Wilson AA, Bloomfield P, Sarusi B, Vasdev N, Bell T, Garcia A, Houle S. New detection configuration for low activity levels of PET tracers during the analysis of plasma samples. Applied Radiation and Isotopes : Including Data, Instrumentation and Methods For Use in Agriculture, Industry and Medicine. 151: 317-330. PMID 31376719 DOI: 10.1016/J.Apradiso.2019.05.025  1
2019 Dahl K, Garcia A, Stephenson NA, Vasdev N. "In-loop" F-fluorination: A proof-of-concept study. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 31083778 DOI: 10.1002/Jlcr.3751  1
2019 Dahl K, Bernard-Gauthier V, Nag S, Varnäs K, Narayanaswami V, Mahdi Moein M, Arakawa R, Vasdev N, Halldin C. Synthesis and preclinical evaluation of [F]FSL25.1188, a reversible PET radioligand for monoamine oxidase-B. Bioorganic & Medicinal Chemistry Letters. PMID 31060887 DOI: 10.1016/J.Bmcl.2019.04.040  0.01
2019 Liang SH, Wang L, Stephenson NA, Rotstein BH, Vasdev N. Facile F labeling of non-activated arenes via a spirocyclic iodonium(III) ylide method and its application in the synthesis of the mGluR PET radiopharmaceutical [F]FPEB. Nature Protocols. PMID 30980032 DOI: 10.1038/S41596-019-0149-3  1
2019 Moriguchi S, Wilson AA, Miler L, Rusjan PM, Vasdev N, Kish SJ, Rajkowska G, Wang J, Bagby M, Mizrahi R, Varughese B, Houle S, Meyer JH. Monoamine Oxidase B Total Distribution Volume in the Prefrontal Cortex of Major Depressive Disorder: An [11C]SL25.1188 Positron Emission Tomography Study. Jama Psychiatry. PMID 30840042 DOI: 10.1001/Jamapsychiatry.2019.0044  1
2019 Chen Z, Mori W, Deng X, Cheng R, Ogasawara D, Zhang G, Schafroth MA, Dahl K, Fu H, Hatori A, Shao T, Zhang Y, Yamasaki T, Zhang X, Rong J, ... ... Vasdev N, et al. Design, synthesis and evaluation of reversible and irreversible monoacylglycerol lipase positron emission tomography (PET) tracers using a 'tail switching' strategy on a piperazinyl azetidine skeleton. Journal of Medicinal Chemistry. PMID 30829483 DOI: 10.1021/Acs.Jmedchem.8B01778  1
2019 Narayanaswami V, Drake LR, Brooks AF, Meyer JH, Houle S, Kilbourn MR, Scott PJH, Vasdev N. Classics in Neuroimaging: Development of PET Tracers for Imaging Monoamine Oxidases. Acs Chemical Neuroscience. PMID 30789704 DOI: 10.1021/Acschemneuro.9B00081  1
2019 Deng X, Rong J, Wang L, Vasdev N, Zhang L, Josephson L, Liang SH. Chemie der Positronenemissionstomographie: Aktuelle Fortschritte bei 11C‐, 18F‐, 13N‐ und 15O‐Markierungsreaktionen Angewandte Chemie. 131: 2604-2631. DOI: 10.1002/Ange.201805501  1
2018 Collier TL, Dahl K, Stephenson NA, Holland JP, Riley A, Liang SH, Vasdev N. Recent applications of a single quadrupole mass spectrometer in C, F and radiometal chemistry. Journal of Fluorine Chemistry. 210: 46-55. PMID 30410189 DOI: 10.1016/J.Jfluchem.2018.02.009  1
2018 Josephson L, Stratman N, Liu Y, Qian F, Liang SH, Vasdev N, Patel S. The Binding of BF-227-Like Benzoxazoles to Human α-Synuclein and Amyloid β Peptide Fibrils. Molecular Imaging. 17: 1536012118796297. PMID 30213230 DOI: 10.1177/1536012118796297  1
2018 Narayanaswami V, Dahl K, Bernard-Gauthier V, Josephson L, Cumming P, Vasdev N. Emerging PET Radiotracers and Targets for Imaging of Neuroinflammation in Neurodegenerative Diseases: Outlook Beyond TSPO. Molecular Imaging. 17: 1536012118792317. PMID 30203712 DOI: 10.1177/1536012118792317  1
2018 Varlow C, Szames D, Dahl K, Bernard-Gauthier V, Vasdev N. Fluorine-18: an untapped resource in inorganic chemistry. Chemical Communications (Cambridge, England). PMID 30191929 DOI: 10.1039/C8Cc04751K  0.01
2018 Deng X, Rong J, Wang L, Vasdev N, Zhang L, Josephson L, Liang S. Chemistry for Positron Emission Tomography: Recent Advances in 11C-, 18F-, 13N- and 15O-labeling Reactions. Angewandte Chemie (International Ed. in English). PMID 30054961 DOI: 10.1002/Anie.201805501  1
2018 Cheng R, Mori W, Ma L, Alhouayek M, Hatori A, Zhang Y, Ogasawara D, Yuan G, Chen Z, Zhang X, Shi H, Yamasaki T, Xie L, Kumata K, Fujinaga M, ... ... Vasdev N, et al. In vitro and in vivo evaluation ofC-labeled azetidine-carboxylates for imaging monoacylglycerol lipase by PET imaging studies. Journal of Medicinal Chemistry. PMID 29481079 DOI: 10.1021/Acs.Jmedchem.7B01400  1
2018 Krishnan HS, Bernard-Gauthier V, Placzek MS, Dahl K, Narayanaswami V, Livni E, Chen Z, Yang J, Collier TL, Ran C, Hooker JM, Liang SH, Vasdev N. A metal protein-attenuating compound for PET neuroimaging: Synthesis and preclinical evaluation of [11C]PBT2. Molecular Pharmaceutics. PMID 29298483 DOI: 10.1021/Acs.Molpharmaceut.7B00936  1
2017 Collier TL, Liang SH, Mann JJ, Vasdev N, Kumar JSD. Microfluidic radiosynthesis of [F]FEMPT, a high affinity PET radiotracer for imaging serotonin receptors. Beilstein Journal of Organic Chemistry. 13: 2922-2927. PMID 29564020 DOI: 10.3762/Bjoc.13.285  1
2017 Bernard-Gauthier V, Lepage M, Waengler B, Bailey JA, Liang SH, Perrin D, Vasdev N, Schirrmacher R. Recent advances in fluorine-18 radiochemistry: Focus on B-18F, Si-18F, Al-18F and C-18F radiofluorination via spirocyclic iodonium ylides. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 29284673 DOI: 10.2967/Jnumed.117.197095  1
2017 Cumming P, Burgher B, Patkar O, Breakspear M, Vasdev N, Thomas P, Liu GJ, Banati R. Sifting through the surfeit of neuroinflammation tracers. Journal of Cerebral Blood Flow and Metabolism : Official Journal of the International Society of Cerebral Blood Flow and Metabolism. 271678X17748786. PMID 29256293 DOI: 10.1177/0271678X17748786  1
2017 Bernard-Gauthier V, Collier TL, Liang SH, Vasdev N. Discovery of PET radiopharmaceuticals at the academia-industry interface. Drug Discovery Today. Technologies. 25: 19-26. PMID 29233263 DOI: 10.1016/J.Ddtec.2017.09.001  1
2017 Yuan G, Jankins TC, Patrick CG, Philbrook P, Sears O, Hatfield S, Sitkovsky M, Vasdev N, Liang SH, Ondrechen MJ, Pollastri MP, Jones GB. Fluorinated Adenosine A2A Receptor Antagonists Inspired by Preladenant as Potential Cancer Immunotherapeutics. International Journal of Medicinal Chemistry. 2017: 4852537. PMID 29201461 DOI: 10.1155/2017/4852537  1
2017 Collier TL, Maresca KP, Normandin MD, Richardson P, McCarthy TJ, Liang SH, Waterhouse RN, Vasdev N. Brain Penetration of the ROS1/ALK Inhibitor Lorlatinib Confirmed by PET. Molecular Imaging. 16: 1536012117736669. PMID 29067878 DOI: 10.1177/1536012117736669  1
2017 Makaretz SJ, Quimby M, Collins J, Makris N, McGinnis S, Schultz A, Vasdev N, Johnson KA, Dickerson BC. Flortaucipir tau PET imaging in semantic variant primary progressive aphasia. Journal of Neurology, Neurosurgery, and Psychiatry. PMID 28986472 DOI: 10.1136/Jnnp-2017-316409  1
2017 Lin SF, Bois F, Holden D, Nabulsi N, Pracitto R, Gao H, Kapinos M, Teng JK, Shirali A, Ropchan J, Carson RE, Elmore CS, Vasdev N, Huang Y. The Search for a Subtype-Selective PET Imaging Agent for the GABAA Receptor Complex: Evaluation of the Radiotracer [(11)C]ADO in Nonhuman Primates. Molecular Imaging. 16: 1536012117731258. PMID 28929924 DOI: 10.1177/1536012117731258  0.01
2017 Kanthan M, Cumming P, Hooker JM, Vasdev N. Classics in Neuroimaging: Imaging the Dopaminergic Pathway with PET. Acs Chemical Neuroscience. PMID 28719177 DOI: 10.1021/Acschemneuro.7B00252  1
2017 Krishnan H, Ma L, Vasdev N, Liang S. ¹⁸F-Labeling of Sensitive Biomolecules for Positron Emission Tomography. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28704575 DOI: 10.1002/Chem.201701581  0.01
2017 Dahl K, Collier TL, Chang R, Zhang X, Sadovski O, Liang SH, Vasdev N. "In-Loop" [(11) C]CO2 -Fixation: Prototype and Proof-of-Concept. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 28600835 DOI: 10.1002/Jlcr.3528  1
2017 Collier TL, Normandin MD, Stephenson NA, Livni E, Liang SH, Wooten DW, Esfahani SA, Stabin MG, Mahmood U, Chen J, Wang W, Maresca K, Waterhouse RN, El Fakhri G, Richardson P, ... Vasdev N, et al. Synthesis and preliminary PET imaging of (11)C and (18)F isotopologues of the ROS1/ALK inhibitor lorlatinib. Nature Communications. 8: 15761. PMID 28594000 DOI: 10.1038/Ncomms15761  1
2017 Ma L, Placzek MS, Hooker JM, Vasdev N, Liang SH. [(11)C]Cyanation of arylboronic acids in aqueous solutions. Chemical Communications (Cambridge, England). PMID 28580477 DOI: 10.1039/C7Cc02886E  1
2017 Vasdev N, Alavi A. Novel PET Radiotracers with Potential Clinical Applications. Pet Clinics. 12: xi-xii. PMID 28576174 DOI: 10.1016/J.Cpet.2017.04.002  0.01
2017 Wang L, Cheng R, Fujinaga M, Yang J, Zhang Y, Hatori A, Kumata K, Yang J, Vasdev N, Du Y, Ran C, Zhang MR, Liang SH. A Facile Radiolabeling of [(18)F]FDPA via Spirocyclic Iodonium Ylides: Preliminary PET Imaging Studies in Preclinical Models of Neuroinflammation. Journal of Medicinal Chemistry. PMID 28530834 DOI: 10.1021/Acs.Jmedchem.7B00432  1
2017 Hu K, Patnaik D, Collier TL, Lee KN, Gao H, Swoyer MR, Rotstein BH, Krishnan HS, Liang SH, Wang J, Yan Z, Hooker JM, Vasdev N, Haggarty SJ, Ngai MY. Development of [(18)F]Maleimide-Based Glycogen Synthase Kinase-3β Ligands for Positron Emission Tomography Imaging. Acs Medicinal Chemistry Letters. 8: 287-292. PMID 28337318 DOI: 10.1021/Acsmedchemlett.6B00405  1
2017 Xia C, Makaretz SJ, Caso C, McGinnis S, Gomperts SN, Sepulcre J, Gomez-Isla T, Hyman BT, Schultz A, Vasdev N, Johnson KA, Dickerson BC. Association of In Vivo [18F]AV-1451 Tau PET Imaging Results With Cortical Atrophy and Symptoms in Typical and Atypical Alzheimer Disease. Jama Neurology. PMID 28241163 DOI: 10.1001/Jamaneurol.2016.5755  1
2017 Collier TL, Yokell DL, Livni E, Rice PA, Celen S, Serdons K, Neelamegam R, Bormans G, Harris D, Walji A, Hostetler ED, Bennacef I, Vasdev N. cGMP Production of the Radiopharmaceutical [(18) F]MK-6240 for PET imaging of Human Neurofibrillary Tangles. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 28185305 DOI: 10.1002/Jlcr.3496  1
2017 Khotavivattana T, Calderwood S, Verhoog S, Pfeifer L, Preshlock S, Vasdev N, Collier TL, Gouverneur V. Synthesis and Reactivity of (18)F-Labeled α,α-Difluoro-α-(aryloxy)acetic Acids. Organic Letters. PMID 28085289 DOI: 10.1021/Acs.Orglett.6B03730  1
2017 Krishnan HS, Ma L, Vasdev N, Liang SH. Frontispiece: 18F‐Labeling of Sensitive Biomolecules for Positron Emission Tomography Chemistry: a European Journal. 23. DOI: 10.1002/Chem.201786262  1
2016 Yuan G, Wang F, Stephenson NA, Wang L, Rotstein BH, Vasdev N, Tang P, Liang SH. Metal-free (18)F-labeling of aryl-CF2H via nucleophilic radiofluorination and oxidative C-H activation. Chemical Communications (Cambridge, England). PMID 27917423 DOI: 10.1039/C6Cc07913J  1
2016 Wooten D, Guehl NJ, Verwer EE, Shoup TM, Yokell DL, Zubcevik N, Vasdev N, Zafonte RD, Johnson KA, El Fakhri G, Normandin MD. Pharmacokinetic evaluation of the tau PET radiotracer [18F]T807 ([18F]AV-1451) in human subjects. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 27660144 DOI: 10.2967/Jnumed.115.170910  1
2016 Ding Y, Gao H, Zhang Y, Li Y, Vasdev N, Gao Y, Chen Y, Zhang Q. Alantolactone selectively ablates acute myeloid leukemia stem and progenitor cells. Journal of Hematology & Oncology. 9: 93. PMID 27658462 DOI: 10.1186/S13045-016-0327-5  0.01
2016 Gomperts SN, Locascio JJ, Makaretz SJ, Schultz A, Caso C, Vasdev N, Sperling R, Growdon JH, Dickerson BC, Johnson K. Tau Positron Emission Tomographic Imaging in the Lewy Body Diseases. Jama Neurology. PMID 27654968 DOI: 10.1001/Jamaneurol.2016.3338  1
2016 Rotstein BH, Placzek MS, Krishnan HS, Pekošak A, Collier TL, Wang C, Liang SH, Burstein ES, Hooker JM, Vasdev N. Preclinical PET Neuroimaging of [11C]Bexarotene. Molecular Imaging. 15. PMID 27553293 DOI: 10.1177/1536012116663054  1
2016 Vasdev N, Collier TL. Design and Prototype of an Automated Column-Switching HPLC System for Radiometabolite Analysis. Pharmaceuticals (Basel, Switzerland). 9. PMID 27548189 DOI: 10.3390/Ph9030051  1
2016 Yuan G, Jones GB, Vasdev N, Liang SH. Radiosynthesis and preliminary PET evaluation of (18)F-labeled 2-(1-(3-fluorophenyl)-2-oxo-5-(pyrimidin-2-yl)-1,2-dihydropyridin-3-yl)benzonitrile for imaging AMPA receptors. Bioorganic & Medicinal Chemistry Letters. PMID 27546294 DOI: 10.1016/J.Bmcl.2016.07.078  1
2016 Rotstein BH, Wang L, Liu RY, Patteson J, Kwan EE, Vasdev N, Liang SH. Mechanistic Studies and Radiofluorination of Structurally Diverse Pharmaceuticals with Spirocyclic Iodonium(III) Ylides. Chemical Science. 7: 4407-4417. PMID 27540460 DOI: 10.1039/C6Sc00197A  1
2016 Shi H, Braun A, Wang L, Liang SH, Vasdev N, Ritter T. Synthesis of (18) F-Difluoromethylarenes from Aryl (Pseudo) Halides. Angewandte Chemie (International Ed. in English). PMID 27491349 DOI: 10.1002/Anie.201604106  1
2016 Liang SH, Chen JM, Normandin MD, Chang JS, Chang GC, Taylor CK, Trapa P, Plummer MS, Para KS, Conn EL, Lopresti-Morrow L, Lanyon LF, Cook JM, Richter KE, Nolan CE, ... ... Vasdev N, et al. Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging. Angewandte Chemie (International Ed. in English). PMID 27355874 DOI: 10.1002/Anie.201603797  1
2016 Wang L, Mori W, Cheng R, Yui J, Hatori A, Ma L, Zhang Y, Rotstein BH, Fujinaga M, Shimoda Y, Yamasaki T, Xie L, Nagai Y, Minamimoto T, Higuchi M, ... Vasdev N, et al. Synthesis and Preclinical Evaluation of Sulfonamido-based [(11)C-Carbonyl]-Carbamates and Ureas for Imaging Monoacylglycerol Lipase. Theranostics. 6: 1145-59. PMID 27279908 DOI: 10.7150/Thno.15257  1
2016 Rotstein BH, Liang SH, Placzek MS, Hooker JM, Gee AD, Dollé F, Wilson AA, Vasdev N. (11)C[double bond, length as m-dash]O bonds made easily for positron emission tomography radiopharmaceuticals. Chemical Society Reviews. PMID 27276357 DOI: 10.1039/C6Cs00310A  1
2016 Kassenbrock A, Vasdev N, Liang SH. Selected PET Radioligands for Ion Channel Linked Neuroreceptor Imaging: Focus on GABA, NMDA and nACh Receptors. Current Topics in Medicinal Chemistry. PMID 26975506 DOI: 10.2174/1568026616666160315142457  1
2015 Boros E, Bowen AM, Josephson L, Vasdev N, Holland JP. Chelate-free metal ion binding and heat-induced radiolabeling of iron oxide nanoparticles. Chemical Science. 6: 225-236. PMID 28553472 DOI: 10.1039/C4Sc02778G  1
2015 Calderwood S, Collier TL, Gouverneur V, Liang SH, Vasdev N. Synthesis of (18)F-Arenes from Spirocyclic Iodonium(III) Ylides via Continuous-Flow Microfluidics. Journal of Fluorine Chemistry. 178: 249-253. PMID 27512233 DOI: 10.1016/J.Jfluchem.2015.08.006  1
2015 Liang SH, Vasdev N. Total Radiosynthesis: Thinking outside "the box". Australian Journal of Chemistry. 68: 1319-1328. PMID 27512156 DOI: 10.1071/Ch15406  1
2015 Rashidian M, Wang L, Eden JG, Jacobsen JT, Hossain I, Wang Q, Victora GD, Vasdev N, Ploegh H, Liang SH. Enzyme-Mediated Modification of Single-Domain Antibodies for Imaging Modalities with Different Characteristics. Angewandte Chemie (International Ed. in English). PMID 26630549 DOI: 10.1002/Anie.201507596  1
2015 Johnson KA, Schultz A, Betensky RA, Becker JA, Sepulcre J, Rentz D, Mormino E, Chhatwal J, Amariglio R, Papp K, Marshall G, Albers M, Mauro S, Pepin L, Alverio J, ... ... Vasdev N, et al. Tau PET imaging in aging and early Alzheimer's disease. Annals of Neurology. PMID 26505746 DOI: 10.1002/Ana.24546  1
2015 Wang L, Yui J, Wang Q, Zhang Y, Mori W, Shimoda Y, Fujinaga M, Kumata K, Yamasak TI, Hatori A, Rotstein BH, Collier TL, Ran C, Vasdev N, Zhang MR, et al. Synthesis and preliminary PET imaging studies of a FAAH radiotracer ([(11)C]MPPO) based on α-ketoheterocyclic scaffold. Acs Chemical Neuroscience. PMID 26505525 DOI: 10.1021/Acschemneuro.5B00248  1
2015 Liang SH, Southon AG, Fraser BH, Krause-Heuer AM, Zhang B, Shoup TM, Lewis R, Volitakis I, Han Y, Greguric I, Bush AI, Vasdev N. Novel Fluorinated 8-Hydroxyquinoline Based Metal Ionophores for Exploring the Metal Hypothesis of Alzheimer's Disease. Acs Medicinal Chemistry Letters. 6: 1025-9. PMID 26396692 DOI: 10.1021/Acsmedchemlett.5B00281  1
2015 Marquié M, Normandin MD, Vanderburg CR, Costantino IM, Bien EA, Rycyna LG, Klunk WE, Mathis CA, Ikonomovic MD, Debnath ML, Vasdev N, Dickerson BC, Gomperts SN, Growdon JH, Johnson KA, et al. Validating novel tau positron emission tomography tracer [F-18]-AV-1451 (T807) on postmortem brain tissue. Annals of Neurology. PMID 26344059 DOI: 10.1002/Ana.24517  1
2015 Jacobson O, Weiss I, Wang L, Wang Z, Yang X, Dewhurst A, Ma Y, Zhu G, Niu G, Kiesewetter DO, Vasdev N, Liang S, Chen X. 18F-labeled Single-Stranded DNA Aptamer for PET Imaging of Protein Tyrosine Kinase-7 Expression. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 26315836 DOI: 10.2967/Jnumed.115.160960  1
2015 Wang L, Jacobson O, Avdic D, Rotstein BH, Weiss ID, Collier L, Chen X, Vasdev N, Liang SH. Ortho-Stabilized (18) F-Azido Click Agents and their Application in PET Imaging with Single-Stranded DNA Aptamers. Angewandte Chemie (International Ed. in English). PMID 26308650 DOI: 10.1002/Anie.201505927  1
2015 Rotstein BH, Liang SH, Belov VV, Livni E, Levine DB, Bonab AA, Papisov MI, Perlis RH, Vasdev N. Practical Radiosynthesis and Preclinical Neuroimaging of [11C]isradipine, a Calcium Channel Antagonist. Molecules (Basel, Switzerland). 20: 9550-9. PMID 26016546 DOI: 10.3390/Molecules20069550  1
2015 Liang SH, Holland JP, Stephenson NA, Kassenbrock A, Rotstein BH, Daignault CP, Lewis R, Collier L, Hooker JM, Vasdev N. PET neuroimaging studies of [(18)F]CABS13 in a double transgenic mouse model of Alzheimer's disease and nonhuman primates. Acs Chemical Neuroscience. 6: 535-41. PMID 25776827 DOI: 10.1021/Acschemneuro.5B00055  1
2015 Stephenson NA, Holland JP, Kassenbrock A, Yokell DL, Livni E, Liang SH, Vasdev N. Iodonium ylide-mediated radiofluorination of 18F-FPEB and validation for human use. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 56: 489-92. PMID 25655630 DOI: 10.2967/Jnumed.114.151332  1
2015 Heidari P, Deng F, Esfahani SA, Leece AK, Shoup TM, Vasdev N, Mahmood U. Pharmacodynamic imaging guides dosing of a selective estrogen receptor degrader. Clinical Cancer Research : An Official Journal of the American Association For Cancer Research. 21: 1340-7. PMID 25609068 DOI: 10.1158/1078-0432.Ccr-14-1178  1
2015 Hicks JW, Sadovski O, Parkes J, Houle S, Hay BA, Carter RL, Wilson AA, Vasdev N. Radiosynthesis and ex vivo evaluation of [(18)F]-(S)-3-(6-(3-fluoropropoxy)benzo[d]isoxazol-3-yl)-5-(methoxymethyl)oxazolidin-2-one for imaging MAO-B with PET. Bioorganic & Medicinal Chemistry Letters. 25: 288-91. PMID 25488845 DOI: 10.1016/J.Bmcl.2014.11.048  1
2015 Shoup TM, Bonab AA, Wilson AA, Vasdev N. Synthesis and preclinical evaluation of [¹⁸F]FCHC for neuroimaging of fatty acid amide hydrolase. Molecular Imaging and Biology : Mib : the Official Publication of the Academy of Molecular Imaging. 17: 257-63. PMID 25273322 DOI: 10.1007/S11307-014-0789-1  1
2015 Dickerson B, Makaretz S, Caso C, Stepanovic M, McGinnis SM, Xia C, Schultz AP, Vasdev N, Johnson KA. Imaging tau pathology in vivo in ftld with [18F] T807 PET Alzheimers & Dementia. 11: 545. DOI: 10.1016/J.Jalz.2015.06.690  1
2014 Liang SH, Yokell DL, Normandin MD, Rice PA, Jackson RN, Shoup TM, Brady TJ, Fakhri GE, Collier TL, Vasdev N. First Human Use of a Radiopharmaceutical Prepared by Continuous-Flow Microfluidic Radiofluorination: Proof of Concept with the Tau Imaging Agent [(18)F]T807. Molecular Imaging. 13: 7290201400025. PMID 28650281 DOI: 10.2310/7290.2014.00025  1
2014 Liang SH, Yokell DL, Jackson RN, Rice PA, Callahan R, Johnson KA, Alagille D, Tamagnan G, Collier TL, Vasdev N. Microfluidic continuous-flow radiosynthesis of [(18)F]FPEB suitable for human PET imaging. Medchemcomm. 5: 432-435. PMID 25431646 DOI: 10.1039/C3Md00335C  1
2014 Liang SH, Yokell DL, Normandin MD, Rice PA, Jackson RN, Shoup TM, Brady TJ, El Fakhri G, Collier TL, Vasdev N. First human use of a radiopharmaceutical prepared by continuous-flow microfluidic radiofluorination: proof of concept with the tau imaging agent [18F]T807. Molecular Imaging. 13. PMID 25248283 DOI: 10.2310/7290.2014.00025  1
2014 Liang SH, Vasdev N. C(sp³)-¹⁸F bond formation by transition-metal-based [¹⁸F]fluorination. Angewandte Chemie (International Ed. in English). 53: 11416-8. PMID 25243361 DOI: 10.1002/Anie.201407065  1
2014 Rotstein BH, Stephenson NA, Vasdev N, Liang SH. Spirocyclic hypervalent iodine(III)-mediated radiofluorination of non-activated and hindered aromatics. Nature Communications. 5: 4365. PMID 25007318 DOI: 10.1038/Ncomms5365  1
2014 Rotstein BH, Wey HY, Shoup TM, Wilson AA, Liang SH, Hooker JM, Vasdev N. PET imaging of fatty acid amide hydrolase with [(18)F]DOPP in nonhuman primates. Molecular Pharmaceutics. 11: 3832-8. PMID 25004399 DOI: 10.1021/Mp500316H  1
2014 Hicks JW, Parkes J, Tong J, Houle S, Vasdev N, Wilson AA. Radiosynthesis and ex vivo evaluation of [(11)C-carbonyl]carbamate- and urea-based monoacylglycerol lipase inhibitors. Nuclear Medicine and Biology. 41: 688-94. PMID 24969632 DOI: 10.1016/J.Nucmedbio.2014.05.001  1
2014 Rotstein BH, Hooker JM, Woo J, Collier TL, Brady TJ, Liang SH, Vasdev N. Synthesis of [(11)C]Bexarotene by Cu-Mediated [(11)C]Carbon Dioxide Fixation and Preliminary PET Imaging. Acs Medicinal Chemistry Letters. 5: 668-72. PMID 24944741 DOI: 10.1021/Ml500065Q  1
2014 Holland JP, Vasdev N. Charting the mechanism and reactivity of zirconium oxalate with hydroxamate ligands using density functional theory: implications in new chelate design. Dalton Transactions (Cambridge, England : 2003). 43: 9872-84. PMID 24722728 DOI: 10.1039/C4Dt00733F  1
2014 Rusjan PM, Wilson AA, Miler L, Fan I, Mizrahi R, Houle S, Vasdev N, Meyer JH. Kinetic modeling of the monoamine oxidase B radioligand [¹¹C]SL25.1188 in human brain with high-resolution positron emission tomography. Journal of Cerebral Blood Flow and Metabolism : Official Journal of the International Society of Cerebral Blood Flow and Metabolism. 34: 883-9. PMID 24517979 DOI: 10.1038/Jcbfm.2014.34  1
2014 Holland JP, Liang SH, Rotstein BH, Collier TL, Stephenson NA, Greguric I, Vasdev N. Alternative approaches for PET radiotracer development in Alzheimer's disease: imaging beyond plaque. Journal of Labelled Compounds & Radiopharmaceuticals. 57: 323-31. PMID 24327420 DOI: 10.1002/Jlcr.3158  1
2014 Shoup TM, McCauley JP, Lee DF, Chen R, Normandin MD, Bonab AA, El Fakhri G, Vasdev N. Synthesis of the dopamine D2/D3 receptor agonist (+)-PHNO via supercritical fluid chromatography: Preliminary PET imaging study with [3-11C]-(+)PHNO Tetrahedron Letters. 55: 682-685. DOI: 10.1016/J.Tetlet.2013.11.113  1
2014 Johnson KA, Schultz A, Becker A, Hyman B, Rentz D, Sepulcre J, Vasdev N, Sperling R, Brady T. Tau Pet Using F18-T807: Initial Experience In Normal Elderly And Ad Dementia Alzheimers & Dementia. 10: 242. DOI: 10.1016/J.Jalz.2014.04.365  1
2014 Liang SH, Vasdev N. C(sp3)-18F-Bindungsbildung durch übergangsmetallvermittelte [18F]Fluorierung Angewandte Chemie. 126: 11600-11602. DOI: 10.1002/Ange.201407065  1
2013 Shoup TM, Yokell DL, Rice PA, Jackson RN, Livni E, Johnson KA, Brady TJ, Vasdev N. A concise radiosynthesis of the tau radiopharmaceutical, [(18) F]T807. Journal of Labelled Compounds & Radiopharmaceuticals. 56: 736-40. PMID 24339014 DOI: 10.1002/Jlcr.3098  1
2013 Liang SH, Collier TL, Rotstein BH, Lewis R, Steck M, Vasdev N. Rapid microfluidic flow hydrogenation for reduction or deprotection of 18F-labeled compounds. Chemical Communications (Cambridge, England). 49: 8755-7. PMID 23948863 DOI: 10.1039/C3Cc45166F  1
2013 Hicks JW, Parkes J, Sadovski O, Tong J, Houle S, Vasdev N, Wilson AA. Synthesis and preclinical evaluation of [11C-carbonyl]PF-04457845 for neuroimaging of fatty acid amide hydrolase. Nuclear Medicine and Biology. 40: 740-6. PMID 23731552 DOI: 10.1016/J.Nucmedbio.2013.04.008  1
2013 Sadovski O, Hicks JW, Parkes J, Raymond R, Nobrega J, Houle S, Cipriano M, Fowler CJ, Vasdev N, Wilson AA. Development and characterization of a promising fluorine-18 labelled radiopharmaceutical for in vivo imaging of fatty acid amide hydrolase. Bioorganic & Medicinal Chemistry. 21: 4351-7. PMID 23712084 DOI: 10.1016/J.Bmc.2013.04.077  1
2013 Rotstein BH, Liang SH, Holland JP, Collier TL, Hooker JM, Wilson AA, Vasdev N. 11CO2 fixation: a renaissance in PET radiochemistry. Chemical Communications (Cambridge, England). 49: 5621-9. PMID 23673726 DOI: 10.1039/C3Cc42236D  1
2013 Holland JP, Cumming P, Vasdev N. PET radiopharmaceuticals for probing enzymes in the brain. American Journal of Nuclear Medicine and Molecular Imaging. 3: 194-216. PMID 23638333  1
2013 Vasdev N, Green DE, Vines DC, McLarty K, McCormick PN, Moran MD, Houle S, Wilson AA, Reilly RM. Positron-emission tomography imaging of the TSPO with [18F]FEPPA in a preclinical breast cancer model Cancer Biotherapy and Radiopharmaceuticals. 28: 254-259. PMID 23350894 DOI: 10.1089/Cbr.2012.1196  1
2013 Wilson AA, Hicks JW, Sadovski O, Parkes J, Tong J, Houle S, Fowler CJ, Vasdev N. Radiosynthesis and evaluation of [¹¹C-carbonyl]-labeled carbamates as fatty acid amide hydrolase radiotracers for positron emission tomography. Journal of Medicinal Chemistry. 56: 201-9. PMID 23214511 DOI: 10.1021/Jm301492Y  1
2012 Carroll L, Perumal M, Vasdev N, Robins E, Aboagye EO. Radiosynthesis and in vivo tumor uptake of 2-deoxy-2-[(18)F]fluoro-myo-inositol. Bioorganic & Medicinal Chemistry Letters. 22: 6148-50. PMID 22944120 DOI: 10.1016/J.Bmcl.2012.08.022  1
2012 Holland JP, Cumming P, Vasdev N. PET of signal transduction pathways in cancer. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 53: 1333-6. PMID 22879078 DOI: 10.2967/Jnumed.112.105387  1
2012 Moran MD, Wilson AA, Elmore CS, Parkes J, Ng A, Sadovski O, Graff A, Daskalakis ZJ, Houle S, Chapdelaine MJ, Vasdev N. Development of new carbon-11 labelled radiotracers for imaging GABA A- and GABA B-benzodiazepine receptors Bioorganic and Medicinal Chemistry. 20: 4482-4488. PMID 22717238 DOI: 10.1016/J.Bmc.2012.05.046  1
2012 Hicks JW, Wilson AA, Rubie EA, Woodgett JR, Houle S, Vasdev N. Towards the preparation of radiolabeled 1-aryl-3-benzyl ureas: Radiosynthesis of [(11)C-carbonyl] AR-A014418 by [(11)C]CO(2) fixation. Bioorganic & Medicinal Chemistry Letters. 22: 2099-101. PMID 22321216 DOI: 10.1016/J.Bmcl.2011.12.139  1
2012 Vasdev N, Cao P, Oosten EMV, Wilson AA, Houle S, Hao G, Sun X, Slavine NV, Alhasan M, Antich PP, Bonte FJ, Kulkarni PV. Synthesis and PET imaging studies of [18F]2-fluoroquinolin-8-ol ([18F]CABS13) in transgenic mouse models of Alzheimer's disease Medchemcomm. 3: 1228-1230. DOI: 10.1039/C2Md20075A  1
2012 Kulkarni P, Alhasan M, Slavine N, Chiguru S, Hao G, Vasdev N, Thomas P, Bonte F, Sun X. Assessment of disease progression in Alzheimer's transgenic mice by PET imaging with F-18 quinoline Alzheimers & Dementia. 8: 155. DOI: 10.1016/J.Jalz.2012.05.417  0.01
2011 Hicks JW, Lough AJ, Wilson AA, Vasdev N. (E)-2-(2-Methyl-cyclo-hexyl-idene)hydrazinecarbothio-amide. Acta Crystallographica. Section E, Structure Reports Online. 67: o3005. PMID 22220022 DOI: 10.1107/S1600536811042486  1
2011 McLarty K, Moran MD, Scollard DA, Chan C, Sabha N, Mukherjee J, Guha A, McLaurin J, Nitz M, Houle S, Wilson AA, Reilly RM, Vasdev N. Comparisons of [18F]-1-deoxy-1-fluoro-scyllo-inositol with [18F]-FDG for PET imaging of inflammation, breast and brain cancer xenografts in athymic mice. Nuclear Medicine and Biology. 38: 953-9. PMID 21982567 DOI: 10.1016/J.Nucmedbio.2011.02.017  1
2011 Vasdev N, Sadovski O, Moran MD, Parkes J, Meyer JH, Houle S, Wilson AA. Development of new radiopharmaceuticals for imaging monoamine oxidase B. Nuclear Medicine and Biology. 38: 933-43. PMID 21982565 DOI: 10.1016/J.Nucmedbio.2011.03.003  1
2011 Stephenson KA, Wilson AA, Houle S, Vasdev N. Synthesis and in vitro evaluation of derivatives of the β₁-adrenergic receptor antagonist HX-CH 44. Bioorganic & Medicinal Chemistry Letters. 21: 5506-9. PMID 21783363 DOI: 10.1016/J.Bmcl.2011.06.106  1
2011 Vasdev N, Dorff PN, O'Neil JP, Chin FT, Hanrahan S, VanBrocklin HF. Metabolic stability of 6,7-dialkoxy-4-(2-, 3- and 4-[18F]fluoroanilino)quinazolines, potential EGFR imaging probes. Bioorganic & Medicinal Chemistry. 19: 2959-65. PMID 21478021 DOI: 10.1016/J.Bmc.2011.03.032  1
2011 Louie AS, Vasdev N, Valliant JF. Preparation, characterization, and screening of a high affinity organometallic probe for α-adrenergic receptors. Journal of Medicinal Chemistry. 54: 3360-7. PMID 21428421 DOI: 10.1021/Jm2001162  1
2011 Wilson AA, Garcia A, Parkes J, Houle S, Tong J, Vasdev N. [11C]CURB: Evaluation of a novel radiotracer for imaging fatty acid amide hydrolase by positron emission tomography. Nuclear Medicine and Biology. 38: 247-53. PMID 21315280 DOI: 10.1016/J.Nucmedbio.2010.08.001  1
2011 Wilson AA, Garcia A, Houle S, Sadovski O, Vasdev N. Synthesis and application of isocyanates radiolabeled with carbon-11. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 259-64. PMID 21207622 DOI: 10.1002/Chem.201002345  1
2011 Van Oosten EM, Gerken M, Hazendonk P, Shank R, Houle S, Wilson AA, Vasdev N. Regioselective ring opening of 2-methylaziridine derivatives with 18F- and 19F-fluoride Tetrahedron Letters. 52: 4114-4116. DOI: 10.1016/J.Tetlet.2011.05.139  1
2011 Kulkarni P, Arora V, Chiguru S, Hao G, Gupta A, Slavine N, Qu B, Vasdev N, Sun X, Bennett M, Antich P, Bonte F. PET imaging of Alzheimer's transgenic mice at an early age with F-18 quinoline Alzheimers & Dementia. 7. DOI: 10.1016/J.Jalz.2011.05.021  0.01
2011 Vasdev N, Sadovski O, Garcia A, Dollé F, Meyer JH, Houle S, Wilson AA. Radiosynthesis of [11C]SL25.1188 via [11C]CO2 fixation for imaging monoamine oxidase B Journal of Labelled Compounds and Radiopharmaceuticals. 54: 678-680. DOI: 10.1002/Jlcr.1908  1
2011 Moran MD, Wilson AA, Stableford WT, Wong M, Garcia A, Houle S, Vasdev N. A rapid one-step radiosynthesis of [11C]-d-threo-methylphenidate Journal of Labelled Compounds and Radiopharmaceuticals. 54: 168-170. DOI: 10.1002/Jlcr.1824  1
2010 Lough AJ, Hicks JW, Valliant JF, Wilson AA, Vasdev N. N-(4-Meth-oxy-phen-yl)-N'-(5-nitro-1,3-thia-zol-2-yl)urea. Acta Crystallographica. Section E, Structure Reports Online. 66: o2339. PMID 21588684 DOI: 10.1107/S1600536810032186  1
2010 Hicks JW, VanBrocklin HF, Wilson AA, Houle S, Vasdev N. Radiolabeled small molecule protein kinase inhibitors for imaging with PET or SPECT. Molecules (Basel, Switzerland). 15: 8260-78. PMID 21079565 DOI: 10.3390/Molecules15118260  1
2010 Vasdev N, Moran MD, Tuononen HM, Chirakal R, Suontamo RJ, Bain AD, Schrobilgen GJ. NMR spectroscopic evidence for the intermediacy of XeF(3)(-) in XeF(2)/F(-) exchange, attempted syntheses and thermochemistry of XeF(3)(-) salts, and theoretical studies of the XeF(3)(-) anion. Inorganic Chemistry. 49: 8997-9004. PMID 20799721 DOI: 10.1021/Ic101275M  1
2010 Gerretsen P, Graff-Guerrero A, Menon M, Pollock BG, Kapur S, Vasdev N, Houle S, Mamo D. Is desire for social relationships mediated by the serotonergic system in the prefrontal cortex? An [(18)F]setoperone PET study. Social Neuroscience. 5: 375-83. PMID 20198536 DOI: 10.1080/17470911003589309  1
2010 Wilson AA, Garcia A, Houle S, Vasdev N. Direct fixation of [(11)C]-CO(2) by amines: formation of [(11)C-carbonyl]-methylcarbamates. Organic & Biomolecular Chemistry. 8: 428-32. PMID 20066280 DOI: 10.1039/B916419G  1
2010 Vasdev N, Sadovski O, Parkes J, Moran MD, Meyer JH, Houle S, Wilson AA. Development of New PET radiopharmaceuticals for imaging monoamine oxidase-B Neuroimage. 52. DOI: 10.1016/J.Neuroimage.2010.04.201  1
2010 Kulkarni PV, Vasdev N, Arora V, Hao G, Long M, Slavine N, Qu B, Sun X, Bennett M, Antich PP, Bonte FJ. PET imaging of Alzheimer's disease (AD) transgenic mice with F-18 labeled 8-hydroxy quinoline Alzheimers & Dementia. 6. DOI: 10.1016/J.Jalz.2010.05.017  0.01
2009 Vasdev N, Chio J, van Oosten EM, Nitz M, McLaurin J, Vines DC, Houle S, Reilly RM, Wilson AA. Synthesis and preliminary biological evaluations of [18F]-1-deoxy-1-fluoro-scyllo-inositol. Chemical Communications (Cambridge, England). 5527-9. PMID 19753345 DOI: 10.1039/B913317H  1
2009 van Oosten EM, Wilson AA, Stephenson KA, Mamo DC, Pollock BG, Mulsant BH, Yudin AK, Houle S, Vasdev N. An improved radiosynthesis of the muscarinic M2 radiopharmaceutical, [18F]FP-TZTP. Applied Radiation and Isotopes : Including Data, Instrumentation and Methods For Use in Agriculture, Industry and Medicine. 67: 611-6. PMID 19186063 DOI: 10.1016/J.Apradiso.2008.12.015  1
2009 Vasdev N, van Oosten EM, Stephenson KA, Zadikian N, Yudin AK, Lough AJ, Houle S, Wilson AA. [18F]Fluoroamines via ring-opening of N-Cbz-2-methylaziridine with [18F]-fluoride Tetrahedron Letters. 50: 544-547. DOI: 10.1016/J.Tetlet.2008.11.074  1
2009 Wilson AA, Garcia A, Houle S, Vasdev N. Utility of commercial radiosynthetic modules in captive solvent [11C]‐methylation reactions Journal of Labelled Compounds and Radiopharmaceuticals. 52: 490-492. DOI: 10.1002/Jlcr.1618  1
2008 Vasdev N, Kulkarni PV, Wilson AA, Houle S, Lough AJ. 4-Bromo-8-methoxy-quinoline. Acta Crystallographica. Section E, Structure Reports Online. 64: o1117. PMID 21202628 DOI: 10.1107/S1600536808014591  1
2008 van Oosten EM, Lough AJ, Vasdev N. N-Isopropyl-benzamide. Acta Crystallographica. Section E, Structure Reports Online. 64: o1005. PMID 21202531 DOI: 10.1107/S1600536808012804  1
2008 Stephenson KA, van Oosten EM, Wilson AA, Meyer JH, Houle S, Vasdev N. Synthesis and preliminary evaluation of [(18)F]-fluoro-(2S)-Exaprolol for imaging cerebral beta-adrenergic receptors with PET. Neurochemistry International. 53: 173-9. PMID 18675864 DOI: 10.1016/J.Neuint.2008.06.013  1
2008 Stephenson KA, Wilson AA, Meyer JH, Houle S, Vasdev N. Facile radiosynthesis of fluorine-18 labeled beta-blockers. Synthesis, radiolabeling, and ex vivo biodistribution of [18F]-(2S and 2R)-1-(1-fluoropropan-2-ylamino)-3-(m-tolyloxy)propan-2-ol. Journal of Medicinal Chemistry. 51: 5093-100. PMID 18656910 DOI: 10.1021/Jm800227H  1
2008 Wilson AA, Garcia A, Parkes J, McCormick P, Stephenson KA, Houle S, Vasdev N. Radiosynthesis and initial evaluation of [18F]-FEPPA for PET imaging of peripheral benzodiazepine receptors. Nuclear Medicine and Biology. 35: 305-14. PMID 18355686 DOI: 10.1016/J.Nucmedbio.2007.12.009  1
2008 Vasdev N, LaRonde FJ, Woodgett JR, Garcia A, Rubie EA, Meyer JH, Houle S, Wilson AA. Rationally designed PKA inhibitors for positron emission tomography: Synthesis and cerebral biodistribution of N-(2-(4-bromocinnamylamino)ethyl)-N-[11C]methyl-isoquinoline-5-sulfonamide. Bioorganic & Medicinal Chemistry. 16: 5277-84. PMID 18346896 DOI: 10.1016/J.Bmc.2008.03.013  1
2008 Vasdev N, Stephenson KA, Oosten EMv, Meyer JH, Houle S, Wilson AA. Recent advances towards imaging cerebral β-adrenergic receptors with PET Neuroimage. 41. DOI: 10.1016/J.Neuroimage.2008.04.165  1
2007 Vasdev N, Seeman P, Garcia A, Stableford WT, Nobrega JN, Houle S, Wilson AA. Syntheses and in vitro evaluation of fluorinated naphthoxazines as dopamine D2/D3 receptor agonists: radiosynthesis, ex vivo biodistribution and autoradiography of [(18)F]F-PHNO. Nuclear Medicine and Biology. 34: 195-203. PMID 17307127 DOI: 10.1016/J.Nucmedbio.2006.11.001  1
2007 Vasdev N, Wilson AA, Houle S, Lough AJ. N‐(4‐Methoxy­benz­yl)‐N′‐(5‐nitro‐1,3‐thia­zol‐2‐yl)urea (AR‐A014418) Acta Crystallographica Section E-Structure Reports Online. 63. DOI: 10.1107/S1600536807010215  1
2006 Vasdev N, Natesan S, Galineau L, Garcia A, Stableford WT, McCormick P, Seeman P, Houle S, Wilson AA. Radiosynthesis, ex vivo and in vivo evaluation of [11C]preclamol as a partial dopamine D2 agonist radioligand for positron emission tomography. Synapse (New York, N.Y.). 60: 314-8. PMID 16786538 DOI: 10.1002/Syn.20304  1
2006 McCormick PN, Ginovart N, Vasdev N, Seeman P, Kapur S, Wilson AA. Isoflurane increases both the specific binding ratio and sensitivity to amphetamine challenge of [11C]-(+)-PHNO Neuroimage. 31. DOI: 10.1016/J.Neuroimage.2006.04.023  1
2005 Vasdev N, Garcia A, Stableford WT, Young AB, Meyer JH, Houle S, Wilson AA. Synthesis and ex vivo evaluation of carbon-11 labelled N-(4-methoxybenzyl)-N'-(5-nitro-1,3-thiazol-2-yl)urea ([11C]AR-A014418): a radiolabelled glycogen synthase kinase-3beta specific inhibitor for PET studies. Bioorganic & Medicinal Chemistry Letters. 15: 5270-3. PMID 16202587 DOI: 10.1016/J.Bmcl.2005.08.037  1
2005 Vasdev N, Dorff PN, Gibbs AR, Nandanan E, Reid LM, O'Neil JP, VanBrocklin HF. Synthesis of 6-acrylamido-4-(2-[18F]fluoroanilino)quinazoline: A prospective irreversible EGFR binding probe Journal of Labelled Compounds and Radiopharmaceuticals. 48: 109-115. DOI: 10.1002/Jlcr.903  1
2003 Vasdev N, Chirakal R, Ashique R, Schrobilgen GJ, Gulenchyn K. Syntheses of [18F]5-fluoro-3-nitro-L-tyrosine Journal of Fluorine Chemistry. 121: 9-14. DOI: 10.1016/S0022-1139(02)00334-2  1
2002 Vasdev N, Pointner BE, Chirakal R, Schrobilgen GJ. On the preparation of fluorine-18 labelled XeF(2) and chemical exchange between fluoride ion and XeF(2). Journal of the American Chemical Society. 124: 12863-8. PMID 12392433 DOI: 10.1021/Ja020604Y  1
2002 Vasdev N, Pointner BE, Chirakal R, Schrobilgen GJ. On the preparation of fluorine-18 labelled XeF2 and chemical exchange between fluoride ion and XeF2 Journal of the American Chemical Society. 124: 12863-12868. DOI: 10.1021/ja020604y  1
2002 Chirakal R, Vasdev N, Asselin MC, Schrobilgen GJ, Nahmias C. The effect of aromatic fluorine substitution in L-DOPA on the in vivo behaviour of [18F]2-, [18F]5- and [18F]6-fluoro-L-DOPA in the human brain Journal of Fluorine Chemistry. 115: 33-39. DOI: 10.1016/S0022-1139(02)00025-8  1
2001 Vasdev N, Chirakal R, Schrobilgen GJ, Nahmias C. Selectivity of elemental fluorine towards L-tyrosine and L-α-methyltyrosine in acidic media and the syntheses of their [18F]3-fluoro and [18F]3,5-difluoro derivatives Journal of Fluorine Chemistry. 111: 17-25. DOI: 10.1016/S0022-1139(01)00406-7  1
1999 Chirakal R, Vasdev N, Schrobilgen GJ, Nahmias C. Radiochemical and NMR spectroscopic investigation of the solvent effect on the electrophilic elemental fluorination of L-DOPA: Synthesis of [ 18F ]5-fluoro-L-DOPA Journal of Fluorine Chemistry. 99: 87-94. DOI: 10.1016/S0022-1139(99)00123-2  1
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