| Year |
Citation |
Score |
| 2022 |
Cunningham MJ, Bock HA, Serrano IC, Bechand B, Vidyadhara DJ, Bonniwell EM, Lankri D, Duggan P, Nazarova AL, Cao AB, Calkins MM, Khirsariya P, Hwu C, Katritch V, Chandra SS, ... ... Sames D, et al. Pharmacological Mechanism of the Non-hallucinogenic 5-HT Agonist Ariadne and Analogs. Acs Chemical Neuroscience. PMID 36521179 DOI: 10.1021/acschemneuro.2c00597 |
0.76 |
|
| 2022 |
Pazos M, Dibello E, Mesa JM, Sames D, Comini MA, Seoane G, Carrera I. Iboga Inspired -Indolylethyl-Substituted Isoquinuclidines as a Bioactive Scaffold: Chemoenzymatic Synthesis and Characterization as GDNF Releasers and Antitrypanosoma Agents. Molecules (Basel, Switzerland). 27. PMID 35164094 DOI: 10.3390/molecules27030829 |
0.783 |
|
| 2021 |
Bhowmik S, Galeta J, Havel V, Nelson M, Faouzi A, Bechand B, Ansonoff M, Fiala T, Hunkele A, Kruegel AC, Pintar JE, Majumdar S, Javitch JA, Sames D. Site selective C-H functionalization of Mitragyna alkaloids reveals a molecular switch for tuning opioid receptor signaling efficacy. Nature Communications. 12: 3858. PMID 34158473 DOI: 10.1038/s41467-021-23736-2 |
0.766 |
|
| 2020 |
Rodríguez P, Urbanavicius J, Prieto JP, Fabius S, Reyes AL, Havel V, Sames D, Scorza C, Carrera I. A Single Administration of the Atypical Psychedelic Ibogaine or its Metabolite Noribogaine Induces an Antidepressant-like Effect in Rats. Acs Chemical Neuroscience. PMID 32330007 DOI: 10.1021/Acschemneuro.0C00152 |
0.664 |
|
| 2019 |
Marton S, González B, Rodríguez-Bottero S, Miquel E, Martínez-Palma L, Pazos M, Prieto JP, Rodríguez P, Sames D, Seoane G, Scorza C, Cassina P, Carrera I. Ibogaine Administration Modifies GDNF and BDNF Expression in Brain Regions Involved in Mesocorticolimbic and Nigral Dopaminergic Circuits. Frontiers in Pharmacology. 10: 193. PMID 30890941 DOI: 10.3389/Fphar.2019.00193 |
0.762 |
|
| 2017 |
Henke A, Kovalyova Y, Dunn M, Dreier D, Gubernator NG, Dincheva I, Hwu C, Sebej P, Ansorge MS, Sulzer D, Sames D. Toward Serotonin Fluorescent False Neurotransmitters: Development of Fluorescent Dual Serotonin and Vesicular Monoamine Transporter Substrates for Visualizing Serotonin Neurons. Acs Chemical Neuroscience. PMID 29281252 DOI: 10.1021/Acschemneuro.7B00320 |
0.309 |
|
| 2017 |
Boltaev U, Meyer Y, Tolibzoda F, Jacques T, Gassaway M, Xu Q, Wagner F, Zhang YL, Palmer M, Holson E, Sames D. Multiplex quantitative assays indicate a need for reevaluating reported small-molecule TrkB agonists. Science Signaling. 10. PMID 28831019 DOI: 10.1126/Scisignal.Aal1670 |
0.768 |
|
| 2016 |
Genovino J, Sames D, Hamann LG, Touré BB. Accessing Drug Metabolites via Transition-Metal Catalyzed C-H Oxidation: Liver as Synthetic Inspiration. Angewandte Chemie (International Ed. in English). PMID 27723189 DOI: 10.1002/Anie.201602644 |
0.308 |
|
| 2016 |
Pereira DB, Schmitz Y, Mészáros J, Merchant P, Hu G, Li S, Henke A, Lizardi-Ortiz JE, Karpowicz RJ, Morgenstern TJ, Sonders MS, Kanter E, Rodriguez PC, Mosharov EV, Sames D, et al. Fluorescent false neurotransmitter reveals functionally silent dopamine vesicle clusters in the striatum. Nature Neuroscience. PMID 26900925 DOI: 10.1038/Nn.4252 |
0.634 |
|
| 2016 |
Genovino J, Sames D, Hamann LG, Touré BB. Die Erschließung von Wirkstoffmetaboliten durch übergangsmetallkatalysierte C-H-Oxidation: die Leber als Inspiration für die Synthese Angewandte Chemie. 128: 14430-14451. DOI: 10.1002/Ange.201602644 |
0.318 |
|
| 2015 |
Gassaway MM, Jacques TL, Kruegel AC, Karpowicz RJ, Li X, Li S, Myer Y, Sames D. Deconstructing the Iboga Alkaloid Skeleton: Potentiation of FGF2-induced Glial Cell Line-Derived Neurotrophic Factor Release by a Novel Compound. Acs Chemical Biology. PMID 26517751 DOI: 10.1021/Acschembio.5B00678 |
0.772 |
|
| 2015 |
Kruegel AC, Rakshit S, Li X, Sames D. Constructing Iboga alkaloids via C-H bond functionalization: examination of the direct and catalytic union of heteroarenes and isoquinuclidine alkenes. The Journal of Organic Chemistry. 80: 2062-71. PMID 25633249 DOI: 10.1021/Jo5018102 |
0.409 |
|
| 2014 |
Genovino J, Sames D, Touré BB. Access to drug metabolites via C-H functionalization: Copper-catalyzed aerobic oxidation of N,N-dimethylalkylamines in complex pharmaceuticals Tetrahedron Letters. DOI: 10.1016/J.Tetlet.2014.11.037 |
0.308 |
|
| 2013 |
Genovino J, Lütz S, Sames D, Touré BB. Complementation of biotransformations with chemical C-H oxidation: copper-catalyzed oxidation of tertiary amines in complex pharmaceuticals. Journal of the American Chemical Society. 135: 12346-52. PMID 23875728 DOI: 10.1021/Ja405471H |
0.342 |
|
| 2013 |
Hu G, Henke A, Karpowicz RJ, Sonders MS, Farrimond F, Edwards R, Sulzer D, Sames D. New fluorescent substrate enables quantitative and high-throughput examination of vesicular monoamine transporter 2 (VMAT2). Acs Chemical Biology. 8: 1947-54. PMID 23859623 DOI: 10.1021/Cb400259N |
0.351 |
|
| 2013 |
Karpowicz RJ, Dunn M, Sulzer D, Sames D. APP+, a fluorescent analogue of the neurotoxin MPP+, is a marker of catecholamine neurons in brain tissue, but not a fluorescent false neurotransmitter. Acs Chemical Neuroscience. 4: 858-69. PMID 23647019 DOI: 10.1021/Cn400038U |
0.311 |
|
| 2013 |
Rodriguez PC, Pereira DB, Borgkvist A, Wong MY, Barnard C, Sonders MS, Zhang H, Sames D, Sulzer D. Fluorescent dopamine tracer resolves individual dopaminergic synapses and their activity in the brain. Proceedings of the National Academy of Sciences of the United States of America. 110: 870-5. PMID 23277566 DOI: 10.1073/Pnas.1213569110 |
0.646 |
|
| 2013 |
Joo JM, Guo P, Sames D. C-H bonds as ubiquitous functionality: preparation of multiple regioisomers of arylated 1,2,4-triazoles via C-H arylation. The Journal of Organic Chemistry. 78: 738-43. PMID 23276283 DOI: 10.1021/Jo3021677 |
0.414 |
|
| 2012 |
Vadola PA, Sames D. Catalytic coupling of arene C-H bonds and alkynes for the synthesis of coumarins: substrate scope and application to the development of neuroimaging agents. The Journal of Organic Chemistry. 77: 7804-14. PMID 22768913 DOI: 10.1021/Jo3006842 |
0.807 |
|
| 2012 |
Vadola PA, Carrera I, Sames D. C-H bond functionalization via hydride transfer: formation of α-arylated piperidines and 1,2,3,4-tetrahydroisoquinolines via stereoselective intramolecular amination of benzylic C-H bonds. The Journal of Organic Chemistry. 77: 6689-702. PMID 22672002 DOI: 10.1021/Jo300635M |
0.787 |
|
| 2011 |
Guo P, Joo JM, Rakshit S, Sames D. C-H arylation of pyridines: high regioselectivity as a consequence of the electronic character of C-H bonds and heteroarene ring. Journal of the American Chemical Society. 133: 16338-41. PMID 21939181 DOI: 10.1021/Ja206022P |
0.415 |
|
| 2011 |
Lee M, Tremblay MS, Jockusch S, Turro NJ, Sames D. Intermolecular energy transfer from Tb3+ to Eu3+ in aqueous aggregates and on the surface of human cells. Organic Letters. 13: 2802-5. PMID 21563789 DOI: 10.1021/Ol200328P |
0.597 |
|
| 2010 |
Rodriguez PC, Yee DJ, Sames D. Expanding the use of fluorogenic enzyme reporter substrates to imaging metabolic flux changes: the activity measurement of 5α-steroid reductase in intact mammalian cells. Acs Chemical Biology. 5: 1045-52. PMID 20863068 DOI: 10.1021/Cb100196N |
0.777 |
|
| 2010 |
Muirhead KE, Froemming M, Li X, Musilek K, Conway SJ, Sames D, Gunn-Moore FJ. (-)-CHANA, a fluorogenic probe for detecting amyloid binding alcohol dehydrogenase HSD10 activity in living cells. Acs Chemical Biology. 5: 1105-14. PMID 20836522 DOI: 10.1021/Cb100199M |
0.765 |
|
| 2010 |
Joo JM, Touré BB, Sames D. C-H bonds as ubiquitous functionality: a general approach to complex arylated imidazoles via regioselective sequential arylation of all three C-H bonds and regioselective N-alkylation enabled by SEM-group transposition. The Journal of Organic Chemistry. 75: 4911-20. PMID 20608749 DOI: 10.1021/Jo100727J |
0.425 |
|
| 2010 |
Lee M, Gubernator NG, Sulzer D, Sames D. Development of pH-responsive fluorescent false neurotransmitters. Journal of the American Chemical Society. 132: 8828-30. PMID 20540519 DOI: 10.1021/Ja101740K |
0.446 |
|
| 2010 |
SAMES D, POLT R. ChemInform Abstract: Piperidine Triols via Enantioselective Alkylation and Osmylation of Alanine Schiff Base Esters. Cheminform. 26: no-no. DOI: 10.1002/CHIN.199540222 |
0.567 |
|
| 2009 |
Vadola PA, Sames D. C-H bond functionalization via hydride transfer: direct coupling of unactivated alkynes and sp(3) C-H bonds catalyzed by platinum tetraiodide. Journal of the American Chemical Society. 131: 16525-8. PMID 19852462 DOI: 10.1021/Ja906480W |
0.804 |
|
| 2009 |
Zhang H, Gubernator NG, Yue M, Staal RG, Mosharov EV, Pereira D, Balsanek V, Vadola PA, Mukherjee B, Edwards RH, Sulzer D, Sames D. Dopamine release at individual presynaptic terminals visualized with FFNs. Journal of Visualized Experiments : Jove. PMID 19721412 DOI: 10.3791/1562 |
0.75 |
|
| 2009 |
McQuaid KM, Long JZ, Sames D. C-H bond functionalization via hydride transfer: synthesis of dihydrobenzopyrans from ortho-vinylaryl akyl ethers. Organic Letters. 11: 2972-5. PMID 19548698 DOI: 10.1021/Ol900915P |
0.729 |
|
| 2009 |
Gubernator NG, Zhang H, Staal RG, Mosharov EV, Pereira DB, Yue M, Balsanek V, Vadola PA, Mukherjee B, Edwards RH, Sulzer D, Sames D. Fluorescent false neurotransmitters visualize dopamine release from individual presynaptic terminals. Science (New York, N.Y.). 324: 1441-4. PMID 19423778 DOI: 10.1126/Science.1172278 |
0.751 |
|
| 2009 |
Goikhman R, Jacques TL, Sames D. C-H bonds as ubiquitous functionality: a general approach to complex arylated pyrazoles via sequential regioselective C-arylation and N-alkylation enabled by SEM-group transposition. Journal of the American Chemical Society. 131: 3042-8. PMID 19206533 DOI: 10.1021/Ja8096114 |
0.802 |
|
| 2009 |
McQuaid KM, Sames D. C-H bond functionalization via hydride transfer: Lewis acid catalyzed alkylation reactions by direct intramolecular coupling of sp3 C-H bonds and reactive alkenyl oxocarbenium intermediates. Journal of the American Chemical Society. 131: 402-3. PMID 19099474 DOI: 10.1021/Ja806068H |
0.743 |
|
| 2008 |
Halim M, Yee DJ, Sames D. Imaging induction of cytoprotective enzymes in intact human cells: coumberone, a metabolic reporter for human AKR1C enzymes reveals activation by panaxytriol, an active component of red ginseng. Journal of the American Chemical Society. 130: 14123-8. PMID 18826220 DOI: 10.1021/Ja801245Y |
0.784 |
|
| 2008 |
Tremblay MS, Lee M, Sames D. A luminescent sensor for tyrosine phosphorylation. Organic Letters. 10: 5-8. PMID 18069839 DOI: 10.1021/Ol701920X |
0.595 |
|
| 2007 |
Froemming MK, Sames D. Harnessing functional plasticity of enzymes: a fluorogenic probe for imaging 17beta-HSD10 dehydrogenase, an enzyme involved in Alzheimer's and Parkinson's diseases. Journal of the American Chemical Society. 129: 14518-22. PMID 17958419 DOI: 10.1021/Ja072601X |
0.767 |
|
| 2007 |
Gribkov DV, Pastine SJ, Schnürch M, Sames D. Ruthenium catalyzed decarbonylative arylation at sp3 carbon centers in pyrrolidine and piperidine heterocycles. Journal of the American Chemical Society. 129: 11750-5. PMID 17803274 DOI: 10.1021/Ja072577N |
0.754 |
|
| 2007 |
Halim M, Tremblay MS, Jockusch S, Turro NJ, Sames D. Transposing molecular fluorescent switches into the near-IR: development of luminogenic reporter substrates for redox metabolism. Journal of the American Chemical Society. 129: 7704-5. PMID 17542585 DOI: 10.1021/Ja071311D |
0.584 |
|
| 2007 |
Tremblay MS, Halim M, Sames D. Cocktails of Tb(3+) and Eu(3+) complexes: a general platform for the design of ratiometric optical probes. Journal of the American Chemical Society. 129: 7570-7. PMID 17518468 DOI: 10.1021/Ja070867Y |
0.536 |
|
| 2007 |
Wang X, Gribkov DV, Sames D. Phosphine-free palladium-catalyzed C-H bond arylation of free (N-H)-indoles and pyrroles. The Journal of Organic Chemistry. 72: 1476-9. PMID 17288392 DOI: 10.1021/Jo061979V |
0.388 |
|
| 2007 |
Sames D, Pastine S, Gribkov D. trans-Selective sp3 C-H Bond Arylation of Pyrrolidines and Piperidines Synfacts. 2007: 0181-0181. DOI: 10.1055/s-2006-955850 |
0.709 |
|
| 2007 |
Jockusch S, Zheng Q, He GS, Pudavar HE, Yee DJ, Balsanek V, Halim M, Sames D, Prasad PN, Turro NJ. Two-photon excitation of fluorogenic probes for redox metabolism: Dramatic enhancement of optical contrast ratio by two-photon excitation Journal of Physical Chemistry C. 111: 8872-8877. DOI: 10.1021/Jp067430H |
0.77 |
|
| 2007 |
Lane BS, Brown aMA, Sames D. Direct Palladium-Catalyzed C-2 and C-3 Arylation of Indoles: A Mechanistic Rationale for Regioselectivity [J. Am. Chem. Soc. 2005, 127, 8050−8057]. Journal of the American Chemical Society. 129: 241-241. DOI: 10.1021/Ja0699790 |
0.344 |
|
| 2006 |
Pastine SJ, Gribkov DV, Sames D. sp3 C-H bond arylation directed by amidine protecting group: alpha-arylation of pyrrolidines and piperidines. Journal of the American Chemical Society. 128: 14220-1. PMID 17076471 DOI: 10.1021/Ja064481J |
0.745 |
|
| 2006 |
Tremblay MS, Sames D. Synthesis of luminescent heterometallic bis-lanthanide complexes via selective, sequential metallation. Chemical Communications (Cambridge, England). 4116-8. PMID 17024267 DOI: 10.1039/B607949K |
0.53 |
|
| 2006 |
Yee DJ, Balsanek V, Bauman DR, Penning TM, Sames D. Fluorogenic metabolic probes for direct activity readout of redox enzymes: Selective measurement of human AKR1C2 in living cells. Proceedings of the National Academy of Sciences of the United States of America. 103: 13304-9. PMID 16938874 DOI: 10.1073/Pnas.0604672103 |
0.794 |
|
| 2006 |
and BS, Sames D. Diversity Synthesis via C−H Bond Functionalization: Concept-Guided Development of New C-Arylation Methods for Imidazoles [J. Am. Chem. Soc. 2003, 125, 10580−10585]. Journal of the American Chemical Society. 128: 8364-8364. PMID 16787104 DOI: 10.1021/Ja0699642 |
0.346 |
|
| 2006 |
and BS, Sames D. Selective C-Arylation of Free (NH)-Heteroarenes via Catalytic C−H Bond Functionalization [J. Am. Chem. Soc. 2003, 125, 5274−5275]. Journal of the American Chemical Society. 128: 8364-8364. PMID 16787103 DOI: 10.1021/Ja069965U |
0.356 |
|
| 2006 |
Tremblay MS, Zhu Q, Martí AA, Dyer J, Halim M, Jockusch S, Turro NJ, Sames D. Phosphorylation state-responsive lanthanide peptide conjugates: a luminescence switch based on reversible complex reorganization. Organic Letters. 8: 2723-6. PMID 16774241 DOI: 10.1021/Ol060614U |
0.532 |
|
| 2006 |
Touré BB, Lane BS, Sames D. Catalytic C-H arylation of SEM-protected azoles with palladium complexes of NHCs and phosphines. Organic Letters. 8: 1979-82. PMID 16671761 DOI: 10.1021/Ol053021C |
0.37 |
|
| 2006 |
Godula K, Sames D. C-H bond functionalization in complex organic synthesis. Science (New York, N.Y.). 312: 67-72. PMID 16601184 DOI: 10.1126/Science.1114731 |
0.706 |
|
| 2006 |
Sezen B, Sames D. Oxidative C-arylation of free (NH)-heterocycles via direct sp3 C-H bond functionalization [J. Am. Chem. Soc. 2004, 126, 13244-13246]. Journal of the American Chemical Society. 128: 3102. PMID 16506793 DOI: 10.1021/Ja069957D |
0.36 |
|
| 2006 |
Sezen B, Sames D. Selective and catalytic arylation of N-phenylpyrrolidine: (sp3) C-H bond functionalization in the absence of a directing group [J. Am. Chem. Soc. 2005, 127, 5284-5285]. Journal of the American Chemical Society. 128: 3102. PMID 16506792 DOI: 10.1021/Ja0699586 |
0.371 |
|
| 2006 |
Froemming MK, Sames D. Fluoromorphic substrates for fatty acid metabolism: highly sensitive probes for mammalian medium-chain acyl-CoA dehydrogenase. Angewandte Chemie (International Ed. in English). 45: 637-42. PMID 16365837 DOI: 10.1002/Anie.200502675 |
0.758 |
|
| 2006 |
Godula K, Sezen aB, Sames D. Site-Specific Phenylation of Pyridine Catalyzed by Phosphido-Bridged Ruthenium Dimer Complexes: A Prototype for C−H Arylation of Electron-Deficient Heteroarenes [J. Am. Chem. Soc. 2005, 127, 3648−3649]. Journal of the American Chemical Society. 128: 3102-3102. DOI: 10.1021/Ja069956L |
0.648 |
|
| 2005 |
Pastine SJ, Sames D. Room temperature intramolecular hydro-O-alkylation of aldehydes: sp3 C-H functionalization via a Lewis acid catalyzed tandem 1,5-hydride transfer/cyclization. Organic Letters. 7: 5429-31. PMID 16288523 DOI: 10.1021/Ol0522283 |
0.741 |
|
| 2005 |
Pastine SJ, McQuaid KM, Sames D. Room temperature hydroalkylation of electron-deficient olefins: sp3 C-H functionalization via a lewis acid-catalyzed intramolecular redox event. Journal of the American Chemical Society. 127: 12180-1. PMID 16131169 DOI: 10.1021/Ja053337F |
0.799 |
|
| 2005 |
Tremblay MS, Sames D. A new fluorogenic transformation: development of an optical probe for coenzyme Q. Organic Letters. 7: 2417-20. PMID 15932212 DOI: 10.1021/Ol0507569 |
0.553 |
|
| 2005 |
Lane BS, Brown MA, Sames D. Direct palladium-catalyzed C-2 and C-3 arylation of indoles: a mechanistic rationale for regioselectivity. Journal of the American Chemical Society. 127: 8050-7. PMID 15926829 DOI: 10.1021/Ja043273T |
0.39 |
|
| 2005 |
Sezen B, Sames D. Selective and catalytic arylation of N-phenylpyrrolidine: sp3 C-H bond functionalization in the absence of a directing group. Journal of the American Chemical Society. 127: 5284-5. PMID 15826142 DOI: 10.1021/Ja050269O |
0.384 |
|
| 2005 |
Wang X, Lane BS, Sames D. Direct C-arylation of free (NH)-indoles and pyrroles catalyzed by Ar-Rh(III) complexes assembled in situ. Journal of the American Chemical Society. 127: 4996-7. PMID 15810815 DOI: 10.1021/Ja050279P |
0.372 |
|
| 2005 |
Chen G, Yee DJ, Gubernator NG, Sames D. Design of optical switches as metabolic indicators: new fluorogenic probes for monoamine oxidases (MAO A and B). Journal of the American Chemical Society. 127: 4544-5. PMID 15796498 DOI: 10.1021/Ja0428457 |
0.788 |
|
| 2005 |
Godula K, Sezen B, Sames D. Site-specific phenylation of pyridine catalyzed by phosphido-bridged ruthenium dimer complexes: a prototype for C-H arylation of electron-deficient heteroarenes. Journal of the American Chemical Society. 127: 3648-9. PMID 15771470 DOI: 10.1021/Ja042510P |
0.698 |
|
| 2004 |
Sezen B, Sames D. Oxidative C-arylation of free (NH)-heterocycles via direct (sp3) C-H bond functionalization. Journal of the American Chemical Society. 126: 13244-6. PMID 15479077 DOI: 10.1021/Ja045402B |
0.412 |
|
| 2004 |
Lane BS, Sames D. Direct C-H bond arylation: selective palladium-catalyzed C2-arylation of N-substituted indoles. Organic Letters. 6: 2897-900. PMID 15330642 DOI: 10.1021/Ol0490072 |
0.387 |
|
| 2004 |
DeBoef B, Pastine SJ, Sames D. Cross-coupling of sp(3) C-H bonds and alkenes: catalytic cyclization of alkene-amide substrates. Journal of the American Chemical Society. 126: 6556-7. PMID 15161275 DOI: 10.1021/Ja049111E |
0.813 |
|
| 2004 |
Yee DJ, Balsanek V, Sames D. New tools for molecular imaging of redox metabolism: development of a fluorogenic probe for 3 alpha-hydroxysteroid dehydrogenases. Journal of the American Chemical Society. 126: 2282-3. PMID 14982413 DOI: 10.1021/Ja039799F |
0.782 |
|
| 2004 |
Youn SW, Pastine SJ, Sames D. Ru(III)-catalyzed cyclization of arene-alkene substrates via intramolecular electrophilic hydroarylation. Organic Letters. 6: 581-4. PMID 14961628 DOI: 10.1021/ol036385i |
0.698 |
|
| 2003 |
Slovin SF, Ragupathi G, Musselli C, Olkiewicz K, Verbel D, Kuduk SD, Schwarz JB, Sames D, Danishefsky S, Livingston PO, Scher HI. Fully synthetic carbohydrate-based vaccines in biochemically relapsed prostate cancer: clinical trial results with alpha-N-acetylgalactosamine-O-serine/threonine conjugate vaccine. Journal of Clinical Oncology : Official Journal of the American Society of Clinical Oncology. 21: 4292-8. PMID 14645418 DOI: 10.1200/JCO.2003.04.112 |
0.491 |
|
| 2003 |
Pastine SJ, Sames D. Concise synthesis of the chemopreventitive agent (+/-)-deguelin via a key 6-endo hydroarylation. Organic Letters. 5: 4053-5. PMID 14572247 DOI: 10.1021/Ol035419J |
0.704 |
|
| 2003 |
Sezen B, Sames D. Cobalt-catalyzed arylation of azole heteroarenes via direct C-H bond functionalization. Organic Letters. 5: 3607-10. PMID 14507184 DOI: 10.1021/Ol035313O |
0.405 |
|
| 2003 |
Sezen B, Sames D. Diversity synthesis via C-H bond functionalization: concept-guided development of new C-arylation methods for imidazoles. Journal of the American Chemical Society. 125: 10580-5. PMID 12940740 DOI: 10.1021/Ja036157J |
0.399 |
|
| 2003 |
Chen G, Heim A, Riether D, Yee D, Milgrom Y, Gawinowicz MA, Sames D. Reactivity of functional groups on the protein surface: development of epoxide probes for protein labeling. Journal of the American Chemical Society. 125: 8130-3. PMID 12837082 DOI: 10.1021/Ja034287M |
0.774 |
|
| 2003 |
Sezen B, Sames D. Selective C-arylation of free (NH)-heteroarenes via catalytic C-H bond functionalization. Journal of the American Chemical Society. 125: 5274-5. PMID 12720429 DOI: 10.1021/Ja034848+ |
0.402 |
|
| 2003 |
Pastine SJ, Youn SW, Sames D. Pt(IV)-catalyzed cyclization of arene-alkyne substrates via intramolecular electrophilic hydroarylation. Organic Letters. 5: 1055-8. PMID 12659572 DOI: 10.1021/Ol034177K |
0.713 |
|
| 2003 |
Pastine SJ, Youn SW, Sames D. Pt(IV)-catalyzed cyclization of arene-alkyne substrates via C-H bond functionalization Tetrahedron. 59: 8859-8868. DOI: 10.1016/J.Tet.2003.05.003 |
0.733 |
|
| 2002 |
Sezen B, Franz R, Sames D. C-C bond formation via C-H bond activation: catalytic arylation and alkenylation of alkane segments. Journal of the American Chemical Society. 124: 13372-3. PMID 12418875 DOI: 10.1021/Ja027891Q |
0.387 |
|
| 2002 |
Dangel BD, Godula K, Youn SW, Sezen B, Sames D. C-C bond formation via C-H bond activation: synthesis of the core of teleocidin B4. Journal of the American Chemical Society. 124: 11856-7. PMID 12358522 DOI: 10.1021/Ja027311P |
0.797 |
|
| 2002 |
Coltart DM, Royyuru AK, Williams LJ, Glunz PW, Sames D, Kuduk SD, Schwarz JB, Chen XT, Danishefsky SJ, Live DH. Principles of mucin architecture: structural studies on synthetic glycopeptides bearing clustered mono-, di-, tri-, and hexasaccharide glycodomains. Journal of the American Chemical Society. 124: 9833-44. PMID 12175243 DOI: 10.1021/Ja020208F |
0.721 |
|
| 2002 |
Johnson JA, Li N, Sames D. Total synthesis of (-)-rhazinilam: asymmetric C[bond]H bond activation via the use of a chiral auxiliary. Journal of the American Chemical Society. 124: 6900-3. PMID 12059212 DOI: 10.1021/Ja026130K |
0.39 |
|
| 2001 |
Dangel BD, Johnson JA, Sames D. Selective functionalization of amino acids in water: a synthetic method via catalytic C-H bond activation. Journal of the American Chemical Society. 123: 8149-50. PMID 11506585 DOI: 10.1021/Ja016280F |
0.794 |
|
| 2001 |
Havranek M, Moreira R, Sames D. New fluorogenic probes for oxygen and carbene transfer: a sensitive assay for single bead-supported catalysts. Journal of the American Chemical Society. 123: 3927-31. PMID 11457142 DOI: 10.1021/Ja003786+ |
0.688 |
|
| 2000 |
Moreira RF, Wehn PM, Sames D. Highly Regioselective Oxygenation of C-H Bonds: Diamidomanganese Constructs with Attached Substrates as Catalyst Models Financial support has been provided by Columbia University and the Camille and Henry Dreyfus Foundation. P.M.W. acknowledges the REU-NSF program for summer support. We also thank Dr. J. B. Schwarz (manuscript preparation) and Dr. Y. Itagaki (mass spectrometry). Angewandte Chemie (International Ed. in English). 39: 1618-1621. PMID 10820453 DOI: 10.1002/(Sici)1521-3773(20000502)39:9<1618::Aid-Anie1618>3.0.Co;2-M |
0.681 |
|
| 2000 |
Johnson JA, Sames D. C-H bond activation of hydrocarbon segments in complex organic molecules: Total synthesis of the antimitotic rhazinilam [18] Journal of the American Chemical Society. 122: 6321-6322. DOI: 10.1021/Ja0003223 |
0.35 |
|
| 2000 |
Moreira R, Wehn P, Sames D. Hoch regioselektive Oxygenierung von CHBindungen: Diamidmangankomplexe mit angebundenem Substrat als Katalysatormodelle Angewandte Chemie. 112: 1696-1699. DOI: 10.1002/(Sici)1521-3757(20000502)112:9<1696::Aid-Ange1696>3.0.Co;2-3 |
0.637 |
|
| 1999 |
Ragupathi G, Slovin SF, Adluri S, Sames D, Kim IJ, Kim HM, Spassova M, Bornmann WG, Lloyd KO, Scher HI, Livingston PO, Danishefsky SJ. A Fully Synthetic Globo H Carbohydrate Vaccine Induces a Focused Humoral Response in Prostate Cancer Patients: A Proof of Principle. Angewandte Chemie (International Ed. in English). 38: 563-566. PMID 29711780 DOI: 10.1002/(Sici)1521-3773(19990215)38:4<563::Aid-Anie563>3.0.Co;2-3 |
0.469 |
|
| 1999 |
Live DH, Williams LJ, Kuduk SD, Schwarz JB, Glunz PW, Chen XT, Sames D, Kumar RA, Danishefsky SJ. Probing cell-surface architecture through synthesis: an NMR-determined structural motif for tumor-associated mucins. Proceedings of the National Academy of Sciences of the United States of America. 96: 3489-93. PMID 10097062 DOI: 10.1073/Pnas.96.7.3489 |
0.531 |
|
| 1999 |
Polt R, Sames D, Chruma J. Glycosidase inhibitors: Synthesis of enantiomerically pure aza-sugars from Schiff base amino esters via tandem reduction-alkenylation and osmylation Journal of Organic Chemistry. 64: 6147-6158. DOI: 10.1021/Jo9820115 |
0.618 |
|
| 1999 |
Glunz PW, Hintermann S, Schwarz JB, Kuduk SD, Chen XT, Williams LJ, Sames D, Danishefsky SJ, Kudryashov V, Lloyd KO. Probing cell surface 'glyco-architecture' through total synthesis. Immunological consequences of a human blood group determinant in a clustered mucin-like context [6] Journal of the American Chemical Society. 121: 10636-10637. DOI: 10.1021/Ja992309S |
0.533 |
|
| 1999 |
Schwarz JB, Kuduk SD, Chen XT, Sames D, Glunz PW, Danishefsky SJ. A broadly applicable method for the efficient synthesis of α-O-linked glycopeptides and clustered sialic acid residues Journal of the American Chemical Society. 121: 2662-2673. DOI: 10.1021/Ja9833265 |
0.545 |
|
| 1999 |
Ragupathi G, Slovin SF, Adluri S, Sames D, Kim IJ, Kim HM, Spassova M, Bornmann WG, Lloyd KO, Scher HI, Livingston PO, Danishefsky SJ. Ein totalsynthetischer Globo-H-Kohlenhydrat-Impfstoff verursacht eine gezielte humorale Immunantwort bei Prostatakrebs-Patienten: der Beweis des Prinzips Angewandte Chemie. 111: 590-594. DOI: 10.1002/(Sici)1521-3757(19990215)111:4<590::Aid-Ange590>3.0.Co;2-A |
0.481 |
|
| 1998 |
Kuduk SD, Schwarz JB, Chen X, Glunz PW, Sames D, Ragupathi G, Livingston PO, Danishefsky SJ. Synthetic and Immunological Studies on Clustered Modes of Mucin-Related Tn and TF O-Linked Antigens: The Preparation of a Glycopeptide-Based Vaccine for Clinical Trials against Prostate Cancer† Journal of the American Chemical Society. 120: 12474-12485. DOI: 10.1021/Ja9825128 |
0.556 |
|
| 1997 |
Sames D, Chen XT, Danishefsky SJ. Convergent total synthesis of a tumour-associated mucin motif. Nature. 389: 587-91. PMID 9335496 DOI: 10.1038/39292 |
0.527 |
|
| 1997 |
Dangel B, Clarke M, Haley J, Sames D, Polt R. Amino acid-derived ligands for transition metals: Catalysis via a minimalist interpretation of a metalloprotein Journal of the American Chemical Society. 119: 10865-10866. DOI: 10.1021/Ja972135J |
0.756 |
|
| 1997 |
Chruma JJ, Sames D, Polt R. General method for the synthesis of N-methyl amino acids and N-alkyl amino esters from O'Donnell's Schiff bases Tetrahedron Letters. 38: 5085-5086. DOI: 10.1016/S0040-4039(97)01132-5 |
0.595 |
|
| 1995 |
Sames D, Polt R. Piperidine Triols via Enantioselective Alkylation and Osmylation of Alanine Schiff Base Esters Synlett. 1995: 552-554. DOI: 10.1055/S-1995-5282 |
0.613 |
|
| 1995 |
Sames D, Liu Y, DeYoung L, Polt R. Preparation of monosilyl acetals from esters via iBu2AlH reduction and trapping with N-(trimethylsilyl)imidazole. Addition of allyltrimethylsilane to yield homoallylic alcohols or ethers Journal of Organic Chemistry. 60: 2153-2159. DOI: 10.1021/Jo00112A039 |
0.537 |
|
| 1994 |
Sames D, Polt R. An enantioselective synthesis of N-methylfucosamine via tandem C-C/C-O bond formation Journal of Organic Chemistry. 59: 4596-4601. DOI: 10.1021/Jo00095A039 |
0.64 |
|
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