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Scott C. Eagon, Ph.D. - Publications

Affiliations: 
2014- California Polytechnic State University, San Luis Obispo, CA, United States 
Area:
Synthetic Organic & Medicinal Chemistry
Website:
https://eagonlab.github.io/about_Dr_Eagon.html
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31 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Viswanathan NK, Chirgwin ME, Gibbs J, Kalaj BN, Durham S, Tran J, Gomez M, Lazaro H, Chen M, Mansfield CR, Derbyshire ER, Eagon S. Synthesis and Activity of β-Carboline Antimalarials Targeting the Plasmodium falciparum Heat Shock 90 Protein. Bioorganic & Medicinal Chemistry Letters. 129410. PMID 37478957 DOI: 10.1016/j.bmcl.2023.129410  0.771
2021 Eagon S, Howland M, Heying M, Callant E, Brar N, Pompa E, Mallari JP. Identification of Plasmodium falciparum falcilysin inhibitors by a virtual screen. Bioorganic & Medicinal Chemistry Letters. 52: 128394. PMID 34606998 DOI: 10.1016/j.bmcl.2021.128394  0.251
2021 Eagon S, Hammill JT, Fitzsimmons K, Sienko N, Nguyen B, Law J, Manjunath A, Wilkinson SP, Thompson K, Elizabeth Glidden J, Rice AL, Falade MO, Kimball JJ, DiBernardo C, Kiplin Guy R. Antimalarial Activity of 2,6-Dibenzylidenecyclohexanone Derivatives. Bioorganic & Medicinal Chemistry Letters. 128216. PMID 34157390 DOI: 10.1016/j.bmcl.2021.128216  0.771
2021 Zhang L, Howland M, Hilgenfeld R, Anderson MO, Eagon S. Identification of Non-Covalent SARS-CoV-2 Main Protease Inhibitors by a Virtual Screen of Commercially Available Drug-Like Compounds. Bioorganic & Medicinal Chemistry Letters. 127990. PMID 33775840 DOI: 10.1016/j.bmcl.2021.127990  0.599
2021 Kahlon G, Lira R, Masvlov N, Pompa E, Brar N, Eagon S, Anderson MO, Andaya A, Chance JP, Fejzic H, Keniston A, Huynh N, Celis N, Vidal B, Trieu N, et al. Corrigendum to "Structure guided development of potent piperazine-derived hydroxamic acid inhibitors targeting falcilysin" [Bioorg. Med. Chem. Lett. 32 (2021) 127683]. Bioorganic & Medicinal Chemistry Letters. 37: 127836. PMID 33588181 DOI: 10.1016/j.bmcl.2021.127836  0.59
2021 Everson N, Bach J, Hammill JT, Falade MO, Rice AL, Guy RK, Eagon S. Identification of Plasmodium falciparum heat shock 90 inhibitors via molecular docking. Bioorganic & Medicinal Chemistry Letters. 35: 127818. PMID 33513390 DOI: 10.1016/j.bmcl.2021.127818  0.794
2020 Kahlon G, Lira R, Masvlov N, Pompa E, Brar N, Eagon S, Anderson MO, Andaya A, Chance JP, Fejzic H, Keniston A, Vidal B, Trieu N, Rodriguez P, Mallari JP. Structure Guided Development of Potent Piperazine-Derived Hydroxamic Acid Inhibitors Targeting Falcilysin. Bioorganic & Medicinal Chemistry Letters. 127683. PMID 33227414 DOI: 10.1016/j.bmcl.2020.127683  0.63
2020 Eagon S, Hammill JT, Sigal MS, Ahn KJ, Tryhorn JE, Koch G, Belanger B, Chaplan CA, Loop L, Kashtanova AS, Yniguez K, Lazaro H, Wilkinson SP, Rice A, Falade M, et al. Synthesis and structure-activity relationship of dual-stage antimalarial pyrazolo[3,4-b]pyridines. Journal of Medicinal Chemistry. PMID 32945666 DOI: 10.1021/Acs.Jmedchem.0C01152  0.676
2020 Eagon S, Hammill JT, Bach J, Everson N, Sisley TA, Walls MJ, Durham S, Pillai DR, Falade MO, Rice AL, Kimball JJ, Lazaro H, DiBernardo C, Kiplin Guy R. Antimalarial activity of tetrahydro-β-carbolines targeting the ATP binding pocket of the Plasmodium falciparum heat shock 90 protein. Bioorganic & Medicinal Chemistry Letters. 30: 127502. PMID 32822760 DOI: 10.1016/J.Bmcl.2020.127502  0.743
2020 Masters L, Eagon S, Heying M. Evaluation of consensus scoring methods for AutoDock Vina, smina and idock. Journal of Molecular Graphics & Modelling. 96: 107532. PMID 31991303 DOI: 10.1016/J.Jmgm.2020.107532  0.348
2019 Law J, Manjunath A, Schioldager R, Eagon S. Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines. Journal of Visualized Experiments : Jove. PMID 31282901 DOI: 10.3791/59896  0.766
2019 Bowen LR, Li DJ, Nola DT, Anderson MO, Heying M, Groves AT, Eagon S. Identification of potential Zika virus NS2B-NS3 protease inhibitors via docking, molecular dynamics and consensus scoring-based virtual screening. Journal of Molecular Modeling. 25: 194. PMID 31209577 DOI: 10.1007/S00894-019-4076-6  0.634
2019 Everson N, Yniguez K, Loop L, Lazaro H, Belanger B, Koch G, Bach J, Manjunath A, Schioldager R, Law J, Grabenauer M, Eagon S. Microwave synthesis of 1-aryl-1H-pyrazole-5-amines Tetrahedron Letters. 60: 72-74. DOI: 10.1016/J.Tetlet.2018.11.060  0.661
2017 Durham SD, Sierra B, Gomez MJ, Tran JK, Anderson MO, Whittington-Davis NA, Eagon S. Synthesis of β-carbolines via a silver-mediated oxidation of tetrahydro-β-carbolines Tetrahedron Letters. 58: 2747-2750. DOI: 10.1016/J.Tetlet.2017.05.098  0.781
2016 Bayih AG, Folefoc A, Mohon AN, Eagon S, Anderson M, Pillai DR. In vitro and in vivo anti-malarial activity of novel harmine-analog heat shock protein 90 inhibitors: a possible partner for artemisinin. Malaria Journal. 15: 579. PMID 27903279 DOI: 10.1186/S12936-016-1625-7  0.639
2015 Eagon S, Anderson MO. ChemInform Abstract: Microwave-Assisted Synthesis of Tetrahydro-β-carbolines and β-Carbolines. Cheminform. 46: no-no. DOI: 10.1002/CHIN.201504165  0.333
2014 Eagon S, Anderson MO. Microwave-assisted synthesis of tetrahydro-β-carbolines and β-carbolines European Journal of Organic Chemistry. 2014: 1653-1665. DOI: 10.1002/Ejoc.201301580  0.679
2012 Saavedra JZ, Resendez A, Rovira A, Eagon S, Haddenham D, Singaram B. Reaction of InCl3 with various reducing agents: InCl3-NaBH4-mediated reduction of aromatic and aliphatic nitriles to primary amines. The Journal of Organic Chemistry. 77: 221-8. PMID 22148510 DOI: 10.1021/Jo201809A  0.799
2012 Bailey CL, Murphy CL, Clary JW, Eagon S, Gould N, Singaram B. Reaction of grignard reagents with diisopropylaminoborane. Synthesis of alkyl, aryl, heteroaryl and allyl boronic acids from organo(diisopropyl)- aminoborane by a simple hydrolysis Heterocycles. 86: 331-341. DOI: 10.3987/Com-12-S(N)14  0.805
2012 Saavedra JZ, Resendez A, Rovira A, Eagon S, Haddenham D, Singaram B. Reaction of InCl 3 with various reducing agents: InCl 3-NaBH 4-mediated reduction of aromatic and aliphatic nitriles to primary amines Journal of Organic Chemistry. 77: 221-228. DOI: 10.1021/jo201809a  0.78
2011 Haddenham D, Bailey CL, Vu C, Nepomuceno G, Eagon S, Pasumansky L, Singaram B. Lithium aminoborohydrides 17. Palladium catalyzed borylation of aryl iodides, bromides, and triflates with diisopropylaminoborane prepared from lithium diisopropylaminoborohydride Tetrahedron. 67: 576-583. DOI: 10.1016/J.Tet.2010.11.065  0.806
2011 Haddenham D, Bailey CL, Vu C, Nepomuceno G, Eagon S, Pasumansky L, Singaram B. ChemInform Abstract: Lithium Aminoborohydrides. Part 17. Palladium Catalyzed Borylation of Aryl Iodides, Bromides, and Triflates with Diisopropylaminoborane Prepared from Lithium Diisopropylaminoborohydride. Cheminform. 42: no-no. DOI: 10.1002/CHIN.201122191  0.385
2011 Eagon S, Ball-Jones N, Haddenham D, Saavedra J, DeLieto C, Buckman M, Singaram B. ChemInform Abstract: Enantioselective Reduction of α-Substituted Ketones Mediated by the Boronate Ester TarB-NO2. Cheminform. 42: no-no. DOI: 10.1002/CHIN.201112070  0.379
2010 Eagon S, DeLieto C, McDonald WJ, Haddenham D, Saavedra J, Kim J, Singaram B. Mild and expedient asymmetric reductions of α,β-unsaturated alkenyl and alkynyl ketones by TarB-NO2 and mechanistic investigations of ketone reduction. The Journal of Organic Chemistry. 75: 7717-25. PMID 21033682 DOI: 10.1021/Jo101530F  0.793
2010 Eagon S, Delieto C, McDonald WJ, Haddenham D, Saavedra J, Kim J, Singaram B. Mild and expedient asymmetric reductions of α,β-unsaturated alkenyl and alkynyl ketones by TarB-NO2 and mechanistic investigations of ketone reduction Journal of Organic Chemistry. 75: 7717-7725. DOI: 10.1021/jo101530f  0.779
2010 Eagon S, Ball-Jones N, Haddenham D, Saavedra J, Delieto C, Buckman M, Singaram B. Enantioselective reduction of α-substituted ketones mediated by the boronate ester TarB-NO2 Tetrahedron Letters. 51: 6418-6421. DOI: 10.1016/J.Tetlet.2010.09.146  0.795
2009 Haddenham D, Pasumansky L, DeSoto J, Eagon S, Singaram B. Reductions of aliphatic and aromatic nitriles to primary amines with diisopropylaminoborane Journal of Organic Chemistry. 74: 1964-1970. PMID 19191712 DOI: 10.1021/Jo8023329  0.788
2009 Eagon S, Kim J, Singaram B. ChemInform Abstract: Mild and Practical Reductions of Prochiral Ketones to Chiral Alcohols Using the Chiral Boronic Ester TarB-H. Cheminform. 40. DOI: 10.1002/CHIN.200915067  0.348
2008 Eagon S, Kim J, Singaram B. Mild and practical reductions of prochiral ketones to chiral alcohols using the chiral boronic ester TarB-H Synthesis. 3874-3876. DOI: 10.1055/S-0028-1083605  0.737
2008 Eagon S, Kim J, Yan K, Haddenham D, Singaram B. ChemInform Abstract: Asymmetric Reductions Using the Chiral Boronic Ester TarB—H: A Practical and Inexpensive Procedure for Synthesizing Chiral Alcohols. Cheminform. 39. DOI: 10.1002/CHIN.200814031  0.668
2007 Eagon S, Kim J, Yan K, Haddenham D, Singaram B. Asymmetric reductions using the chiral boronic ester TarB-H: a practical and inexpensive procedure for synthesizing chiral alcohols Tetrahedron Letters. 48: 9025-9029. DOI: 10.1016/J.Tetlet.2007.10.075  0.791
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