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Anna K. Mapp, Ph.D. - Publications

Affiliations: 
Chemistry, Medicinal Chemsitry University of Michigan, Ann Arbor, Ann Arbor, MI 
Area:
Chemical biology
Website:
https://www.chem.lsa.umich.edu/chem/faculty/facultyDetail.php?Uniqname=amapp

85 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2024 Pattelli ON, Valdivia EM, Beyersdorf MS, Regan CS, Rivas M, Hebert KA, Merajver SD, Cierpicki T, Mapp AK. A Lipopeptidomimetic of Transcriptional Activation Domains Selectively Disrupts Med25 Protein-Protein Interactions. Angewandte Chemie (International Ed. in English). e202400781. PMID 38527936 DOI: 10.1002/anie.202400781  0.474
2023 Liu Y, Joy ST, Henley MJ, Croskey A, Yates JA, Merajver SD, Mapp AK. Inhibition of CREB Binding and Function with a Dual-Targeting Ligand. Biochemistry. PMID 38086054 DOI: 10.1021/acs.biochem.3c00469  0.384
2023 Breen ME, Joy ST, Baruti OJ, Beyersdorf MS, Henley MJ, De Salle SN, Ycas PD, Croskey A, Cierpicki T, Pomerantz WCK, Mapp AK. Garcinolic acid distinguishes between GACKIX domains and modulates interaction networks. Chembiochem : a European Journal of Chemical Biology. e202300439. PMID 37525583 DOI: 10.1002/cbic.202300439  0.392
2023 Pattelli ON, Valdivia EM, Beyersdorf MS, Regan CS, Rivas M, Merajver SD, Cierpicki T, Mapp AK. A lipopeptidomimetic of transcriptional activation domains selectively disrupts Med25 PPIs. Biorxiv : the Preprint Server For Biology. PMID 36993479 DOI: 10.1101/2023.03.24.534168  0.457
2022 Peiffer AL, Garlick JM, Joy ST, Mapp AK, Brooks CL. Allostery in the dynamic coactivator domain KIX occurs through minor conformational micro-states. Plos Computational Biology. 18: e1009977. PMID 35452454 DOI: 10.1371/journal.pcbi.1009977  0.35
2021 Joy ST, Henley MJ, De Salle SN, Beyersdorf MS, Vock IW, Huldin AJL, Mapp AK. A Dual-Site Inhibitor of CBP/p300 KIX is a Selective and Effective Modulator of Myb. Journal of the American Chemical Society. PMID 34491719 DOI: 10.1021/jacs.1c04432  0.393
2021 Garlick JM, Sturlis SM, Bruno PA, Yates JA, Peiffer AL, Liu Y, Goo L, Bao L, De Salle SN, Tamayo-Castillo G, Brooks CL, Merajver SD, Mapp AK. Norstictic Acid Is a Selective Allosteric Transcriptional Regulator. Journal of the American Chemical Society. PMID 34137598 DOI: 10.1021/jacs.1c03258  0.438
2020 Henley MJ, Linhares BM, Morgan BS, Cierpicki T, Fierke CA, Mapp AK. Unexpected specificity within dynamic transcriptional protein-protein complexes. Proceedings of the National Academy of Sciences of the United States of America. PMID 33077600 DOI: 10.1073/pnas.2013244117  0.455
2020 Annand JR, Henderson AR, Cole KS, Maurais AJ, Becerra J, Liu Y, Weerapana E, Koehler AN, Mapp AK, Schindler CS. Gibberellin JRA-003: A Selective Inhibitor of Nuclear Translocation of IKKα. Acs Medicinal Chemistry Letters. 11: 1913-1918. PMID 33062173 DOI: 10.1021/Acsmedchemlett.9B00613  0.33
2020 Huang H, Howard CA, Zari S, Cho HJ, Shukla S, Li H, Ndoj J, González-Alonso P, Nikolaidis C, Abbott J, Rogawski DS, Potopnyk MA, Kempinska K, Miao H, Purohit T, ... ... Mapp A, et al. Covalent inhibition of NSD1 histone methyltransferase. Nature Chemical Biology. PMID 32868895 DOI: 10.1038/S41589-020-0626-6  0.46
2020 Garlick JM, Mapp AK. Selective Modulation of Dynamic Protein Complexes. Cell Chemical Biology. 27: 986-997. PMID 32783965 DOI: 10.1016/J.Chembiol.2020.07.019  0.407
2020 Strunk BS, Steinfeld N, Lee S, Jin N, Muñoz-Rivera C, Meeks G, Thomas A, Akemann C, Mapp AK, MacGurn JA, Weisman LS. Roles for a lipid phosphatase in the activation of its opposing lipid kinase. Molecular Biology of the Cell. mbcE18090556. PMID 32583743 DOI: 10.1091/Mbc.E18-09-0556  0.369
2019 Joiner CM, Breen ME, Mapp AK. Electron-deficient p-benzoyl-L-phenylalanine derivatives increase covalent chemical capture yields for protein-protein interactions. Protein Science : a Publication of the Protein Society. PMID 30977234 DOI: 10.1002/Pro.3621  0.799
2018 Rabuck-Gibbons JN, Lodge JM, Mapp AK, Ruotolo BT. Collision-Induced Unfolding Reveals Unique Fingerprints for Remote Protein Interaction Sites in the KIX Regulation Domain. Journal of the American Society For Mass Spectrometry. PMID 30136215 DOI: 10.1007/S13361-018-2043-6  0.525
2018 Henderson AR, Henley MJ, Foster NJ, Peiffer AL, Beyersdorf MS, Stanford KD, Sturlis SM, Linhares BM, Hill ZB, Wells JA, Cierpicki T, Brooks CL, Fierke CA, Mapp AK. Conservation of coactivator engagement mechanism enables small-molecule allosteric modulators. Proceedings of the National Academy of Sciences of the United States of America. PMID 30127017 DOI: 10.1073/Pnas.1806202115  0.538
2018 Breen ME, Mapp AK. Modulating the masters: chemical tools to dissect CBP and p300 function. Current Opinion in Chemical Biology. 45: 195-203. PMID 30025258 DOI: 10.1016/J.Cbpa.2018.06.005  0.472
2018 Lodge JM, Majmudar CY, Clayton J, Mapp AK. Covalent chemical co-chaperones of the p300/CBP GACKIX domain. Chembiochem : a European Journal of Chemical Biology. PMID 29939485 DOI: 10.1002/Cbic.201800173  0.84
2018 Jennings LE, Schiedel M, Hewings DS, Picaud S, Laurin CMC, Bruno PA, Bluck JP, Scorah AR, See L, Reynolds JK, Moroglu M, Mistry IN, Hicks A, Guzanov P, Clayton J, ... ... Mapp AK, et al. BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability. Bioorganic & Medicinal Chemistry. PMID 29776834 DOI: 10.1016/J.Bmc.2018.05.003  0.371
2018 Ouimet CM, Dawod M, Grinias J, Assimon VA, Lodge J, Mapp AK, Gestwicki JE, Kennedy RT. Protein cross-linking capillary electrophoresis at increased throughput for a range of protein-protein interactions. The Analyst. PMID 29565056 DOI: 10.1039/C7An02098H  0.404
2017 Cesa LC, Shao H, Srinivasan SR, Tse E, Jain C, Zuiderweg ERP, Southworth DR, Mapp AK, Gestwicki JE. X-Linked Inhibitor of Apoptosis Protein (XIAP) is a Client of Heat Shock Protein 70 (Hsp70) and a Biomarker of its Inhibition. The Journal of Biological Chemistry. PMID 29255093 DOI: 10.1074/Jbc.Ra117.000634  0.316
2017 Pricer R, Gestwicki JE, Mapp AK. From Fuzzy to Function: The New Frontier of Protein-Protein Interactions. Accounts of Chemical Research. 50: 584-589. PMID 28945413 DOI: 10.1021/Acs.Accounts.6B00565  0.503
2016 Joiner CM, Breen ME, Clayton J, Mapp AK. A Bifunctional Amino Acid Enables Both Covalent Chemical Capture and Isolation of in Vivo Protein-Protein Interactions. Chembiochem : a European Journal of Chemical Biology. PMID 27966261 DOI: 10.1002/Cbic.201600578  0.815
2016 Bruno PA, Morriss-Andrews A, Henderson AR, Brooks CL, Mapp AK. A Synthetic Loop Replacement Peptide That Blocks Canonical NF-κB Signaling. Angewandte Chemie (International Ed. in English). PMID 27791341 DOI: 10.1002/Anie.201607990  0.327
2016 Dugan A, Majmudar CY, Pricer RE, Niessen S, Lancia JK, Fung HY, Cravatt BF, Mapp AK. Discovery of enzymatic targets of transcriptional activators via in vivo covalent chemical capture. Journal of the American Chemical Society. PMID 27611834 DOI: 10.1021/Jacs.6B07680  0.835
2016 Dugan A, Pricer R, Katz M, Mapp AK. TRIC: Capturing the direct cellular targets of promoter-bound transcriptional activators. Protein Science : a Publication of the Protein Society. PMID 27213278 DOI: 10.1002/Pro.2951  0.53
2015 Mapp AK, Pricer R, Sturlis S. Targeting transcription is no longer a quixotic quest. Nature Chemical Biology. 11: 891-4. PMID 26575226 DOI: 10.1038/Nchembio.1962  0.435
2015 Cesa LC, Mapp AK, Gestwicki JE. Direct and Propagated Effects of Small Molecules on Protein-Protein Interaction Networks. Frontiers in Bioengineering and Biotechnology. 3: 119. PMID 26380257 DOI: 10.3389/Fbioe.2015.00119  0.396
2015 Annand JR, Bruno PA, Mapp AK, Schindler CS. Synthesis and biological evaluation of pharbinilic acid and derivatives as NF-κB pathway inhibitors. Chemical Communications (Cambridge, England). 51: 8990-3. PMID 25932702 DOI: 10.1039/C5Cc02918J  0.34
2014 Wang N, Lodge JM, Fierke CA, Mapp AK. Dissecting allosteric effects of activator-coactivator complexes using a covalent small molecule ligand. Proceedings of the National Academy of Sciences of the United States of America. 111: 12061-6. PMID 25049401 DOI: 10.1073/Pnas.1406033111  0.722
2014 Law SM, Gagnon JK, Mapp AK, Brooks CL. Prepaying the entropic cost for allosteric regulation in KIX. Proceedings of the National Academy of Sciences of the United States of America. 111: 12067-72. PMID 25002472 DOI: 10.1073/Pnas.1405831111  0.445
2014 Lodge JM, Rettenmaier TJ, Wells JA, Pomerantz WC, Mapp AK. FP Tethering: a screening technique to rapidly identify compounds that disrupt protein-protein interactions. Medchemcomm. 5: 370-375. PMID 24795804 DOI: 10.1039/C3Md00356F  0.827
2014 Højfeldt JW, Cruz-Rodríguez O, Imaeda Y, Van Dyke AR, Carolan JP, Mapp AK, Iñiguez-Lluhí JA. Bifunctional ligands allow deliberate extrinsic reprogramming of the glucocorticoid receptor. Molecular Endocrinology (Baltimore, Md.). 28: 249-59. PMID 24422633 DOI: 10.1210/Me.2013-1343  0.783
2014 Lancia JK, Nwokoye A, Dugan A, Joiner C, Pricer R, Mapp AK. Sequence context and crosslinking mechanism affect the efficiency of in vivo capture of a protein-protein interaction. Biopolymers. 101: 391-7. PMID 24037947 DOI: 10.1002/Bip.22395  0.787
2014 Xie X, Piao L, Cavey GS, Old M, Teknos TN, Mapp AK, Pan Q. Phosphorylation of Nanog is essential to regulate Bmi1 and promote tumorigenesis. Oncogene. 33: 2040-52. PMID 23708658 DOI: 10.1038/Onc.2013.173  0.362
2013 Merrins MJ, Van Dyke AR, Mapp AK, Rizzo MA, Satin LS. Direct measurements of oscillatory glycolysis in pancreatic islet β-cells using novel fluorescence resonance energy transfer (FRET) biosensors for pyruvate kinase M2 activity. The Journal of Biological Chemistry. 288: 33312-22. PMID 24100037 DOI: 10.1074/Jbc.M113.508127  0.775
2013 Wang N, Majmudar CY, Pomerantz WC, Gagnon JK, Sadowsky JD, Meagher JL, Johnson TK, Stuckey JA, Brooks CL, Wells JA, Mapp AK. Ordering a dynamic protein via a small-molecule stabilizer. Journal of the American Chemical Society. 135: 3363-6. PMID 23384013 DOI: 10.1021/Ja3122334  0.812
2012 Majmudar CY, Højfeldt JW, Arevang CJ, Pomerantz WC, Gagnon JK, Schultz PJ, Cesa LC, Doss CH, Rowe SP, Vásquez V, Tamayo-Castillo G, Cierpicki T, Brooks CL, Sherman DH, Mapp AK. Sekikaic acid and lobaric acid target a dynamic interface of the coactivator CBP/p300. Angewandte Chemie (International Ed. in English). 51: 11258-62. PMID 23042634 DOI: 10.1002/Anie.201206815  0.789
2012 Thompson AD, Dugan A, Gestwicki JE, Mapp AK. Fine-tuning multiprotein complexes using small molecules. Acs Chemical Biology. 7: 1311-20. PMID 22725693 DOI: 10.1021/Cb300255P  0.425
2012 Pomerantz WC, Wang N, Lipinski AK, Wang R, Cierpicki T, Mapp AK. Profiling the dynamic interfaces of fluorinated transcription complexes for ligand discovery and characterization. Acs Chemical Biology. 7: 1345-50. PMID 22725662 DOI: 10.1021/Cb3002733  0.839
2012 Taylor CE, Pan Q, Mapp AK. Synergistic enhancement of the potency and selectivity of small molecule transcriptional inhibitors. Acs Medicinal Chemistry Letters. 3: 30-34. PMID 22368762 DOI: 10.1021/Ml200186R  0.424
2012 Yu J, Meijer EW, Booker SJ, Mapp AK, Jamison TF, Aube J, Wasielewski MR, Schuster DI, Snyder SA, Tang Y, Chang CJ, Glorius F, Feringa B. Arthur C. Cope Scholar Awards and Eli Lilly Award Angewandte Chemie. 51: 8693-8694. DOI: 10.1002/Anie.201204828  0.473
2011 Krishnamurthy M, Dugan A, Nwokoye A, Fung YH, Lancia JK, Majmudar CY, Mapp AK. Caught in the act: covalent cross-linking captures activator-coactivator interactions in vivo. Acs Chemical Biology. 6: 1321-6. PMID 21977905 DOI: 10.1021/Cb200308E  0.828
2011 Højfeldt JW, Van Dyke AR, Mapp AK. Transforming ligands into transcriptional regulators: building blocks for bifunctional molecules. Chemical Society Reviews. 40: 4286-94. PMID 21701709 DOI: 10.1039/C1Cs15050B  0.834
2011 Wands AM, Wang N, Lum JK, Hsieh J, Fierke CA, Mapp AK. Transient-state kinetic analysis of transcriptional activator·DNA complexes interacting with a key coactivator. The Journal of Biological Chemistry. 286: 16238-45. PMID 21317429 DOI: 10.1074/Jbc.M110.207589  0.805
2011 Mapp A. Human disease and transcriptional misregulation have strengthened Biopolymers. 95: iii. PMID 21031499 DOI: 10.1002/Bip.21554  0.314
2011 Bates CA, Pomerantz WC, Mapp AK. Transcriptional tools: Small molecules for modulating CBP KIX-dependent transcriptional activators. Biopolymers. 95: 17-23. PMID 20882601 DOI: 10.1002/Bip.21548  0.857
2010 Danowitz AM, Taylor CE, Shrikian TM, Mapp AK. Palladium-catalyzed [3,3]-rearrangement for the facile synthesis of allenamides. Organic Letters. 12: 2574-7. PMID 20438110 DOI: 10.1021/Ol1007845  0.748
2010 Lee LW, Mapp AK. Transcriptional switches: chemical approaches to gene regulation. The Journal of Biological Chemistry. 285: 11033-8. PMID 20147748 DOI: 10.1074/Jbc.R109.075044  0.54
2009 Lee LW, Taylor CE, Desaulniers JP, Zhang M, Højfeldt JW, Pan Q, Mapp AK. Inhibition of ErbB2(Her2) expression with small molecule transcription factor mimics. Bioorganic & Medicinal Chemistry Letters. 19: 6233-6. PMID 19782563 DOI: 10.1016/J.Bmcl.2009.08.090  0.499
2009 Majmudar CY, Lee LW, Lancia JK, Nwokoye A, Wang Q, Wands AM, Wang L, Mapp AK. Impact of nonnatural amino acid mutagenesis on the in vivo function and binding modes of a transcriptional activator. Journal of the American Chemical Society. 131: 14240-2. PMID 19764747 DOI: 10.1021/Ja904378Z  0.828
2009 Majmudar CY, Wang B, Lum JK, Håkansson K, Mapp AK. A high-resolution interaction map of three transcriptional activation domains with a key coactivator from photo-cross-linking and multiplexed mass spectrometry. Angewandte Chemie (International Ed. in English). 48: 7021-4. PMID 19681084 DOI: 10.1002/Anie.200902669  0.848
2009 Bao L, Gorin MA, Zhang M, Ventura AC, Pomerantz WC, Merajver SD, Teknos TN, Mapp AK, Pan Q. Preclinical development of a bifunctional cancer cell homing, PKCepsilon inhibitory peptide for the treatment of head and neck cancer. Cancer Research. 69: 5829-34. PMID 19567682 DOI: 10.1158/0008-5472.Can-08-3465  0.765
2009 Majmudar CY, Labut AE, Mapp AK. Tra1 as a screening target for transcriptional activation domain discovery. Bioorganic & Medicinal Chemistry Letters. 19: 3733-5. PMID 19497740 DOI: 10.1016/J.Bmcl.2009.05.045  0.848
2009 Aminoff D, Bochar DA, Fuller AA, Mapp AK, Showalter HD, Kirchhoff PD. Research into selective biomarkers of erythrocyte exposure to organophosphorus compounds. Analytical Biochemistry. 392: 155-61. PMID 19497294 DOI: 10.1016/J.Ab.2009.05.049  0.599
2009 Buhrlage SJ, Bates CA, Rowe SP, Minter AR, Brennan BB, Majmudar CY, Wemmer DE, Al-Hashimi H, Mapp AK. Amphipathic small molecules mimic the binding mode and function of endogenous transcription factors. Acs Chemical Biology. 4: 335-44. PMID 19348463 DOI: 10.1021/Cb900028J  0.826
2009 Casey RJ, Desaulniers JP, Hojfeldt JW, Mapp AK. Expanding the repertoire of small molecule transcriptional activation domains. Bioorganic & Medicinal Chemistry. 17: 1034-43. PMID 18334300 DOI: 10.1016/J.Bmc.2008.02.045  0.79
2009 Buhrlage SJ, Chen B, Mapp AK. A flexible synthetic route to isoxazolidine β-proline analogs Tetrahedron. 65: 3305-3313. DOI: 10.1016/J.Tet.2008.12.062  0.637
2008 Mapp A, Romesberg FE. Several novel approaches to developing therapeutics that target both bacterial and human proteins. Current Opinion in Chemical Biology. 12: 387-8. PMID 18707019 DOI: 10.1016/J.Cbpa.2008.08.003  0.331
2008 Rowe SP, Mapp AK. Assessing the permissiveness of transcriptional activator binding sites. Biopolymers. 89: 578-81. PMID 18253946 DOI: 10.1002/Bip.20946  0.67
2007 Rowe SP, Casey RJ, Brennan BB, Buhrlage SJ, Mapp AK. Transcriptional up-regulation in cells mediated by a small molecule. Journal of the American Chemical Society. 129: 10654-5. PMID 17691790 DOI: 10.1021/Ja0736865  0.837
2007 Lum JK, Wu Z, Mapp AK. Disrupting mediator with a short peptide ligand. Chembiochem : a European Journal of Chemical Biology. 8: 1233-6. PMID 17583546 DOI: 10.1002/Cbic.200700062  0.697
2007 Kiessling LL, Doudna JA, Johnsson K, Mapp AK, Marletta MA, Seeberger PH, Williamson JR, Wedde SG. A higher degree of difficulty. Acs Chemical Biology. 2: 197-9. PMID 17455890 DOI: 10.1021/Cb7000846  0.432
2007 Mapp AK, Ansari AZ. A TAD further: exogenous control of gene activation. Acs Chemical Biology. 2: 62-75. PMID 17243784 DOI: 10.1021/Cb600463W  0.484
2006 Lum JK, Majmudar CY, Ansari AZ, Mapp AK. Converting inactive peptides into potent transcriptional activators. Acs Chemical Biology. 1: 639-43. PMID 17175579 DOI: 10.1021/Cb600363N  0.846
2006 Ferguson ML, Senecal TD, Groendyke TM, Mapp AK. [3,3]-rearrangements of phosphonium ylides. Journal of the American Chemical Society. 128: 4576-7. PMID 16594686 DOI: 10.1021/Ja058746Q  0.655
2005 Buhrlage SJ, Brennan BB, Minter AR, Mapp AK. Stereochemical promiscuity in artificial transcriptional activators. Journal of the American Chemical Society. 127: 12456-7. PMID 16144370 DOI: 10.1021/Ja0536567  0.834
2005 Majmudar CY, Mapp AK. Chemical approaches to transcriptional regulation. Current Opinion in Chemical Biology. 9: 467-74. PMID 16122970 DOI: 10.1016/J.Cbpa.2005.08.012  0.852
2005 Lum JK, Mapp AK. Artificial transcriptional activation domains. Chembiochem : a European Journal of Chemical Biology. 6: 1311-5. PMID 15973758 DOI: 10.1002/Cbic.200500036  0.721
2005 Lu Z, Rowe SP, Brennan BB, Davis SE, Metzler RE, Nau JJ, Majmudar CY, Mapp AK, Ansari AZ. Unraveling the mechanism of a potent transcriptional activator. The Journal of Biological Chemistry. 280: 29689-98. PMID 15886204 DOI: 10.1074/Jbc.M504895200  0.849
2005 Fuller AA, Chen B, Minter AR, Mapp AK. Succinct synthesis of beta-amino acids via chiral isoxazolines. Journal of the American Chemical Society. 127: 5376-83. PMID 15826175 DOI: 10.1021/Ja0431713  0.782
2005 Majmudar CY, Lum JK, Prasov L, Mapp AK. Functional specificity of artificial transcriptional activators. Chemistry & Biology. 12: 313-21. PMID 15797215 DOI: 10.1016/J.Chembiol.2005.01.014  0.854
2004 Mapp AK. Finding their groove; bifunctional molecules arrest growth of cancer cells. Chemistry & Biology. 11: 1480-2. PMID 15555997 DOI: 10.1016/J.Chembiol.2004.11.002  0.343
2004 Minter AR, Brennan BB, Mapp AK. A small molecule transcriptional activation domain. Journal of the American Chemical Society. 126: 10504-5. PMID 15327284 DOI: 10.1021/Ja0473889  0.854
2004 Fuller AA, Chen B, Minter AR, Mapp AK. Synthesis and structural characteristics of geminally disubstituted β-amino acids Synlett. 1409-1413. DOI: 10.1055/S-2004-829051  0.778
2004 Mapp AK, Ansari AZ, Wu Z, Lu Z. Modulating Transcription with Artificial Regulators Handbook of Experimental Pharmacology. 166: 535-571. DOI: 10.1007/978-3-642-18932-6_18  0.457
2003 Wu Z, Belanger G, Brennan BB, Lum JK, Minter AR, Rowe SP, Plachetka A, Majmudar CY, Mapp AK. Targeting the transcriptional machinery with unique artificial transcriptional activators. Journal of the American Chemical Society. 125: 12390-1. PMID 14531665 DOI: 10.1021/Ja036685V  0.823
2003 Mapp AK. Regulating transcription: a chemical perspective. Organic & Biomolecular Chemistry. 1: 2217-20. PMID 12945688 DOI: 10.1039/B302656F  0.386
2003 Minter AR, Fuller AA, Mapp AK. A concise approach to structurally diverse beta-amino acids. Journal of the American Chemical Society. 125: 6846-7. PMID 12783519 DOI: 10.1021/Ja0298747  0.773
2002 Ansari AZ, Mapp AK. Modular design of artificial transcription factors. Current Opinion in Chemical Biology. 6: 765-72. PMID 12470729 DOI: 10.1016/S1367-5931(02)00377-0  0.398
2001 Ansari AZ, Mapp AK, Nguyen DH, Dervan PB, Ptashne M. Towards a minimal motif for artificial transcriptional activators. Chemistry & Biology. 8: 583-92. PMID 11410377 DOI: 10.1016/S1074-5521(01)00037-0  0.775
2000 Mapp AK, Ansari AZ, Ptashne M, Dervan PB. Activation of gene expression by small molecule transcription factors. Proceedings of the National Academy of Sciences of the United States of America. 97: 3930-5. PMID 10760265 DOI: 10.1073/Pnas.97.8.3930  0.66
2000 Mapp AK, Dervan PB. Preparation of thioesters for the ligation of peptides with non-native substrates Tetrahedron Letters. 41: 9451-9454. DOI: 10.1016/S0040-4039(00)01600-2  0.478
1999 Mapp AK, Heathcock CH. Total Synthesis of Myxalamide A. The Journal of Organic Chemistry. 64: 23-27. PMID 11674080 DOI: 10.1021/Jo9813742  0.472
1996 Marshall KA, Mapp AK, Heathcock CH. Synthesis of a 2,7-dioxatricyclo[4.2.1.03,8]nonane: A model study for possible application in a synthesis of dictyoxetane Journal of Organic Chemistry. 61: 9135-9145. DOI: 10.1021/Jo961680K  0.395
1996 Caron S, Stoermer D, Mapp AK, Heathcock CH. Total synthesis of zaragozic acid A (squalestatin S1). Synthesis of the relay compound Journal of Organic Chemistry. 61: 9126-9134. DOI: 10.1021/Jo961534E  0.427
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