Year |
Citation |
Score |
2017 |
Haney SL, Wills VS, Wiemer DF, Holstein SA. Recent Advances in the Development of Mammalian Geranylgeranyl Diphosphate Synthase Inhibitors. Molecules (Basel, Switzerland). 22. PMID 28555000 DOI: 10.3390/Molecules22060886 |
0.629 |
|
2017 |
Wills VS, Metzger JI, Allen C, Varney ML, Wiemer DF, Holstein SA. Bishomoisoprenoid triazole bisphosphonates as inhibitors of geranylgeranyl diphosphate synthase. Bioorganic & Medicinal Chemistry. PMID 28302510 DOI: 10.1016/J.Bmc.2017.02.066 |
0.626 |
|
2016 |
Matthiesen RA, Wills VS, Metzger JI, Holstein SA, Wiemer DF. Stereoselective Synthesis of Homoneryl and Homogeranyl Triazole Bisphosphonates. The Journal of Organic Chemistry. PMID 27648672 DOI: 10.1021/Acs.Joc.6B01693 |
0.633 |
|
2016 |
Wills VS, Zhou X, Allen C, Holstein SA, Wiemer DF. Stereocontrolled regeneration of olefins from epoxides. Tetrahedron Letters. 57: 1335-1337. PMID 26955189 DOI: 10.1016/J.Tetlet.2016.02.041 |
0.467 |
|
2016 |
Allen C, Metzger JI, Wills VS, Tong H, Kortagere S, Wiemer DF, Holstein SA. Synergistic Inhibition of Geranylgeranyl Diphosphate Synthase By a Mixture of Olefin Stereoisomers Blood. 128: 2320-2320. DOI: 10.1182/Blood.V128.22.2320.2320 |
0.671 |
|
2015 |
Wills VS, Allen C, Holstein SA, Wiemer DF. Potent Triazole Bisphosphonate Inhibitor of Geranylgeranyl Diphosphate Synthase. Acs Medicinal Chemistry Letters. 6: 1195-8. PMID 26713103 DOI: 10.1021/Acsmedchemlett.5B00334 |
0.603 |
|
2014 |
Zhou X, Ferree SD, Wills VS, Born EJ, Tong H, Wiemer DF, Holstein SA. Geranyl and neryl triazole bisphosphonates as inhibitors of geranylgeranyl diphosphate synthase. Bioorganic & Medicinal Chemistry. 22: 2791-8. PMID 24726306 DOI: 10.1016/J.Bmc.2014.03.014 |
0.665 |
|
2014 |
Wills VS, Allen C, Born EJ, Zhou X, Wiemer DF, Holstein SA. A Novel Class of Geranylgeranyl Diphosphate Synthase Inhibitors: Structure-Activity Relationships of Homoisoprenoid Triazoles in Myeloma Cells Blood. 124: 2156-2156. DOI: 10.1182/Blood.V124.21.2156.2156 |
0.666 |
|
2013 |
Ferree SD, Zhou X, Wills VS, Born EJ, Tong H, Wiemer DF, Holstein SA. Synthesis and Structure-Function Relationship Of Novel Triazole Phosphonates As Inhibitors Of Rab Geranylgeranyl Transferase Blood. 122: 4223-4223. DOI: 10.1182/Blood.V122.21.4223.4223 |
0.681 |
|
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