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Christopher D. Vanderwal - Publications

Affiliations: 
Chemistry University of California, Irvine, Irvine, CA 
Area:
Organic and Synthetic
Website:
http://www.faculty.uci.edu/profile.cfm?faculty_id=5265

93 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Niman SW, Buono R, Fruman DA, Vanderwal CD. Synthesis of a Complex Brasilicardin Analogue Utilizing a Cobalt-Catalyzed MHAT-Induced Radical Bicyclization Reaction. Organic Letters. PMID 37141632 DOI: 10.1021/acs.orglett.3c01019  0.406
2023 Chung J, Capani JS, Göhl M, Roosen PC, Vanderwal CD. Enantioselective Syntheses of Wickerols A and B. Journal of the American Chemical Society. 145: 6486-6497. PMID 36883956 DOI: 10.1021/jacs.3c00448  0.383
2023 Dwulet NC, Chahine Z, Le Roch KG, Vanderwal CD. An Enantiospecific Synthesis of Isoneoamphilectane Confirms Its Strained Tricyclic Structure. Journal of the American Chemical Society. 145: 3716-3726. PMID 36730688 DOI: 10.1021/jacs.2c13137  0.317
2022 Roosen PC, Karns AS, Ellis BD, Vanderwal CD. Evolution of a Short and Stereocontrolled Synthesis of (+)-7,20-Diisocyanoadociane. The Journal of Organic Chemistry. 87: 1398-1420. PMID 34990544 DOI: 10.1021/acs.joc.1c02700  0.386
2021 Dwulet NC, Ramella V, Vanderwal CD. Soft Enolization of 3-Substituted Cycloalkanones Exhibits Significantly Improved Regiocontrol vs Hard Enolization Conditions. Organic Letters. 23: 9616-9619. PMID 34870436 DOI: 10.1021/acs.orglett.1c03844  0.314
2021 Johnson LK, Niman SW, Vrubliauskas D, Vanderwal CD. Stereocontrolled Synthesis and Structural Revision of Plebeianiol A. Organic Letters. 23: 9569-9573. PMID 34851132 DOI: 10.1021/acs.orglett.1c03791  0.388
2021 Vrubliauskas D, Gross BM, Vanderwal CD. Stereocontrolled Radical Bicyclizations of Oxygenated Precursors Enable Short Syntheses of Oxidized Abietane Diterpenoids. Journal of the American Chemical Society. PMID 33555176 DOI: 10.1021/jacs.0c13300  0.322
2021 Pak BS, Supantanapong N, Vanderwal CD. The Recurring Roles of Chlorine in Synthetic and Biological Studies of the Lissoclimides. Accounts of Chemical Research. PMID 33544578 DOI: 10.1021/acs.accounts.0c00866  0.306
2020 Ramella V, Roosen PC, Vanderwal CD. Concise Formal Synthesis of the Pseudopterosins via Anionic Oxy-Cope/Transannular Michael Addition Cascade. Organic Letters. PMID 32077289 DOI: 10.1021/Acs.Orglett.0C00486  0.465
2020 Vrubliauskas D, Vanderwal CD. Cobalt-Catalyzed Hydrogen Atom Transfer Induces Bicyclizations that Tolerate Electron-rich and -deficient Intermediate Alkenes. Angewandte Chemie (International Ed. in English). PMID 31991035 DOI: 10.1002/Anie.202000252  0.375
2019 Karns AS, Ellis BD, Roosen PC, Chahine Z, Le Roch KG, Vanderwal CD. Concise Synthesis of the Antiplasmodial Isocyanoterpene 7,20-Diisocyanoadociane. Angewandte Chemie (International Ed. in English). PMID 31270921 DOI: 10.1002/Anie.201906834  0.484
2019 Michalak SE, Nam S, Kwon DM, Horne DA, Vanderwal CD. A Chlorine-Atom-Controlled Terminal-Epoxide-Initiated Bicyclization Cascade Enables a Synthesis of the Potent Cytotoxins Haterumaimides J and K. Journal of the American Chemical Society. PMID 31129963 DOI: 10.1021/Jacs.9B04702  0.447
2019 Balaguer FA, Mühlethaler T, Estévez-Gallego J, Calvo E, Giménez-Abián JF, Risinger AL, Sorensen EJ, Vanderwal CD, Altmann KH, Mooberry SL, Steinmetz MO, Oliva MÁ, Prota AE, Díaz JF. Crystal Structure of the Cyclostreptin-Tubulin Adduct: Implications for Tubulin Activation by Taxane-Site Ligands. International Journal of Molecular Sciences. 20. PMID 30897704 DOI: 10.3390/Ijms20061392  0.497
2019 Pellegrino S, Meyer M, Könst ZA, Holm M, Voora VK, Kashinskaya D, Zanette C, Mobley DL, Yusupova G, Vanderwal CD, Blanchard SC, Yusupov M. Understanding the role of intermolecular interactions between lissoclimides and the eukaryotic ribosome. Nucleic Acids Research. PMID 30759226 DOI: 10.1093/Nar/Gkz053  0.379
2018 Ellis BD, Milligan JC, White AR, Duong V, Altman PX, Mohammed L, Crump MP, Crosby J, Luo R, Vanderwal CD, Tsai SC. An Oxetane-based Polyketide Surrogate to Probe Substrate Binding in a Polyketide Synthase. Journal of the American Chemical Society. PMID 29620883 DOI: 10.1021/Jacs.7B11793  0.344
2017 Schwarzwalder GM, Vanderwal CD. Strategies for the Synthesis of the Halenaquinol and Xestoquinol Families of Natural Products. European Journal of Organic Chemistry. 2017: 1567-1577. PMID 29527124 DOI: 10.1002/Ejoc.201601418  0.399
2017 White AM, Dao K, Vrubliauskas D, Könst ZA, Pierens GK, Mandi A, Andrews KT, Skinner-Adams TS, Clarke ME, Narbutas PT, Sim DC, Cheney KL, Kurtan T, Garson MJ, Vanderwal CD. A Catalyst-controlled Stereoselective Synthesis Secures the Structure of the Antimalarial Isocyanoterpene Pustulosaisonitrile-1. The Journal of Organic Chemistry. PMID 29124922 DOI: 10.1021/Acs.Joc.7B02421  0.323
2017 Könst ZA, Szklarski AR, Pellegrino S, Michalak SE, Meyer M, Zanette C, Cencic R, Nam S, Voora VK, Horne DA, Pelletier J, Mobley DL, Yusupova G, Yusupov M, Vanderwal CD. Synthesis facilitates an understanding of the structural basis for translation inhibition by the lissoclimides. Nature Chemistry. 9: 1140-1149. PMID 29064494 DOI: 10.1038/Nchem.2800  0.783
2017 Ellis BD, Vanderwal CD. Hughes and Gleason's Virosaine A-Appreciating the Art in Synthesis. Angewandte Chemie (International Ed. in English). PMID 29024223 DOI: 10.1002/Anie.201708051  0.505
2017 Herzon SB, Vanderwal CD. Introduction: Natural Product Synthesis. Chemical Reviews. 117: 11649-11650. PMID 28950704 DOI: 10.1021/Acs.Chemrev.7B00520  0.46
2017 Hong AY, Vanderwal CD. A Sequential Cycloaddition Strategy for the Synthesis of Alsmaphorazine B Traces a Path Through a Family of Alstonia Alkaloids. Tetrahedron. 73: 4160-4171. PMID 28943664 DOI: 10.1016/J.Tet.2016.11.004  0.446
2017 White A, Kozlowski R, Tsai SC, Vanderwal CD. A Direct Synthesis of Highly Substituted π-Rich Aromatic Heterocycles from Oxetanes. Angewandte Chemie (International Ed. in English). PMID 28662280 DOI: 10.1002/Anie.201704119  0.546
2017 Daub ME, Roosen PC, Vanderwal CD. General Approaches to Structurally Diverse Isocyanoditerpenes. The Journal of Organic Chemistry. PMID 28402638 DOI: 10.1021/Acs.Joc.7B00448  0.325
2017 Daub ME, Prudhomme J, Ben Mamoun C, Le Roch KG, Vanderwal CD. Antimalarial Properties of Simplified Kalihinol Analogues. Acs Medicinal Chemistry Letters. 8: 355-360. PMID 28337330 DOI: 10.1021/Acsmedchemlett.7B00013  0.375
2017 Mai D, Uchenik D, Vanderwal C. Efforts Toward a Synthesis of Crotogoudin and Crotobarin Synlett. 28: 1758-1762. DOI: 10.1055/S-0036-1588560  0.473
2017 Ellis BD, Vanderwal CD. Virosain A nach Hughes und Gleason - die Kunst der Synthese Angewandte Chemie. 129: 14128-14130. DOI: 10.1002/Ange.201708051  0.316
2016 Schwarzwalder GM, Scott DR, Vanderwal CD. A Synthesis of Exiguaquinol Dessulfate. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27673578 DOI: 10.1002/Chem.201604506  0.431
2016 Roosen PC, Vanderwal CD. A Formal Enantiospecific Synthesis of 7,20-Diisocyanoadociane. Angewandte Chemie (International Ed. in English). PMID 27162155 DOI: 10.1002/Anie.201603581  0.519
2016 White AR, Duggan BM, Tsai SC, Vanderwal CD. The Alga Ochromonas danica Produces Bromosulfolipids. Organic Letters. PMID 26889956 DOI: 10.1021/Acs.Orglett.6B00230  0.301
2016 Horn EJ, Silverston JS, Vanderwal CD. A Failed Late-Stage Epimerization Thwarts an Approach to Ineleganolide. The Journal of Organic Chemistry. PMID 26863401 DOI: 10.1021/Acs.Joc.5B02550  0.656
2016 Chung WJ, Vanderwal CD. Stereoselective Halogenation in Natural Product Synthesis. Angewandte Chemie (International Ed. in English). PMID 26833878 DOI: 10.1002/Anie.201506388  0.638
2015 Quinn RK, Könst ZA, Michalak SE, Schmidt Y, Szklarski AR, Flores AR, Nam S, Horne DA, Vanderwal CD, Alexanian EJ. Site-Selective Aliphatic C-H Chlorination Using N-Chloroamides Enables a Synthesis of Chlorolissoclimide. Journal of the American Chemical Society. PMID 26694767 DOI: 10.1021/Jacs.5B12308  0.771
2015 Hong AY, Vanderwal CD. A Synthesis of Alsmaphorazine B Demonstrates the Chemical Feasibility of a New Biogenetic Hypothesis. Journal of the American Chemical Society. 137: 7306-9. PMID 26034815 DOI: 10.1021/Jacs.5B04686  0.393
2015 Pham HV, Karns AS, Vanderwal CD, Houk KN. Computational and experimental investigations of the formal dyotropic rearrangements of himbert arene/allene cycloadducts. Journal of the American Chemical Society. 137: 6956-64. PMID 25961134 DOI: 10.1021/Jacs.5B03718  0.444
2015 Daub ME, Prudhomme J, Le Roch K, Vanderwal CD. Synthesis and potent antimalarial activity of kalihinol B. Journal of the American Chemical Society. 137: 4912-5. PMID 25815413 DOI: 10.1021/Jacs.5B01152  0.383
2014 Atwood BR, Vanderwal CD. Synthetic methodology: catalytic control of chlorination. Nature Chemistry. 7: 99-100. PMID 25615661 DOI: 10.1038/Nchem.2163  0.405
2014 Vogel CV, Pietraszkiewicz H, Sabry OM, Gerwick WH, Valeriote FA, Vanderwal CD. Enantioselective divergent syntheses of several polyhalogenated Plocamium monoterpenes and evaluation of their selectivity for solid tumors. Angewandte Chemie (International Ed. in English). 53: 12205-9. PMID 25220828 DOI: 10.1002/Anie.201407726  0.42
2014 Roosen PC, Vanderwal CD. Investigations into an anionic oxy-cope/transannular conjugate addition approach to 7,20-diisocyanoadociane. Organic Letters. 16: 4368-71. PMID 25105694 DOI: 10.1021/Ol502205M  0.482
2014 Tartakoff SS, Vanderwal CD. A synthesis of the ABC tricyclic core of the clionastatins serves to corroborate their proposed structures. Organic Letters. 16: 1458-61. PMID 24571064 DOI: 10.1021/Ol500265V  0.511
2014 Chung WJ, Carlson JS, Vanderwal CD. General approach to the synthesis of the chlorosulfolipids danicalipin A, mytilipin A, and malhamensilipin A in enantioenriched form. The Journal of Organic Chemistry. 79: 2226-41. PMID 24494597 DOI: 10.1021/Jo5000829  0.663
2014 Chung WJ, Vanderwal CD. Approaches to the chemical synthesis of the chlorosulfolipids. Accounts of Chemical Research. 47: 718-28. PMID 24400674 DOI: 10.1021/Ar400246W  0.662
2014 Lam JK, Joseph SB, Vanderwal CD. A Zincke aldehyde approach to gelsemine Tetrahedron Letters. 56: 3165-3168. DOI: 10.1016/J.Tetlet.2014.12.089  0.649
2014 Chung W, Carlson JS, Vanderwal CD. ChemInform Abstract: General Approach to the Synthesis of the Chlorosulfolipids Danicalipin A (I), Mytilipin A (II), and Malhamensilipin A (III) in Enantioenriched Form. Cheminform. 45: no-no. DOI: 10.1002/chin.201434213  0.483
2013 Schwarzwalder GM, Steinhardt SE, Pham HV, Houk KN, Vanderwal CD. Synthesis of the tetracyclic core of exiguaquinol. Organic Letters. 15: 6014-7. PMID 24219829 DOI: 10.1021/Ol402905N  0.814
2013 Lam JK, Pham HV, Houk KN, Vanderwal CD. Computation and experiment reveal that the ring-rearrangement metathesis of Himbert cycloadducts can be subject to kinetic or thermodynamic control. Journal of the American Chemical Society. 135: 17585-94. PMID 24111571 DOI: 10.1021/Ja409618P  0.675
2013 Chung WJ, Carlson JS, Bedke DK, Vanderwal CD. A synthesis of the chlorosulfolipid mytilipin A via a longest linear sequence of seven steps. Angewandte Chemie (International Ed. in English). 52: 10052-5. PMID 23929596 DOI: 10.1002/Anie.201304565  0.624
2013 Schmidt Y, Lam JK, Pham HV, Houk KN, Vanderwal CD. Studies on the Himbert intramolecular arene/allene Diels-Alder cycloaddition. Mechanistic studies and expansion of scope to all-carbon tethers. Journal of the American Chemical Society. 135: 7339-48. PMID 23634642 DOI: 10.1021/Ja4025963  0.697
2012 Lam JK, Schmidt Y, Vanderwal CD. Complex polycyclic scaffolds by metathesis rearrangement of Himbert arene/allene cycloadducts. Organic Letters. 14: 5566-9. PMID 23067058 DOI: 10.1021/Ol302680M  0.702
2012 Michels TD, Dowling MS, Vanderwal CD. A synthesis of echinopine B. Angewandte Chemie (International Ed. in English). 51: 7572-6. PMID 22711188 DOI: 10.1002/Anie.201203147  0.765
2012 Pham HV, Martin DB, Vanderwal CD, Houk KN. The Intramolecular Diels-Alder Reaction of Tryptamine-Derived Zincke Aldehydes Is a Stepwise Process. Chemical Science (Royal Society of Chemistry : 2010). 2012: 1650-1655. PMID 22611483 DOI: 10.1039/C2Sc01072K  0.614
2012 Martin DB, Nguyen LQ, Vanderwal CD. Syntheses of strychnine, norfluorocurarine, dehydrodesacetylretuline, and valparicine enabled by intramolecular cycloadditions of Zincke aldehydes. The Journal of Organic Chemistry. 77: 17-46. PMID 22168233 DOI: 10.1021/Jo2020246  0.641
2012 Martin DBC, Vanderwal CD. A short synthesis of strychnine from pyridine Total Synthesis of Natural Products: At the Frontiers of Organic Chemistry. 2147483647: 67-102. DOI: 10.1007/978-3-642-34065-9_4  0.369
2011 Vanderwal CD. Reactivity and synthesis inspired by the Zincke ring-opening of pyridines. The Journal of Organic Chemistry. 76: 9555-67. PMID 21877712 DOI: 10.1021/Jo201625E  0.582
2011 Paton RS, Steinhardt SE, Vanderwal CD, Houk KN. Unraveling the mechanism of cascade reactions of zincke aldehydes. Journal of the American Chemical Society. 133: 3895-905. PMID 21351736 DOI: 10.1021/Ja107988B  0.786
2011 Bedke DK, Vanderwal CD. Chlorosulfolipids: structure, synthesis, and biological relevance. Natural Product Reports. 28: 15-25. PMID 21125121 DOI: 10.1039/C0Np00044B  0.362
2011 Martin DBC, Vanderwal CD. Synthesis of Strychnine Synfacts. 2011: 463-463. DOI: 10.1055/S-0030-1259793  0.494
2011 Martin DBC, Vanderwal CD. A synthesis of strychnine by a longest linear sequence of six steps Chemical Science. 2: 649-651. DOI: 10.1039/C1Sc00009H  0.482
2010 Steinhardt SE, Vanderwal CD. Synthetic strategy: without a trace. Nature Chemistry. 2: 254-6. PMID 21124503 DOI: 10.1038/Nchem.602  0.78
2010 Dowling MS, Vanderwal CD. Ring-closing metathesis of allylsilanes as a flexible strategy toward cyclic terpenes. short syntheses of teucladiol, isoteucladiol, poitediol, and dactylol and an attempted synthesis of caryophyllene. The Journal of Organic Chemistry. 75: 6908-22. PMID 20836562 DOI: 10.1021/Jo101439H  0.816
2010 Michels TD, Kier MJ, Kearney AM, Vanderwal CD. Concise formal synthesis of porothramycins A and B via Zincke pyridinium ring-opening/ring-closing cascade. Organic Letters. 12: 3093-5. PMID 20527899 DOI: 10.1021/Ol101035P  0.803
2010 Martin DB, Vanderwal CD. Concise synthesis of (-)-nakadomarin A. Angewandte Chemie (International Ed. in English). 49: 2830-2. PMID 20301158 DOI: 10.1002/Anie.201000045  0.596
2010 Bedke DK, Shibuya GM, Pereira AR, Gerwick WH, Vanderwal CD. A concise enantioselective synthesis of the chlorosulfolipid malhamensilipin A. Journal of the American Chemical Society. 132: 2542-3. PMID 20141139 DOI: 10.1021/Ja910809C  0.818
2010 Pereira AR, Byrum T, Shibuya GM, Vanderwal CD, Gerwick WH. Structure revision and absolute configuration of malhamensilipin A from the freshwater chrysophyte Poterioochromonas malhamensis. Journal of Natural Products. 73: 279-83. PMID 20099812 DOI: 10.1021/Np900672H  0.769
2010 Bedke DK, Shibuya GM, Pereira AR, Gerwick WH, Vanderwal CD. Enantioselective Synthesis of Malhamensilipin A Synfacts. 2010: 559-559. DOI: 10.1055/S-0029-1219700  0.509
2010 Martin DBC, Vanderwal CD. ChemInform Abstract: Concise Synthesis of (-)-Nakadomarin A. Cheminform. 41: no-no. DOI: 10.1002/chin.201029239  0.38
2010 Soenen DR, Vanderwal CD. ChemInform Abstract: Synthesis of Dialkyl Ether by Addition to Alkenes Cheminform. 41. DOI: 10.1002/chin.201015224  0.432
2010 Martin D, Vanderwal C. Kurze Synthese von (−)-Nakadomarin A Angewandte Chemie. 122: 2893-2895. DOI: 10.1002/Ange.201000045  0.427
2009 Dowling MS, Vanderwal CD. Ring-closing metathesis of allylsilanes/electrophilic desilylation to prepare exo-methylidenecycloalkanes. Short syntheses of teucladiol and poitediol. Journal of the American Chemical Society. 131: 15090-1. PMID 19788178 DOI: 10.1021/Ja906241W  0.794
2009 Steinhardt SE, Vanderwal CD. Complex polycyclic lactams from pericyclic cascade reactions of Zincke aldehydes. Journal of the American Chemical Society. 131: 7546-7. PMID 19449870 DOI: 10.1021/Ja902439F  0.825
2009 Bedke DK, Shibuya GM, Pereira A, Gerwick WH, Haines TH, Vanderwal CD. Relative stereochemistry determination and synthesis of the major chlorosulfolipid from Ochromonas danica. Journal of the American Chemical Society. 131: 7570-2. PMID 19445461 DOI: 10.1021/Ja902138W  0.8
2009 Martin DB, Vanderwal CD. Efficient access to the core of the Strychnos, Aspidosperma and Iboga alkaloids. A short synthesis of norfluorocurarine. Journal of the American Chemical Society. 131: 3472-3. PMID 19236094 DOI: 10.1021/Ja900640V  0.619
2009 Bedke DK, Vanderwal CD. Organic chemistry: Chlorine lends a helping hand. Nature. 457: 548-9. PMID 19177122 DOI: 10.1038/457548A  0.432
2009 Kanady JS, Nguyen JD, Ziller JW, Vanderwal CD. Synthesis and characterization of all four diastereomers of 3,4-dichloro-2-pentanol, motifs relevant to the chlorosulfolipids. The Journal of Organic Chemistry. 74: 2175-8. PMID 19161314 DOI: 10.1021/Jo802390E  0.58
2009 Michels TD, Rhee JU, Vanderwal CD. ChemInform Abstract: Synthesis of δ-Tributylstannyl-α,β,γ,δ-Unsaturated Aldehydes from Pyridines. Cheminform. 40. DOI: 10.1002/chin.200912184  0.769
2008 Michels TD, Rhee JU, Vanderwal CD. Synthesis of delta-tributylstannyl-alpha,beta,gamma,delta-unsaturated aldehydes from pyridines. Organic Letters. 10: 4787-90. PMID 18817407 DOI: 10.1021/Ol8020435  0.811
2008 Shibuya GM, Kanady JS, Vanderwal CD. Stereoselective dichlorination of allylic alcohol derivatives to access key stereochemical arrays of the chlorosulfolipids. Journal of the American Chemical Society. 130: 12514-8. PMID 18717563 DOI: 10.1021/Ja804167V  0.796
2008 Steinhardt SE, Silverston JS, Vanderwal CD. Stereocontrolled synthesis of Z-dienes via an unexpected pericyclic cascade rearrangement of 5-amino-2,4-pentadienals. Journal of the American Chemical Society. 130: 7560-1. PMID 18505251 DOI: 10.1021/Ja8028125  0.831
2008 Bai R, Vanderwal CD, Díaz JF, Hamel E. Interaction of a cyclostreptin analogue with the microtubule taxoid site: the covalent reaction rapidly follows binding. Journal of Natural Products. 71: 370-4. PMID 18298077 DOI: 10.1021/Np800056M  0.366
2008 Vanderwal CD, Jacobsen EN. ChemInform Abstract: Alk-2-enoic Acid Esters Cheminform. 39. DOI: 10.1002/chin.200849251  0.42
2008 Vanderwal CD, Jacobsen EN. ChemInform Abstract: Alk-2-enoic Acids Cheminform. 39. DOI: 10.1002/chin.200843262  0.393
2007 Buey RM, Calvo E, Barasoain I, Pineda O, Edler MC, Matesanz R, Cerezo G, Vanderwal CD, Day BW, Sorensen EJ, López JA, Andreu JM, Hamel E, Díaz JF. Cyclostreptin binds covalently to microtubule pores and lumenal taxoid binding sites. Nature Chemical Biology. 3: 117-25. PMID 17206139 DOI: 10.1038/Nchembio853  0.502
2006 Kearney AM, Vanderwal CD. Synthesis of nitrogen heterocycles by the ring opening of pyridinium salts. Angewandte Chemie (International Ed. in English). 45: 7803-6. PMID 17072923 DOI: 10.1002/Anie.200602996  0.472
2006 Edler MC, Buey RM, Gussio R, Marcus AI, Vanderwal CD, Sorensen EJ, Díaz JF, Giannakakou P, Hamel E. Erratum: Cyclostreptin (FR182877), an antitumor tubulin-polymerizing agent deficient in enhancing tubulin assembly despite its high affinity for the taxoid site (Biochemistry (August 30, 2005) 44, 34 (11525-11538)) Biochemistry. 45. DOI: 10.1021/Bi068009M  0.489
2005 Edler MC, Buey RM, Gussio R, Marcus AI, Vanderwal CD, Sorensen EJ, Díaz JF, Giannakakou P, Hamel E. Cyclostreptin (FR182877), an antitumor tubulin-polymerizing agent deficient in enhancing tubulin assembly despite its high affinity for the taxoid site. Biochemistry. 44: 11525-38. PMID 16114889 DOI: 10.1021/Bi050660M  0.526
2004 Vanderwal CD, Jacobsen EN. Enantioselective formal hydration of alpha,beta-unsaturated imides by Al-catalyzed conjugate addition of oxime nucleophiles. Journal of the American Chemical Society. 126: 14724-5. PMID 15535689 DOI: 10.1021/Ja045563F  0.593
2004 Vanderwal CD, Sorensen EJ. Chapter 1 A remarkable architectural self-construction process is discovered in a synthesis of FR182877 Strategies and Tactics in Organic Synthesis. 5: 1-50. DOI: 10.1016/S1874-6004(04)80024-8  0.6
2003 Adam GC, Vanderwal CD, Sorensen EJ, Cravatt BF. (-)-FR182877 is a potent and selective inhibitor of carboxylesterase-1. Angewandte Chemie (International Ed. in English). 42: 5480-4. PMID 14618582 DOI: 10.1002/Anie.200352576  0.498
2003 Vanderwal CD, Vosburg DA, Weiler S, Sorensen EJ. An enantioselective synthesis of FR182877 provides a chemical rationalization of its structure and affords multigram quantities of its direct precursor. Journal of the American Chemical Society. 125: 5393-407. PMID 12720453 DOI: 10.1021/Ja021472B  0.813
2002 Vosburg DA, Vanderwal CD, Sorensen EJ. A synthesis of (+)-FR182877, featuring tandem transannular Diels-Alder reactions inspired by a postulated biogenesis. Journal of the American Chemical Society. 124: 4552-3. PMID 11971689 DOI: 10.1021/Ja025885O  0.818
2001 Vanderwal CD, Vosburg DA, Sorensen EJ. Intramolecular allenolate acylations in studies toward a synthesis of FR182877. Organic Letters. 3: 4307-10. PMID 11784204 DOI: 10.1021/Ol016994V  0.816
2001 Vanderwal CD, Vosburg DA, Sorensen EJ. Intramolecular allenolate acylations in studies toward a synthesis of FR182877 Organic Letters. 3: 4307-4310. DOI: 10.1021/ol016994v  0.801
1999 Vanderwal CD, Vosburg DA, Weiler S, Sorensen EJ. Postulated biogenesis of WS9885B and progress toward an enantioselective synthesis. Organic Letters. 1: 645-8. PMID 10823194 DOI: 10.1021/Ol990723R  0.782
1996 Friesen RW, Vanderwal C. Total synthesis of (±)-dihydrokawain-5-ol. Regioselective monoprotection of vicinal syn-diols derived from the iodocyclofunctionalization of α-allenic alcohols Journal of Organic Chemistry. 61: 9103-9110. DOI: 10.1021/Jo961653U  0.322
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