| Year |
Citation |
Score |
| 2022 |
Gannam ZTK, Jamali H, Kweon OS, Herrington J, Shillingford SR, Papini C, Gentzel E, Lolis E, Bennett AM, Ellman JA, Anderson KS. Defining the structure-activity relationship for a novel class of allosteric MKP5 inhibitors. European Journal of Medicinal Chemistry. 243: 114712. PMID 36116232 DOI: 10.1016/j.ejmech.2022.114712 |
0.663 |
|
| 2020 |
Gannam ZTK, Min K, Shillingford SR, Zhang L, Herrington J, Abriola L, Gareiss PC, Pantouris G, Tzouvelekis A, Kaminski N, Zhang X, Yu J, Jamali H, Ellman JA, Lolis E, et al. An allosteric site on MKP5 reveals a strategy for small-molecule inhibition. Science Signaling. 13. PMID 32843541 DOI: 10.1126/Scisignal.Aba3043 |
0.605 |
|
| 2018 |
Tjin CC, Wissner RF, Jamali H, Schepartz A, Ellman JA. Synthesis and Biological Evaluation of an Indazole-Based Selective Protein Arginine Deiminase 4 (PAD4) Inhibitor. Acs Medicinal Chemistry Letters. 9: 1013-1018. PMID 30344909 DOI: 10.1021/Acsmedchemlett.8B00283 |
0.606 |
|
| 2016 |
Jamali H, Khan HA, Tjin CC, Ellman JA. Cellular Activity of New Small Molecule Protein Arginine Deiminase 3 (PAD3) Inhibitors. Acs Medicinal Chemistry Letters. 7: 847-51. PMID 27660689 DOI: 10.1021/Acsmedchemlett.6B00215 |
0.575 |
|
| 2016 |
Wilson DL, Meininger I, Strater Z, Steiner S, Tomlin F, Wu J, Jamali H, Krappmann D, Götz MG. Synthesis and Evaluation of Macrocyclic Peptide Aldehydes as Potent and Selective Inhibitors of the 20S Proteasome. Acs Medicinal Chemistry Letters. 7: 250-5. PMID 26985310 DOI: 10.1021/acsmedchemlett.5b00401 |
0.476 |
|
| 2015 |
Jamali H, Khan HA, Stringer JR, Chowdhury S, Ellman JA. Identification of multiple structurally distinct, nonpeptidic small molecule inhibitors of protein arginine deiminase 3 using a substrate-based fragment method. Journal of the American Chemical Society. 137: 3616-21. PMID 25742366 DOI: 10.1021/Jacs.5B00095 |
0.661 |
|
| Show low-probability matches. |